Page last updated: 2024-08-16

5-methylurapidil and prazosin

5-methylurapidil has been researched along with prazosin in 91 studies

Research

Studies (91)

TimeframeStudies, this research(%)All Research%
pre-19903 (3.30)18.7374
1990's54 (59.34)18.2507
2000's32 (35.16)29.6817
2010's2 (2.20)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Foglar, R; Horie, K; Obika, K; Ogawa, S; Sakamoto, A; Shibata, K; Tsujimoto, G1
Bondinell, WE; Hieble, JP; Ruffolo, RR1
Ballard, S; Blagg, J; Fox, D; Kenny, B1
Chang, DJ; Clarke, DE; Daniels, DV; Ford, AP; Gever, JR; Jasper, JR; Lesnick, JD1
Arredondo, NF; Bantle, GW; Blue, DR; Clarke, DE; DeSousa, A; Elworthy, TR; Ford, AP; Gross, LM; Kava, MS; Lesnick, JD; Morgans, DJ; Ozer, RS; Palmer, WS; Pfister, JR; Repke, DB; Romero, M; Sandoval, L; Sjogren, EB; Talamás, FX; Vazquez, A; Vimont, RL; Williams, TJ; Wu, H; Zhu, QM1
Bach, C; Bhakta, S; Chan, HW; Chang, DJ; Chang, TK; Clarke, DE; Daniels, DV; Eglen, RM; Ford, AP; Jasper, JR; Khare, R; Kosaka, AH; Lesnick, JD; Salazar, FH; Shieh, IS; Yamanishi, SS1
Gaivin, RJ; Gonzalez-Cabrera, P; Perez, DM; Ross, SA; Waugh, DJ; Yun, J; Zuscik, MJ1
Pedretti, A; Testa, B; Villa, L; Vistoli, G1
Etgen, AM; Karkanias, GB; Petitti, N1
Kojima, C; Satoh, M; Takayanagi, I2
Hiramatsu, Y; Kigoshi, S; Muramatsu, I; Muraoka, R1
Blue, DR; Clarke, DE; Vimont, RL1
Insel, PA; Jackson, CA; Michel, MC1
Alcántara Hernández, R; García-Sáinz, JA; González-Espinosa, C; Macias-Silva, M; Olivares-Reyes, A; Romero-Avila, MT1
García-Sáinz, JA; Torres-Márquez, ME; Villalobos-Molina, R1
Bolaños, FJ; Gozlan, H; Hamon, M; Laporte, AM; Schechter, LE; Vergé, D1
Bell, K; Insel, PA; Klijn, K; Slivka, SR1
Singer, EA; Valenta, B1
Beller, KD; Boer, R; Sanders, KH; Walter, B1
Gross, G; Hanft, G1
Gross, G; Hanft, G; Mehdorn, HM1
Gross, G; Hanft, G; Rugevics, C1
Duan, D; Fermini, B; Nattel, S1
Guh, JH; Ko, FN; Teng, CM; Wu, YC; Yu, SM1
Chueh, SC; Guh, JH; Ko, FN; Teng, CM1
Bigg, DC; Koek, W; Sleight, AJ1
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H1
Guarneri, L; Leonardi, A; Poggesi, E; Simonazzi, I; Taddei, C; Testa, R1
Hua, Z; Wang, XL; Zhang, Y1
Aston, N; Chess-Williams, R; Couldwell, C1
Guh, JH; Ko, FN; Teng, CM1
García-Sáinz, JA; Gutiérrez-Venegas, G1
Gross, G; Hanft, G; Michel, MC1
Carter, AJ; Greengrass, PM; Kenny, BA; Naylor, AM; Read, AM; Wyllie, MG1
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T1
Docherty, JR; Kearns, S; O'Rourke, M1
Hayashi, H; Hiraoka, Y; Muramatsu, I; Ohmura, T; Sakamoto, S1
Drescher, P; Knes, JM; Madsen, PO; Rauch, D1
Aghajanian, GK; Marek, GJ1
Deng, XF; Varma, DR1
Badia, A; Giraldo, J; Tabernero, A; Vila, E; Vivas, NM1
Chiba, T; Fukutomi, J; Hattori, K; Maruyama, K; Nagatomo, T; Takeda, M; Yamaguchi, M1
