7-hydroxy-2-n,n-dipropylaminotetralin and quinpirole

7-hydroxy-2-n,n-dipropylaminotetralin has been researched along with quinpirole in 64 studies

Research

Studies (64)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's42 (65.63)18.2507
2000's20 (31.25)29.6817
2010's2 (3.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burris, KD; Filtz, TM; Kung, HF; Kung, MP; Molinoff, PB; Pacheco, MA1
Griffon, N; Lévesque, D; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P1
Foulon, C; Kung, HF; Kung, MP1
Dörfler, M; Gmeiner, P; Hamperl, K; Hübner, H; Tschammer, N1
Bonifazi, A; Burzynski, C; Donthamsetti, P; Free, RB; Janowsky, A; Javitch, JA; Keck, TM; Kumar, V; Michino, M; Newman, AH; Schweppe, C; Shi, L; Sibley, DR; Zou, MF1
Bergstrom, DA; Gonzalez, AM; Huang, KX; Kreiss, DS; Sibley, DR; Walters, JR1
Middlemiss, DN; Reavill, C; Storey, VJ1
Malmberg, A; Mohell, N1
Ahlenius, S; Alster, P; Hillegaart, V; Uvnäs-Moberg, K2
Cox, RF; Freedman, JE; Greif, GJ; Liu, JC; Waszczak, BL1
Carlsson, A; Huff, RM; Kling-Petersen, T; Svensson, K; Waters, N1
Alam, AM; Starr, MS1
Nishi, S; Yamada, S; Yokoo, H1
Caine, SB; Koob, GF1
Furukawa, T; Kurashima, M; Nagashima, M; Shirakawa, K; Yamada, K1
Bristow, LJ; Hutson, PH; Patel, S; Ragan, CI; Seabrook, GR1
Misu, Y; Okumura, F; Sato, K; Ueda, H1
Barnhart, WJ; Lehman, DA; Nestler, EJ; Self, DW1
Franklin, SR; Tang, AH1
Ashmeade, T; Routledge, C; Taylor, S; Thorn, L1
Depoortere, R; Perrault, G; Sanger, DJ1
Domae, M; Furukawa, T; Inoue, T; Kurashima, M; Nagashima, M; Shirakawa, K; Yamada, K1
Cools, AR; Kitamura, M; Kobayashi, M; Koshikawa, N1
Ellerbrock, BR; Fici, GJ; Sethy, VH; Wu, H1
Mignot, E; Nishino, S; Reid, MS; Sampathkumaran, R; Siegel, JM; Tafti, M1
Freeman, KA; Mao, A; Tallarida, RJ1
Kamei, J; Ohsawa, M1
Cho, S; Hadjiconstantinou, M; Neff, NH1
Coronas, V; Jourdan, F; Liang, JJ; Moyse, E; Srivastava, LK1
Andersen, SL; Dumont, NL; Teicher, MH1
Badia, A; Clos, MV; García-Sanz, A; Vivas, NM1
Bonardi, CM; Hitchcott, PK; Phillips, GD1
Dall'olio, R; Gandolfi, O; Rimondini, R1
Mohell, N1
Dziedzicka-Wasylewska, M; Maj, J; Rogoz, R; Rogóz, Z1
Reggers, J; Terry, P; Tirelli, E1
Hagan, JJ; Hatcher, JP1
Mach, RH; Nader, MA; Sinnott, RS1
Cook, CD; Picker, MJ; Rodefer, JS1
Brown, RE; Dastur, FN; McGregor, IS1
Honda, K; Mignot, E; Nishino, S; Riehl, J1
Ahmad, B; Darmani, NA; Zhao, W1
Maj, J; Rogóz, Z; Skuza, G1
Hillefors, M; von Euler, G1
Alling, KL; Katz, JL1
Brus, R; Kostrzewa, RM; Nowak, P; Oswiecimska, J; Szkilnik, R1
Badia, A; Clos, MV; García-Sanz, A1
Bridges, RS; Byrnes, EM; Byrnes, JJ1
Butelman, ER; Kreek, MJ1
Garcia-Ladona, J; Wicke, K1
Okuyama, S; Takamori, K; Yoshida, S1
Dlaboga, D; Dziedzicka-Wasylewska, M; Maj, J; Rogoz, Z; Skuza, G1
Rogóz, Z; Skuza, G1
Dall'Olio, R; Gaggi, R; Gandolfi, O; Tanda, O; Voltattorni, M1
Kayir, H; Uzbay, IT1
Heidbreder, CA; Shilliam, CS1
Cooper, SJ; Genn, RF; Higgs, S1
Beardsley, PM; Cook, CD1
Blaha, CD; Forster, GL; Hendry, IA; Holgate, J; Leck, KJ; Matthaei, KI1
Blessing, WW; Hagan, JJ; Heidbreder, CA; Ootsuka, Y1
Greedy, B; Grundt, P; Husbands, SM; Koffarnus, MN; Newman, AH; Woods, JH1
Collo, G; Missale, C; Spano, P; Zanetti, S1
Yoshida, N; Yoshikawa, T1

