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5-methylurapidil and phenylephrine

5-methylurapidil has been researched along with phenylephrine in 61 studies

Research

Studies (61)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's35 (57.38)18.2507
2000's24 (39.34)29.6817
2010's2 (3.28)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, DJ; Clarke, DE; Daniels, DV; Ford, AP; Gever, JR; Jasper, JR; Lesnick, JD1
Endoh, M; Norota, I; Takanashi, M1
Gross, G; Ravens, U; Wang, XL; Wettwer, E1
Moriya, M; Takayanagi, I1
Kow, LM; Pfaff, DW1
Johns, EJ; Sattar, MA2
Abdul Sattar, M; Johns, EJ1
Han, C; Yu, GS1
Duan, D; Fermini, B; Nattel, S1
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H1
Aston, N; Chess-Williams, R; Couldwell, C1
Guh, JH; Ko, FN; Teng, CM1
García-Sáinz, JA; Gutiérrez-Venegas, G1
Buisson-Defferier, S; Hibert, M; van den Buuse, M1
Carter, AJ; Greengrass, PM; Kenny, BA; Naylor, AM; Read, AM; Wyllie, MG1
Lepor, H; Shapiro, E; Tang, R1
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T1
Drescher, P; Knes, JM; Madsen, PO; Rauch, D1
Vargas, HM; Zhou, L1
Chess-Williams, R; Furukawa, K; Uchiyama, T1
Haynes, JM; Hill, SJ1
Forster, C1
Deng, XF; Varma, DR1
Ibarra, M; López-Guerrero, JJ; Terrón, JA; Villalobos-Molina, R1
Andersen, GO; Enger, M; Osnes, JB; Skomedal, T1
Hussain, MB; Marshall, I2
Daniel, EE; Gaspar, V; Kwan, CY; Low, AM; Lu-Chao, H1
Hasegawa, Y; Ono, H; Wada, T1
Avkiran, M; Yasutake, M; Yokoyama, H1
Li, W; Wang, XL; Zhang, Y1
Errasti, AE; Rothlin, RP; Sardi, SP; Torres, RM; Velo, MP1
Davies, MG; Hagen, PO; Huynh, TT1
Berkowitz, DE; Booth, JV; Cozart, KL; D'Amico, EB; El-Moalem, H; Funk, BL; Marucci, L; Page, SO; Richardson, CD; Rudner, XL; Schwinn, DA; Winters, B1
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM1
Saxena, PR; Valdivia, LF; Villalón, CM; Willems, EW1
De Vries, P; Heiligers, JP; Kapoor, K; Saxena, PR; Tom, B; Villalón, CM; Willems, EW1
Hillier, C; Jarajapu, YP; MacDonald, A1
Koike, K; Yamamoto, Y1
Dyer, DC; Ioudina, MV1
Arévalo-León, LE; Gallardo-Ortíz, IA; Urquiza-Marín, H; Villalobos-Molina, R1
Chalothorn, D; Gonzalez-Cabrera, PJ; McCune, DF; Perez, DM; Piascik, MT; Rorabaugh, BR; Ross, SA; Yun, J1
Abdullah, NA; Armenia, A; Helmi, A; Johns, EJ; Munavvar, AS1
Baber, SR; Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD1
Ding, X; McCune, DF; Murray, PA; Perez, DM; Sohn, JT1
Gao, Y; Huang, Z; Wu, LL; Yu, GY; Zhang, YY1
Cunha, FQ; de Andrade, CR; de Godoy, MA; de Oliveira, AM; de Souza, HP; Eberlin, MN; Fukada, SY; Haddad, R; Laurindo, FR; Olivon, VC1
Doze, VA; Hillman, KL; Porter, JE1
Abdullah, NA; Johns, EJ; Khan, AH; Sattar, MA1
Akinaga, J; Buratini, J; Castilho, A; Kamikihara, SY; Lima, V; Mueller, A; Nojimoto, FD; Pupo, AS1
Cheevers, CV; Donello, JE; Gil, DW1
Abdullah, NA; Johns, EJ; Khan, MA; Sattar, MA1
Asbun-Bojalil, J; Castillo-Henkel, C; Castillo-Hernández, MC; Cervantes-Cruz, J; Cruz-Domínguez, MP; Miliar-García, A; Montes-Cortés, DH; Reséndiz-Ramírez, AC; Villalobos-Molina, R1
Abdullah, NA; Armenia, A; Johns, EJ; Khan, MA; Sattar, MA1
Clair, DK; García-Cazarín, ML; Piascik, MT; Smith, JL1
Doze, VA; Hillman, KL; Lei, S; Porter, JE1
Abdullah, NA; Johns, EJ; Kazi, RN; Khan, AH; Munavvar, AS1
Chu, CC; Lin, MT; Shieh, JP; Wang, JJ1
Baker, AJ; Cowley, PM; Myagmar, BE; Simpson, PC; Singh, A; Swigart, PM; Thomas, RC1
Johns, EJ; Kazi, RN; Sattar, MA1