Hussain, MB; Marshall, I2
Daniel, EE; Gaspar, V; Kwan, CY; Low, AM; Lu-Chao, H1
Hasegawa, Y; Ono, H; Wada, T1
Kadavil, EA; Oriowo, MA; Yousif, M1
Avkiran, M; Yasutake, M; Yokoyama, H1
Foster, HE; Latifpour, J; Nishi, K; Saito, M; Weiss, RM; Yoshida, M1
Dang, H; Gruber, DD; Scofield, MA; Shimozono, M; Wangemann, P1
Hattori, K; Makara, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Suzuki, M; Tsuchiya, M; Watanabe, K1
Demenge, P; Godin-Ribuot, D; Joyeux, M; Patel, A; Ribuot, C; Yellon, DM1
Hiraoka, Y; Kato, H; Morikawa, K; Muramatsu, I; Nagata, O; Ohmura, T; Oshita, M; Taniguchi, T; Watanabe, Y1
Errasti, AE; Rothlin, RP; Sardi, SP; Torres, RM; Velo, MP1
Amobi, N; Coker, C; Guillebaud, J; Mulvin, D; Smith, IC1
Davies, MG; Hagen, PO; Huynh, TT1
Berkowitz, DE; Booth, JV; Cozart, KL; D'Amico, EB; El-Moalem, H; Funk, BL; Marucci, L; Page, SO; Richardson, CD; Rudner, XL; Schwinn, DA; Winters, B1
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM1
García-Sáinz, JA; Gottfried-Blackmore, A; Romero-Avila, MT; Vázquez-Prado, J1
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K1
Saxena, PR; Valdivia, LF; Villalón, CM; Willems, EW1
De Vries, P; Heiligers, JP; Kapoor, K; Saxena, PR; Tom, B; Villalón, CM; Willems, EW1
Coats, P; Hillier, C; Jarajapu, YP; MacDonald, A; McGrath, JC1
Hillier, C; Jarajapu, YP; MacDonald, A1
Koike, K; Yamamoto, Y2
García-Sáinz, JA; González-Espinosa, C; González-Espinosa, D; Mora-Rodríguez, DM; Romero-Avila, MT1
D'Ocon, P; Gisbert, R; Ivorra, MD; Noguera, MA; Ziani, K1
Brodde, OE; Dhein, S; Giessler, C; Silber, RE; Wangemann, T1
Dyer, DC; Ioudina, MV1
Horinouchi, T; Koike, K; Shibano, M; Tanaka, Y; Yamamoto, Y1
Alcaide, C; González-Juanatey, JR; Iglesias, MJ; Lago, F; Piñeiro, R1
Koss, MC; Yu, Y2
Hillier, C; MacDonald, A; Zacharia, J2
Eltze, M; Jähnichen, S; Pertz, HH1
Chen, K; Chen, M; Han, C; Lu, Z; Song, Y; Yan, J; Zhang, Y1
Alewood, D; Chen, Z; Kamikihara, SY; Lewis, RJ; Lima, V; Minneman, KP; Mueller, A; Pupo, AS; Raymundi, V1
Ding, X; McCune, DF; Murray, PA; Perez, DM; Sohn, JT1
Hallberg, M; Lindblom, J; Magnusson, K; Nyberg, F; Petrovska, R; Uhlén, S1
Raasmaja, A; York, DA1
Cunha, FQ; de Andrade, CR; de Godoy, MA; de Oliveira, AM; de Souza, HP; Eberlin, MN; Fukada, SY; Haddad, R; Laurindo, FR; Olivon, VC1
Doze, VA; Hillman, KL; Porter, JE1
Akinaga, J; Buratini, J; Castilho, A; Kamikihara, SY; Lima, V; Mueller, A; Nojimoto, FD; Pupo, AS1
Clair, DK; García-Cazarín, ML; Piascik, MT; Smith, JL1
Chu, CC; Lin, MT; Shieh, JP; Wang, JJ1
Du, H; He, L; Ren, J; Wang, S1
Bockman, CS; Dang, HK; Gruber, DD; Scofield, MA; Wangemann, P; Witt, KM1
Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD1

