7-hydroxy-2-n,n-dipropylaminotetralin has been researched along with quinpirole in 64 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 42 (65.63) | 18.2507 |
2000's | 20 (31.25) | 29.6817 |
2010's | 2 (3.13) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Burris, KD; Filtz, TM; Kung, HF; Kung, MP; Molinoff, PB; Pacheco, MA | 1 |
Griffon, N; Lévesque, D; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P | 1 |
Foulon, C; Kung, HF; Kung, MP | 1 |
Dörfler, M; Gmeiner, P; Hamperl, K; Hübner, H; Tschammer, N | 1 |
Bonifazi, A; Burzynski, C; Donthamsetti, P; Free, RB; Janowsky, A; Javitch, JA; Keck, TM; Kumar, V; Michino, M; Newman, AH; Schweppe, C; Shi, L; Sibley, DR; Zou, MF | 1 |
Bergstrom, DA; Gonzalez, AM; Huang, KX; Kreiss, DS; Sibley, DR; Walters, JR | 1 |
Middlemiss, DN; Reavill, C; Storey, VJ | 1 |
Malmberg, A; Mohell, N | 1 |
Ahlenius, S; Alster, P; Hillegaart, V; Uvnäs-Moberg, K | 2 |
Cox, RF; Freedman, JE; Greif, GJ; Liu, JC; Waszczak, BL | 1 |
Carlsson, A; Huff, RM; Kling-Petersen, T; Svensson, K; Waters, N | 1 |
Alam, AM; Starr, MS | 1 |
Nishi, S; Yamada, S; Yokoo, H | 1 |
Caine, SB; Koob, GF | 1 |
Furukawa, T; Kurashima, M; Nagashima, M; Shirakawa, K; Yamada, K | 1 |
Bristow, LJ; Hutson, PH; Patel, S; Ragan, CI; Seabrook, GR | 1 |
Misu, Y; Okumura, F; Sato, K; Ueda, H | 1 |
Barnhart, WJ; Lehman, DA; Nestler, EJ; Self, DW | 1 |
Franklin, SR; Tang, AH | 1 |
Ashmeade, T; Routledge, C; Taylor, S; Thorn, L | 1 |
Depoortere, R; Perrault, G; Sanger, DJ | 1 |
Domae, M; Furukawa, T; Inoue, T; Kurashima, M; Nagashima, M; Shirakawa, K; Yamada, K | 1 |
Cools, AR; Kitamura, M; Kobayashi, M; Koshikawa, N | 1 |
Ellerbrock, BR; Fici, GJ; Sethy, VH; Wu, H | 1 |
Mignot, E; Nishino, S; Reid, MS; Sampathkumaran, R; Siegel, JM; Tafti, M | 1 |
Freeman, KA; Mao, A; Tallarida, RJ | 1 |
Kamei, J; Ohsawa, M | 1 |
Cho, S; Hadjiconstantinou, M; Neff, NH | 1 |
Coronas, V; Jourdan, F; Liang, JJ; Moyse, E; Srivastava, LK | 1 |
Andersen, SL; Dumont, NL; Teicher, MH | 1 |
Badia, A; Clos, MV; García-Sanz, A; Vivas, NM | 1 |
Bonardi, CM; Hitchcott, PK; Phillips, GD | 1 |
Dall'olio, R; Gandolfi, O; Rimondini, R | 1 |
Mohell, N | 1 |
Dziedzicka-Wasylewska, M; Maj, J; Rogoz, R; Rogóz, Z | 1 |
Reggers, J; Terry, P; Tirelli, E | 1 |
Hagan, JJ; Hatcher, JP | 1 |
Mach, RH; Nader, MA; Sinnott, RS | 1 |
Cook, CD; Picker, MJ; Rodefer, JS | 1 |
Brown, RE; Dastur, FN; McGregor, IS | 1 |
Honda, K; Mignot, E; Nishino, S; Riehl, J | 1 |
Ahmad, B; Darmani, NA; Zhao, W | 1 |
Maj, J; Rogóz, Z; Skuza, G | 1 |
Hillefors, M; von Euler, G | 1 |
Alling, KL; Katz, JL | 1 |
Brus, R; Kostrzewa, RM; Nowak, P; Oswiecimska, J; Szkilnik, R | 1 |
Badia, A; Clos, MV; García-Sanz, A | 1 |
Bridges, RS; Byrnes, EM; Byrnes, JJ | 1 |
Butelman, ER; Kreek, MJ | 1 |
Garcia-Ladona, J; Wicke, K | 1 |
Okuyama, S; Takamori, K; Yoshida, S | 1 |
Dlaboga, D; Dziedzicka-Wasylewska, M; Maj, J; Rogoz, Z; Skuza, G | 1 |
Rogóz, Z; Skuza, G | 1 |
Dall'Olio, R; Gaggi, R; Gandolfi, O; Tanda, O; Voltattorni, M | 1 |