Other Studies

61 other study(ies) available for 5-methylurapidil and phenylephrine

ArticleYear
Pharmacological pleiotropism of the human recombinant alpha1A-adrenoceptor: implications for alpha1-adrenoceptor classification.
    British journal of pharmacology, 1997, Volume: 121, Issue:6

    Topics: Adrenergic Agents; Animals; CHO Cells; Cloning, Molecular; Cricetinae; Humans; Inositol Phosphates; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins

1997
Role of alpha 1A adrenoceptor subtype in production of the positive inotropic effect mediated via myocardial alpha 1 adrenoceptors in the rabbit papillary muscle: influence of selective alpha 1A subtype antagonists WB 4101 and 5-methylurapidil.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical

1992
Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect?
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dihydropyridines; Electrophysiology; Heart; Membrane Potentials; Myocardium; Phenylephrine; Piperazines; Propranolol; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical

1991
Alpha 1A-adrenoceptors in rabbit bronchus.
    European journal of pharmacology, 1991, Sep-17, Volume: 202, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Bronchi; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha

1991
Functional analyses of alpha 1-adrenoceptor subtypes in rat hypothalamic ventromedial nucleus neurons.
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Hypothalamus, Middle; In Vitro Techniques; Neurons; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

1995
Evidence for an alpha 1-adrenoceptor subtype mediating adrenergic vasoconstriction in Wistar normotensive and stroke-prone spontaneously hypertensive rat kidney.
    Journal of cardiovascular pharmacology, 1994, Volume: 23, Issue:2

    Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Cerebrovascular Disorders; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Renal Circulation; Sympathetic Nervous System; Vasoconstriction

1994
Alpha 1-adrenoceptor subtypes mediating adrenergic vasoconstriction in kidney, one-clip Goldblatt and deoxycorticosterone acetate-salt hypertensive rats.
    Journal of cardiovascular pharmacology, 1994, Volume: 24, Issue:3

    Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Clonidine; Desoxycorticosterone; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Hypertension, Renovascular; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Vasoconstriction

1994
Role of alpha 1A- and alpha 1B-adrenoceptors in phenylephrine-induced positive inotropic response in isolated rat left atrium.
    Journal of cardiovascular pharmacology, 1994, Volume: 24, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Inositol Phosphates; Male; Myocardial Contraction; Phenethylamines; Phenylephrine; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Tetralones

1994
Alpha-adrenergic control of volume-regulated Cl- currents in rabbit atrial myocytes. Characterization of a novel ionic regulatory mechanism.
    Circulation research, 1995, Volume: 77, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Atrial Function; Autonomic Nervous System; Calcium Channel Blockers; Chloride Channels; Dihydropyridines; Electrophysiology; Heart Atria; In Vitro Techniques; Ion Channels; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical

1995
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine

1995
Alpha 1A-adrenoceptor subtype mediates contraction of the rat urethra.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:6