Reviews

2 review(s) available for 5-methylurapidil and prazosin

ArticleYear
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Humans; Molecular Biology; Molecular Structure; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1995
Pharmacological options in the treatment of benign prostatic hyperplasia.
    Journal of medicinal chemistry, 1997, Apr-25, Volume: 40, Issue:9

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Controlled Clinical Trials as Topic; Endothelins; Enzyme Inhibitors; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1997

Other Studies

89 other study(ies) available for 5-methylurapidil and prazosin

ArticleYear
KMD-3213, a novel, potent, alpha 1a-adrenoceptor-selective antagonist: characterization using recombinant human alpha 1-adrenoceptors and native tissues.
    Molecular pharmacology, 1995, Volume: 48, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Calcium; Cell Line; CHO Cells; Clonidine; Cloning, Molecular; Cricetinae; Humans; Indoles; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Sulfonamides; Tamsulosin

1995
Pharmacological pleiotropism of the human recombinant alpha1A-adrenoceptor: implications for alpha1-adrenoceptor classification.
    British journal of pharmacology, 1997, Volume: 121, Issue:6

    Topics: Adrenergic Agents; Animals; CHO Cells; Cloning, Molecular; Cricetinae; Humans; Inositol Phosphates; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins

1997
N-arylpiperazinyl-N'-propylamino derivatives of heteroaryl amides as functional uroselective alpha 1-adrenoceptor antagonists.
    Journal of medicinal chemistry, 1997, Aug-15, Volume: 40, Issue:17

    Topics: Adolescent; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Adult; Aged; Amides; Animals; Binding, Competitive; Humans; Male; Middle Aged; Models, Chemical; Muscle, Smooth; Piperazines; Prazosin; Propylamines; Prostatic Hyperplasia; Rabbits; Rats; Structure-Activity Relationship; Urinary Bladder

1997
Molecular cloning, genomic characterization and expression of novel human alpha1A-adrenoceptor isoforms.
    FEBS letters, 1998, Jan-30, Volume: 422, Issue:2

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Base Sequence; CHO Cells; Cloning, Molecular; Cricetinae; Gene Library; Humans; Inositol Phosphates; Male; Molecular Sequence Data; Polymerase Chain Reaction; Prostate; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins; RNA, Messenger; Sequence Alignment; Sequence Homology, Amino Acid; Transfection

1998
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists.
    The Journal of biological chemistry, 2001, Jul-06, Volume: 276, Issue:27

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cell Membrane; Clonidine; Conserved Sequence; Cricetinae; Dihydropyridines; Dioxanes; Humans; Imidazoles; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Phenylalanine; Piperazines; Prazosin; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship

2001
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005
Estradiol selectively regulates alpha 1B-noradrenergic receptors in the hypothalamus and preoptic area.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:10

    Topics: Animals; Clonidine; Cyclic AMP; Dioxanes; Estradiol; Female; Hypothalamus; Ovariectomy; Piperazines; Prazosin; Preoptic Area; Rats; Receptors, Adrenergic

1992
Characterization of alpha 1-adrenoceptor subtypes labeled by [3H]prazosin in single cells prepared from rabbit thoracic aorta.
    European journal of pharmacology, 1992, Oct-06, Volume: 221, Issue:1

    Topics: Animals; Aorta, Thoracic; Binding Sites; Calcium; Clonidine; Dioxanes; In Vitro Techniques; Methoxamine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Spiperone

1992
5-Methylurapidil may discriminate between alpha 1-adrenoceptors with a high affinity for WB4101 in rat lung.
    British journal of pharmacology, 1992, Volume: 105, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; In Vitro Techniques; Lung; Male; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1992
Evidence for a noradrenergic innervation to alpha 1A-adrenoceptors in rat kidney.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Calcium Channels; Clonidine; In Vitro Techniques; Kidney; Male; Nitrendipine; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Vasoconstriction

1992
Pharmacological characterization of contractile responses induced by alpha 1-agonists, norepinephrine and clonidine, by selective antagonists of their subtypes in rabbit thoracic aorta.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rabbits

1992
Expression of renal alpha 1-adrenergic receptor subtypes in established hypertension.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:6

    Topics: Animals; Dihydropyridines; Hypertension; In Vitro Techniques; Kidney; Kidney Medulla; Male; Membranes; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic, alpha

1992
Species heterogeneity of hepatic alpha 1-adrenoceptors: alpha 1A-, alpha 1B- and alpha 1C-subtypes.
    Biochemical and biophysical research communications, 1992, Jul-31, Volume: 186, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Blotting, Northern; Cells, Cultured; Guinea Pigs; Inositol 1,4,5-Trisphosphate; Kinetics; Liver; Norepinephrine; Piperazines; Prazosin; Propranolol; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; RNA; Species Specificity

