8-hydroxy-2-(di-n-propylamino)tetralin and citalopram

8-hydroxy-2-(di-n-propylamino)tetralin has been researched along with citalopram in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.45)18.7374
1990's24 (34.78)18.2507
2000's30 (43.48)29.6817
2010's13 (18.84)24.3611
2020's1 (1.45)2.80

Authors

AuthorsStudies
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B1
Bojarski, AJ; Duszyńska, B; Grychowska, K; Jastrzębska-Więsek, M; Lenda, T; Marciniec, K; Maślankiewicz, A; Nowak, G; Partyka, A; Pawłowski, M; Satała, G; Siwek, A; Wesołowska, A; Wróbel, D; Zajdel, P1
Araya-Maturana, R; Fierro, A; González-Lira, C; Iturriaga-Vásquez, P; Ortiz-Severin, J; Pessoa-Mahana, CD; Pessoa-Mahana, H; Reyes-Parada, M; Saitz-Barría, C; Silva-Matus, P; Zapata-Torres, G1
Fu, Y; Gong, Q; Huang, J; Huang, Y; Li, J; Li, X; Mao, F; Wang, H; Xu, Y; You, H; Zhang, D; Zhang, H; Zhu, J1
Maj, J; Moryl, E1
Dawson, IM; Hodgkiss, JP; Kelly, JS1
Engberg, G1
Barzizza, A; Maura, G; Raiteri, M1
Ciesielski, L; Gobaille, S; Isel, F; Mandel, P; Molina, V1
Arborelius, L; Grillner, P; Hacksell, U; Hertel, P; Höök, BB; Nomikos, GG; Svensson, TH1
Kreiss, DS; Lucki, I; Wieland, S1
Butcher, SP; Kelly, JS; Lawrence, JA; Olverman, HJ; Shirakawa, K1
Hyttel, J; Sánchez, C1
Gobbi, M; Mennini, T; Palacios, JM; Pompeiano, M; Regondi, MC1
Artigas, F; Celada, P; Romero, L1
Bramante, M; Invernizzi, R; Samanin, R2
Blatt, GJ; Chen, JC; Galler, JR; Rosene, DL; Volicer, L1
Hjorth, S; Sharp, T1
Hjorth, S1
Moryl, E; Papp, M; Przegaliński, E1
Arborelius, L; Grillner, P; Hacksell, U; Hertel, P; Höök, BB; Nomikos, GG; Salmi, P; Svensson, TH1
Afkhami-Dastjerdian, S; Carli, M; Reader, TA1
Aguerre, S; Berton, O; Chaouloff, F; Kulikov, A; Mormede, P; Ramos, A1
Leander, JD; Wolff, MC1
Ishikane, T1
Evenden, JL1
Jeanningros, R; Kulikov, A; Moreau, X1
Fache, MP; Faudon, M; Héry, F; Héry, M; Sémont, A1
Caccia, S; De Deurwaerdère, P; Lucas, G1
Bosker, FJ; Cremers, TI; de Boer, P; den Boer, JA; Mørk, A; Spoelstra, EN; Westerink, BH; Wikström, HV1
Auerbach, SB; Ma, Z; Tao, R1
Assié, MB; Koek, W1
Chen, F; Lawrence, AJ1
Ross, SB; Stenfors, C; Yu, H1
