7-methoxytacrine has been researched along with physostigmine in 4 studies
Studies (7-methoxytacrine) | Trials (7-methoxytacrine) | Recent Studies (post-2010) (7-methoxytacrine) | Studies (physostigmine) | Trials (physostigmine) | Recent Studies (post-2010) (physostigmine) |
---|---|---|---|---|---|
52 | 1 | 28 | 6,230 | 252 | 331 |
Protein | Taxonomy | 7-methoxytacrine (IC50) | physostigmine (IC50) |
---|---|---|---|
Acetylcholinesterase | Electrophorus electricus (electric eel) | 0.1666 | |
Acetylcholinesterase | Tetronarce californica (Pacific electric ray) | 0.3023 | |
Cholinesterase | Homo sapiens (human) | 0.3055 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.2 | |
Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Acetylcholinesterase | Mus musculus (house mouse) | 0.0269 | |
Acetylcholinesterase | Homo sapiens (human) | 0.0853 | |
Acetylcholinesterase | Bos taurus (cattle) | 0.7197 | |
Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 1.1821 | |
Acetylcholinesterase | Gallus gallus (chicken) | 0.02 | |
Acetylcholinesterase | Rattus norvegicus (Norway rat) | 0.0416 | |
Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Cholinesterase | Equus caballus (horse) | 0.4081 | |
Cholinesterase | Mus musculus (house mouse) | 0.28 | |
Acyl-CoA:cholesterol acyltransferase | Oryctolagus cuniculus (rabbit) | 0.0189 | |
Carboxylic ester hydrolase | Rattus norvegicus (Norway rat) | 0.018 | |
Carboxylic ester hydrolase | Equus caballus (horse) | 1.263 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (25.00) | 18.7374 |
1990's | 2 (50.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (25.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Musílková, J; Tucek, S | 1 |
Menini, C; Rektor, I; Silva-Barrat, C; Svejdová, M | 1 |
Herink, J; Hrdina, V; Koupilová, M | 1 |
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA; Shafiullah, M | 1 |
4 other study(ies) available for 7-methoxytacrine and physostigmine
Article | Year |
---|---|
The binding of cholinesterase inhibitors tacrine (tetrahydroaminoacridine) and 7-methoxytacrine to muscarinic acetylcholine receptors in rat brain in the presence of eserine.
Topics: Animals; Binding, Competitive; Cerebellum; Cerebral Cortex; Cholinesterase Inhibitors; Female; Kinetics; Physostigmine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tacrine | 1991 |
Unexpected potentializing effect of a tacrine derivative (9-amino-7-methoxy-1,2,3,4 tetrahydroacridine) upon the non-epileptic myoclonus in baboons Papio papio.
Topics: Animals; Atropine; Drug Synergism; Epilepsies, Myoclonic; Myoclonus; Papio; Physostigmine; Tacrine | 1990 |
Effects of tetrahydroaminoacridine (tacrine) derivatives and physostigmine in convulsions induced by pentylenetetrazol.
Topics: Aminoacridines; Animals; Cholinesterase Inhibitors; Male; Pentylenetetrazole; Physostigmine; Rats; Rats, Inbred Strains; Seizures; Tacrine | 1989 |
Pretreatment for acute exposure to diisopropylfluorophosphate: in vivo efficacy of various acetylcholinesterase inhibitors.
Topics: Amiloride; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocytes; Female; Humans; Inhibitory Concentration 50; Isoflurophate; Male; Methylene Blue; Metoclopramide; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Tacrine; Tiapride Hydrochloride | 2011 |