1992
Alpha 1-adrenoceptor subtypes in aorta (alpha 1A) and liver (alpha 1B).
    European journal of pharmacology, 1991, Mar-25, Volume: 206, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Liver; Membranes; Muscle, Smooth, Vascular; Phosphatidylinositols; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha

1991
[3H]5-methyl-urapidil labels 5-HT1A receptors and alpha 1-adrenoceptors in the rat CNS. In vitro binding and autoradiographic studies.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding, Competitive; Brain; In Vitro Techniques; Kinetics; Male; Membranes; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1991
Renal alpha 1-adrenergic receptor subtypes: MDCK-D1 cells, but not rat cortical membranes possess a single population of receptors.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Binding, Competitive; Cell Membrane; Clonidine; Dogs; In Vitro Techniques; Kidney; Kidney Cortex; Kidney Tubules; Phosphatidylcholines; Phosphatidylinositols; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Signal Transduction; Tissue Distribution

1991
Hypotensive effects of 8-hydroxy-2-(di-n-propylamino)tetralin and 5-methylurapidil following stereotaxic microinjection into the ventral medulla of the rat.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Blood Pressure; Dioxanes; Dopamine Antagonists; Heart Rate; Male; Medulla Oblongata; Microinjections; Naphthalenes; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Spiperone; Spiro Compounds; Stereotaxic Techniques; Tetrahydronaphthalenes

1990
Is blockade of alpha 1-adrenoceptors favourable in hypotension induced by stimulation of serotonin1A receptors in conscious dogs?
    Drugs, 1990, Volume: 40 Suppl 4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Heart Rate; Male; Piperazines; Prazosin; Rats; Receptors, Serotonin; Stimulation, Chemical; Swine; Tetrahydronaphthalenes

1990
Subclassification of alpha 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Dioxanes; Heart; In Vitro Techniques; Male; Myocardium; Phenethylamines; Phentolamine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1989
Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue.
    European journal of pharmacology, 1989, Oct-10, Volume: 169, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Humans; In Vitro Techniques; Phenethylamines; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Tetralones

1989
5-Methyl-urapidil discriminates between subtypes of the alpha 1-adrenoceptor.
    European journal of pharmacology, 1988, Jul-07, Volume: 151, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; In Vitro Techniques; Male; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tissue Distribution

1988
Alpha-adrenergic control of volume-regulated Cl- currents in rabbit atrial myocytes. Characterization of a novel ionic regulatory mechanism.
    Circulation research, 1995, Volume: 77, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Atrial Function; Autonomic Nervous System; Calcium Channel Blockers; Chloride Channels; Dihydropyridines; Electrophysiology; Heart Atria; In Vitro Techniques; Ion Channels; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical

1995
Pharmacological evaluation of N-methyl-actinodaphnine, a new vascular alpha-adrenoceptor antagonist, isolated from Illigera luzonensis.
    European journal of pharmacology, 1995, Jun-06, Volume: 279, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Cells, Cultured; Dioxolanes; Drugs, Chinese Herbal; Female; Guinea Pigs; Inositol Phosphates; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperazines; Prazosin; Rats; Rats, Wistar; Spleen; Trachea; Vas Deferens

1995
Characterization of alpha 1-adrenoceptor subtypes in tension response of human prostate to electrical field stimulation.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Adrenergic Antagonists; Animals; Clonidine; Electric Stimulation; Humans; Hyperplasia; In Vitro Techniques; Isometric Contraction; Male; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens; Yohimbine

1995
Binding of antipsychotic drugs at alpha 1A- and alpha 1B-adrenoceptors: risperidone is selective for the alpha 1B-adrenoceptors.
    European journal of pharmacology, 1993, Jul-20, Volume: 238, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Binding Sites; Dioxanes; Hippocampus; In Vitro Techniques; Isoxazoles; Male; Phentolamine; Piperazines; Piperidines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Risperidone; Spleen

1993
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine

1995
Mediation of noradrenaline-induced contractions of rat aorta by the alpha 1B-adrenoceptor subtype.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Computer Simulation; Hippocampus; In Vitro Techniques; Liver; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Regression Analysis; Spiperone; Stereoisomerism; Sulfonamides

1995
Altered alpha 1-adrenoceptor density and alpha 1A/alpha 1B ratio in rat hearts after propranolol treatment.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1994, Volume: 15, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Myocardium; Piperazines; Prazosin; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

1994
Alpha 1A-adrenoceptor subtype mediates contraction of the rat urethra.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:6

    Topics: Aminoquinolines; Animals; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetrahydroisoquinolines; Urethra