Other Studies

64 other study(ies) available for 7-hydroxy-2-n,n-dipropylaminotetralin and quinpirole

ArticleYear
Lack of discrimination by agonists for D2 and D3 dopamine receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1995, Volume: 12, Issue:4

    Topics: Cell Line; Cell Membrane; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydronaphthalenes

1995
A functional test identifies dopamine agonists selective for D3 versus D2 receptors.
    Neuroreport, 1995, Jan-26, Volume: 6, Issue:2

    Topics: Animals; CHO Cells; Cricetinae; Dopamine Agents; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3

1995
Synthesis of (R,S)-2'-trans-7-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'- propenyl)-amino]tetralin (trans-7-OH-PIPAT): a new D3 dopamine receptor ligand.
    Journal of medicinal chemistry, 1993, May-14, Volume: 36, Issue:10

    Topics: Binding Sites; Dopamine Agents; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Stereoisomerism; Tetrahydronaphthalenes

1993
Novel D3 selective dopaminergics incorporating enyne units as nonaromatic catechol bioisosteres: synthesis, bioactivity, and mutagenesis studies.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Catechols; Cyclic AMP; Humans; Molecular Structure; Mutagenesis; Protein Binding; Receptors, Dopamine D3; Structure-Activity Relationship

2008
Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Animals; Benzimidazoles; Binding Sites; Chemistry Techniques, Synthetic; CHO Cells; Cricetulus; Humans; Ligands; Models, Molecular; Molecular Dynamics Simulation; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship

2016
Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Aminoquinolines; Animals; Apomorphine; Azepines; Benzothiazoles; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Male; Neurons; Phenethylamines; Piperidines; Pramipexole; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Substantia Nigra; Tetrahydronaphthalenes; Thiazoles; Thiophenes; Transfection

1995
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
    Neuropharmacology, 1995, Volume: 34, Issue:4

    Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes

1995
Characterization of [3H]quinpirole binding to human dopamine D2A and D3 receptors: effects of ions and guanine nucleotides.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:2

    Topics: Animals; Binding, Competitive; Ergolines; Guanylyl Imidodiphosphate; Humans; Magnesium; Male; Mice; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Sodium; Tetrahydronaphthalenes

1995
Suggestive evidence for a DA D3 receptor-mediated increase in the release of oxytocin in the male rat.
    Neuroreport, 1995, Jun-19, Volume: 6, Issue:9

    Topics: Animals; Bromocriptine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Oxytocin; Prolactin; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sex Factors; Tetrahydronaphthalenes

