Page last updated: 2024-09-03

a 71623 and sincalide

a 71623 has been researched along with sincalide in 10 studies

Compound Research Comparison

Studies
(a 71623)
Trials
(a 71623)
Recent Studies (post-2010)
(a 71623)
Studies
(sincalide)
Trials
(sincalide)
Recent Studies (post-2010) (sincalide)
27024,01572533

Protein Interaction Comparison

ProteinTaxonomya 71623 (IC50)sincalide (IC50)
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.0006
Cholecystokinin receptor type AHomo sapiens (human)0.0006
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.001
Gastrin/cholecystokinin type B receptorMus musculus (house mouse)0.0008
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.0004

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (70.00)18.2507
2000's2 (20.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Comstock, JM; Julien, R; Kaiser, F; Pierson, ME; Rosamond, JD; Simmons, RD1
Figlewicz, DP; Green, PK; Liddle, RA; Nadzan, AM; Porte, D; Sipols, AJ; Woods, SC1
Asin, KE; Bednarz, L; Craig, R; Cullen, MJ; Gore, PA; Montana, WE; Nadzan, AM; Nikkel, AL; Shiosaki, K1
Buéno, L; Gué, M; Junien, JL; Tabis, N; Tekamp, A1
Bell, RH; Longnecker, DS; Povoski, SP; Roebuck, BD; Zhou, W2
Bianchi, BR; Lin, CW; Miller, TR; Witte, DG1
Giralt, M; Vergara, P2
Bouali-Benazzouz, R; Covita, J; Egron, K; Favereaux, A; Fossat, P; Gundlach, AL; Landry, M; López-González, MJ; Ma, S; Roca-Lapirot, O; Trigilio, G1

Other Studies

10 other study(ies) available for a 71623 and sincalide

ArticleYear
CCK peptides with combined features of hexa- and tetrapeptide CCK-A agonists.
    Journal of medicinal chemistry, 2000, Jun-15, Volume: 43, Issue:12

    Topics: Animals; Appetite Depressants; Binding, Competitive; Body Weight; Cerebral Cortex; Eating; In Vitro Techniques; Male; Oligopeptides; Pancreas; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Structure-Activity Relationship; Synaptosomes

2000
Intraventricular CCK-8 reduces single meal size in the baboon by interaction with type-A CCK receptors.
    The American journal of physiology, 1992, Volume: 263, Issue:4 Pt 2

    Topics: Animals; Blood Glucose; Cholecystokinin; Eating; Fasting; Injections, Intraventricular; Insulin; Male; Oligopeptides; Papio; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1992
Behavioral effects of A71623, a highly selective CCK-A agonist tetrapeptide.
    The American journal of physiology, 1992, Volume: 263, Issue:1 Pt 2

    Topics: Animals; Anorexia; Behavior, Animal; Body Weight; Cholecystokinin; Circadian Rhythm; Eating; Food Deprivation; Male; Motor Activity; Peptides; Rats; Rats, Inbred Strains; Sincalide; Tetragastrin; Time Factors

1992
Cholecystokinin blockade of emotional stress- and CRF-induced colonic motor alterations in rats: role of the amygdala.
    Brain research, 1994, Sep-26, Volume: 658, Issue:1-2

    Topics: Amygdala; Animals; Colon; Corticotropin-Releasing Hormone; Gastrointestinal Motility; Ibotenic Acid; Injections, Intraventricular; Male; Oligopeptides; Rats; Rats, Wistar; Sincalide; Stress, Psychological; Tetragastrin

1994
Growth of azaserine-induced putative preneoplastic nodules in the rat pancreas is mediated specifically by way of cholecystokinin-A receptors.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Animals; Azaserine; Carcinogens; Cell Division; Cholecystokinin; Male; Pancreas; Pancreatic Neoplasms; Peptide Fragments; Precancerous Conditions; Rats; Rats, Inbred Lew; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1994
Stimulation of growth of azaserine-induced putative preneoplastic lesions in rat pancreas is mediated specifically by way of cholecystokinin-A receptors.
    Cancer research, 1993, Sep-01, Volume: 53, Issue:17

    Topics: Animals; Azaserine; Cholecystokinin; Chronic Disease; Male; Organ Size; Pancreas; Pancreatic Neoplasms; Pancreatitis; Peptide Fragments; Precancerous Conditions; Rats; Rats, Inbred Lew; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1993
Peripheral cholecystokinin type A receptors mediate oxytocin secretion in vivo.
    Regulatory peptides, 1993, Jan-22, Volume: 43, Issue:1-2

    Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Injections, Intraperitoneal; Male; Oligopeptides; Oxytocin; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1993
Both afferent and efferent nerves are implicated in cholecytokinin motor actions in the small intestine of the rat.
    Regulatory peptides, 1999, May-31, Volume: 81, Issue:1-3

    Topics: Anesthetics, Local; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Devazepide; Duodenum; Gastrins; Hexamethonium; Hormone Antagonists; Intestinal Mucosa; Intestine, Small; Jejunum; Lidocaine; Male; Neurons, Afferent; Neurons, Efferent; Nitroarginine; Oligopeptides; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Tetragastrin

1999
Inhibition by CCK of ascending contraction elicited by mucosal stimulation in the duodenum of the rat.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Atropine; Benzodiazepinones; Cholecystokinin; Depression, Chemical; Devazepide; Duodenum; Electric Stimulation; Enteric Nervous System; Enzyme Inhibitors; Gastrins; Hexamethonium; Intestinal Mucosa; Male; Muscle Contraction; Nicotinic Antagonists; Nitroarginine; Oligopeptides; Parasympatholytics; Peristalsis; Phentolamine; Phenylurea Compounds; Propranolol; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Receptors, Vasoactive Intestinal Peptide; Sincalide; Tetragastrin; Vasoactive Intestinal Peptide

2000
Acquisition of analgesic properties by the cholecystokinin (CCK)/CCK2 receptor system within the amygdala in a persistent inflammatory pain condition.
    Pain, 2019, Volume: 160, Issue:2

    Topics: Amygdala; Animals; Cholecystokinin; Dark Adaptation; Disease Models, Animal; Exploratory Behavior; Freund's Adjuvant; Gastrins; Glutamate Decarboxylase; Inflammation; Male; Neurons; Nociception; Pain; Pain Threshold; Periaqueductal Gray; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Signal Transduction; Sincalide; Tetragastrin

2019