1994
Functional identification of alpha 1-adrenoceptor subtypes in human prostate: comparison with those in rat vas deferens and spleen.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Animals; Clonidine; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens

1994
Characterization of the alpha 1B-adrenergic receptors of chicken hepatocytes. Signal transduction and actions.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1993, Volume: 106, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Chickens; Epinephrine; In Vitro Techniques; Liver; Membranes; Norepinephrine; Pertussis Toxin; Phenylephrine; Phosphatidylinositols; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Signal Transduction; Thermodynamics; Virulence Factors, Bordetella

1993
Radioligand binding studies of alpha 1-adrenoceptor subtypes in rat heart.
    British journal of pharmacology, 1994, Volume: 111, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cadmium; Cadmium Chloride; Calcium; Chlorides; Clonidine; Epinephrine; Heart Ventricles; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

1994
Effect of alpha 1 adrenoceptor antagonists on prostatic pressure and blood pressure in the anesthetized dog.
    Urology, 1994, Volume: 44, Issue:1

    Topics: Adrenergic alpha-Antagonists; Affinity Labels; Anesthesia, Endotracheal; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Doxazosin; Male; Models, Biological; Phenylephrine; Piperazines; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin

1994
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
    The Clinical investigator, 1993, Volume: 72, Issue:1

    Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine

1993
Investigation of the actions of chloroethylclonidine in rat aorta.
    British journal of pharmacology, 1995, Volume: 115, Issue:8

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Cystamine; Dioxanes; Dose-Response Relationship, Drug; Drug Synergism; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxathiins; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spiperone; Xylazine; Yohimbine

1995
Identification of alpha 1-adrenoceptor subtypes in the rabbit prostate.
    Journal of autonomic pharmacology, 1995, Volume: 15, Issue:4

    Topics: Acetonitriles; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Male; Muscle Contraction; Norepinephrine; Piperazines; Prazosin; Prostate; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha-1

1995
Contrast medium induced renal vasoconstriction, role of alpha receptors.
    Scandinavian journal of urology and nephrology. Supplementum, 1995, Volume: 172

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Contrast Media; Dose-Response Relationship, Drug; Drug Interactions; Phenylephrine; Piperazines; Prazosin; Rabbits; Radiography; Receptors, Adrenergic, alpha-1; Renal Artery; Sulfonamides; Tamsulosin; Vasoconstriction; Vasoconstrictor Agents

1995
Alpha 1B-adrenoceptor-mediated excitation of piriform cortical interneurons.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Action Potentials; Adrenergic alpha-Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cerebral Cortex; Dioxanes; In Vitro Techniques; Interneurons; Male; Norepinephrine; Oxathiins; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Risperidone; Spiperone

1996
Alpha 1D-adrenoceptors do not contribute to inotropic responses of neonatal rat myocardium.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Aorta; Cell Membrane; Cerebral Cortex; Heart Ventricles; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Phenylephrine; Piperazines; Prazosin; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstrictor Agents; Ventricular Function

1997
Use of the operational model of agonism and [3H]prazosin binding to assess altered responsiveness of alpha1-adrenoceptors in the vas deferens of spontaneously hypertensive rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Vas Deferens

1997
Two district alpha(1)-adrenoceptor subtypes in the human prostate: assessment by radioligand binding assay using 3H-prazosin.
    General pharmacology, 1996, Volume: 27, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Binding, Competitive; Dioxanes; Humans; In Vitro Techniques; Kinetics; Male; Nifedipine; Phentolamine; Piperazines; Prazosin; Prostate; Protein Binding; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tritium

1996
Characterization of alpha1-adrenoceptor subtypes mediating contractions to phenylephrine in rat thoracic aorta, mesenteric artery and pulmonary artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dioxanes; Dioxins; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Indoramin; Isometric Contraction; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Oxathiins; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spiro Compounds; Vasoconstrictor Agents

1997
Characterization of alpha-adrenoceptors in canine mesenteric vein.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dogs; Female; Male; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Yohimbine

1997
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord

1997
Heterogeneity of alpha 1-adrenoceptor subtypes mediating noradrenaline-induced contractions of the rat superior mesenteric artery.
    Pharmacology, 1998, Volume: 56, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Mesenteric Artery, Superior; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spiperone; Vasoconstriction; Vasoconstrictor Agents

