7-hydroxy-2-n,n-dipropylaminotetralin and sulpiride

7-hydroxy-2-n,n-dipropylaminotetralin has been researched along with sulpiride in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's15 (65.22)18.2507
2000's7 (30.43)29.6817
2010's1 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burris, KD; Filtz, TM; Kung, HF; Kung, MP; Molinoff, PB; Pacheco, MA1
Diaz, J; Giros, B; Lévesque, D; Martres, MP; Morgat, JL; Pilon, C; Schott, D; Schwartz, JC; Sokoloff, P; Souil, E1
Cooper, SJ; Gilbert, DB; Millar, J1
Middlemiss, DN; Reavill, C; Storey, VJ1
De Souza, EB; Grigoriadis, DE; Levant, B1
Booze, RM; Wallace, DR1
Misu, Y; Okumura, F; Sato, K; Ueda, H1
Izenwasser, S; Katz, JL1
Buell, G; Hussy, N; Jones, KA; North, RA; Werner, P1
Cools, AR; Kitamura, M; Kobayashi, M; Koshikawa, N1
Freeman, KA; Mao, A; Tallarida, RJ1
Coronas, V; Jourdan, F; Liang, JJ; Moyse, E; Srivastava, LK1
Costall, B; Neill, JC; Smith, AG1
Audinot, V; Cussac, D; Dubuffet, T; Lavielle, G; Loutz, A; Millan, MJ; Newman-Tancredi, A1
Ahmad, B; Darmani, NA; Zhao, W1
Hillefors, M; von Euler, G1
Okuyama, S; Takamori, K; Yoshida, S1
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH1
Gomes, P; Hopfer, U; Jose, PA; Pedrosa, R; Soares-da-Silva, P1
Barik, S; de Beaurepaire, R1
Cummins, R; Gnoffo, Z; Kew, JN; Roberts, C1
Dai, Z; Kang, L; Ma, L; Wang, L1
Ananthan, S; Głowacka, U; Kosmowska, B; Ossowska, K; Wardas, J1

Other Studies

23 other study(ies) available for 7-hydroxy-2-n,n-dipropylaminotetralin and sulpiride

ArticleYear
Lack of discrimination by agonists for D2 and D3 dopamine receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1995, Volume: 12, Issue:4

    Topics: Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes

1995
Identification, characterization, and localization of the dopamine D3 receptor in rat brain using 7-[3H]hydroxy-N,N-di-n-propyl-2-aminotetralin.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Sep-01, Volume: 89, Issue:17

    Topics: Animals; Brain; Brain Mapping; Cell Membrane; Cells, Cultured; Drug Design; Gene Expression; In Vitro Techniques; Male; Nucleic Acid Hybridization; Rats; Rats, Inbred Strains; Receptors, Dopamine; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes

1992
The putative dopamine D3 agonist, 7-OH-DPAT, reduces dopamine release in the nucleus accumbens and electrical self-stimulation to the ventral tegmentum.
    Brain research, 1995, May-29, Volume: 681, Issue:1-2

    Topics: Animals; Dopamine; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Electrodes, Implanted; Female; Male; Nucleus Accumbens; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Stimulation; Sulpiride; Tetrahydronaphthalenes; Ventral Tegmental Area

1995
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
    Neuropharmacology, 1995, Volume: 34, Issue:4

    Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes

1995
Relative affinities of dopaminergic drugs at dopamine D2 and D3 receptors.
    European journal of pharmacology, 1995, May-24, Volume: 278, Issue:3

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Caudate Nucleus; Cerebellum; CHO Cells; Cricetinae; Dopamine Agents; Iodine Radioisotopes; Male; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sensitivity and Specificity; Sulpiride; Tetrahydronaphthalenes

1995
Dopamine D2 and D3 receptors in the rat striatum and nucleus accumbens: use of 7-OH-DPAT and [125I]-iodosulpride.
    Synapse (New York, N.Y.), 1995, Volume: 19, Issue:1

    Topics: Animals; Autoradiography; Binding, Competitive; Cell Membrane; Corpus Striatum; Dopamine Agonists; Iodine Radioisotopes; Kinetics; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes

1995
6-OHDA-induced lesion of the nigrostriatal dopaminergic neurons potentiates the inhibitory effect of 7-OHDPAT, a selective D3 agonist, on acetylcholine release during striatal microdialysis in conscious rats.
    Brain research, 1994, Aug-29, Volume: 655, Issue:1-2

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dopamine Agonists; Male; Medial Forebrain Bundle; Microdialysis; Neostriatum; Oxidopamine; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes

1994
7-OH-DPAT antagonizes dopamine D2 receptor-inhibited adenylyl cyclase activity.
    Life sciences, 1994, Volume: 55, Issue:14

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Binding, Competitive; Colforsin; Dopamine; Dopamine D2 Receptor Antagonists; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes; Tritium

1994
D2, D3, and D4 dopamine receptors couple to G protein-regulated potassium channels in Xenopus oocytes.
    Molecular pharmacology, 1996, Volume: 49, Issue:4