Kayir, H; Uzbay, IT | 1 |
Heidbreder, CA; Shilliam, CS | 1 |
Cooper, SJ; Genn, RF; Higgs, S | 1 |
Beardsley, PM; Cook, CD | 1 |
Blaha, CD; Forster, GL; Hendry, IA; Holgate, J; Leck, KJ; Matthaei, KI | 1 |
Blessing, WW; Hagan, JJ; Heidbreder, CA; Ootsuka, Y | 1 |
Greedy, B; Grundt, P; Husbands, SM; Koffarnus, MN; Newman, AH; Woods, JH | 1 |
Collo, G; Missale, C; Spano, P; Zanetti, S | 1 |
Yoshida, N; Yoshikawa, T | 1 |
64 other study(ies) available for 7-hydroxy-2-n,n-dipropylaminotetralin and quinpirole
Article | Year |
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Lack of discrimination by agonists for D2 and D3 dopamine receptors.
Topics: Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes | 1995 |
A functional test identifies dopamine agonists selective for D3 versus D2 receptors.
Topics: Animals; CHO Cells; Cricetinae; Dopamine Agents; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3 | 1995 |
Synthesis of (R,S)-2'-trans-7-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'- propenyl)-amino]tetralin (trans-7-OH-PIPAT): a new D3 dopamine receptor ligand.
Topics: Binding Sites; Dopamine Agents; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Stereoisomerism; Tetrahydronaphthalenes | 1993 |
Novel D3 selective dopaminergics incorporating enyne units as nonaromatic catechol bioisosteres: synthesis, bioactivity, and mutagenesis studies.
Topics: Catechols; Cyclic AMP; Humans; Molecular Structure; Mutagenesis; Protein Binding; Receptors, Dopamine D3; Structure-Activity Relationship | 2008 |
Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.
Topics: Animals; Benzimidazoles; Binding Sites; Chemistry Techniques, Synthetic; CHO Cells; Cricetulus; Humans; Ligands; Models, Molecular; Molecular Dynamics Simulation; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship | 2016 |
Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities.
Topics: Aminoquinolines; Animals; Apomorphine; Azepines; Benzothiazoles; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Male; Neurons; Phenethylamines; Piperidines; Pramipexole; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Substantia Nigra; Tetrahydronaphthalenes; Thiazoles; Thiophenes; Transfection | 1995 |
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes | 1995 |
Characterization of [3H]quinpirole binding to human dopamine D2A and D3 receptors: effects of ions and guanine nucleotides.
Topics: Animals; Binding, Competitive; Ergolines; Guanylyl Imidodiphosphate; Humans; Magnesium; Male; Mice; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sodium; Tetrahydronaphthalenes | 1995 |
Suggestive evidence for a DA D3 receptor-mediated increase in the release of oxytocin in the male rat.
Topics: Animals; Bromocriptine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Oxytocin; Prolactin; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sex Factors; Tetrahydronaphthalenes | 1995 |
The putative dopamine D3 receptor agonist 7-OH-DPAT: lack of mesolimbic selectivity.