1998
Alpha1-adrenergic stimulation of sarcolemmal Na+-H+ exchanger activity in rat ventricular myocytes: evidence for selective mediation by the alpha1A-adrenoceptor subtype.
    Circulation research, 1998, Jun-01, Volume: 82, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cattle; Clonidine; Dioxanes; Heart Ventricles; Humans; Imidazoles; Kinetics; Myocardium; Phenylephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sarcolemma; Sodium-Hydrogen Exchangers; Tetrahydronaphthalenes

1998
Characterization, localization and distribution of alpha1 adrenoceptor subtype in male rabbit urethra.
    The Journal of urology, 1998, Volume: 160, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Autoradiography; Dioxanes; Immunohistochemistry; Male; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1; Spiperone; Urethra

1998
Alpha1A-adrenergic receptors mediate vasoconstriction of the isolated spiral modiolar artery in vitro.
    Hearing research, 1998, Volume: 119, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arteries; Cochlea; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gerbillinae; Nitric Oxide Synthase; Nitroarginine; Norepinephrine; Piperazines; Polymerase Chain Reaction; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; RNA; Vasoconstriction; Yohimbine

1998
Discrimination of alpha1-adrenoceptor subtypes in rat aorta and prostate.
    Pharmacology, 1998, Volume: 57, Issue:2

    Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vasoconstriction; Vasodilator Agents

1998
Infarct size-reducing effect of heat stress and alpha1 adrenoceptors in rats.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Heat Stress Disorders; Heat-Shock Proteins; HSP72 Heat-Shock Proteins; Infarction; Male; Myocardial Ischemia; Organ Culture Techniques; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reperfusion Injury

1998
Binding and functional characterization of alpha1-adrenoceptor subtypes in the rat prostate.
    European journal of pharmacology, 1999, Jan-29, Volume: 366, Issue:1

    Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Prostate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tritium

1999
Characterization of alpha1-adrenoceptor subtypes mediating vasoconstriction in human umbilical vein.
    British journal of pharmacology, 1999, Volume: 126, Issue:2

    Topics: Adrenergic Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Humans; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Umbilical Veins; Vasoconstriction; Vasoconstrictor Agents

1999
Functional characterization of alpha1-adrenoceptor subtypes in longitudinal and circular muscle of human vas deferens.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Alkylating Agents; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenoxybenzamine; Piperazines; Prazosin; Receptors, Adrenergic; Spiperone; Vas Deferens

1999
Functional characterization of alpha1-adrenergic receptors in experimental vein grafts.
    The Journal of surgical research, 1999, Jun-01, Volume: 84, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Carotid Artery, Common; Dioxanes; GTP-Binding Proteins; Jugular Veins; Male; Osmolar Concentration; Pertussis Toxin; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Virulence Factors, Bordetella

1999
Subtype specific regulation of human vascular alpha(1)-adrenergic receptors by vessel bed and age.
    Circulation, 1999, Dec-07, Volume: 100, Issue:23

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Aging; Aorta; Arteries; Celiac Artery; Dopamine Antagonists; Female; Femoral Artery; Gene Expression; Hepatic Artery; Humans; Iliac Artery; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; Phenylephrine; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Renal Artery; RNA, Messenger; Saphenous Vein; Spiperone; Splenic Artery; Vasoconstriction

1999
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured

1999
Protein kinase C-mediated phosphorylation and desensitization of human alpha(1b)-adrenoceptors.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Animals; Binding, Competitive; Calcium; Cell Line; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Inositol Phosphates; Membranes; Norepinephrine; Phentolamine; Phosphorylation; Piperazines; Prazosin; Precipitin Tests; Protein Kinase C; Radioligand Assay; Receptors, Adrenergic, alpha-1; RNA, Messenger; Sulfur Radioisotopes; Tetradecanoylphorbol Acetate; Tritium

1999
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
    European journal of pharmacology, 2000, Jan-03, Volume: 387, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine

2000
Alpha(1)-adrenoceptor subtypes mediating contractions of the rat mesenteric artery.
    European journal of pharmacology, 2000, Apr-21, Volume: 395, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Indoles; Indoramin; Male; Mesenteric Arteries; Methoxamine; Oxathiins; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents

2000
The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation.
    British journal of pharmacology, 2001, Volume: 132, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Carotid Artery, External; Dogs; Female; Imidazoles; Indoles; Isoindoles; Male; Phenylephrine; Piperazines; Prazosin; Quinolizines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Regional Blood Flow; Vasoconstriction

