acea 1011 has been researched along with licostinel in 4 studies
Studies (acea 1011) | Trials (acea 1011) | Recent Studies (post-2010) (acea 1011) | Studies (licostinel) | Trials (licostinel) | Recent Studies (post-2010) (licostinel) |
---|---|---|---|---|---|
12 | 0 | 1 | 49 | 1 | 0 |
Protein | Taxonomy | acea 1011 (IC50) | licostinel (IC50) |
---|---|---|---|
Glutamate receptor ionotropic, NMDA 2D | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 3B | Homo sapiens (human) | 0.0059 | |
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | 0.766 | |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.766 | |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | 0.766 | |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | 0.766 | |
Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 1 | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 2A | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 2B | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 2C | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 2D | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 3A | Homo sapiens (human) | 0.0059 | |
Glutamate receptor ionotropic, NMDA 3B | Rattus norvegicus (Norway rat) | 0.0068 | |
Glutamate receptor ionotropic, NMDA 3A | Rattus norvegicus (Norway rat) | 0.0068 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cai, SX; Dinsmore, CM; Glenn, AG; Guastella, J; Huang, JC; Ilyin, V; Keana, JF; Kher, SM; Lü, Y; Mouser, PL | 1 |
Matsumoto, RR; Nguyen, D; Truong, DD | 1 |
Keana, JF; Ludwig, P; Martin, H; McAllister, A; Warner, DS; Weber, E | 1 |
Balster, RL; Compton, AD; Holcomb, JD; McCallum, SE; Porter, JH; Varvel, SA; Wiley, JL | 1 |
4 other study(ies) available for acea 1011 and licostinel
Article | Year |
---|---|
Synthesis and structure-activity relationships of substituted 1,4-dihydroquinoxaline-2,3-diones: antagonists of N-methyl-D-aspartate (NMDA) receptor glycine sites and non-NMDA glutamate receptors.
Topics: Animals; Excitatory Amino Acid Antagonists; Magnetic Resonance Spectroscopy; Membrane Potentials; Oocytes; Quinoxalines; Rats; Receptors, Glutamate; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Xenopus | 1995 |
Strychnine-insensitive glycine site antagonists attenuate a cardiac arrest-induced movement disorder.
Topics: Animals; Anticonvulsants; Behavior, Animal; Cardiopulmonary Resuscitation; Central Nervous System; Dose-Response Relationship, Drug; Felbamate; Heart Arrest; Male; Myoclonus; Phenylcarbamates; Propylene Glycols; Pyrrolidinones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Stereoisomerism; Strychnine | 1995 |
In vivo models of cerebral ischemia: effects of parenterally administered NMDA receptor glycine site antagonists.
Topics: Animals; Brain Ischemia; Male; Nervous System; Neuroprotective Agents; Quinoxalines; Rats; Rats, Wistar; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate | 1995 |
Effects of modulation of NMDA neurotransmission on response rate and duration in a conflict procedure in rats.
Topics: 2-Amino-5-phosphonovalerate; Acetamides; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reward; Synaptic Transmission | 1998 |