    Topics: Aminoquinolines; Animals; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetrahydroisoquinolines; Urethra

1994
Functional identification of alpha 1-adrenoceptor subtypes in human prostate: comparison with those in rat vas deferens and spleen.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Animals; Clonidine; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens

1994
Characterization of the alpha 1B-adrenergic receptors of chicken hepatocytes. Signal transduction and actions.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1993, Volume: 106, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Chickens; Epinephrine; In Vitro Techniques; Liver; Membranes; Norepinephrine; Pertussis Toxin; Phenylephrine; Phosphatidylinositols; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Signal Transduction; Thermodynamics; Virulence Factors, Bordetella

1993
Differential cardiovascular effects of 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT), flesinoxan, 5-methyl-urapidil and MDL 75,608A in conscious spontaneously hypertensive rats.
    Fundamental & clinical pharmacology, 1993, Volume: 7, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Dioxanes; Heart Rate; Hypertension; Injections, Intraventricular; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Spiro Compounds

1993
Effect of alpha 1 adrenoceptor antagonists on prostatic pressure and blood pressure in the anesthetized dog.
    Urology, 1994, Volume: 44, Issue:1

    Topics: Adrenergic alpha-Antagonists; Affinity Labels; Anesthesia, Endotracheal; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Doxazosin; Male; Models, Biological; Phenylephrine; Piperazines; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin

1994
The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle.
    The Prostate, 1993, Volume: 22, Issue:4

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylephrine; Piperazines; Prostate; Receptors, Adrenergic, alpha

1993
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
    The Clinical investigator, 1993, Volume: 72, Issue:1

    Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine

1993
Contrast medium induced renal vasoconstriction, role of alpha receptors.
    Scandinavian journal of urology and nephrology. Supplementum, 1995, Volume: 172

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Contrast Media; Dose-Response Relationship, Drug; Drug Interactions; Phenylephrine; Piperazines; Prazosin; Rabbits; Radiography; Receptors, Adrenergic, alpha-1; Renal Artery; Sulfonamides; Tamsulosin; Vasoconstriction; Vasoconstrictor Agents

1995
alpha1-Adrenoceptor subtypes mediating antinatriuresis in Wistar and stroke-prone spontaneously hypertensive rats.
    European journal of pharmacology, 1995, Dec-29, Volume: 294, Issue:2-3

    Topics: Animals; Clonidine; Diuresis; Hypertension; Male; Natriuresis; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1

1995
Vascular alpha 1D-adrenoceptors have a role in the pressor response to phenylephrine in the pithed rat.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Imidazoles; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes

1996
Alpha 1B-adrenoceptor subtype mediating the phenylephrine-induced contractile response in rabbit corpus cavernosum penis.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Male; Penile Erection; Penis; Phenylephrine; Piperazines; Rabbits

1996
Alpha-adrenoceptor mediated responses of the cauda epididymis of the guinea-pig.
    British journal of pharmacology, 1996, Volume: 119, Issue:6

    Topics: Animals; Calcium; Cyclic AMP; Epididymis; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha; Xylazine

1996
Interaction of 5-methyl-urapidil with alpha 1-adrenoceptors in canine blood vessels: impact of pacing-induced heart failure.
    European journal of pharmacology, 1996, Dec-27, Volume: 318, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Cardiac Pacing, Artificial; Dogs; Heart Failure; Hindlimb; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Piperazines; Saphenous Vein; Vasoconstrictor Agents

1996
Alpha 1D-adrenoceptors do not contribute to inotropic responses of neonatal rat myocardium.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Aorta; Cell Membrane; Cerebral Cortex; Heart Ventricles; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Phenylephrine; Piperazines; Prazosin; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstrictor Agents; Ventricular Function

1997
Evidence for an age-dependent functional expression of alpha 1D-adrenoceptors in the rat vasculature.
    European journal of pharmacology, 1997, Mar-19, Volume: 322, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Aging; Animals; Blood Pressure; Blood Vessels; Clonidine; Male; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