2001
Alpha1-adrenoceptor subtypes mediating vasoconstriction in the carotid circulation of anaesthetized pigs: possible avenues for antimigraine drug development.
    Cephalalgia : an international journal of headache, 2001, Volume: 21, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dose-Response Relationship, Drug; Female; Hemodynamics; Infusions, Intra-Arterial; Migraine Disorders; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Swine; Vasoconstriction

2001
Functional characterization of alpha(1)-adrenoceptor subtypes in human skeletal muscle resistance arteries.
    British journal of pharmacology, 2001, Volume: 133, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Arteries; Clonidine; Dose-Response Relationship, Drug; Humans; Imidazoles; In Vitro Techniques; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vasoconstriction

2001
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction

2001
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
    European journal of pharmacology, 2001, Jul-20, Volume: 424, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction

2001
Molecular cloning and functional expression of the guinea pig alpha(1a)-adrenoceptor.
    European journal of pharmacology, 2001, Aug-31, Volume: 426, Issue:3

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cloning, Molecular; COS Cells; DNA, Complementary; Dose-Response Relationship, Drug; Epinephrine; Gene Expression; Guinea Pigs; Methoxamine; Molecular Sequence Data; Norepinephrine; Oxathiins; Oxymetazoline; Phentolamine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sulfonamides; Tamsulosin; Tritium

2001
alpha(1)-Adrenoceptor subtypes in the mouse mesenteric artery and abdominal aorta.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Abdominal; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mesenteric Arteries; Mice; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction

2001
Modulatory role of a constitutively active population of alpha(1D)-adrenoceptors in conductance arteries.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Arteries; Calcium; Clonidine; Dose-Response Relationship, Drug; Female; Iliac Artery; Mesenteric Arteries; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance

2002
Noradrenaline-induced contraction of human saphenous vein and human internal mammary artery: involvement of different alpha-adrenoceptor subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Clonidine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Mammary Arteries; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Regression Analysis; Saphenous Vein; Yohimbine

2002
Pharmacological characterization of alpha1-adrenoceptor subtypes in the bovine tail artery.
    Journal of veterinary pharmacology and therapeutics, 2002, Volume: 25, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tail; Tetrahydronaphthalenes; Vasoconstriction

2002
Pharmacological characterization of alpha1-adrenoceptor in mouse iliac artery.
    European journal of pharmacology, 2002, Dec-05, Volume: 456, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Iliac Artery; In Vitro Techniques; Male; Mice; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction

2002
Doxazosin induces apoptosis in cardiomyocytes cultured in vitro by a mechanism that is independent of alpha1-adrenergic blockade.
    Circulation, 2003, Jan-07, Volume: 107, Issue:1

    Topics: 3T3 Cells; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Apoptosis; Calcineurin Inhibitors; Cell Survival; Cells, Cultured; Doxazosin; Heart; Humans; Mice; Myocardium; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley

2003
Functional characterization of alpha-adrenoceptors mediating pupillary dilation in rats.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic Fibers; Animals; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Injections, Intravenous; Male; Mydriasis; Norepinephrine; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Pupil; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Yohimbine

2003
Studies of alpha-adrenoceptor antagonists on sympathetic mydriasis in rabbits.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2003, Volume: 19, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Isoquinolines; Male; Mydriasis; Mydriatics; Naphthyridines; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Pupil; Rabbits; Sympathetic Nervous System

2003
Alpha1-adrenoceptor subtypes involved in vasoconstrictor responses to exogenous and neurally released noradrenaline in rat femoral resistance arteries.
    British journal of pharmacology, 2004, Volume: 141, Issue:6

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cocaine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

2004
Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery.
    European journal of pharmacology, 2004, Mar-19, Volume: 488, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Arteries; Clonidine; Dioxins; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Pyrimidinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tail

2004
Different roles of alpha1-adrenoceptor subtypes in mediating cardiomyocyte protein synthesis in neonatal rats.
    Clinical and experimental pharmacology & physiology, 2004, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Cell Enlargement; Cells, Cultured; Dioxanes; Indoles; Leucine; Muscle Proteins; Myocytes, Cardiac; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2004
Pharmacological characterization of alpha1-adrenoceptors in mouse isolated femoral small arteries.
    European journal of pharmacology, 2004, Oct-25, Volume: 503, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