1995
The putative dopamine D3 receptor agonist 7-OH-DPAT: lack of mesolimbic selectivity.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: Animals; Caudate Nucleus; Dopamine Agonists; Dose-Response Relationship, Drug; Electrophysiology; Ergolines; Injections, Intravenous; Iontophoresis; Male; Neostriatum; Neurons; Nucleus Accumbens; Patch-Clamp Techniques; Putamen; Quinpirole; Rats; Rats, Sprague-Dawley; Stereoisomerism; Substantia Nigra; Tetrahydronaphthalenes; Ventral Tegmental Area

1994
Behavioral and neurochemical data suggest functional differences between dopamine D2 and D3 receptors.
    European journal of pharmacology, 1994, Oct-03, Volume: 263, Issue:3

    Topics: Analysis of Variance; Animals; Apomorphine; Benzothiazoles; CHO Cells; Cricetinae; Cricetulus; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Microdialysis; Mitogens; Motor Activity; Piperidines; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Thiazoles; Transfection

1994
Bimodal effects of dopamine D2 receptor agonists on zero Mg(2+)-induced epileptiform activity in the rat cingulate cortex slice.
    Experimental brain research, 1994, Volume: 102, Issue:1

    Topics: Animals; Benzazepines; Dopamine D2 Receptor Antagonists; Epilepsy; Ergolines; Evoked Potentials; Female; Gyrus Cinguli; In Vitro Techniques; Lisuride; Magnesium; Male; Oxazines; Phenethylamines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes

1994
Differential effects of dopamine agonists on evoked dopamine release from slices of striatum and nucleus accumbens in rats.
    Brain research, 1994, Jun-13, Volume: 648, Issue:1

    Topics: Animals; Apomorphine; Dopamine; Dopamine Agonists; Electric Stimulation; Ergolines; In Vitro Techniques; Male; Neostriatum; Nerve Endings; Nucleus Accumbens; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

1994
Modulation of cocaine self-administration in the rat through D-3 dopamine receptors.
    Science (New York, N.Y.), 1993, Jun-18, Volume: 260, Issue:5115

    Topics: Animals; Apomorphine; Cocaine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Self Administration; Tetrahydronaphthalenes

1993
Effects of putative dopamine D3 receptor agonists, 7-OH-DPAT, and quinpirole, on yawning, stereotypy, and body temperature in rats.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Body Temperature; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Tetrahydronaphthalenes; Yawning

1995
Functional relevance of dopamine receptors.
    Trends in pharmacological sciences, 1995, Volume: 16, Issue:12

    Topics: Antipsychotic Agents; Dopamine Agonists; Dopamine Antagonists; Ergolines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia; Tetrahydronaphthalenes

1995
L-DOPA inhibits spontaneous acetylcholine release from the striatum of experimental Parkinson's model rats.
    Brain research, 1995, Nov-06, Volume: 698, Issue:1-2

    Topics: Acetylcholine; Analysis of Variance; Animals; Corpus Striatum; Disease Models, Animal; Dopamine Agonists; Drug Synergism; Ergolines; Levodopa; Male; Oxidopamine; Parkinson Disease, Secondary; Quinpirole; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes

1995
Opposite modulation of cocaine-seeking behavior by D1- and D2-like dopamine receptor agonists.
    Science (New York, N.Y.), 1996, Mar-15, Volume: 271, Issue:5255

    Topics: Animals; Behavior, Addictive; Behavior, Animal; Benzazepines; Caffeine; Cocaine; Dopamine Agonists; Ergolines; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Recurrence; Reinforcement, Psychology; Substance-Related Disorders; Tetrahydronaphthalenes

1996
Dopamine agonists facilitate footshock-elicited locomotion in rats, and suppress level-press responding for food.
    Psychopharmacology, 1995, Volume: 121, Issue:4

    Topics: Animals; Apomorphine; Clonidine; Conditioning, Operant; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Locomotion; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes

1995
Elucidation of D3 receptor function in vivo: do D3 receptors mediate inhibition of dopamine neuronal activity?
    Biochemical Society transactions, 1996, Volume: 24, Issue:1

    Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Male; Mice; Mice, Inbred Strains; Microdialysis; Neurons; Nucleus Accumbens; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