1997
Alpha 1-adrenoceptor mediated activation of Na/K/2Cl cotransport and K+ channels in the rat heart involves different receptor subtypes.
    Research communications in molecular pathology and pharmacology, 1997, Volume: 96, Issue:3

    Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Bumetanide; Carrier Proteins; Chlorides; Clonidine; Heart; In Vitro Techniques; Male; Myocardium; Phenylephrine; Piperazines; Potassium; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sodium; Sodium-Potassium-Chloride Symporters

1997
Characterization of alpha1-adrenoceptor subtypes mediating contractions to phenylephrine in rat thoracic aorta, mesenteric artery and pulmonary artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dioxanes; Dioxins; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Indoramin; Isometric Contraction; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Oxathiins; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spiro Compounds; Vasoconstrictor Agents

1997
Characterization of alpha-adrenoceptors in canine mesenteric vein.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dogs; Female; Male; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Yohimbine

1997
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord

1997
Alpha1-adrenergic stimulation of sarcolemmal Na+-H+ exchanger activity in rat ventricular myocytes: evidence for selective mediation by the alpha1A-adrenoceptor subtype.
    Circulation research, 1998, Jun-01, Volume: 82, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cattle; Clonidine; Dioxanes; Heart Ventricles; Humans; Imidazoles; Kinetics; Myocardium; Phenylephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sarcolemma; Sodium-Hydrogen Exchangers; Tetrahydronaphthalenes

1998
Altered alpha 1-adrenoceptor subtypes mediated cardiac function after treatment of propranolol to rats.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1997, Volume: 18, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Clonidine; Heart Rate; Male; Myocardial Contraction; Phenylephrine; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Stimulation, Chemical

1997
Characterization of alpha1-adrenoceptor subtypes mediating vasoconstriction in human umbilical vein.
    British journal of pharmacology, 1999, Volume: 126, Issue:2

    Topics: Adrenergic Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Humans; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Umbilical Veins; Vasoconstriction; Vasoconstrictor Agents

1999
Functional characterization of alpha1-adrenergic receptors in experimental vein grafts.
    The Journal of surgical research, 1999, Jun-01, Volume: 84, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Carotid Artery, Common; Dioxanes; GTP-Binding Proteins; Jugular Veins; Male; Osmolar Concentration; Pertussis Toxin; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Virulence Factors, Bordetella

1999
Subtype specific regulation of human vascular alpha(1)-adrenergic receptors by vessel bed and age.
    Circulation, 1999, Dec-07, Volume: 100, Issue:23

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Aging; Aorta; Arteries; Celiac Artery; Dopamine Antagonists; Female; Femoral Artery; Gene Expression; Hepatic Artery; Humans; Iliac Artery; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; Phenylephrine; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Renal Artery; RNA, Messenger; Saphenous Vein; Spiperone; Splenic Artery; Vasoconstriction

1999
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured

1999
Alpha(1)-adrenoceptor subtypes mediating contractions of the rat mesenteric artery.
    European journal of pharmacology, 2000, Apr-21, Volume: 395, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Indoles; Indoramin; Male; Mesenteric Arteries; Methoxamine; Oxathiins; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents

2000
The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation.
    British journal of pharmacology, 2001, Volume: 132, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Carotid Artery, External; Dogs; Female; Imidazoles; Indoles; Isoindoles; Male; Phenylephrine; Piperazines; Prazosin; Quinolizines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Regional Blood Flow; Vasoconstriction

2001
Alpha1-adrenoceptor subtypes mediating vasoconstriction in the carotid circulation of anaesthetized pigs: possible avenues for antimigraine drug development.
    Cephalalgia : an international journal of headache, 2001, Volume: 21, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dose-Response Relationship, Drug; Female; Hemodynamics; Infusions, Intra-Arterial; Migraine Disorders; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Swine; Vasoconstriction

