7-hydroxy-2-n,n-dipropylaminotetralin and raclopride

7-hydroxy-2-n,n-dipropylaminotetralin has been researched along with raclopride in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (60.00)18.2507
2000's8 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Foulon, C; Kung, HF; Kung, MP1
Malmberg, A; Mohell, N1
Mignot, E; Nishino, S; Reid, MS; Sampathkumaran, R; Siegel, JM; Tafti, M1
Dijkstra, D; Farde, L; Hall, H; Halldin, C; Pauli, S; Pugsley, TA; Sedvall, G; Sokoloff, P; Wikström, H; Wise, LD1
Fernandez, AG; O'Neill, MF; Palacios, JM; Silvestre, JS1
Creese, I; Florijn, WJ; Tarazi, FI1
Gallagher, DW; McInerney, S; Primus, RJ; Shaw, K; Tallman, JF; Thurkauf, A; Xu, J; Yevich, E1
Ahlenius, S; Wanderoy, MH; Westlind-Danielsson, A1
Mohell, N1
Costall, B; Neill, JC; Smith, AG1
Ballard, C; Burn, D; Court, JA; Jaros, E; Johnson, M; Lloyd, S; Marshall, EF; McKeith, IG; Perry, EK; Perry, RH; Piggott, MA; Thomas, N1
Brown, RE; Dastur, FN; McGregor, IS1
Boulay, D; Depoortere, R; Perrault, G; Sanger, DJ1
Hillefors, M; von Euler, G1
Ahlenius, S; Eltayb, A; Lindblom, S; Oerther, S1
Berra, R; Flores, G; Gómez, Mde J; Nadeau, R; Rousseau, G; Suárez, J1
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH1
Chu, TC; He, Q; Potter, DE1
Cooper, SJ; Genn, RF; Higgs, S1
Chu, E; Chu, J; Chu, TC; Socci, RR1

Other Studies

20 other study(ies) available for 7-hydroxy-2-n,n-dipropylaminotetralin and raclopride

ArticleYear
Synthesis of (R,S)-2'-trans-7-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'- propenyl)-amino]tetralin (trans-7-OH-PIPAT): a new D3 dopamine receptor ligand.
    Journal of medicinal chemistry, 1993, May-14, Volume: 36, Issue:10

    Topics: Binding Sites; Dopamine Agents; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Stereoisomerism; Tetrahydronaphthalenes

1993
Characterization of [3H]quinpirole binding to human dopamine D2A and D3 receptors: effects of ions and guanine nucleotides.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:2

    Topics: Animals; Binding, Competitive; Ergolines; Guanylyl Imidodiphosphate; Humans; Magnesium; Male; Mice; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sodium; Tetrahydronaphthalenes

1995
Local administration of dopaminergic drugs into the ventral tegmental area modulates cataplexy in the narcoleptic canine.
    Brain research, 1996, Sep-09, Volume: 733, Issue:1

    Topics: Amygdala; Animals; Azepines; Cataplexy; Disease Models, Animal; Dogs; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Electroencephalography; Electromyography; Electrooculography; Female; Globus Pallidus; Male; Microdialysis; Pons; Putamen; Quinpirole; Raclopride; Reticular Formation; Salicylamides; Sleep, REM; Tetrahydronaphthalenes; Ventral Tegmental Area

1996
Autoradiographic localisation of D3-dopamine receptors in the human brain using the selective D3-dopamine receptor agonist (+)-[3H]PD 128907.
    Psychopharmacology, 1996, Volume: 128, Issue:3

    Topics: Adult; Autoradiography; Benzopyrans; Brain Chemistry; Dopamine Agonists; Dopamine Antagonists; Female; Guanosine Triphosphate; Humans; Male; Middle Aged; Oxazines; Raclopride; Receptors, Dopamine; Salicylamides; Tetrahydronaphthalenes

1996
Effects of a range of dopamine receptor agonists and antagonists on ethanol intake in the rat.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Alcohol Drinking; Animals; Benzazepines; Dopamine Agonists; Dopamine Antagonists; Male; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes

1996
Dopamine receptor subtypes: differential regulation after 8 months treatment with antipsychotic drugs.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Benzazepines; Brain; Clozapine; Corpus Striatum; Haloperidol; Iodine Radioisotopes; Male; Organ Specificity; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Spiperone; Tetrahydronaphthalenes; Time Factors; Tritium; Up-Regulation