Jeanningros, R; Mazzola-Pomietto, P; Moreau, X1
Ase, AR; Descarries, L; Hen, R; Reader, TA; Riad, M1
Jensen, JB; Mikkelsen, JD; Mørk, A1
Allikmets, L; Matto, V; Pruus, K; Rudissaar, R; Vaarmann, A1
Bobula, B; Hess, G; Tokarski, K; Zahorodna, A1
Kehr, J; Yoshitake, T1
Arborelius, L; Hawks, BW; Nemeroff, CB; Owens, MJ; Plotsky, PM1
Chouvet, G; El Mansari, M; Haddjeri, N; Renaud, B; Sánchez, C1
Höglund, AU; Kommalage, M1
Grandoso, L; Pineda, J; Torrecilla, M; Ugedo, L1
Ma, Z; McCarley, RW; McKenna, JT; Strecker, RE; Tao, R; Thakkar, MM1
Isgor, C; Ma, Z; Pearson, E; Tao, R1
Hess, G; Zahorodna, A1
Coppinger, D; Maciag, D; Paul, IA1
Andrews, AM; Chenu, F; David, DJ; Deltheil, T; Gardier, AM; Guiard, BP; Hamon, M; Hen, R; Lanfumey, L; Le Maître, E; Leroux-Nicollet, I; Renoir, T; Sokoloff, P1
Burke, TF; Hensler, JG; Rossi, DV1
Adrien, J; Alexandre, C; Léna, C; Popa, D1
Craighead, M; Gartside, SE; Grant, EJ; Ingram, CD; Johnson, DA1
Hummel, R; Jacobsen, JP; Mirza, N; Nielsen, EØ; Redrobe, JP; Weikop, P1
Chidori, S; Egashira, N; Fujiwara, M; Hasebe, N; Higashihara, F; Iwasaki, K; Koushi, E; Matsuda, T; Mishima, K; Nishimura, R; Oishi, R1
El Yacoubi, M; Hamon, M; Hanoun, N; Lanfumey, L; Lesch, KP; Melfort, M; Païzanis, E; Renoir, T; Saurini, F1
Günther, L; Jähkel, M; Liebscher, S; Oehler, J1
Charnay, Y; Fagret, D; Ginovart, N; Hamon, M; Hen, R; Ibáñez, V; Lanfumey, L; Millet, P; Moulin-Sallanon, M; Perret, P1
Blendy, JA; Gur, TL; Mombereau, C; Onksen, J1
Hadley, JK; Halliwell, JV1
Chen, CP; Esiri, MM; Francis, PT; Lai, MK; Tsang, SW; Wong, PT1
Amar, M; Callebert, J; Fossier, P; Moreau, AW1
Khatri, N; Lin, RC; Paul, IA; Simpson, KL1
Seyfried, CA; van Amsterdam, C1
Bishop, C; Conti, MM; Lindenbach, D; Ostock, CY; Palumbo, N; Vilceus, N1
Gong, WG; Ren, QG; Wang, YJ; Xu, L; Zhang, ZJ; Zhou, QD1
Bruzos-Cidón, C; Llamosas, N; Rodríguez, JJ; Torrecilla, M; Ugedo, L1
Chiba, H; Kanno, Y; Kitta, T; Mitsui, T; Moriya, K; Ohmura, Y; Shinohara, N; Yoshioka, M1
Aguilar-Magaña, D; Atzori, M; Canto-Bustos, M; Cervantes-Ramírez, V; Góngora-Alfaro, JL; Pérez-Padilla, EA; Pineda, JC; Salgado, H1

