aa 861 and calcimycin
aa 861 has been researched along with calcimycin in 17 studies
Research
Studies (17)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 12 (70.59) | 18.7374 |
1990's | 4 (23.53) | 18.2507 |
2000's | 1 (5.88) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Kanamaru, K; Matsumoto, T; Murata, Y; Sugiyama, Y | 1 |
Boot, JR; Edwards, D; Herbert, CA; Robinson, C | 1 |
Adachi, H; Aoki, E; Honda, T; Noguchi, M; Onishi, S; Sato, S; Torizuka, K | 1 |
Kohno, SW; Nanbu, F; Negi, H; Ohata, K; Taira, M; Yamamura, H | 1 |
Bonta, IL; Elliott, GR; van Hilten, JA | 2 |
Fujimoto, K; Itoh, H; Kanamaru, K; Kubo, Y; Waga, S | 1 |
Kobayashi, K; Mizoguchi, Y; Morisawa, S; Sakagami, Y; Seki, S; Yamamoto, S | 2 |
Colombo, C; Dotson, R; Ghai, G; Kimble, EF; Ku, EC; Lee, WH; Oglesby, TD; Raychaudhuri, A; Wasley, JW | 1 |
Schulz, R; Seeger, W | 1 |
Niwa, Y; Ohashi, T; Ozaki, Y | 1 |
Mita, H; Shida, T; Yui, Y | 1 |
Hirai, A; Saito, H; Tamura, Y; Yoshida, S | 1 |
Fujimoto, K; Kobayashi, T; Kubo, K; Matsuzawa, Y; Okada, K; Shinozaki, S; Sugane, K | 1 |
Bye, A; Robinson, C; Summers, JA | 1 |
Other Studies
17 other study(ies) available for aa 861 and calcimycin
Article | Year |
---|---|
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Endothelium-derived relaxation of the pregnant and nonpregnant canine uterine artery.
Topics: Acetylcholine; Animals; Benzoquinones; Calcimycin; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Evaluation Studies as Topic; Female; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Nitric Oxide; Pregnancy; Pregnancy, Animal; Uterus; Vasoconstriction | 1992 |
In vitro modulation of the eosinophil-dependent enhancement of the permeability of the bronchial mucosa.
Topics: Animals; Benzoquinones; Bronchi; Calcimycin; Cattle; Culture Techniques; Cytochalasin B; Diffusion Chambers, Culture; Dimethyl Sulfoxide; Eosinophils; Guinea Pigs; Lipoxygenase Inhibitors; Male; Mucous Membrane; Neutrophils; Permeability; Radioimmunoassay; Serum Albumin, Bovine | 1991 |
Effect of AA861, a 5-lipoxygenase inhibitor, on amylase secretion from rat pancreatic acini.
Topics: Amylases; Animals; Arachidonate Lipoxygenases; Benzoquinones; Bombesin; Calcimycin; Carbachol; Cholecystokinin; In Vitro Techniques; Indomethacin; Kinetics; Lipoxygenase Inhibitors; Male; Pancreas; Quinones; Rats; Rats, Inbred Strains; Sincalide; Tetradecanoylphorbol Acetate | 1988 |
Effect of AA-861, a selective 5-lipoxygenase inhibitor, on models of allergy in several species.
Topics: Animals; Asthma; Benzoquinones; Calcimycin; Chromatography, High Pressure Liquid; Female; Guinea Pigs; Histamine; Histamine Release; Hypersensitivity; Lipoxygenase Inhibitors; Macaca; Macaca mulatta; Male; Mites; Quinones; Radioimmunoassay; Rats; Rats, Inbred Strains; Species Specificity; SRS-A | 1988 |
Endogenous lipoxygenase metabolites mediate A23187 induced macrophage cytostasis towards P815 tumor cells in vitro.
Topics: Animals; Antineoplastic Agents; Benzoquinones; Calcimycin; Lipoxygenase; Lipoxygenase Inhibitors; Macrophage Activation; Masoprocol; Mice; Quinones; Tumor Cells, Cultured | 1989 |
Endothelium-dependent relaxation of human basilar arteries.
Topics: Acetylcholine; Adult; Aged; Basilar Artery; Benzoquinones; Calcimycin; Child; Child, Preschool; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Indomethacin; Lipoxygenase Inhibitors; Male; Middle Aged; Mixed Function Oxygenases; Muscle Contraction; Muscle Relaxation; Pyridines; Quinones | 1989 |
Release of leukotriene B4 from rat Kupffer cells.