1997
II. Localization and characterization of dopamine D4 binding sites in rat and human brain by use of the novel, D4 receptor-selective ligand [3H]NGD 94-1.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: Animals; Autoradiography; Brain; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Imidazoles; Male; Pyrimidines; Raclopride; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides; Tetrahydronaphthalenes; Tritium

1997
Dopamine D2 receptor upregulation in rat neostriatum following in vivo infusion of forskolin.
    Neuroreport, 1997, Sep-08, Volume: 8, Issue:13

    Topics: Animals; Cerebral Ventricles; Colforsin; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; In Vitro Techniques; Infusions, Parenteral; Male; Neostriatum; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Tetrahydronaphthalenes; Up-Regulation

1997
Agonist and inverse agonist activity at the dopamine D3 receptor measured by guanosine 5'--gamma-thio-triphosphate--35S- binding.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:1

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Mice; Pertussis Toxin; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes; Virulence Factors, Bordetella

1998
The dopamine D3/D2 receptor agonist 7-OH-DPAT induces cognitive impairment in the marmoset.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 63, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Callithrix; Cognition; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Female; Male; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydronaphthalenes; Yohimbine

1999
Striatal dopaminergic markers in dementia with Lewy bodies, Alzheimer's and Parkinson's diseases: rostrocaudal distribution.
    Brain : a journal of neurology, 1999, Volume: 122 ( Pt 8)

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Autoradiography; Corpus Striatum; Dementia; Dopamine; Female; Homovanillic Acid; Humans; Lewy Bodies; Male; Mazindol; Middle Aged; Parkinson Disease; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes; Tritium

1999
Dopaminergic modulation of rat pup ultrasonic vocalizations.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Animals, Newborn; Benzazepines; Body Temperature; Body Temperature Regulation; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Male; Motor Activity; Quinpirole; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Tetrahydronaphthalenes; Vocalization, Animal

1999
Decreased locomotor activity after microinjection of dopamine D2/D3 receptor agonists and antagonists into lobule 9/10 of the cerebellum: a D3 receptor mediated effect?
    Progress in neuro-psychopharmacology & biological psychiatry, 2000, Volume: 24, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Male; Microinjections; Motor Activity; Quinolines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2000
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
    Neurochemistry international, 2001, Volume: 38, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes

2001
Additive hypothermic effects of the 5-HT1A receptor agonist 8-OH-DPAT and the dopamine D2/3 receptor agonist 7-OH-DPAT in the rat.
    Acta physiologica Scandinavica, 2001, Volume: 172, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dopamine Agonists; Hypothermia; Male; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Tetrahydronaphthalenes

2001
Functional and autoradiographic characterization of dopamine D2-like receptors in the guinea pig heart.
    Canadian journal of physiology and pharmacology, 2002, Volume: 80, Issue:6

    Topics: Adenylyl Cyclases; Animals; Autoradiography; Benzamides; Blood Pressure; Blotting, Western; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Guinea Pigs; Heart Rate; In Vitro Techniques; Kinetics; Male; Membranes; Myocardium; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Tetrahydronaphthalenes

2002
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
    Psychopharmacology, 2003, Volume: 166, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes

2003
Biodegradable calcium phosphate nanoparticles as a new vehicle for delivery of a potential ocular hypotensive agent.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2002, Volume: 18, Issue:6

    Topics: Animals; Aqueous Humor; Biodegradation, Environmental; Calcium Phosphates; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Delivery Systems; Female; Intraocular Pressure; Male; Nanotechnology; Ocular Hypertension; Pigmentation; Rabbits; Raclopride; Tetrahydronaphthalenes

2002
The effects of 7-OH-DPAT, quinpirole and raclopride on licking for sucrose solutions in the non-deprived rat.
    Behavioural pharmacology, 2003, Volume: 14, Issue:8

    Topics: Animals; Dopamine Agonists; Dopamine Antagonists; Feeding Behavior; Male; Quinpirole; Raclopride; Rats; Sucrose; Taste; Tetrahydronaphthalenes

2003
7-OH-DPAT-induced inhibition of norepinephrine release in PC12 cells.
    Pharmacology, 2004, Volume: 70, Issue:3

    Topics: Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Gene Expression; Immunoblotting; Immunochemistry; Nerve Growth Factor; Norepinephrine; PC12 Cells; Potassium Chloride; Raclopride; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Reverse Transcriptase Polymerase Chain Reaction; Tetrahydronaphthalenes

2004