Page last updated: 2024-09-03

a 68930 and dihydrexidine

a 68930 has been researched along with dihydrexidine in 5 studies

Compound Research Comparison

Studies
(a 68930)
Trials
(a 68930)
Recent Studies (post-2010)
(a 68930)
Studies
(dihydrexidine)
Trials
(dihydrexidine)
Recent Studies (post-2010) (dihydrexidine)
6321999521

Protein Interaction Comparison

ProteinTaxonomya 68930 (IC50)dihydrexidine (IC50)
DRattus norvegicus (Norway rat)0.0096
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0448

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's2 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Laiter, S; Mailman, RB; Mottola, DM; Nichols, DE; Tropsha, A; Watts, VJ; Wyrick, SD1
Bone, RG; Villar, HO1
Deveney, AM; Waddington, JL1
Isacson, R; Kull, B; Salmi, P; Wahlestedt, C1
Colago, EE; Mania, I; Molosh, AI; Pickel, VM; Rainnie, DG1

Other Studies

5 other study(ies) available for a 68930 and dihydrexidine

ArticleYear
Conformational analysis of D1 dopamine receptor agonists: pharmacophore assessment and receptor mapping.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Adenylyl Cyclases; Animals; Brain; Computer Simulation; Dopamine; Dopamine Agonists; Ligands; Molecular Conformation; Molecular Structure; Phenanthridines; Rats; Receptors, Dopamine D1; Software; Structure-Activity Relationship

1996
Discriminating D1 and D2 agonists with a hydrophobic similarity index.
    Journal of molecular graphics, 1995, Volume: 13, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Benzazepines; Chemical Phenomena; Chemistry, Physical; Chromans; Dopamine Agonists; Drug Design; Ergolines; Indoles; Ligands; Lisuride; Models, Molecular; Phenanthridines; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2

1995
Psychopharmacological distinction between novel full-efficacy "D1-like" dopamine receptor agonists.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:2

    Topics: Animals; Behavior, Animal; Chromans; Dopamine Agonists; Locomotion; Male; Phenanthridines; Radioligand Assay; Rats; Rats, Sprague-Dawley

1997
A 68930 and dihydrexidine inhibit locomotor activity and d-amphetamine-induced hyperactivity in rats: a role of inhibitory dopamine D(1/5) receptors in the prefrontal cortex?
    Neuroscience, 2004, Volume: 124, Issue:1

    Topics: Animals; Benzazepines; Chromans; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Gene Expression; Hyperkinesis; Male; Motor Activity; Neural Inhibition; Phenanthridines; Prefrontal Cortex; Proto-Oncogene Proteins c-fos; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Stereotypic Movement Disorder

2004
Dopamine D1 receptors co-distribute with N-methyl-D-aspartic acid type-1 subunits and modulate synaptically-evoked N-methyl-D-aspartic acid currents in rat basolateral amygdala.
    Neuroscience, 2006, Oct-27, Volume: 142, Issue:3

    Topics: Amygdala; Analysis of Variance; Animals; Benzazepines; Chromans; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Lysine; Male; Microscopy, Immunoelectron; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Phenanthridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, N-Methyl-D-Aspartate; Synapses

2006