Topics: Animals; Caudate Nucleus; Dopamine Agonists; Dose-Response Relationship, Drug; Electrophysiology; Ergolines; Injections, Intravenous; Iontophoresis; Male; Neostriatum; Neurons; Nucleus Accumbens; Patch-Clamp Techniques; Putamen; Quinpirole; Rats; Rats, Sprague-Dawley; Stereoisomerism; Substantia Nigra; Tetrahydronaphthalenes; Ventral Tegmental Area | 1994 |
Behavioral and neurochemical data suggest functional differences between dopamine D2 and D3 receptors.
Topics: Analysis of Variance; Animals; Apomorphine; Benzothiazoles; CHO Cells; Cricetinae; Cricetulus; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Microdialysis; Mitogens; Motor Activity; Piperidines; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Thiazoles; Transfection | 1994 |
Bimodal effects of dopamine D2 receptor agonists on zero Mg(2+)-induced epileptiform activity in the rat cingulate cortex slice.
Topics: Animals; Benzazepines; Dopamine D2 Receptor Antagonists; Epilepsy; Ergolines; Evoked Potentials; Female; Gyrus Cinguli; In Vitro Techniques; Lisuride; Magnesium; Male; Oxazines; Phenethylamines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes | 1994 |
Differential effects of dopamine agonists on evoked dopamine release from slices of striatum and nucleus accumbens in rats.
Topics: Animals; Apomorphine; Dopamine; Dopamine Agonists; Electric Stimulation; Ergolines; In Vitro Techniques; Male; Neostriatum; Nerve Endings; Nucleus Accumbens; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 1994 |
Modulation of cocaine self-administration in the rat through D-3 dopamine receptors.
Topics: Animals; Apomorphine; Cocaine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Self Administration; Tetrahydronaphthalenes | 1993 |
Effects of putative dopamine D3 receptor agonists, 7-OH-DPAT, and quinpirole, on yawning, stereotypy, and body temperature in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Body Temperature; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Tetrahydronaphthalenes; Yawning | 1995 |
Functional relevance of dopamine receptors.
Topics: Antipsychotic Agents; Dopamine Agonists; Dopamine Antagonists; Ergolines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Tetrahydronaphthalenes | 1995 |
L-DOPA inhibits spontaneous acetylcholine release from the striatum of experimental Parkinson's model rats.
Topics: Acetylcholine; Analysis of Variance; Animals; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Drug Synergism; Ergolines; Levodopa; Male; Oxidopamine; Parkinson Disease, Secondary; Quinpirole; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes | 1995 |
Opposite modulation of cocaine-seeking behavior by D1- and D2-like dopamine receptor agonists.
Topics: Animals; Behavior, Addictive; Behavior, Animal; Benzazepines; Caffeine; Cocaine; Dopamine Agonists; Ergolines; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Recurrence; Reinforcement, Psychology; Substance-Related Disorders; Tetrahydronaphthalenes | 1996 |
Dopamine agonists facilitate footshock-elicited locomotion in rats, and suppress level-press responding for food.
Topics: Animals; Apomorphine; Clonidine; Conditioning, Operant; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Locomotion; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes | 1995 |
Elucidation of D3 receptor function in vivo: do D3 receptors mediate inhibition of dopamine neuronal activity?
Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Male; Mice; Mice, Inbred Strains; Microdialysis; Neurons; Nucleus Accumbens; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 1996 |
Effects of selective serotonin and dopamine agonists on plasma levels of glucose, insulin and glucagon in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Glucose; Bromocriptine; Buspirone; Dopamine Agonists; Ergolines; Glucagon; Insulin; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Tetrahydronaphthalenes | 1996 |
Behavioural effects in the rat of the putative dopamine D3 receptor agonist 7-OH-DPAT: comparison with quinpirole and apomorphine.
Topics: Animals; Apomorphine; Behavior, Animal; Conditioning, Operant; Dopamine Agonists; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Rats, Wistar; Self Administration; Stereotyped Behavior; Tetrahydronaphthalenes | 1996 |
Inhibitory effects of putative dopamine D3 receptor agonists, 7-OH-DPAT and quinpirole, on prolactin secretion in rats.