1996
Effects of selective serotonin and dopamine agonists on plasma levels of glucose, insulin and glucagon in the rat.
    Neuroendocrinology, 1996, Volume: 63, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Glucose; Bromocriptine; Buspirone; Dopamine Agonists; Ergolines; Glucagon; Insulin; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Tetrahydronaphthalenes

1996
Behavioural effects in the rat of the putative dopamine D3 receptor agonist 7-OH-DPAT: comparison with quinpirole and apomorphine.
    Psychopharmacology, 1996, Volume: 124, Issue:3

    Topics: Animals; Apomorphine; Behavior, Animal; Conditioning, Operant; Dopamine Agonists; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Rats, Wistar; Self Administration; Stereotyped Behavior; Tetrahydronaphthalenes

1996
Inhibitory effects of putative dopamine D3 receptor agonists, 7-OH-DPAT and quinpirole, on prolactin secretion in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: alpha-Methyltyrosine; Animals; Body Temperature; Depression, Chemical; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estradiol; Male; Methyltyrosines; Prolactin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase; Yawning

1996
Behavioural effects of 7-OH-DPAT are solely due to stimulation of dopamine D2 receptors in the shell of the nucleus accumbens; turning behaviour.
    European journal of pharmacology, 1996, Jul-25, Volume: 308, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzazepines; Benzopyrans; Domperidone; Dopamine Agonists; Dopamine Antagonists; Male; Movement; Nucleus Accumbens; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Sulpiride; Tetrahydronaphthalenes

1996
D2 and D1 dopaminergic activity of 7-OH-DPAT.
    Brain research, 1996, Sep-09, Volume: 733, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Cells, Cultured; Cerebellum; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Indans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetrahydronaphthalenes

1996
Local administration of dopaminergic drugs into the ventral tegmental area modulates cataplexy in the narcoleptic canine.
    Brain research, 1996, Sep-09, Volume: 733, Issue:1

    Topics: Amygdala; Animals; Azepines; Cataplexy; Disease Models, Animal; Dogs; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Electroencephalography; Electromyography; Electrooculography; Female; Globus Pallidus; Male; Microdialysis; Pons; Putamen; Quinpirole; Raclopride; Reticular Formation; Salicylamides; Sleep, REM; Tetrahydronaphthalenes; Ventral Tegmental Area

1996
Transient loss of dopamine autoreceptor control in the presence of highly potent dopamine agonists.
    Life sciences, 1996, Volume: 59, Issue:21

    Topics: Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Male; Phenethylamines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes

1996
Effects of diabetes on methamphetamine-induced place preference in mice.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: Animals; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Male; Methamphetamine; Mice; Mice, Inbred ICR; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Streptozocin; Tetrahydronaphthalenes

1996
Regulation of tyrosine hydroxylase and aromatic L-amino acid decarboxylase by dopaminergic drugs.
    European journal of pharmacology, 1997, Apr-04, Volume: 323, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Aromatic-L-Amino-Acid Decarboxylases; Benzazepines; Brain; Bromocriptine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Mesencephalon; Mice; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase

1997
Identification and localization of dopamine receptor subtypes in rat olfactory mucosa and bulb: a combined in situ hybridization and ligand binding radioautographic approach.
    Journal of chemical neuroanatomy, 1997, Volume: 12, Issue:4

    Topics: Animals; Autoradiography; Benzazepines; Binding Sites; Binding, Competitive; Domperidone; Dopamine Agonists; Dopamine Antagonists; In Situ Hybridization; Iodine Radioisotopes; Male; Olfactory Bulb; Olfactory Mucosa; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sulpiride; Tetrahydronaphthalenes

1997
Developmental differences in dopamine synthesis inhibition by (+/-)-7-OH-DPAT.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Age Factors; Animals; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Female; Levodopa; Nucleus Accumbens; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Salicylamides; Tetrahydronaphthalenes

