Page last updated: 2024-09-03

a 68930 and quinpirole

a 68930 has been researched along with quinpirole in 6 studies

Compound Research Comparison

Studies
(a 68930)
Trials
(a 68930)
Recent Studies (post-2010)
(a 68930)
Studies
(quinpirole)
Trials
(quinpirole)
Recent Studies (post-2010) (quinpirole)
632192,2130367

Protein Interaction Comparison

ProteinTaxonomya 68930 (IC50)quinpirole (IC50)
D(2) dopamine receptorRattus norvegicus (Norway rat)0.1

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's0 (0.00)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Laiter, S; Mailman, RB; Mottola, DM; Nichols, DE; Tropsha, A; Watts, VJ; Wyrick, SD1
Bone, RG; Villar, HO1
Ahlenius, S; Karlsson, T; Salmi, P1
Ahlenius, S; Jimenez, P; Salmi, P1
Adachi, K; Hasegawa, M; Ikeda, H; Koshikawa, N; Nakamura, S; Waddington, JL1
Hamann, M; Lange, N; Richter, A; Shashidharan, P1

Other Studies

6 other study(ies) available for a 68930 and quinpirole

ArticleYear
Conformational analysis of D1 dopamine receptor agonists: pharmacophore assessment and receptor mapping.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Adenylyl Cyclases; Animals; Brain; Computer Simulation; Dopamine; Dopamine Agonists; Ligands; Molecular Conformation; Molecular Structure; Phenanthridines; Rats; Receptors, Dopamine D1; Software; Structure-Activity Relationship

1996
Discriminating D1 and D2 agonists with a hydrophobic similarity index.
    Journal of molecular graphics, 1995, Volume: 13, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Benzazepines; Chemical Phenomena; Chemistry, Physical; Chromans; Dopamine Agonists; Drug Design; Ergolines; Indoles; Ligands; Lisuride; Models, Molecular; Phenanthridines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2

1995
Antagonism by SCH 23390 of clozapine-induced hypothermia in the rat.
    European journal of pharmacology, 1994, Feb-21, Volume: 253, Issue:1-2

    Topics: Amphetamines; Animals; Benzazepines; Body Temperature; Body Temperature Regulation; Chromans; Clonidine; Clozapine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Hypothermia; Injections, Subcutaneous; Male; Oxotremorine; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Salicylamides; Serotonin Antagonists

1994
Evidence for specific involvement of dopamine D1 and D2 receptors in the regulation of body temperature in the rat.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Animals; Benzazepines; Body Temperature Regulation; Chromans; Dopamine Agents; Dopamine D2 Receptor Antagonists; Drug Interactions; Ergolines; Injections, Subcutaneous; Male; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides

1993
SK&F 83959 and non-cyclase-coupled dopamine D1-like receptors in jaw movements via dopamine D1-like/D2-like receptor synergism.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Anesthesia; Animals; Chromans; Dopamine Agonists; Drug Combinations; Drug Interactions; Jaw; Male; Muscle Contraction; Muscle, Skeletal; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine

1999
Behavioural and pharmacological examinations in a transgenic mouse model of early-onset torsion dystonia.
    Pharmacology, biochemistry, and behavior, 2011, Volume: 97, Issue:4

    Topics: Amphetamines; Animals; Anxiety; Behavior, Animal; Carbidopa; Chromans; Disease Models, Animal; Dystonia; Levodopa; Locomotion; Mice; Mice, Transgenic; Quinpirole; Raclopride

2011