Topics: alpha-Methyltyrosine; Animals; Body Temperature; Depression, Chemical; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estradiol; Male; Methyltyrosines; Prolactin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase; Yawning | 1996 |
Behavioural effects of 7-OH-DPAT are solely due to stimulation of dopamine D2 receptors in the shell of the nucleus accumbens; turning behaviour.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Benzopyrans; Domperidone; Dopamine Agonists; Dopamine Antagonists; Male; Movement; Nucleus Accumbens; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes | 1996 |
D2 and D1 dopaminergic activity of 7-OH-DPAT.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Cells, Cultured; Cerebellum; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Indans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes | 1996 |
Local administration of dopaminergic drugs into the ventral tegmental area modulates cataplexy in the narcoleptic canine.
Topics: Amygdala; Animals; Azepines; Cataplexy; Disease Models, Animal; Dogs; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Electroencephalography; Electromyography; Electrooculography; Female; Globus Pallidus; Male; Microdialysis; Pons; Putamen; Quinpirole; Raclopride; Reticular Formation; Salicylamides; Sleep, REM; Tetrahydronaphthalenes; Ventral Tegmental Area | 1996 |
Transient loss of dopamine autoreceptor control in the presence of highly potent dopamine agonists.
Topics: Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Male; Phenethylamines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes | 1996 |
Effects of diabetes on methamphetamine-induced place preference in mice.
Topics: Animals; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Male; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Streptozocin; Tetrahydronaphthalenes | 1996 |
Regulation of tyrosine hydroxylase and aromatic L-amino acid decarboxylase by dopaminergic drugs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aromatic-L-Amino-Acid Decarboxylases; Benzazepines; Brain; Bromocriptine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Mesencephalon; Mice; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase | 1997 |
Identification and localization of dopamine receptor subtypes in rat olfactory mucosa and bulb: a combined in situ hybridization and ligand binding radioautographic approach.
Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Binding, Competitive; Domperidone; Dopamine Agonists; Dopamine Antagonists; In Situ Hybridization; Iodine Radioisotopes; Male; Olfactory Bulb; Olfactory Mucosa; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes | 1997 |
Developmental differences in dopamine synthesis inhibition by (+/-)-7-OH-DPAT.
Topics: Age Factors; Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Levodopa; Nucleus Accumbens; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Salicylamides; Tetrahydronaphthalenes | 1997 |
D2 dopamine receptors and modulation of spontaneous acetylcholine (ACh) release from rat striatal synaptosomes.
Topics: Acetylcholine; Animals; Benzamides; CHO Cells; Cricetinae; Dopamine Agonists; Humans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Presynaptic; Synaptosomes; Tetrahydronaphthalenes | 1997 |
Enhanced stimulus-reward learning by intra-amygdala administration of a D3 dopamine receptor agonist.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amygdala; Animals; Conditioning, Operant; Discrimination Learning; Dopamine Agonists; Injections; Male; Photic Stimulation; Quinpirole; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Reward; Tetrahydronaphthalenes | 1997 |
Effects of competitive and non-competitive NMDA receptor antagonists on behavioral responses induced by 7-OH-DPAT and quinpirole in rats.
Topics: 2-Amino-5-phosphonovalerate; Animals; Dizocilpine Maleate; Dopamine Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Neostriatum; Nucleus Accumbens; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spiperone; Tetrahydronaphthalenes | 1997 |
Agonist and inverse agonist activity at the dopamine D3 receptor measured by guanosine 5'--gamma-thio-triphosphate--35S- binding.
Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Mice; Pertussis Toxin; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes; Virulence Factors, Bordetella | 1998 |
Effect of antidepressant drugs administered repeatedly on the dopamine D3 receptors in the rat brain.
Topics: Administration, Oral; Amitriptyline; Animals; Antidepressive Agents; Autoradiography; Brain; Citalopram; Dopamine Agonists; Imipramine; Injections, Subcutaneous; Male; Mianserin; Motor Activity; Nucleus Accumbens; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 1998 |
Dopamine 'D2-like' receptor agonists in combination with cocaine: absence of interactive effects on locomotor activity.