1997
D2 dopamine receptors and modulation of spontaneous acetylcholine (ACh) release from rat striatal synaptosomes.
    British journal of pharmacology, 1997, Volume: 122, Issue:2

    Topics: Acetylcholine; Animals; Benzamides; CHO Cells; Cricetinae; Dopamine Agonists; Humans; Male; Neostriatum; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Presynaptic; Synaptosomes; Tetrahydronaphthalenes

1997
Enhanced stimulus-reward learning by intra-amygdala administration of a D3 dopamine receptor agonist.
    Psychopharmacology, 1997, Volume: 133, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amygdala; Animals; Conditioning, Operant; Discrimination Learning; Dopamine Agonists; Injections; Male; Photic Stimulation; Quinpirole; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Reward; Tetrahydronaphthalenes

1997
Effects of competitive and non-competitive NMDA receptor antagonists on behavioral responses induced by 7-OH-DPAT and quinpirole in rats.
    Pharmacological research, 1997, Volume: 36, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Dizocilpine Maleate; Dopamine Agonists; Excitatory Amino Acid Antagonists; Male; Motor Activity; Neostriatum; Nucleus Accumbens; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spiperone; Tetrahydronaphthalenes

1997
Agonist and inverse agonist activity at the dopamine D3 receptor measured by guanosine 5'--gamma-thio-triphosphate--35S- binding.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:1

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Mice; Pertussis Toxin; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Tetrahydronaphthalenes; Virulence Factors, Bordetella

1998
Effect of antidepressant drugs administered repeatedly on the dopamine D3 receptors in the rat brain.
    European journal of pharmacology, 1998, Jun-12, Volume: 351, Issue:1

    Topics: Administration, Oral; Amitriptyline; Animals; Antidepressive Agents; Autoradiography; Brain; Citalopram; Dopamine Agonists; Imipramine; Injections, Subcutaneous; Male; Mianserin; Motor Activity; Nucleus Accumbens; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

1998
Dopamine 'D2-like' receptor agonists in combination with cocaine: absence of interactive effects on locomotor activity.
    Behavioural pharmacology, 1997, Volume: 8, Issue:2-3

    Topics: Animals; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Motor Activity; Phenethylamines; Quinpirole; Receptors, Dopamine D2; Tetrahydronaphthalenes

1997
The effects of dopamine D3/D2 receptor agonists on intracranial self stimulation in the rat.
    Psychopharmacology, 1998, Volume: 140, Issue:4

    Topics: Animals; Area Under Curve; Brain; Dopamine Agonists; Injections, Subcutaneous; Male; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Stimulation; Tetrahydronaphthalenes

1998
Dopamine D2/D3 receptors modulate cocaine's reinforcing and discriminative stimulus effects in rhesus monkeys.
    Drug and alcohol dependence, 1999, Apr-01, Volume: 54, Issue:2

    Topics: Analysis of Variance; Animals; Appetitive Behavior; Behavior, Addictive; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Macaca mulatta; Male; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Tetrahydronaphthalenes; Time Factors

1999
Selective attenuation of the antinociceptive effects of mu opioids by the putative dopamine D3 agonist 7-OH-DPAT.
    Psychopharmacology, 1999, Volume: 144, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesics, Opioid; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cycloparaffins; Dopamine Agonists; Dopamine Antagonists; Drug Antagonism; Male; Morphine; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Spiperone; Tetrahydronaphthalenes

1999
Dopaminergic modulation of rat pup ultrasonic vocalizations.
    European journal of pharmacology, 1999, Oct-08, Volume: 382, Issue:2

    Topics: Animals; Animals, Newborn; Benzazepines; Body Temperature; Body Temperature Regulation; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Male; Motor Activity; Quinpirole; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Tetrahydronaphthalenes; Vocalization, Animal

1999
Dopamine D3 agonists into the substantia nigra aggravate cataplexy but do not modify sleep.
    Neuroreport, 1999, Nov-26, Volume: 10, Issue:17