Topics: Animals; Benzoquinones; Calcimycin; Cells, Cultured; Kupffer Cells; Leukotriene B4; Lipoxygenase Inhibitors; Male; Platelet Activating Factor; Quinones; Rats; Rats, Inbred Strains; Zymosan | 1989 |
Characterization of CGS 8515 as a selective 5-lipoxygenase inhibitor using in vitro and in vivo models.
Topics: Animals; Arachidonate Lipoxygenases; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Biotransformation; Blood Platelets; Calcimycin; Dexamethasone; Guinea Pigs; Humans; Hydroxyeicosatetraenoic Acids; Indomethacin; Leukocytes; Leukotriene B4; Lipoxygenase Inhibitors; Male; Naphthoquinones; ortho-Aminobenzoates; Pleurisy; Quinones; Rats; Rats, Inbred Strains; Sheep | 1988 |
Release of peptide leukotrienes from rat Kupffer cells.
Topics: Animals; Benzoquinones; Calcimycin; Kinetics; Kupffer Cells; Leukotriene E4; Lipoxygenase Inhibitors; Quinones; Rats; Rats, Inbred Strains; Reference Values; SRS-A | 1988 |
Release of leukotrienes into the perfusate of calcium-ionophore stimulated rabbit lungs. Influence of 5-lipoxygenase inhibitors.
Topics: 6-Ketoprostaglandin F1 alpha; Animals; Arachidonate Lipoxygenases; Aspirin; Benzoquinones; Blood Pressure; Calcimycin; Dose-Response Relationship, Drug; Epoprostenol; Leukotriene B4; Lipoxygenase Inhibitors; Lung; Perfusion; Pulmonary Artery; Quinones; Rabbits; Secretory Rate; SRS-A | 1986 |
A comparative study on the effects of inhibitors of the lipoxygenase pathway on neutrophil function. Inhibitory effects on neutrophil function may not be attributed to inhibition of the lipoxygenase pathway.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Benzoquinones; Calcimycin; Chemotaxis, Leukocyte; Epoprostenol; Humans; Hydroxides; Hydroxyl Radical; Leukotriene B4; Lipoxygenase Inhibitors; Masoprocol; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases A; Phospholipases A2; Platelet Activating Factor; Quinones; Tetradecanoylphorbol Acetate; Umbelliferones | 1986 |
Effect of AA-861, a 5-lipoxygenase inhibitor, on leukotriene synthesis in human polymorphonuclear leukocytes and on cyclooxygenase and 12-lipoxygenase activities in human platelets.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Blood Platelets; Calcimycin; Diethylcarbamazine; Humans; Leukotriene B4; Lipoxygenase Inhibitors; Neutrophils; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Quinones; SRS-A | 1986 |
Specific lipoxygenase inhibition reverses macrophage cytotasis towards P815 tumor cells in vitro induced by the calcium ionophore A23187.
Topics: Animals; Arachidonate Lipoxygenases; Benzoquinones; Calcimycin; Cytotoxicity, Immunologic; Female; Lipoxygenase Inhibitors; Macrophages; Masoprocol; Mice; Mice, Inbred BALB C; Neoplasms, Experimental; Quinones | 1988 |
The 5-lipoxygenase products can modulate the synthesis of platelet-activating factor (alkyl-acetyl GPC) in Ca-ionophore A23187-stimulated rat peritoneal macrophages.
Topics: Acetophenones; Animals; Arachidonic Acids; Benzoquinones; Calcimycin; Carbon Radioisotopes; Dose-Response Relationship, Drug; Hydroxyeicosatetraenoic Acids; In Vitro Techniques; Leukotrienes; Lipid Peroxides; Macrophages; Male; Platelet Activating Factor; Quinones; Rats; Rats, Inbred Strains | 1985 |
Neutrophil elastase inhibitor reduces asthmatic responses in allergic sheep.
Topics: Airway Resistance; Animals; Antigens; Asthma; Benzoquinones; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Calcimycin; Glycine; Heterocyclic Compounds; Leukocyte Elastase; Leukocytes; Leukotriene B4; Masoprocol; Methacholine Chloride; Pancreatic Elastase; Polycyclic Compounds; Sheep; Sulfonamides; Thromboxane B2 | 1995 |
Lipoxygenase inhibitory activity of U-66,858 and its deacetylated metabolite U-68,244 in human whole blood.
Topics: Adult; Benzoquinones; Calcimycin; Female; Humans; Leukotriene B4; Lipoxygenase Inhibitors; Male; Naphthols; Thromboxane A2; Thromboxane B2 | 1994 |