8-hydroxy-2-(di-n-propylamino)tetralin has been researched along with metergoline in 50 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (28.00) | 18.7374 |
1990's | 27 (54.00) | 18.2507 |
2000's | 7 (14.00) | 29.6817 |
2010's | 2 (4.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Glennon, RA | 1 |
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S | 1 |
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J | 1 |
Adham, N; Bard, J; Branchek, TA; Durkin, M; Hartig, PR; Kao, HT; Olsen, M; Schecter, LE; Urquhart, D; Weinshank, RL | 1 |
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR | 1 |
Amlaiky, N; Hen, R; Plassat, JL | 1 |
Arrang, JM; Diaz, J; Leurs, R; Ruat, M; Schwartz, JC; Tardivel-Lacombe, J; Traiffort, E | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R | 1 |
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP | 1 |
Beleta, J; Doménech, T; Palacios, JM | 1 |
Bach, T; Krobert, KA; Kvingedal, AM; Levy, FO; Syversveen, T | 1 |
Bai, F; Johnstone, EM; Little, SP; Nelson, DL; Su, C; Varga, G; Yin, T | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Lepailleur, A; Rochais, C; Thirumaran, SL | 1 |
Flores, CM; Hulihan-Giblin, BA; Kellar, KJ; Lumpkin, MD; Mulroney, SE | 1 |
Jackson, HC; Nutt, DJ | 1 |
Murphy, AZ; Murphy, RM; Zemlan, FP | 1 |
Eide, PK; Hole, K | 1 |
Davies, M; Fletcher, PJ | 1 |
Kuno, S; Mizuta, E; Yamaguchi, M | 1 |
Lucot, JB | 1 |
Ramage, AG | 1 |
Nanry, KP; Tilson, HA | 1 |
Cervo, L; Grignaschi, G; Nowakowska, E; Samanin, R | 1 |
Bagdy, G; Murphy, DL; Szemeredi, K | 1 |
Appel, JB; Cunningham, KA | 1 |
Feuerstein, TJ; Hertting, G; Lupp, A | 1 |
Houston, DS; Vanhoutte, PM | 1 |
Berendsen, HH; Broekkamp, CL; Oosterloo, SK; van Delft, AM | 1 |
Eide, PK; Tjølsen, A | 1 |
Bockaert, J; Kemp, DE; Sebben, M; Weiss, S | 1 |
Lis, EV; Martin, GE | 1 |
Svensson, L | 1 |
Ahlenius, S; Larsson, K | 1 |
Baudrie, V; Bluet-Pajot, MT; Broqua, P; Chaouloff, F; Laude, D; Schmidt, B | 1 |
Rusak, B; Ying, SW | 1 |
Kellar, KJ; Lumpkin, MD; Mulroney, SE; Shemer, A; Skudlarek, C | 1 |
Dean, RR; Edgar, DM; Heller, HC; Miller, JD; Prosser, RA | 1 |
Clifton, PG; Dourish, CT; Vickers, SP | 1 |
Del Prete, E; Lutz, TA; Scharrer, E; Walzer, B | 1 |
Cattaneo, MG; Fesce, R; Vicentini, LM | 1 |
Gean, PW; Lu, KT | 1 |
Evenden, JL | 1 |
Dinardo, LA; Dudley, TE; Glass, JD | 1 |
Hrupka, BJ; Langhans, W | 1 |
Choi, S; Fernstrom, JD; Jonak, E | 1 |
Centurión, D; Gupta, S; MaassenVanDenBrink, A; Mehotra, S; Sánchez-López, A; Villalón, CM | 1 |
Beckman, D; da Cunha, IC; Faria, MS; Lopes, AP; Marino-Neto, J; Paschoalini, MA; Steffens, SM | 1 |
Francl, JM; Glass, JD; Guinn, J; Kaur, G | 1 |
2 review(s) available for 8-hydroxy-2-(di-n-propylamino)tetralin and metergoline
Article | Year |
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Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
Structure-activity relationships of serotonin 5-HT
Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship | 2019 |
48 other study(ies) available for 8-hydroxy-2-(di-n-propylamino)tetralin and metergoline
Article | Year |
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Cloning and characterisation of the human 5-HT5A serotonin receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection | 1994 |
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase.
Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction | 1993 |
Cloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Colforsin; Dose-Response Relationship, Drug; Gene Library; Guinea Pigs; Humans; Indoles; Lymphocytes; Molecular Sequence Data; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Serotonin; Serotonin Receptor Agonists; Spiperone; Sulfonamides; Sumatriptan; Tissue Distribution | 1993 |
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection | 1993 |
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists | 1993 |
Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.
Topics: Amino Acid Sequence; Animals; Base Sequence; Blotting, Northern; Brain; CHO Cells; Cricetinae; Cyclic AMP; DNA; Genomic Library; Kinetics; Lysergic Acid Diethylamide; Mianserin; Molecular Sequence Data; Multigene Family; Oligodeoxyribonucleotides; Organ Specificity; Rats; Receptors, Serotonin; Restriction Mapping; Serotonin; Serotonin Receptor Agonists; Transfection | 1993 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents | 1996 |
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b).
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid | 1997 |
Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist.
Topics: Benzamides; Binding, Competitive; Gene Expression; HeLa Cells; Humans; Kinetics; Ligands; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Tritium | 1997 |
The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution.
Topics: Adenylyl Cyclases; Alternative Splicing; Binding, Competitive; Brain; Cell Line; Cloning, Organism; Genetic Variation; Humans; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution | 2001 |
Molecular cloning and pharmacological characterization of the guinea pig 5-HT1E receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Chickens; Cloning, Molecular; Cricetinae; Dose-Response Relationship, Drug; Gerbillinae; Guinea Pigs; Haplorhini; Humans; Molecular Sequence Data; Protein Binding; Rabbits; Receptors, Serotonin; Serotonin Agents; Swine | 2004 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Stimulation of serotonin1A receptors increases release of prolactin in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Male; Metergoline; Methysergide; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Time Factors | 1992 |
Are 5-HT receptors or beta-adrenoceptors involved in idazoxan-induced food and water intake?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Betaxolol; Dioxanes; Dose-Response Relationship, Drug; Drinking; Eating; Idazoxan; Male; Metergoline; Propanolamines; Propranolol; Quinolizines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Serotonin; Stereoisomerism | 1992 |
Role of spinal serotonin1 receptor subtypes in thermally and mechanically elicited nociceptive reflexes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hot Temperature; Indoles; Male; Metergoline; Nociceptors; Physical Stimulation; Piperazines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Reflex; Spinal Cord | 1992 |
Interactions between serotonin and substance P in the spinal regulation of nociception.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Indoles; Injections, Spinal; Male; Metergoline; Mice; Mice, Inbred Strains; Neurons; Pain; Serotonin; Serotonin Antagonists; Skin Temperature; Spinal Cord; Substance P; Tetrahydronaphthalenes | 1991 |
A pharmacological analysis of the eating response induced by 8-OH-DPAT injected into the dorsal raphé nucleus reveals the involvement of a dopaminergic mechanism.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine; Drug Interactions; Eating; Haloperidol; Injections; Male; Metergoline; Naphthalenes; Propranolol; Raphe Nuclei; Rats; Rats, Inbred Strains; Spiperone; Tetrahydronaphthalenes | 1990 |
Behavioural effects of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) in monkeys.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Macaca fascicularis; Male; Metergoline; Naphthalenes; Tetrahydronaphthalenes | 1990 |
Effects of serotonin antagonists on motion sickness and its suppression by 8-OH-DPAT in cats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Dose-Response Relationship, Drug; Ergolines; Female; Metergoline; Motion Sickness; Piperazines; Propranolol; Serotonin Antagonists; Stereoisomerism; Tetrahydronaphthalenes | 1990 |
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes | 1988 |
The role of 5HT1A receptors in the modulation of the acoustic startle reflex in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Metergoline; Methoxydimethyltryptamines; Quipazine; Rats; Rats, Inbred F344; Receptors, Serotonin; Reflex, Startle; Serotonin Antagonists; Tetrahydronaphthalenes | 1989 |
1-(3-Trifluoromethylphenyl) piperazine (TFMPP) in the ventral tegmental area reduces the effect of desipramine in the forced swimming test in rats: possible role of serotonin receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Depression; Desipramine; Injections; Male; Metergoline; Piperazines; Rats; Receptors, Serotonin; Swimming; Tegmentum Mesencephali; Tetrahydronaphthalenes | 1989 |
Marked increases in plasma catecholamine concentrations precede hypotension and bradycardia caused by 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT) in conscious rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Catecholamines; Epinephrine; Heart Rate; Male; Metergoline; Naphthalenes; Norepinephrine; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes | 1989 |
Possible 5-hydroxytryptamine1 (5-HT1) receptor involvement in the stimulus properties of 1-(m-trifluoromethylphenyl)piperazine (TFMPP).