    Topics: Animals; Cataplexy; Dogs; Dopamine Agonists; Dose-Response Relationship, Drug; Electroencephalography; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Sleep; Sleep Stages; Substantia Nigra; Tetrahydronaphthalenes; Time Factors; Ventral Tegmental Area

1999
The role of D2 and D3 dopamine receptors in the mediation of emesis in Cryptotis parva (the least shrew).
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12

    Topics: Analysis of Variance; Animals; Apomorphine; Benzopyrans; Brain Chemistry; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Indans; Male; Oxazines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Shrews; Species Specificity; Sulpiride; Tetrahydronaphthalenes; Vomiting

1999
The anticataleptic effect of 7-OH-DPAT: are dopamine D3 receptors involved?
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12

    Topics: Animals; Antipsychotic Agents; Brain Chemistry; Catalepsy; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Fluphenazine; Haloperidol; Hyperkinesis; Levodopa; Locomotion; Male; Naphthalenes; Pyrrolidines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reserpine; Tetrahydronaphthalenes

1999
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
    Neurochemistry international, 2001, Volume: 38, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes

2001
Discriminative stimulus effects of putative D3 dopamine receptor agonists in rats.
    Behavioural pharmacology, 2000, Volume: 11, Issue:6

    Topics: Animals; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Male; Oxazines; Perception; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2000
7-OH-DPAT, unlike quinpirole, does not prime a yawning response in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:1

    Topics: Animals; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Yawning

2000
Differential effect of quinpirole and 7-OH-DPAT on the spontaneous [(3)H]-dopamine efflux from rat striatal synaptosomes.
    Synapse (New York, N.Y.), 2001, Volume: 40, Issue:1

    Topics: Animals; Benzopyrans; Calcium; Calcium Channels; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Male; Neostriatum; Oxazines; Presynaptic Terminals; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Synaptosomes; Tetrahydronaphthalenes; Tetrodotoxin; Tritium

2001
Increased sensitivity of dopamine systems following reproductive experience in rats.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:3

    Topics: Animals; Conditioning, Operant; Dextroamphetamine; Discrimination Learning; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Neurotransmitter; Receptors, Presynaptic; Tetrahydronaphthalenes

2001
kappa-Opioid receptor agonist-induced prolactin release in primates is blocked by dopamine D(2)-like receptor agonists.
    European journal of pharmacology, 2001, Jul-06, Volume: 423, Issue:2-3

    Topics: Animals; Behavior, Animal; Benzazepines; Benzeneacetamides; Conscious Sedation; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Prolactin; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, kappa; Tetrahydronaphthalenes

2001
The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors.
    European journal of pharmacology, 2001, Jul-20, Volume: 424, Issue:2

    Topics: Animals; Benzopyrans; Binding, Competitive; CHO Cells; Cricetinae; Dendrites; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Neurons; Oxazines; Piperazines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Sulfur Radioisotopes; Tetrahydronaphthalenes

2001
Repeated treatment with imipramine, fluvoxamine and tranylcypromine decreases the number of escape failures by activating dopaminergic systems in a rat learned helplessness test.
    Life sciences, 2001, Sep-07, Volume: 69, Issue:16

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antidepressive Agents; Benzazepines; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Escape Reaction; Fluvoxamine; Helplessness, Learned; Imipramine; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Sulpiride; Tetrahydronaphthalenes; Tranylcypromine

2001
Effect of repeated treatment with tianeptine and fluoxetine on central dopamine D(2) /D(3) receptors.
    Behavioural pharmacology, 2002, Volume: 13, Issue:2

    Topics: Animals; Antidepressive Agents, Second-Generation; Antidepressive Agents, Tricyclic; Autoradiography; Brain Chemistry; Caudate Nucleus; Dextroamphetamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Fluoxetine; Islands of Calleja; Male; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Tetrahydronaphthalenes; Thiazepines

2002
A potential antidepressant activity of SA4503, a selective sigma 1 receptor agonist.
    Behavioural pharmacology, 2002, Volume: 13, Issue:7

