8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine has been researched along with 8-phenyltheophylline in 5 studies
| Studies (8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine) | Trials (8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine) | Recent Studies (post-2010) (8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine) | Studies (8-phenyltheophylline) | Trials (8-phenyltheophylline) | Recent Studies (post-2010) (8-phenyltheophylline) |
|---|---|---|---|---|---|
| 16 | 0 | 3 | 518 | 0 | 11 |
| Protein | Taxonomy | 8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine (IC50) | 8-phenyltheophylline (IC50) |
|---|---|---|---|
| Adenosine receptor A3 | Homo sapiens (human) | 1.25 | |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | 0.2756 | |
| Adenosine receptor A1 | Bos taurus (cattle) | 0.003 | |
| Adenosine receptor A2a | Homo sapiens (human) | 0.454 | |
| Adenosine receptor A2b | Homo sapiens (human) | 0.3125 | |
| Adenosine receptor A2b | Rattus norvegicus (Norway rat) | 1.1 | |
| Adenosine receptor A1 | Homo sapiens (human) | 1.34 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 3 (60.00) | 18.7374 |
| 1990's | 1 (20.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Jacobson, KA; van Galen, PJ; Williams, M | 1 |
| Barone, S; Bradbury, BJ; Campagne, JM; Daly, JW; Jacobson, KA; Kammula, U; Kiriasis, L; Neumeyer, JL; Pfleiderer, W; Secunda, S | 1 |
| Craig, RH; Daluge, SM; Earl, CQ; Linden, J; Patel, A | 1 |
| Daly, JW; Jacobson, KA; Kirk, KL; Padgett, W; Ukena, D | 1 |
| Jacobson, KA; Kim, HS; Kim, SA; Linden, J; Marshall, MA; Melman, N; Müller, CE | 1 |
1 review(s) available for 8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine and 8-phenyltheophylline
| Article | Year |
|---|---|
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship | 1992 |
4 other study(ies) available for 8-(4-carboxymethyloxy)phenyl-1,3-dipropylxanthine and 8-phenyltheophylline
| Article | Year |
|---|---|
Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.
Topics: Animals; Binding, Competitive; Chemical Phenomena; Chemistry; In Vitro Techniques; Radioligand Assay; Rats; Receptors, Purinergic; Structure-Activity Relationship; Sulfur; Xanthines | 1989 |
125I-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Affinity Labels; Algorithms; Animals; Binding, Competitive; Brain; Cattle; Humans; Iodine Radioisotopes; Iodobenzenes; Isotope Labeling; Kinetics; Ligands; Membranes; Rats; Rats, Inbred Strains; Receptors, Purinergic; Sodium Chloride; Structure-Activity Relationship; Theophylline; Xanthines | 1988 |
Xanthine functionalized congeners as potent ligands at A2-adenosine receptors.
Topics: Adenylyl Cyclases; Blood Platelets; Humans; Magnetic Resonance Spectroscopy; Mass Spectrometry; Receptors, Purinergic; Structure-Activity Relationship; Xanthines | 1987 |
Structure-activity relationships at human and rat A2B adenosine receptors of xanthine derivatives substituted at the 1-, 3-, 7-, and 8-positions.
Topics: Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Ligands; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2B; Receptors, Purinergic P1; Recombinant Proteins; Structure-Activity Relationship; Xanthines | 2002 |