Other Studies

69 other study(ies) available for 8-hydroxy-2-(di-n-propylamino)tetralin and citalopram

ArticleYear
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT₁A/5-HT₂A/5-HT₇ and dopamine D₂/D₃ receptors.
    European journal of medicinal chemistry, 2013, Volume: 60

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Aripiprazole; Behavior, Animal; Dizocilpine Maleate; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Isoquinolines; Mice; Molecular Structure; Motor Activity; Piperazines; Quinolines; Quinolones; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Structure-Activity Relationship; Sulfonamides

2013
Synthesis, docking and pharmacological evaluation of novel homo- and hetero-bis 3-piperazinylpropylindole derivatives at SERT and 5-HT1A receptor.
    Bioorganic & medicinal chemistry, 2013, Dec-15, Volume: 21, Issue:24

    Topics: Dose-Response Relationship, Drug; Humans; Indoles; Models, Molecular; Molecular Docking Simulation; Molecular Structure; Piperazines; Receptor, Serotonin, 5-HT1A; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship

2013
The novel therapeutic strategy of vilazodone-donepezil chimeras as potent triple-target ligands for the potential treatment of Alzheimer's disease with comorbid depression.
    European journal of medicinal chemistry, 2022, Feb-05, Volume: 229

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Antidepressive Agents; Binding Sites; Brain; Cholinesterase Inhibitors; Depression; Donepezil; Drug Design; Half-Life; Humans; Ligands; Mice; Molecular Docking Simulation; Rats; Rats, Sprague-Dawley; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Vilazodone Hydrochloride

2022
Effects of sertraline and citalopram given repeatedly on the responsiveness of 5-HT receptor subpopulations.
    Journal of neural transmission. General section, 1992, Volume: 88, Issue:2

    Topics: 1-Naphthylamine; 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Body Temperature; Citalopram; Drug Interactions; Exploratory Behavior; Fenfluramine; Male; Motor Activity; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Sertraline; Tetrahydronaphthalenes

1992
An intracellular study of the action of NAN-190 on neurons in the dorsal raphe nucleus of the rat.
    Brain research, 1992, Mar-27, Volume: 576, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Dose-Response Relationship, Drug; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurons; Piperazines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1992
Citalopram and 8-OH-DPAT attenuate nicotine-induced excitation of central noradrenaline neurons.
    Journal of neural transmission. General section, 1992, Volume: 89, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amino Acids; Animals; Citalopram; Injections, Intravenous; Locus Coeruleus; Male; Neurons; Nicotine; Norepinephrine; Rats; Rats, Sprague-Dawley; Serotonin

1992
Activation of presynaptic 5-hydroxytryptamine1-like receptors on glutamatergic terminals inhibits N-methyl-D-aspartate-induced cyclic GMP production in rat cerebellar slices.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium; Cerebellum; Citalopram; Cyclic GMP; Fenfluramine; Glutamates; Glutamic Acid; In Vitro Techniques; Male; Methiothepin; N-Methylaspartate; Potassium; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Inhibition of mouse killing behavior by serotonin-mimetic drugs: effects of partial alterations of serotonin neurotransmission.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Citalopram; Fenclonine; Fluoxetine; Hydroxyindoleacetic Acid; Male; Methoxydimethyltryptamines; Motor Activity; Propylamines; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin; Tetrahydronaphthalenes

1987
5-HT1A receptor antagonists increase the activity of serotonergic cells in the dorsal raphe nucleus in rats treated acutely or chronically with citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Citalopram; Electrophysiology; Extracellular Space; Male; Neurons; Piperazines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Synaptic Transmission

1995
The presence of a serotonin uptake inhibitor alters pharmacological manipulations of serotonin release.
    Neuroscience, 1993, Volume: 52, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Chromatography, High Pressure Liquid; Citalopram; Corpus Striatum; Dialysis; Electrochemistry; Fenfluramine; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Sodium Channels; Tetrodotoxin

1993
Binding of 5-HT1A receptor and 5-HT transporter ligands in rat cortex and hippocampus following cholinergic and serotonergic lesions.
    Brain research, 1993, May-28, Volume: 612, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Carrier Proteins; Cerebral Cortex; Citalopram; Hippocampus; Ibotenic Acid; Kinetics; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Endings; Nerve Tissue Proteins; Parasympathetic Nervous System; Prosencephalon; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Plasma Membrane Transport Proteins

1993
Isolation-induced aggression in mice: effects of 5-hydroxytryptamine uptake inhibitors and involvement of postsynaptic 5-HT1A receptors.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: 1-Naphthylamine; 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Analysis of Variance; Animals; Behavior, Animal; Brain; Citalopram; Dose-Response Relationship, Drug; Fenclonine; Fluoxetine; Fluvoxamine; Male; Mice; Paroxetine; Penbutolol; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Sertraline; Synaptosomes

1994
Differential effects of 5,7-dihydroxytryptamine-induced serotoninergic degeneration of 5-HT1A receptors and 5-HT uptake sites in the rat brain.
    Journal of chemical neuroanatomy, 1994, Volume: 7, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain; Citalopram; Male; Nerve Degeneration; Paroxetine; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reserpine; Serotonin

1994
Reduction of in vivo striatal 5-hydroxytryptamine release by 8-OH-DPAT after inactivation of Gi/G(o) proteins in dorsal raphe nucleus.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Autoreceptors; Citalopram; Corpus Striatum; GTP-Binding Proteins; Male; Pertussis Toxin; Potassium Channels; Propanolamines; Raphe Nuclei; Rats; Rats, Wistar; Serotonin; Thiophenes; Virulence Factors, Bordetella