    Topics: Animals; Base Sequence; Dopamine; Female; GTP-Binding Proteins; Molecular Sequence Data; Oocytes; Pertussis Toxin; Potassium Channels; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Sulpiride; Tetrahydronaphthalenes; Virulence Factors, Bordetella; Xenopus laevis

1996
Behavioural effects of 7-OH-DPAT are solely due to stimulation of dopamine D2 receptors in the shell of the nucleus accumbens; turning behaviour.
    European journal of pharmacology, 1996, Jul-25, Volume: 308, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Benzopyrans; Domperidone; Dopamine Agonists; Dopamine Antagonists; Male; Movement; Nucleus Accumbens; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes

1996
Transient loss of dopamine autoreceptor control in the presence of highly potent dopamine agonists.
    Life sciences, 1996, Volume: 59, Issue:21

    Topics: Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Male; Phenethylamines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes

1996
Identification and localization of dopamine receptor subtypes in rat olfactory mucosa and bulb: a combined in situ hybridization and ligand binding radioautographic approach.
    Journal of chemical neuroanatomy, 1997, Volume: 12, Issue:4

    Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Binding, Competitive; Domperidone; Dopamine Agonists; Dopamine Antagonists; In Situ Hybridization; Iodine Radioisotopes; Male; Olfactory Bulb; Olfactory Mucosa; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes

1997
The dopamine D3/D2 receptor agonist 7-OH-DPAT induces cognitive impairment in the marmoset.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 63, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Callithrix; Cognition; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Female; Male; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydronaphthalenes; Yohimbine

1999
Novel benzopyrano[3,4-c]pyrrole derivatives as potent and selective dopamine D3 receptor antagonist.
    Bioorganic & medicinal chemistry letters, 1999, Jul-19, Volume: 9, Issue:14

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Iodine Radioisotopes; Pyrroles; Pyrrolidines; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Sulpiride; Tetrahydronaphthalenes; Transfection

1999
The role of D2 and D3 dopamine receptors in the mediation of emesis in Cryptotis parva (the least shrew).
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12

    Topics: Analysis of Variance; Animals; Apomorphine; Benzopyrans; Brain Chemistry; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Indans; Male; Oxazines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Shrews; Species Specificity; Sulpiride; Tetrahydronaphthalenes; Vomiting

1999
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
    Neurochemistry international, 2001, Volume: 38, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes

2001
Repeated treatment with imipramine, fluvoxamine and tranylcypromine decreases the number of escape failures by activating dopaminergic systems in a rat learned helplessness test.
    Life sciences, 2001, Sep-07, Volume: 69, Issue:16

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Benzazepines; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Escape Reaction; Fluvoxamine; Helplessness, Learned; Imipramine; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes; Tranylcypromine

2001
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
    Psychopharmacology, 2003, Volume: 166, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes

2003
Gialpha3 protein-coupled dopamine D3 receptor-mediated inhibition of renal NHE3 activity in SHR proximal tubular cells is a PLC-PKC-mediated event.
    American journal of physiology. Renal physiology, 2004, Volume: 287, Issue:5

    Topics: Animals; Calcium; Cell Line; Cholera Toxin; Dopamine Antagonists; Down-Regulation; Flavonoids; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Kidney Tubules, Proximal; Pertussis Toxin; Protein Kinase C; Pyridines; Rats; Rats, Inbred SHR; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, G-Protein-Coupled; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers; Sulpiride; Tetrahydronaphthalenes; Type C Phospholipases

2004
Dopamine D3 modulation of locomotor activity and sleep in the nucleus accumbens and in lobules 9 and 10 of the cerebellum in the rat.
    Progress in neuro-psychopharmacology & biological psychiatry, 2005, Volume: 29, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Amphetamine; Animals; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Female; Haloperidol; Microinjections; Motor Activity; Naphthalenes; Nucleus Accumbens; Pyrrolidines; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sleep; Sulpiride; Tetrahydronaphthalenes

2005
Dopamine D3 receptor modulation of dopamine efflux in the rat nucleus accumbens.
    European journal of pharmacology, 2006, Mar-18, Volume: 534, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Haloperidol; Male; Nitriles; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2006
Different roles of dopamine receptor subtypes in footshock stress-induced enhancement of morphine conditioned place preference.
    Neuroscience letters, 2006, Nov-27, Volume: 409, Issue:1

    Topics: Animals; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Dose-Response Relationship, Drug; Electroshock; Male; Morphine; Narcotics; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stress, Psychological; Sulpiride; Tetrahydronaphthalenes

2006
Pramipexole at a Low Dose Induces Beneficial Effect in the Harmaline-induced Model of Essential Tremor in Rats.
    CNS neuroscience & therapeutics, 2016, Volume: 22, Issue:1

    Topics: Amisulpride; Animals; Anti-Dyskinesia Agents; Benzothiazoles; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Essential Tremor; Haloperidol; Harmaline; Imidazoles; Male; Movement; Nitriles; Pramipexole; Pyridines; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes; Treatment Outcome

2016