Topics: Animals; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Motor Activity; Phenethylamines; Quinpirole; Receptors, Dopamine D2; Tetrahydronaphthalenes | 1997 |
The effects of dopamine D3/D2 receptor agonists on intracranial self stimulation in the rat.
Topics: Animals; Area Under Curve; Brain; Dopamine Agonists; Injections, Subcutaneous; Male; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Stimulation; Tetrahydronaphthalenes | 1998 |
Dopamine D2/D3 receptors modulate cocaine's reinforcing and discriminative stimulus effects in rhesus monkeys.
Topics: Analysis of Variance; Animals; Appetitive Behavior; Behavior, Addictive; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Macaca mulatta; Male; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Tetrahydronaphthalenes; Time Factors | 1999 |
Selective attenuation of the antinociceptive effects of mu opioids by the putative dopamine D3 agonist 7-OH-DPAT.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Opioid; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cycloparaffins; Dopamine Agonists; Dopamine Antagonists; Drug Antagonism; Male; Morphine; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Spiperone; Tetrahydronaphthalenes | 1999 |
Dopaminergic modulation of rat pup ultrasonic vocalizations.
Topics: Animals; Animals, Newborn; Benzazepines; Body Temperature; Body Temperature Regulation; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Male; Motor Activity; Quinpirole; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Tetrahydronaphthalenes; Vocalization, Animal | 1999 |
Dopamine D3 agonists into the substantia nigra aggravate cataplexy but do not modify sleep.
Topics: Animals; Cataplexy; Dogs; Dopamine Agonists; Dose-Response Relationship, Drug; Electroencephalography; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Sleep; Sleep Stages; Substantia Nigra; Tetrahydronaphthalenes; Time Factors; Ventral Tegmental Area | 1999 |
The role of D2 and D3 dopamine receptors in the mediation of emesis in Cryptotis parva (the least shrew).
Topics: Analysis of Variance; Animals; Apomorphine; Benzopyrans; Brain Chemistry; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Indans; Male; Oxazines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Shrews; Species Specificity; Sulpiride; Tetrahydronaphthalenes; Vomiting | 1999 |
The anticataleptic effect of 7-OH-DPAT: are dopamine D3 receptors involved?
Topics: Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Fluphenazine; Haloperidol; Hyperkinesis; Levodopa; Locomotion; Male; Naphthalenes; Pyrrolidines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reserpine; Tetrahydronaphthalenes | 1999 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Discriminative stimulus effects of putative D3 dopamine receptor agonists in rats.
Topics: Animals; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Male; Oxazines; Perception; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 2000 |
7-OH-DPAT, unlike quinpirole, does not prime a yawning response in rats.
Topics: Animals; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Yawning | 2000 |
Differential effect of quinpirole and 7-OH-DPAT on the spontaneous [(3)H]-dopamine efflux from rat striatal synaptosomes.
Topics: Animals; Benzopyrans; Calcium; Calcium Channels; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Neostriatum; Oxazines; Presynaptic Terminals; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Synaptosomes; Tetrahydronaphthalenes; Tetrodotoxin; Tritium | 2001 |
Increased sensitivity of dopamine systems following reproductive experience in rats.
Topics: Animals; Conditioning, Operant; Dextroamphetamine; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Neurotransmitter; Receptors, Presynaptic; Tetrahydronaphthalenes | 2001 |
kappa-Opioid receptor agonist-induced prolactin release in primates is blocked by dopamine D(2)-like receptor agonists.
Topics: Animals; Behavior, Animal; Benzazepines; Benzeneacetamides; Conscious Sedation; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Prolactin; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, kappa; Tetrahydronaphthalenes | 2001 |
The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors.