1994
Chronic treatment with citalopram facilitates the effect of a challenge dose on cortical serotonin output: role of presynaptic 5-HT1A receptors.
    European journal of pharmacology, 1994, Aug-01, Volume: 260, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Analysis of Variance; Animals; Cerebral Cortex; Citalopram; Dialysis; Male; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin

1994
Prenatal protein malnutrition effects on the serotonergic system in the hippocampal formation: an immunocytochemical, ligand binding, and neurochemical study.
    Brain research bulletin, 1994, Volume: 34, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Chromatography, High Pressure Liquid; Citalopram; Female; Fetal Diseases; Hippocampus; Immunohistochemistry; Ligands; Pregnancy; Prenatal Exposure Delayed Effects; Protein-Energy Malnutrition; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin

1994
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism

1993
Serotonin 5-HT1A autoreceptor blockade potentiates the ability of the 5-HT reuptake inhibitor citalopram to increase nerve terminal output of 5-HT in vivo: a microdialysis study.
    Journal of neurochemistry, 1993, Volume: 60, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Chromatography, High Pressure Liquid; Citalopram; Dialysis; Feedback; Hippocampus; Male; Microchemistry; Nerve Endings; Penbutolol; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists

1993
The effect of 5-HT1A receptor ligands in a chronic mild stress model of depression.
    Neuropharmacology, 1995, Volume: 34, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Depressive Disorder; Disease Models, Animal; Imipramine; Male; Rats; Rats, Wistar; Receptors, Serotonin; Time Factors

1995
Extracellular concentrations of serotonin in the dorsal hippocampus after acute and chronic treatment with citalopram.
    Brain research, 1995, Oct-23, Volume: 696, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Extracellular Space; Hippocampus; Infusions, Intravenous; Injections, Intraperitoneal; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

1995
The 5-HT1A receptor antagonist (S)-UH-301 augments the increase in extracellular concentrations of 5-HT in the frontal cortex produced by both acute and chronic treatment with citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Body Temperature; Citalopram; Extracellular Space; Male; Microdialysis; Raphe Nuclei; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Effects of a chronic lithium treatment on cortical serotonin uptake sites and 5-HT1A receptors.
    Neurochemical research, 1997, Volume: 22, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Membrane; Cerebral Cortex; Citalopram; Humans; Hydroxyindoleacetic Acid; Lithium; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Tritium

1997
Central serotonergic systems in the spontaneously hypertensive and Lewis rat strains that differ in the elevated plus-maze test of anxiety.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Behavior, Animal; Citalopram; Female; Hippocampus; Hydroxyindoleacetic Acid; Ketanserin; Male; Mesencephalon; Rats; Rats, Inbred Lew; Rats, Inbred SHR; Receptors, Serotonin; Serotonin; Tritium; Tryptophan Hydroxylase

1997
Selective serotonin reuptake inhibitors potentiate 8-OH-DPAT-induced stimulus control in the pigeon.
    European journal of pharmacology, 1998, Mar-12, Volume: 345, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Columbidae; Conditioning, Operant; Discrimination, Psychological; Drug Synergism; Fluoxetine; Generalization, Stimulus; Imipramine; Male; Neurotransmitter Uptake Inhibitors; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists

1998
[Effects of serotonergic drugs on the up-regulation of dopamine D2 receptors induced by haloperidol in rat striatum].
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1998, Volume: 73, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Dyskinesia Agents; Antipsychotic Agents; Citalopram; Corpus Striatum; Dopamine Antagonists; Haloperidol; Male; Pyrazines; Rats; Rats, Wistar; Receptors, Dopamine D2; Ritanserin; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Up-Regulation

1998
The pharmacology of impulsive behaviour in rats IV: the effects of selective serotonergic agents on a paced fixed consecutive number schedule.
    Psychopharmacology, 1998, Volume: 140, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Impulsive Behavior; Indoles; Male; Metergoline; p-Chloroamphetamine; Rats; Reinforcement, Psychology; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

