Page last updated: 2024-09-04

a 195773 and ketoconazole

a 195773 has been researched along with ketoconazole in 1 studies

Compound Research Comparison

Studies
(a 195773)
Trials
(a 195773)
Recent Studies (post-2010)
(a 195773)
Studies
(ketoconazole)
Trials
(ketoconazole)
Recent Studies (post-2010) (ketoconazole)
13061490120

Protein Interaction Comparison

ProteinTaxonomya 195773 (IC50)ketoconazole (IC50)
Bile salt export pumpHomo sapiens (human)3.4
Steroid 17-alpha-hydroxylase/17,20 lyaseHomo sapiens (human)1.175
Epoxide hydrolase 1 Homo sapiens (human)0.04
ATP-dependent translocase ABCB1Homo sapiens (human)1.058
Cytochrome P450 3A4Homo sapiens (human)0.2303
Cytochrome P450 2D6Homo sapiens (human)2.774
AromataseHomo sapiens (human)1.3026
Cytochrome P450 11B1, mitochondrialHomo sapiens (human)0.4519
Cytochrome P450 11B2, mitochondrialHomo sapiens (human)0.1272
Cytochrome P450 3A5Homo sapiens (human)0.2535
Bifunctional epoxide hydrolase 2Homo sapiens (human)0.04
1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialHomo sapiens (human)0.3
Sterol 14-alpha demethylaseTrypanosoma cruzi strain CL Brener0.014

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cushman, M; Fan, BZ; Han, X; Kong, FS; Li, YX; Liang, JH; Lv, W; Ma, CX; Tian, JC1

Other Studies

1 other study(ies) available for a 195773 and ketoconazole

ArticleYear
Design, synthesis and structure-activity relationships of novel macrolones: Hybrids of 2-fluoro 9-oxime ketolides and carbamoyl quinolones with highly improved activity against resistant pathogens.
    European journal of medicinal chemistry, 2019, May-01, Volume: 169

    Topics: Anti-Bacterial Agents; Dose-Response Relationship, Drug; Drug Design; Drug Resistance, Bacterial; Ketolides; Microbial Sensitivity Tests; Molecular Structure; Oximes; Quinolones; Streptococcus pneumoniae; Streptococcus pyogenes; Structure-Activity Relationship

2019