2004
Differential antagonism by conotoxin rho-TIA of contractions mediated by distinct alpha1-adrenoceptor subtypes in rat vas deferens, spleen and aorta.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Cell Line; Cell Membrane; Conotoxins; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Iodine Radioisotopes; Male; Muscle Contraction; Norepinephrine; Piperazines; Potassium Chloride; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Tetralones; Vas Deferens

2005
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction.
    Anesthesiology, 2005, Volume: 103, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Fentanyl; Hydrogen-Ion Concentration; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Receptors, Adrenergic, alpha-1; Vasoconstriction

2005
Nandrolone treatment decreases the alpha1B-adrenoceptor mRNA level in rat kidney, but not the density of alpha1B-adrenoceptors in cultured MDCK-D1 kidney cells.
    European journal of pharmacology, 2005, Dec-19, Volume: 527, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Animals; Cell Line; Dogs; Down-Regulation; Gene Expression; Kidney; Male; Methiothepin; Nandrolone; Piperazines; Polymerase Chain Reaction; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Androgen; RNA, Messenger; Species Specificity; Tritium

2005
Pharmacological characterization of alpha1- and beta-adrenergic synergism of 5'DII activity in rat brown adipocytes.
    Archives of physiology and biochemistry, 2006, Volume: 112, Issue:1

    Topics: Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Cell Membrane; Drug Synergism; Ethanolamines; Female; Imidazoles; Iodide Peroxidase; Male; Oxathiins; Piperazines; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Rats, Zucker; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Triiodothyronine

2006
Alpha1D-adrenoceptor-induced relaxation on rat carotid artery is impaired during the endothelial dysfunction evoked in the early stages of hyperhomocysteinemia.
    European journal of pharmacology, 2006, Aug-14, Volume: 543, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Hyperhomocysteinemia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Superoxides; Vasoconstriction; Vasodilation

2006
Alpha1A-adrenergic receptors are functionally expressed by a subpopulation of cornu ammonis 1 interneurons in rat hippocampus.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electrophysiology; Hippocampus; In Vitro Techniques; Interneurons; Isoproterenol; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2007
alpha1-Adrenoceptors in proximal segments of tail arteries from control and reserpinised rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 376, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Buspirone; Gene Expression; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Oxymetazoline; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reserpine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sympathectomy; Tail; Tetrahydronaphthalenes

2007
The alpha1D-adrenergic receptor induces vascular smooth muscle apoptosis via a p53-dependent mechanism.
    Molecular pharmacology, 2008, Volume: 74, Issue:4

    Topics: Acetophenones; Adrenergic alpha-1 Receptor Antagonists; Anthracenes; Aorta; Apoptosis; Benzothiazoles; Cells, Cultured; Culture Media, Serum-Free; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitochondria; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Pyridines; Reactive Oxygen Species; Receptors, Adrenergic, alpha-1; Time Factors; Toluene; Tumor Suppressor Protein p53

2008
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats.
    Acta pharmacologica Sinica, 2009, Volume: 30, Issue:9

    Topics: Adrenergic alpha-1 Receptor Antagonists; Anesthesia, Local; Anesthetics, Local; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Methoxamine; Nifedipine; Nitroglycerin; Pain Measurement; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2009
Cell membrane chromatography competitive binding analysis for characterization of α1A adrenoreceptor binding interactions.
    Analytical and bioanalytical chemistry, 2011, Volume: 400, Issue:10

    Topics: Adrenergic alpha-1 Receptor Antagonists; Binding, Competitive; Cell Line; Cell Membrane; Chromatography; Doxazosin; Humans; Methods; Phentolamine; Piperazines; Prazosin; Protein Binding; Quinazolines; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin

2011
Molecular and pharmacological characteristics of the gerbil α(1a)-adrenergic receptor.
    Hearing research, 2012, Volume: 283, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Amino Acid Sequence; Animals; Arteries; Chlorocebus aethiops; Clonidine; Cloning, Molecular; Cochlea; Conserved Sequence; COS Cells; Dioxanes; Dose-Response Relationship, Drug; Gerbillinae; Humans; Mice; Molecular Sequence Data; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Sequence Analysis, Protein; Transfection; Vasoconstriction

2012
Ma huang and alpha subtype adrenoceptors in the cat pulmonary vascular bed.
    Journal of dietary supplements, 2008, Volume: 5, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Ephedra sinica; Female; Lung; Male; Phentolamine; Piperazines; Prazosin; Prospective Studies; Pulmonary Circulation; Receptors, Adrenergic; Vasoconstrictor Agents

2008