aa 861 and calcimycin

aa 861 has been researched along with calcimycin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199012 (70.59)18.7374
1990's4 (23.53)18.2507
2000's1 (5.88)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Kanamaru, K; Matsumoto, T; Murata, Y; Sugiyama, Y1
Boot, JR; Edwards, D; Herbert, CA; Robinson, C1
Adachi, H; Aoki, E; Honda, T; Noguchi, M; Onishi, S; Sato, S; Torizuka, K1
Kohno, SW; Nanbu, F; Negi, H; Ohata, K; Taira, M; Yamamura, H1
Bonta, IL; Elliott, GR; van Hilten, JA2
Fujimoto, K; Itoh, H; Kanamaru, K; Kubo, Y; Waga, S1
Kobayashi, K; Mizoguchi, Y; Morisawa, S; Sakagami, Y; Seki, S; Yamamoto, S2
Colombo, C; Dotson, R; Ghai, G; Kimble, EF; Ku, EC; Lee, WH; Oglesby, TD; Raychaudhuri, A; Wasley, JW1
Schulz, R; Seeger, W1
Niwa, Y; Ohashi, T; Ozaki, Y1
Mita, H; Shida, T; Yui, Y1
Hirai, A; Saito, H; Tamura, Y; Yoshida, S1
Fujimoto, K; Kobayashi, T; Kubo, K; Matsuzawa, Y; Okada, K; Shinozaki, S; Sugane, K1
Bye, A; Robinson, C; Summers, JA1

Other Studies

17 other study(ies) available for aa 861 and calcimycin

ArticleYear
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Endothelium-derived relaxation of the pregnant and nonpregnant canine uterine artery.
    The Journal of reproductive medicine, 1992, Volume: 37, Issue:6

    Topics: Acetylcholine; Animals; Benzoquinones; Calcimycin; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Evaluation Studies as Topic; Female; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Nitric Oxide; Pregnancy; Pregnancy, Animal; Uterus; Vasoconstriction

1992
In vitro modulation of the eosinophil-dependent enhancement of the permeability of the bronchial mucosa.
    British journal of pharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Benzoquinones; Bronchi; Calcimycin; Cattle; Culture Techniques; Cytochalasin B; Diffusion Chambers, Culture; Dimethyl Sulfoxide; Eosinophils; Guinea Pigs; Lipoxygenase Inhibitors; Male; Mucous Membrane; Neutrophils; Permeability; Radioimmunoassay; Serum Albumin, Bovine

1991
Effect of AA861, a 5-lipoxygenase inhibitor, on amylase secretion from rat pancreatic acini.
    Biochimica et biophysica acta, 1988, Jan-18, Volume: 968, Issue:1

    Topics: Amylases; Animals; Arachidonate Lipoxygenases; Benzoquinones; Bombesin; Calcimycin; Carbachol; Cholecystokinin; In Vitro Techniques; Indomethacin; Kinetics; Lipoxygenase Inhibitors; Male; Pancreas; Quinones; Rats; Rats, Inbred Strains; Sincalide; Tetradecanoylphorbol Acetate

1988
Effect of AA-861, a selective 5-lipoxygenase inhibitor, on models of allergy in several species.
    Japanese journal of pharmacology, 1988, Volume: 47, Issue:3

    Topics: Animals; Asthma; Benzoquinones; Calcimycin; Chromatography, High Pressure Liquid; Female; Guinea Pigs; Histamine; Histamine Release; Hypersensitivity; Lipoxygenase Inhibitors; Macaca; Macaca mulatta; Male; Mites; Quinones; Radioimmunoassay; Rats; Rats, Inbred Strains; Species Specificity; SRS-A

1988
Endogenous lipoxygenase metabolites mediate A23187 induced macrophage cytostasis towards P815 tumor cells in vitro.
    Agents and actions, 1989, Volume: 26, Issue:1-2

    Topics: Animals; Antineoplastic Agents; Benzoquinones; Calcimycin; Lipoxygenase; Lipoxygenase Inhibitors; Macrophage Activation; Masoprocol; Mice; Quinones; Tumor Cells, Cultured

1989
Endothelium-dependent relaxation of human basilar arteries.
    Stroke, 1989, Volume: 20, Issue:9

    Topics: Acetylcholine; Adult; Aged; Basilar Artery; Benzoquinones; Calcimycin; Child; Child, Preschool; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Indomethacin; Lipoxygenase Inhibitors; Male; Middle Aged; Mixed Function Oxygenases; Muscle Contraction; Muscle Relaxation; Pyridines; Quinones

1989
Release of leukotriene B4 from rat Kupffer cells.
    Prostaglandins, leukotrienes, and essential fatty acids, 1989, Volume: 36, Issue:3

    Topics: Animals; Benzoquinones; Calcimycin; Cells, Cultured; Kupffer Cells; Leukotriene B4; Lipoxygenase Inhibitors; Male; Platelet Activating Factor; Quinones; Rats; Rats, Inbred Strains; Zymosan