Topics: Animals; Benzopyrans; Binding, Competitive; CHO Cells; Cricetinae; Dendrites; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Neurons; Oxazines; Piperazines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Sulfur Radioisotopes; Tetrahydronaphthalenes | 2001 |
Repeated treatment with imipramine, fluvoxamine and tranylcypromine decreases the number of escape failures by activating dopaminergic systems in a rat learned helplessness test.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Benzazepines; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Escape Reaction; Fluvoxamine; Helplessness, Learned; Imipramine; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes; Tranylcypromine | 2001 |
Effect of repeated treatment with tianeptine and fluoxetine on central dopamine D(2) /D(3) receptors.
Topics: Animals; Antidepressive Agents, Second-Generation; Antidepressive Agents, Tricyclic; Autoradiography; Brain Chemistry; Caudate Nucleus; Dextroamphetamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Fluoxetine; Islands of Calleja; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Tetrahydronaphthalenes; Thiazepines | 2002 |
A potential antidepressant activity of SA4503, a selective sigma 1 receptor agonist.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Male; Motor Activity; Piperazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, sigma; Stereotyped Behavior; Swimming; Tetrahydronaphthalenes | 2002 |
Nafadotride administration increases D1 and D1/D2 dopamine receptor mediated behaviors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Body Temperature; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Exploratory Behavior; Grooming; Male; Motor Activity; Naphthalenes; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Stimulation, Chemical; Tetrahydronaphthalenes | 2002 |
Bromocriptine and quinpirole, but not 7-OH-DPAT or SKF 38393, potentiate the inhibitory effect of L-NAME on ethanol-induced locomotor activity in mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arginine; Bromocriptine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Ethanol; Male; Mice; Motor Activity; NG-Nitroarginine Methyl Ester; Nitric Oxide; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 2003 |
Gradient of dopamine responsiveness to dopamine receptor agonists in subregions of the rat nucleus accumbens.
Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Dopamine; Dose-Response Relationship, Drug; Male; Microdialysis; Nucleus Accumbens; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Time Factors | 2003 |
The effects of 7-OH-DPAT, quinpirole and raclopride on licking for sucrose solutions in the non-deprived rat.
Topics: Animals; Dopamine Agonists; Dopamine Antagonists; Feeding Behavior; Male; Quinpirole; Raclopride; Rats; Sucrose; Taste; Tetrahydronaphthalenes | 2003 |
Modulation of the discriminative stimulus effects of mu opioid agonists in rats: II. Effects of dopamine D2/3 agonists.
Topics: Animals; Appetitive Behavior; Brain; Discrimination Learning; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Heroin; Male; Methadone; Morphine; Motivation; Nalbuphine; Quinolines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Tetrahydronaphthalenes | 2004 |
Gz proteins are functionally coupled to dopamine D2-like receptors in vivo.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Behavior, Animal; Blotting, Western; Body Temperature; Dopamine; Dopamine Agonists; GTP-Binding Protein alpha Subunits; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D2; Serotonin Receptor Agonists; Tetrahydronaphthalenes; Time Factors | 2006 |
Dopamine D2 receptor stimulation inhibits cold-initiated thermogenesis in brown adipose tissue in conscious rats.
Topics: Adaptation, Physiological; Adipose Tissue, Brown; Animals; Body Temperature Regulation; Cold Temperature; Dopamine Agonists; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Statistics, Nonparametric; Sympathetic Fibers, Postganglionic; Tetrahydronaphthalenes; Thermogenesis | 2007 |
The discriminative stimulus effects of dopamine D2- and D3-preferring agonists in rats.
Topics: Animals; Benzimidazoles; Benzothiazoles; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 2009 |
Dopamine D3 receptor-preferring agonists increase dendrite arborization of mesencephalic dopaminergic neurons via extracellular signal-regulated kinase phosphorylation.
Topics: Amphetamine; Animals; Cell Shape; Cells, Cultured; Dendrites; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Mesencephalon; Mice; Nerve Growth Factors; Neurogenesis; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase | 2008 |
The possible involvement of dopamine D3 receptors in the regulation of gastric emptying in rats.
Topics: 2-Naphthylamine; Animals; Benzopyrans; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Furans; Gastric Emptying; Male; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 2010 |