1998
Effects of experimental hypothyroidism on 5-HT1A, 5-HT2A receptors, 5-HT uptake sites and tryptophan hydroxylase activity in mature rat brain1.
    Neuroendocrinology, 1999, Volume: 69, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Brain Chemistry; Citalopram; Hypothyroidism; Ketanserin; Luminescent Measurements; Male; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thyroidectomy; Thyroxine; Triiodothyronine; Tryptophan Hydroxylase

1999
The effects of serotonin on glucocorticoid receptor binding in rat raphe nuclei and hippocampal cells in culture.
    Journal of neurochemistry, 2000, Volume: 74, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Cells, Cultured; Citalopram; Hippocampus; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Glucocorticoid; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

2000
The effect of serotonergic agents on haloperidol-induced striatal dopamine release in vivo: opposite role of 5-HT(2A) and 5-HT(2C) receptor subtypes and significance of the haloperidol dose used.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Corpus Striatum; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Fluorobenzenes; Haloperidol; Indoles; Male; Microdialysis; Phenols; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Desensitisation of 5-HT autoreceptors upon pharmacokinetically monitored chronic treatment with citalopram.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Citalopram; Infusion Pumps; Male; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Time Factors

2000
Differential effect of local infusion of serotonin reuptake inhibitors in the raphe versus forebrain and the role of depolarization-induced release in increased extracellular serotonin.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Dendritic Cells; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Male; Microdialysis; Nucleus Accumbens; Prosencephalon; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Tetrodotoxin

2000
[(3)H]-8-OH-DPAT binding in the rat brain raphe area: involvement of 5-HT(1A) and non-5-HT(1A) receptors.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Brain; Citalopram; Dose-Response Relationship, Drug; Male; Membranes; Piperazines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Tritium

2000
5-HT transporter sites and 5-HT1A and 5-HT3 receptors in Fawn-Hooded rats: a quantitative autoradiography study.
    Alcoholism, clinical and experimental research, 2000, Volume: 24, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain; Carrier Proteins; Central Nervous System Depressants; Citalopram; Ethanol; Imidazoles; Indoles; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Inbred WKY; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin Plasma Membrane Transport Proteins; Species Specificity

2000
Pharmacological characterisation of the decrease in 5-HT synthesis in the mouse brain evoked by the selective serotonin re-uptake inhibitor citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:2

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Animals; Citalopram; Dose-Response Relationship, Drug; Hippocampus; Hypothalamus; Mice; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2001
Chronic effects of triiodothyronine in combination with imipramine on 5-HT transporter, 5-HT(1A) and 5-HT(2A) receptors in adult rat brain.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 24, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Tricyclic; Body Weight; Brain; Carrier Proteins; Citalopram; Depressive Disorder; Drug Administration Schedule; Drug Interactions; Drug Therapy, Combination; Imipramine; Ketanserin; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Thyroid Gland; Time Factors; Triiodothyronine

2001
Regional changes in density of serotonin transporter in the brain of 5-HT1A and 5-HT1B knockout mice, and of serotonin innervation in the 5-HT1B knockout.
    Journal of neurochemistry, 2001, Volume: 78, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Behavior, Animal; Brain; Carrier Proteins; Citalopram; Female; Immunohistochemistry; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Nerve Tissue Proteins; Neurons; Pindolol; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2001
Chronic antidepressant treatments decrease pro-opiomelanocortin mRNA expression in the pituitary gland: effects of acute stress and 5-HT(1A) receptor activation.
    Journal of neuroendocrinology, 2001, Volume: 13, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acute Disease; Animals; Antidepressive Agents; Citalopram; Genes, fos; Immunohistochemistry; In Situ Hybridization; Male; Paraventricular Hypothalamic Nucleus; Pituitary Gland; Pro-Opiomelanocortin; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Restraint, Physical; RNA, Messenger; Seizures; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Stress, Psychological; Swimming

2001
Role of 5-HT1A receptors in the mediation of acute citalopram effects: a 8-OH-DPAT challenge study.
    Progress in neuro-psychopharmacology & biological psychiatry, 2002, Volume: 26, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anxiety; Brain; Citalopram; Drug Synergism; Exploratory Behavior; Female; Hydroxyindoleacetic Acid; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