2001
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction

2001
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
    European journal of pharmacology, 2001, Jul-20, Volume: 424, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction

2001
Pharmacological characterization of alpha1-adrenoceptor subtypes in the bovine tail artery.
    Journal of veterinary pharmacology and therapeutics, 2002, Volume: 25, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tail; Tetrahydronaphthalenes; Vasoconstriction

2002
Evidence for the role of alpha1D- and alpha1A-adrenoceptors in contraction of the rat mesenteric artery.
    Vascular pharmacology, 2003, Volume: 40, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxymetazoline; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

2003
The alpha(1B)-adrenergic receptor decreases the inotropic response in the mouse Langendorff heart model.
    Cardiovascular research, 2003, Dec-01, Volume: 60, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Female; Gene Expression; Heart; Male; Mice; Mice, Transgenic; Myocardial Contraction; Myocytes, Cardiac; Perfusion; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha-1; Stimulation, Chemical

2003
The contribution of adrenoceptor subtype(s) in the renal vasculature of diabetic spontaneously hypertensive rats.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: Animals; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Electric Stimulation; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intravenous; Kidney; Kidney Cortex; Malaysia; Male; Methoxamine; Muscle, Smooth, Vascular; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-1; Streptozocin; Time Factors; Vasoconstriction

2004
Effects of norepinephrine on alpha-subtype receptors in the feline pulmonary vascular bed.
    Critical care medicine, 2004, Volume: 32, Issue:11

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Angiotensin II; Animals; Cats; Clonidine; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation, Preclinical; Ephedrine; Female; Injections, Intra-Arterial; Injections, Intravenous; Male; Norepinephrine; Phenylephrine; Piperazines; Pulmonary Artery; Pulmonary Circulation; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstrictor Agents

2004
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction.
    Anesthesiology, 2005, Volume: 103, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Fentanyl; Hydrogen-Ion Concentration; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Receptors, Adrenergic, alpha-1; Vasoconstriction

2005
Functional alpha(1)-adrenoceptor subtypes in human submandibular glands.
    Journal of dental research, 2006, Volume: 85, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aged; Blotting, Western; Calcium; Cells, Cultured; Female; Humans; Immunohistochemistry; In Situ Hybridization; Male; Middle Aged; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Submandibular Gland; Tissue Distribution

2006
Alpha1D-adrenoceptor-induced relaxation on rat carotid artery is impaired during the endothelial dysfunction evoked in the early stages of hyperhomocysteinemia.
    European journal of pharmacology, 2006, Aug-14, Volume: 543, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Hyperhomocysteinemia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Superoxides; Vasoconstriction; Vasodilation

2006
Alpha1A-adrenergic receptors are functionally expressed by a subpopulation of cornu ammonis 1 interneurons in rat hippocampus.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electrophysiology; Hippocampus; In Vitro Techniques; Interneurons; Isoproterenol; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2007
Influence of cisplatin-induced renal failure on the alpha(1)-adrenoceptor subtype causing vasoconstriction in the kidney of the rat.
    European journal of pharmacology, 2007, Aug-13, Volume: 569, Issue:1-2

    Topics: Amlodipine; Animals; Cisplatin; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Injections, Intraperitoneal; Kidney; Male; Methoxamine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Renal Insufficiency; Vasoconstriction; Vasodilator Agents

2007
alpha1-Adrenoceptors in proximal segments of tail arteries from control and reserpinised rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 376, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Buspirone; Gene Expression; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Oxymetazoline; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reserpine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sympathectomy; Tail; Tetrahydronaphthalenes

2007
Transient allodynia pain models in mice for early assessment of analgesic activity.
    British journal of pharmacology, 2008, Volume: 153, Issue:4