1989
Characterization of CGS 8515 as a selective 5-lipoxygenase inhibitor using in vitro and in vivo models.
    Biochimica et biophysica acta, 1988, Apr-15, Volume: 959, Issue:3

    Topics: Animals; Arachidonate Lipoxygenases; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Biotransformation; Blood Platelets; Calcimycin; Dexamethasone; Guinea Pigs; Humans; Hydroxyeicosatetraenoic Acids; Indomethacin; Leukocytes; Leukotriene B4; Lipoxygenase Inhibitors; Male; Naphthoquinones; ortho-Aminobenzoates; Pleurisy; Quinones; Rats; Rats, Inbred Strains; Sheep

1988
Release of peptide leukotrienes from rat Kupffer cells.
    Biochemical and biophysical research communications, 1988, Oct-14, Volume: 156, Issue:1

    Topics: Animals; Benzoquinones; Calcimycin; Kinetics; Kupffer Cells; Leukotriene E4; Lipoxygenase Inhibitors; Quinones; Rats; Rats, Inbred Strains; Reference Values; SRS-A

1988
Release of leukotrienes into the perfusate of calcium-ionophore stimulated rabbit lungs. Influence of 5-lipoxygenase inhibitors.
    Biochemical pharmacology, 1986, Jan-15, Volume: 35, Issue:2

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Arachidonate Lipoxygenases; Aspirin; Benzoquinones; Blood Pressure; Calcimycin; Dose-Response Relationship, Drug; Epoprostenol; Leukotriene B4; Lipoxygenase Inhibitors; Lung; Perfusion; Pulmonary Artery; Quinones; Rabbits; Secretory Rate; SRS-A

1986
A comparative study on the effects of inhibitors of the lipoxygenase pathway on neutrophil function. Inhibitory effects on neutrophil function may not be attributed to inhibition of the lipoxygenase pathway.
    Biochemical pharmacology, 1986, Oct-15, Volume: 35, Issue:20

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Benzoquinones; Calcimycin; Chemotaxis, Leukocyte; Epoprostenol; Humans; Hydroxides; Hydroxyl Radical; Leukotriene B4; Lipoxygenase Inhibitors; Masoprocol; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases A; Phospholipases A2; Platelet Activating Factor; Quinones; Tetradecanoylphorbol Acetate; Umbelliferones

1986
Effect of AA-861, a 5-lipoxygenase inhibitor, on leukotriene synthesis in human polymorphonuclear leukocytes and on cyclooxygenase and 12-lipoxygenase activities in human platelets.
    Allergy, 1986, Volume: 41, Issue:7

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Arachidonic Acids; Benzoquinones; Blood Platelets; Calcimycin; Diethylcarbamazine; Humans; Leukotriene B4; Lipoxygenase Inhibitors; Neutrophils; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Quinones; SRS-A

1986
Specific lipoxygenase inhibition reverses macrophage cytotasis towards P815 tumor cells in vitro induced by the calcium ionophore A23187.
    Prostaglandins, leukotrienes, and essential fatty acids, 1988, Volume: 34, Issue:3

    Topics: Animals; Arachidonate Lipoxygenases; Benzoquinones; Calcimycin; Cytotoxicity, Immunologic; Female; Lipoxygenase Inhibitors; Macrophages; Masoprocol; Mice; Mice, Inbred BALB C; Neoplasms, Experimental; Quinones

1988
The 5-lipoxygenase products can modulate the synthesis of platelet-activating factor (alkyl-acetyl GPC) in Ca-ionophore A23187-stimulated rat peritoneal macrophages.
    Prostaglandins, leukotrienes, and medicine, 1985, Volume: 18, Issue:3

    Topics: Acetophenones; Animals; Arachidonic Acids; Benzoquinones; Calcimycin; Carbon Radioisotopes; Dose-Response Relationship, Drug; Hydroxyeicosatetraenoic Acids; In Vitro Techniques; Leukotrienes; Lipid Peroxides; Macrophages; Male; Platelet Activating Factor; Quinones; Rats; Rats, Inbred Strains

1985
Neutrophil elastase inhibitor reduces asthmatic responses in allergic sheep.
    Respiration physiology, 1995, Volume: 100, Issue:1

    Topics: Airway Resistance; Animals; Antigens; Asthma; Benzoquinones; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Calcimycin; Glycine; Heterocyclic Compounds; Leukocyte Elastase; Leukocytes; Leukotriene B4; Masoprocol; Methacholine Chloride; Pancreatic Elastase; Polycyclic Compounds; Sheep; Sulfonamides; Thromboxane B2

1995
Lipoxygenase inhibitory activity of U-66,858 and its deacetylated metabolite U-68,244 in human whole blood.
    Agents and actions, 1994, Volume: 41, Issue:1-2

    Topics: Adult; Benzoquinones; Calcimycin; Female; Humans; Leukotriene B4; Lipoxygenase Inhibitors; Male; Naphthols; Thromboxane A2; Thromboxane B2

1994
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