a 68930 has been researched along with dihydrexidine in 5 studies
Studies (a 68930) | Trials (a 68930) | Recent Studies (post-2010) (a 68930) | Studies (dihydrexidine) | Trials (dihydrexidine) | Recent Studies (post-2010) (dihydrexidine) |
---|---|---|---|---|---|
63 | 2 | 19 | 99 | 5 | 21 |
Protein | Taxonomy | a 68930 (IC50) | dihydrexidine (IC50) |
---|---|---|---|
D | Rattus norvegicus (Norway rat) | 0.0096 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 0.0448 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (60.00) | 18.2507 |
2000's | 2 (40.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Laiter, S; Mailman, RB; Mottola, DM; Nichols, DE; Tropsha, A; Watts, VJ; Wyrick, SD | 1 |
Bone, RG; Villar, HO | 1 |
Deveney, AM; Waddington, JL | 1 |
Isacson, R; Kull, B; Salmi, P; Wahlestedt, C | 1 |
Colago, EE; Mania, I; Molosh, AI; Pickel, VM; Rainnie, DG | 1 |
5 other study(ies) available for a 68930 and dihydrexidine
Article | Year |
---|---|
Conformational analysis of D1 dopamine receptor agonists: pharmacophore assessment and receptor mapping.
Topics: Adenylyl Cyclases; Animals; Brain; Computer Simulation; Dopamine; Dopamine Agonists; Ligands; Molecular Conformation; Molecular Structure; Phenanthridines; Rats; Receptors, Dopamine D1; Software; Structure-Activity Relationship | 1996 |
Discriminating D1 and D2 agonists with a hydrophobic similarity index.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Benzazepines; Chemical Phenomena; Chemistry, Physical; Chromans; Dopamine Agonists; Drug Design; Ergolines; Indoles; Ligands; Lisuride; Models, Molecular; Phenanthridines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1995 |
Psychopharmacological distinction between novel full-efficacy "D1-like" dopamine receptor agonists.
Topics: Animals; Behavior, Animal; Chromans; Dopamine Agonists; Locomotion; Male; Phenanthridines; Radioligand Assay; Rats; Rats, Sprague-Dawley | 1997 |
A 68930 and dihydrexidine inhibit locomotor activity and d-amphetamine-induced hyperactivity in rats: a role of inhibitory dopamine D(1/5) receptors in the prefrontal cortex?
Topics: Animals; Benzazepines; Chromans; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Gene Expression; Hyperkinesis; Male; Motor Activity; Neural Inhibition; Phenanthridines; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Stereotypic Movement Disorder | 2004 |
Dopamine D1 receptors co-distribute with N-methyl-D-aspartic acid type-1 subunits and modulate synaptically-evoked N-methyl-D-aspartic acid currents in rat basolateral amygdala.
Topics: Amygdala; Analysis of Variance; Animals; Benzazepines; Chromans; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Lysine; Male; Microscopy, Immunoelectron; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Phenanthridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; Synapses | 2006 |