    Topics: Adrenergic alpha-Antagonists; Amines; Amitriptyline; Analgesics; Animals; Clonidine; Cyclohexanecarboxylic Acids; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Excitatory Amino Acid Antagonists; Gabapentin; gamma-Aminobutyric Acid; Hyperalgesia; Injections, Intraperitoneal; Injections, Spinal; Male; Memantine; Mice; Mice, Inbred C57BL; Morphine; N-Methylaspartate; Pain; Peripheral Nervous System; Phenylephrine; Piperazines; Prostaglandin Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, N-Methyl-D-Aspartate; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Reproducibility of Results; Spinal Cord; Spinal Nerves; Time Factors

2008
Alpha1A- and alpha1D-adrenoceptors are the major functional subtypes of renal alpha1-adrenoceptors in streptozotocin-induced diabetic and normal Sprague-Dawley rats.
    Autonomic & autacoid pharmacology, 2008, Volume: 28, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Kidney; Male; Methoxamine; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Renal Artery; Renal Circulation; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

2008
Evidence of alpha1-adrenoceptor functional changes in omental arteries of patients with end-stage renal disease.
    Autonomic & autacoid pharmacology, 2008, Volume: 28, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Arteries; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Humans; Imines; Kidney Failure, Chronic; Male; Middle Aged; Omentum; Phenylephrine; Piperazines; Piperidines; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Vasoconstriction; Vasoconstrictor Agents

2008
Functional subtypes of renal alpha1-adrenoceptor in diabetic and non-diabetic 2K1C Goldblatt renovascular hypertension.
    Acta pharmacologica Sinica, 2008, Volume: 29, Issue:5

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Clonidine; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension, Renovascular; Kidney; Male; Methoxamine; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Vasoconstriction

2008
The alpha1D-adrenergic receptor induces vascular smooth muscle apoptosis via a p53-dependent mechanism.
    Molecular pharmacology, 2008, Volume: 74, Issue:4

    Topics: Acetophenones; Adrenergic alpha-1 Receptor Antagonists; Anthracenes; Aorta; Apoptosis; Benzothiazoles; Cells, Cultured; Culture Media, Serum-Free; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitochondria; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Pyridines; Reactive Oxygen Species; Receptors, Adrenergic, alpha-1; Time Factors; Toluene; Tumor Suppressor Protein p53

2008
Alpha-1A adrenergic receptor activation increases inhibitory tone in CA1 hippocampus.
    Epilepsy research, 2009, Volume: 84, Issue:2-3

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phenylephrine; Picrotoxin; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sodium Channel Blockers; Somatostatin; Tetrodotoxin; Time Factors

2009
Influence of high dietary sodium intake on the functional subtypes of alpha-adrenoceptors in the renal cortical vasculature of Wistar-Kyoto rats.
    Autonomic & autacoid pharmacology, 2009, Volume: 29, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Body Weight; Clonidine; Drinking; Hydroxylamines; Kidney Cortex; Male; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Sodium; Sodium, Dietary; Urine; Vasoconstriction; Vasoconstrictor Agents

2009
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats.
    Acta pharmacologica Sinica, 2009, Volume: 30, Issue:9

    Topics: Adrenergic alpha-1 Receptor Antagonists; Anesthesia, Local; Anesthetics, Local; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Methoxamine; Nifedipine; Nitroglycerin; Pain Measurement; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2009
The Alpha-1A Adrenergic Receptor in the Rabbit Heart.
    PloS one, 2016, Volume: 11, Issue:6

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Blood Pressure; Brain; Heart Ventricles; Isoproterenol; Liver; Male; Myocardium; Phenylephrine; Piperazines; Protein Binding; Rabbits; Receptors, Adrenergic, alpha-1

2016
Antidiuretic and antinatriuretic response to high salt load in normotensive Wistar-Kyoto rats: Role of alpha-1A-adrenoreceptors.
    Autonomic & autacoid pharmacology, 2017, Volume: 37, Issue:1

    Topics: Animals; Antidiuretic Agents; Arterial Pressure; Insulin; Male; Natriuretic Agents; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Sodium Chloride, Dietary

2017