Page last updated: 2024-09-03

acea 1011 and licostinel

acea 1011 has been researched along with licostinel in 4 studies

Compound Research Comparison

Studies
(acea 1011)
Trials
(acea 1011)
Recent Studies (post-2010)
(acea 1011)
Studies
(licostinel)
Trials
(licostinel)
Recent Studies (post-2010) (licostinel)
12014910

Protein Interaction Comparison

ProteinTaxonomyacea 1011 (IC50)licostinel (IC50)
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.0059
Glutamate receptor 1Rattus norvegicus (Norway rat)0.766
Glutamate receptor 2Rattus norvegicus (Norway rat)0.766
Glutamate receptor 3Rattus norvegicus (Norway rat)0.766
Glutamate receptor 4Rattus norvegicus (Norway rat)0.766
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.0068

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cai, SX; Dinsmore, CM; Glenn, AG; Guastella, J; Huang, JC; Ilyin, V; Keana, JF; Kher, SM; Lü, Y; Mouser, PL1
Matsumoto, RR; Nguyen, D; Truong, DD1
Keana, JF; Ludwig, P; Martin, H; McAllister, A; Warner, DS; Weber, E1
Balster, RL; Compton, AD; Holcomb, JD; McCallum, SE; Porter, JH; Varvel, SA; Wiley, JL1

Other Studies

4 other study(ies) available for acea 1011 and licostinel

ArticleYear
Synthesis and structure-activity relationships of substituted 1,4-dihydroquinoxaline-2,3-diones: antagonists of N-methyl-D-aspartate (NMDA) receptor glycine sites and non-NMDA glutamate receptors.
    Journal of medicinal chemistry, 1995, Oct-27, Volume: 38, Issue:22

    Topics: Animals; Excitatory Amino Acid Antagonists; Magnetic Resonance Spectroscopy; Membrane Potentials; Oocytes; Quinoxalines; Rats; Receptors, Glutamate; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Xenopus

1995
Strychnine-insensitive glycine site antagonists attenuate a cardiac arrest-induced movement disorder.
    European journal of pharmacology, 1995, Mar-06, Volume: 275, Issue:2

    Topics: Animals; Anticonvulsants; Behavior, Animal; Cardiopulmonary Resuscitation; Central Nervous System; Dose-Response Relationship, Drug; Felbamate; Heart Arrest; Male; Myoclonus; Phenylcarbamates; Propylene Glycols; Pyrrolidinones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Stereoisomerism; Strychnine

1995
In vivo models of cerebral ischemia: effects of parenterally administered NMDA receptor glycine site antagonists.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1995, Volume: 15, Issue:2

    Topics: Animals; Brain Ischemia; Male; Nervous System; Neuroprotective Agents; Quinoxalines; Rats; Rats, Wistar; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1995
Effects of modulation of NMDA neurotransmission on response rate and duration in a conflict procedure in rats.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 2-Amino-5-phosphonovalerate; Acetamides; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reward; Synaptic Transmission

1998