Topics: 2-Methyl-4-chlorophenoxyacetic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Discrimination Learning; Dose-Response Relationship, Drug; Indoles; Lysergic Acid Diethylamide; Male; Metergoline; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes | 1986 |
The serotonin (5-HT) autoreceptor in the hippocampus of the rabbit: role of 5-HT biophase concentration.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Mathematics; Metergoline; Methiothepin; Methoxydimethyltryptamines; Methysergide; Phentolamine; Pindolol; Quipazine; Rabbits; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1987 |
Comparison of serotonergic receptor subtypes on the smooth muscle and endothelium of the canine coronary artery.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Ketanserin; Male; Metergoline; Methiothepin; Muscle, Smooth, Vascular; Pindolol; Receptors, Serotonin; Tetrahydronaphthalenes; Vasodilation | 1988 |
Effect of metergoline, fenfluramine, and 8-OHDPAT on catalepsy induced by haloperidol or morphine.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Catalepsy; Drug Interactions; Fenfluramine; Haloperidol; Male; Metergoline; Mice; Morphine; Rats; Rats, Inbred Strains; Serotonin; Tetrahydronaphthalenes | 1988 |
Effects of serotonin receptor antagonists and agonists on the tail-flick response in mice involve altered tail-skin temperature.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Hypothermia, Induced; Male; Metergoline; Methiothepin; Methoxydimethyltryptamines; Mice; Mice, Inbred Strains; Reaction Time; Receptors, Serotonin; Skin Temperature; Tetrahydronaphthalenes | 1988 |
Serotonin 5-HT1 receptors mediate inhibition of cyclic AMP production in neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Brain; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Female; Fetus; Indoles; Ketanserin; Metergoline; Mice; Neurons; Piperidines; Pregnancy; Receptors, Serotonin; Tetrahydronaphthalenes; Vasoactive Intestinal Peptide | 1986 |
Hypotensive action of 8-hydroxy-2-(di-N-propylamino)tetralin (8-OH-DPAT) in spontaneously hypertensive rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Cyproheptadine; Heart Rate; Injections, Intraperitoneal; Injections, Intraventricular; Male; Metergoline; Methiothepin; Naphthalenes; Rats; Rats, Inbred SHR; Tetrahydronaphthalenes | 1985 |
Effects of 8-OH-DPAT, lisuride and some ergot-related compounds on the acoustic startle response in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bromocriptine; Ergolines; Lisuride; Male; Metergoline; Methiothepin; Naphthalenes; Pergolide; Quinpirole; Rats; Rats, Inbred Strains; Reflex, Startle; Tetrahydronaphthalenes | 1985 |
Failure to antagonize the 8-hydroxy-2-di-n-propylamino)tetralin-induced facilitation of male rat sexual behavior by the administration of 5-HT receptor antagonists.
Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Male; Metergoline; Methiothepin; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Sexual Behavior, Animal; Tetrahydronaphthalenes | 1984 |
Are 5-HT1A autoreceptors involved in the inhibitory effect of ipsapirone on cold-elicited thyrotropin secretion?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Glucose; Cold Temperature; Corticosterone; Fenclonine; Hydroxyindoleacetic Acid; Hypothalamus; Male; Metergoline; Pindolol; Proadifen; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Thyrotropin | 1993 |
Effects of serotonergic agonists on firing rates of photically responsive cells in the hamster suprachiasmatic nucleus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Circadian Rhythm; Cricetinae; Light; Male; Metergoline; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus | 1994 |
Tandospirone stimulates prolactin secretion in the rat by an action at serotonin-1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Dose-Response Relationship, Drug; Isoindoles; Male; Metergoline; Piperazines; Prolactin; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists | 1994 |
Serotonin and the mammalian circadian system: I. In vitro phase shifts by serotonergic agonists and antagonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Circadian Rhythm; Dose-Response Relationship, Drug; Electrophysiology; In Vitro Techniques; Iodocyanopindolol; Lysergic Acid Diethylamide; Male; Metergoline; Neurons; Pindolol; Quipazine; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus | 1993 |
Behavioural evidence that d-fenfluramine-induced anorexia in the rat is not mediated by the 5-HT1A receptor subtype.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anorexia; Appetite Depressants; Appetitive Behavior; Drug Interactions; Fenfluramine; Male; Metergoline; Piperazines; Pyridines; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists | 1996 |
The histaminergic, but not the serotoninergic, system mediates amylin's anorectic effect.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amyloid; Animals; Appetite Depressants; Eating; Food Deprivation; Histamine; Histamine Agonists; Islet Amyloid Polypeptide; Male; Metergoline; Methylhistamines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Synaptic Transmission | 1996 |
Evidence for receptor subtype cross-talk in the mitogenic action of serotonin on human small-cell lung carcinoma cells.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium-Calmodulin-Dependent Protein Kinases; Carcinoma, Small Cell; Humans; Lung Neoplasms; Metergoline; Mitogens; Receptors, Serotonin; Serotonin; Temperature; Thymidine; Tumor Cells, Cultured | 1996 |
Endogenous serotonin inhibits epileptiform activity in rat hippocampal CA1 neurons via 5-hydroxytryptamine1A receptor activation.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Barium; Epilepsy; Excitatory Postsynaptic Potentials; Fluoxetine; Hippocampus; In Vitro Techniques; Ketanserin; Male; Membrane Potentials; Metergoline; Neurons; Oxadiazoles; Picrotoxin; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Tryptamines | 1998 |
The pharmacology of impulsive behaviour in rats IV: the effects of selective serotonergic agents on a paced fixed consecutive number schedule.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Impulsive Behavior; Indoles; Male; Metergoline; p-Chloroamphetamine; Rats; Reinforcement, Psychology; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes | 1998 |
In vivo assessment of the midbrain raphe nuclear regulation of serotonin release in the hamster suprachiasmatic nucleus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Brain Chemistry; Chromatography, High Pressure Liquid; Cricetinae; Electric Stimulation; Male; Mesocricetus; Metergoline; Microdialysis; Piperazines; Pyridines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus | 1999 |
A role for serotonin in lipopolysaccharide-induced anorexia in rats.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anorexia; Cisterna Magna; Dose-Response Relationship, Drug; Eating; Lipopolysaccharides; Male; Metergoline; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 2001 |
Serotonin reuptake inhibitors do not prevent 5,7-dihydroxytryptamine-induced depletion of serotonin in rat brain.
Topics: 5-Hydroxytryptophan; 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Animals; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Desipramine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Electrochemistry; Injections, Intraventricular; Male; Metergoline; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Agents; Serotonin Antagonists | 2004 |
Potential vascular alpha1-adrenoceptor blocking properties of an array of 5-HT receptor ligands in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Buspirone; Clozapine; Decerebrate State; Dose-Response Relationship, Drug; Drug Interactions; Ergotamine; Heart Rate; Ketanserin; Lisuride; Male; Metergoline; Methiothepin; Methysergide; Phenylephrine; Piperazines; Pizotyline; Prazosin; Pyridines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Serotonin Antagonists; Serotonin Receptor Agonists; Yohimbine | 2006 |
The effects of metergoline and 8-OH-DPAT injections into arcuate nucleus and lateral hypothalamic area on feeding in female rats during the estrous cycle.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Eating; Estrous Cycle; Feeding Behavior; Female; Hypothalamic Area, Lateral; Metergoline; Nucleus Accumbens; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
On the intrinsic regulation of neuropeptide Y release in the mammalian suprachiasmatic nucleus circadian clock.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Circadian Rhythm; Cricetinae; Electric Stimulation; GABA Agonists; Male; Metergoline; Microdialysis; Motor Activity; Muscimol; Neuropeptide Y; Physical Conditioning, Animal; Radioimmunoassay; Serotonin Antagonists; Serotonin Receptor Agonists; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Suprachiasmatic Nucleus | 2010 |