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Male; Motor Activity; Piperazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, sigma; Stereotyped Behavior; Swimming; Tetrahydronaphthalenes

2002
Nafadotride administration increases D1 and D1/D2 dopamine receptor mediated behaviors.
    Behavioural pharmacology, 2002, Volume: 13, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Body Temperature; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Exploratory Behavior; Grooming; Male; Motor Activity; Naphthalenes; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior; Stimulation, Chemical; Tetrahydronaphthalenes

2002
Bromocriptine and quinpirole, but not 7-OH-DPAT or SKF 38393, potentiate the inhibitory effect of L-NAME on ethanol-induced locomotor activity in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arginine; Bromocriptine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Ethanol; Male; Mice; Motor Activity; NG-Nitroarginine Methyl Ester; Nitric Oxide; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2003
Gradient of dopamine responsiveness to dopamine receptor agonists in subregions of the rat nucleus accumbens.
    European journal of pharmacology, 2003, Sep-12, Volume: 477, Issue:2

    Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Dopamine; Dose-Response Relationship, Drug; Male; Microdialysis; Nucleus Accumbens; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Time Factors

2003
The effects of 7-OH-DPAT, quinpirole and raclopride on licking for sucrose solutions in the non-deprived rat.
    Behavioural pharmacology, 2003, Volume: 14, Issue:8

    Topics: Animals; Dopamine Agonists; Dopamine Antagonists; Feeding Behavior; Male; Quinpirole; Raclopride; Rats; Sucrose; Taste; Tetrahydronaphthalenes

2003
Modulation of the discriminative stimulus effects of mu opioid agonists in rats: II. Effects of dopamine D2/3 agonists.
    Behavioural pharmacology, 2004, Volume: 15, Issue:1

    Topics: Animals; Appetitive Behavior; Brain; Discrimination Learning; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Heroin; Male; Methadone; Morphine; Motivation; Nalbuphine; Quinolines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Tetrahydronaphthalenes

2004
Gz proteins are functionally coupled to dopamine D2-like receptors in vivo.
    Neuropharmacology, 2006, Volume: 51, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenocorticotropic Hormone; Animals; Behavior, Animal; Blotting, Western; Body Temperature; Dopamine; Dopamine Agonists; GTP-Binding Protein alpha Subunits; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nucleus Accumbens; Quinpirole; Receptors, Dopamine D2; Serotonin Receptor Agonists; Tetrahydronaphthalenes; Time Factors

2006
Dopamine D2 receptor stimulation inhibits cold-initiated thermogenesis in brown adipose tissue in conscious rats.
    Neuroscience, 2007, Jun-15, Volume: 147, Issue:1

    Topics: Adaptation, Physiological; Adipose Tissue, Brown; Animals; Body Temperature Regulation; Cold Temperature; Dopamine Agonists; Male; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Statistics, Nonparametric; Sympathetic Fibers, Postganglionic; Tetrahydronaphthalenes; Thermogenesis

2007
The discriminative stimulus effects of dopamine D2- and D3-preferring agonists in rats.
    Psychopharmacology, 2009, Volume: 203, Issue:2

    Topics: Animals; Benzimidazoles; Benzothiazoles; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2009
Dopamine D3 receptor-preferring agonists increase dendrite arborization of mesencephalic dopaminergic neurons via extracellular signal-regulated kinase phosphorylation.
    The European journal of neuroscience, 2008, Volume: 28, Issue:7

    Topics: Amphetamine; Animals; Cell Shape; Cells, Cultured; Dendrites; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Mesencephalon; Mice; Nerve Growth Factors; Neurogenesis; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase

2008
The possible involvement of dopamine D3 receptors in the regulation of gastric emptying in rats.
    Life sciences, 2010, Nov-20, Volume: 87, Issue:19-22

    Topics: 2-Naphthylamine; Animals; Benzopyrans; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Furans; Gastric Emptying; Male; Oxazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

2010