2002
Adaptive changes in the reactivity of 5-HT1A and 5-HT2 receptors induced in rat frontal cortex by repeated imipramine and citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adaptation, Physiological; Administration, Topical; Amphetamines; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Citalopram; Cortical Synchronization; Dose-Response Relationship, Drug; Frontal Lobe; Imipramine; Male; Neurons; Piperazines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT2

2003
Differential effects of (R)-, (R, S)- and (S)-8-hydroxy-2-(di-n-propylamino)tetralin on hippocampal serotonin release and induction of hypothermia in awake rats.
    Life sciences, 2004, Apr-23, Volume: 74, Issue:23

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Chromatography, High Pressure Liquid; Citalopram; Drug Antagonism; Hippocampus; Hypothermia, Induced; Injections, Subcutaneous; Male; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Wakefulness

2004
Increased responsiveness of presumed 5-HT cells to citalopram in adult rats subjected to prolonged maternal separation relative to brief separation.
    Psychopharmacology, 2004, Volume: 176, Issue:3-4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding Sites; Citalopram; Dose-Response Relationship, Drug; Electrophysiology; Female; In Situ Hybridization; Male; Maternal Deprivation; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Pregnancy; Radioligand Assay; Raphe Nuclei; Rats; Receptor, Serotonin, 5-HT1A; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2004
Effects of acute and long-term administration of escitalopram and citalopram on serotonin neurotransmission: an in vivo electrophysiological study in rat brain.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analysis of Variance; Animals; Brain; Citalopram; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Male; Neurons; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

2005
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors

2005
alpha(2)-Adrenoceptor involvement in the in vitro inhibitory effect of citalopram on a subpopulation of rat locus coeruleus neurons.
    European journal of pharmacology, 2005, Jul-04, Volume: 517, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amphetamines; Animals; Bridged Bicyclo Compounds, Heterocyclic; Brimonidine Tartrate; Citalopram; Dose-Response Relationship, Drug; Duloxetine Hydrochloride; Idazoxan; In Vitro Techniques; Locus Coeruleus; Male; Methiothepin; Naloxone; Narcotic Antagonists; Neurons; Norepinephrine; Oxazines; Piperazines; Piperidines; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Opioid, mu; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

2005
Effects on serotonin of (-)nicotine and dimethylphenylpiperazinium in the dorsal raphe and nucleus accumbens of freely behaving rats.
    Neuroscience, 2005, Volume: 135, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Carrier Proteins; Citalopram; Dimethylphenylpiperazinium Iodide; Male; Microdialysis; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Nucleus Accumbens; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Presynaptic; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

2005
Evidence of reuptake inhibition responsible for mecamylamine-evoked increases in extracellular serotonin.
    Brain research, 2006, Feb-16, Volume: 1073-1074

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aconitine; Animals; Citalopram; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Mecamylamine; Microdialysis; Nicotinic Antagonists; Raphe Nuclei; Rats; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Wakefulness

2006
Imipramine and citalopram reverse corticosterone-induced alterations in the effects of the activation of 5-HT(1A) and 5-HT(2) receptors in rat frontal cortex.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2006, Volume: 57, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Antidepressive Agents, Second-Generation; Antidepressive Agents, Tricyclic; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Citalopram; Corticosterone; Depression; Frontal Lobe; Imipramine; Male; Models, Animal; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists; Stress, Psychological

2006
Evidence that the deficit in sexual behavior in adult rats neonatally exposed to citalopram is a consequence of 5-HT1 receptor stimulation during development.
    Brain research, 2006, Dec-13, Volume: 1125, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Citalopram; Female; Male; Pregnancy; Quinoxalines; Rats; Rats, Long-Evans; Reaction Time; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sexual Behavior, Animal; Sexual Dysfunction, Physiological

2006
Brain-derived neurotrophic factor-deficient mice exhibit a hippocampal hyperserotonergic phenotype.
    The international journal of neuropsychopharmacology, 2008, Volume: 11, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain Chemistry; Brain-Derived Neurotrophic Factor; Citalopram; Dose-Response Relationship, Drug; Electrophysiology; Hippocampus; Male; Mice; Mice, Knockout; Microdialysis; Paroxetine; Phenotype; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Synaptic Transmission

