Page last updated: 2024-08-16

5-methylurapidil and rs 17053

5-methylurapidil has been researched along with rs 17053 in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (62.50)18.2507
2000's3 (37.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ballard, S; Blagg, J; Fox, D; Kenny, B1
Chang, DJ; Clarke, DE; Daniels, DV; Ford, AP; Gever, JR; Jasper, JR; Lesnick, JD1
Arredondo, NF; Bantle, GW; Blue, DR; Clarke, DE; DeSousa, A; Elworthy, TR; Ford, AP; Gross, LM; Kava, MS; Lesnick, JD; Morgans, DJ; Ozer, RS; Palmer, WS; Pfister, JR; Repke, DB; Romero, M; Sandoval, L; Sjogren, EB; Talamás, FX; Vazquez, A; Vimont, RL; Williams, TJ; Wu, H; Zhu, QM1
Bach, C; Bhakta, S; Chan, HW; Chang, DJ; Chang, TK; Clarke, DE; Daniels, DV; Eglen, RM; Ford, AP; Jasper, JR; Khare, R; Kosaka, AH; Lesnick, JD; Salazar, FH; Shieh, IS; Yamanishi, SS1
Pedretti, A; Testa, B; Villa, L; Vistoli, G1
Hussain, MB; Marshall, I1
Chen, K; Chen, M; Han, C; Lu, Z; Song, Y; Yan, J; Zhang, Y1
Bagot, K; Chess-Williams, R1

Reviews

1 review(s) available for 5-methylurapidil and rs 17053

ArticleYear
Pharmacological options in the treatment of benign prostatic hyperplasia.
    Journal of medicinal chemistry, 1997, Apr-25, Volume: 40, Issue:9

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Controlled Clinical Trials as Topic; Endothelins; Enzyme Inhibitors; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1997

Other Studies

7 other study(ies) available for 5-methylurapidil and rs 17053

ArticleYear
Pharmacological pleiotropism of the human recombinant alpha1A-adrenoceptor: implications for alpha1-adrenoceptor classification.
    British journal of pharmacology, 1997, Volume: 121, Issue:6

    Topics: Adrenergic Agents; Animals; CHO Cells; Cloning, Molecular; Cricetinae; Humans; Inositol Phosphates; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins

1997
N-arylpiperazinyl-N'-propylamino derivatives of heteroaryl amides as functional uroselective alpha 1-adrenoceptor antagonists.
    Journal of medicinal chemistry, 1997, Aug-15, Volume: 40, Issue:17

    Topics: Adolescent; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Amides; Animals; Binding, Competitive; Humans; Male; Middle Aged; Models, Chemical; Muscle, Smooth; Piperazines; Prazosin; Propylamines; Prostatic Hyperplasia; Rabbits; Rats; Structure-Activity Relationship; Urinary Bladder

1997
Molecular cloning, genomic characterization and expression of novel human alpha1A-adrenoceptor isoforms.
    FEBS letters, 1998, Jan-30, Volume: 422, Issue:2

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cloning, Molecular; Cricetinae; Gene Library; Humans; Inositol Phosphates; Male; Molecular Sequence Data; Polymerase Chain Reaction; Prostate; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins; RNA, Messenger; Sequence Alignment; Sequence Homology, Amino Acid; Transfection

1998
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005
Characterization of alpha1-adrenoceptor subtypes mediating contractions to phenylephrine in rat thoracic aorta, mesenteric artery and pulmonary artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dioxanes; Dioxins; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Indoramin; Isometric Contraction; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Oxathiins; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spiro Compounds; Vasoconstrictor Agents

1997
Different roles of alpha1-adrenoceptor subtypes in mediating cardiomyocyte protein synthesis in neonatal rats.
    Clinical and experimental pharmacology & physiology, 2004, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Cell Enlargement; Cells, Cultured; Dioxanes; Indoles; Leucine; Muscle Proteins; Myocytes, Cardiac; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2004
Alpha(1A/L)-adrenoceptors mediate contraction of the circular smooth muscle of the pig urethra.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Indoles; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperazines; Receptors, Adrenergic, alpha-1; Regression Analysis; Swine; Thymine; Urethra

2006