2008
Differential regulation of serotonin-1A receptor-stimulated [35S]GTP gamma S binding in the dorsal raphe nucleus by citalopram and escitalopram.
    European journal of pharmacology, 2008, Mar-31, Volume: 583, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Binding, Competitive; Citalopram; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Imipramine; In Vitro Techniques; Male; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists

2008
Lasting syndrome of depression produced by reduction in serotonin uptake during postnatal development: evidence from sleep, stress, and behavior.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Apr-02, Volume: 28, Issue:14

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Animals, Newborn; Antidepressive Agents; Behavior, Animal; Choice Behavior; Citalopram; Corticosterone; Depressive Disorder; Disease Models, Animal; Fluoxetine; Food Preferences; Hypothermia; Maze Learning; Mice; Mice, Knockout; Serotonin; Serotonin Plasma Membrane Transport Proteins; Sleep Wake Disorders; Spectrum Analysis; Stress, Physiological; Wakefulness

2008
Glucocorticoid receptor antagonism augments fluoxetine-induced downregulation of the 5-HT transporter.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Autoradiography; Brain; Citalopram; Densitometry; Down-Regulation; Fluoxetine; In Situ Hybridization; Male; Rats; Receptor, Serotonin, 5-HT1A; Receptors, Glucocorticoid; RNA, Messenger; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Agonists; Serotonin Plasma Membrane Transport Proteins; Steroids; Sulfones; Tritium; Tryptophan Hydroxylase

2009
Insensitivity of NMRI mice to selective serotonin reuptake inhibitors in the tail suspension test can be reversed by co-treatment with 5-hydroxytryptophan.
    Psychopharmacology, 2008, Volume: 199, Issue:2

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Citalopram; Dose-Response Relationship, Drug; Fluoxetine; Genotype; Hindlimb Suspension; Hippocampus; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Microdialysis; Motor Activity; Norepinephrine Plasma Membrane Transport Proteins; Prefrontal Cortex; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Species Specificity; Tyrosine 3-Monooxygenase

2008
Delta(9)-tetrahydrocannabinol prolongs the immobility time in the mouse forced swim test: involvement of cannabinoid CB(1) receptor and serotonergic system.
    European journal of pharmacology, 2008, Jul-28, Volume: 589, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Brain; Citalopram; Dose-Response Relationship, Drug; Dronabinol; Injections, Intraperitoneal; Male; Mice; Motor Activity; Phenols; Piperazines; Piperidines; Psychotropic Drugs; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Rimonabant; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Succinimides; Sulfonamides; Swimming

2008
Differential long-term effects of MDMA on the serotoninergic system and hippocampal cell proliferation in 5-HTT knock-out vs. wild-type mice.
    The international journal of neuropsychopharmacology, 2008, Volume: 11, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Proliferation; Citalopram; Electrophysiology; Female; Hallucinogens; Hindlimb Suspension; Hippocampus; Injections, Intraperitoneal; Male; Membranes; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Patch-Clamp Techniques; Raphe Nuclei; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Agents; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Swimming

2008
Effects of chronic citalopram treatment on 5-HT1A and 5-HT2A receptors in group- and isolation-housed mice.
    European journal of pharmacology, 2008, Sep-28, Volume: 593, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antidepressive Agents; Autoradiography; Brain; Brain Chemistry; Citalopram; Data Interpretation, Statistical; Ketanserin; Male; Mice; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Serotonin Antagonists; Social Environment; Social Isolation

2008
Acute and chronic effects of citalopram on 5-HT1A receptor-labeling by [18F]MPPF and -coupling to receptors-G proteins.
    Synapse (New York, N.Y.), 2009, Volume: 63, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoradiography; Brain; Citalopram; Fluorine Radioisotopes; Guanosine 5'-O-(3-Thiotriphosphate); Male; Mice; Mice, Knockout; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists

2009
Differential effects of acute and repeated citalopram in mouse models of anxiety and depression.
    The international journal of neuropsychopharmacology, 2010, Volume: 13, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents, Second-Generation; Anxiety; Chlordiazepoxide; Citalopram; CREB-Binding Protein; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Gene Expression Regulation; Hindlimb Suspension; Hypothermia; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Statistics, Nonparametric

2010
Serotonin modulates glutamatergic transmission in the rat olfactory tubercle.
    The European journal of neuroscience, 2010, Volume: 31, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Olfactory Pathways; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Synaptic Transmission; Tryptamines

2010
Differential involvement of hippocampal serotonin1A receptors and re-uptake sites in non-cognitive behaviors of Alzheimer's disease.
    Psychopharmacology, 2011, Volume: 213, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Aged, 80 and over; Alzheimer Disease; Autopsy; Binding Sites; Citalopram; Female; Follow-Up Studies; Hippocampus; Humans; Ketanserin; Longitudinal Studies; Male; Prospective Studies; Protein Binding; Receptor, Serotonin, 5-HT1A

2011
Serotonergic modulation of LTP at excitatory and inhibitory synapses in the developing rat visual cortex.
    Neuroscience, 2013, May-15, Volume: 238

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Long-Term Potentiation; Neural Inhibition; Pyramidal Cells; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Synapses; Visual Cortex

2013
Lasting neurobehavioral abnormalities in rats after neonatal activation of serotonin 1A and 1B receptors: possible mechanisms for serotonin dysfunction in autistic spectrum disorders.
    Psychopharmacology, 2014, Volume: 231, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Brain; Citalopram; Exploratory Behavior; Female; Freezing Reaction, Cataleptic; Locomotion; Male; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Social Behavior

2014
Mechanism of action of the bimodal antidepressant vilazodone: evidence for serotonin1A-receptor-mediated auto-augmentation of extracellular serotonin output.
    Psychopharmacology, 2014, Volume: 231, Issue:12

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Benzofurans; Brain; Citalopram; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Fluoxetine; Indoles; Male; Paroxetine; Piperazines; Pyridines; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Vilazodone Hydrochloride

2014
Side effect profile of 5-HT treatments for Parkinson's disease and L-DOPA-induced dyskinesia in rats.
    British journal of pharmacology, 2015, Volume: 172, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antiparkinson Agents; Buspirone; Citalopram; Dyskinesia, Drug-Induced; Levodopa; Male; Parkinson Disease; Psychomotor Performance; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Agonists

2015
Escitalopram Ameliorates Forskolin-Induced Tau Hyperphosphorylation in HEK239/tau441 Cells.
    Journal of molecular neuroscience : MN, 2015, Volume: 56, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Citalopram; Colforsin; Cyclic AMP-Dependent Protein Kinases; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; HEK293 Cells; Humans; Phosphorylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-akt; Selective Serotonin Reuptake Inhibitors; tau Proteins

2015
Deletion of GIRK2 Subunit of GIRK Channels Alters the 5-HT1A Receptor-Mediated Signaling and Results in a Depression-Resistant Behavior.
    The international journal of neuropsychopharmacology, 2015, May-08, Volume: 18, Issue:11

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Antidepressive Agents, Second-Generation; Bee Venoms; Citalopram; Depressive Disorder; Disease Models, Animal; Dorsal Raphe Nucleus; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Hippocampus; Male; Mice, Inbred C57BL; Mice, Knockout; Neurogenesis; Neurons; Potassium Channel Blockers; Resilience, Psychological; Serotonin Receptor Agonists

2015
The role of serotonergic mechanism in the rat prefrontal cortex for controlling the micturition reflex: An in vivo microdialysis study.
    Neurourology and urodynamics, 2016, Volume: 35, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Citalopram; Dopamine; Female; Glutamic Acid; Microdialysis; Muscle Contraction; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Reflex; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Urinary Bladder; Urination

2016
Citalopram reduces glutamatergic synaptic transmission in the auditory cortex via activation of 5-HT1A receptors.
    Neuroreport, 2019, 12-18, Volume: 30, Issue:18

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Auditory Cortex; Citalopram; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Piperazines; Pyramidal Cells; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission

2019