5-methylurapidil has been researched along with phenylephrine in 61 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 35 (57.38) | 18.2507 |
2000's | 24 (39.34) | 29.6817 |
2010's | 2 (3.28) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Chang, DJ; Clarke, DE; Daniels, DV; Ford, AP; Gever, JR; Jasper, JR; Lesnick, JD | 1 |
Endoh, M; Norota, I; Takanashi, M | 1 |
Gross, G; Ravens, U; Wang, XL; Wettwer, E | 1 |
Moriya, M; Takayanagi, I | 1 |
Kow, LM; Pfaff, DW | 1 |
Johns, EJ; Sattar, MA | 2 |
Abdul Sattar, M; Johns, EJ | 1 |
Han, C; Yu, GS | 1 |
Duan, D; Fermini, B; Nattel, S | 1 |
Adachi, M; Manita, S; Matsuda, T; Shigenobu, K; Tanaka, H | 1 |
Aston, N; Chess-Williams, R; Couldwell, C | 1 |
Guh, JH; Ko, FN; Teng, CM | 1 |
García-Sáinz, JA; Gutiérrez-Venegas, G | 1 |
Buisson-Defferier, S; Hibert, M; van den Buuse, M | 1 |
Carter, AJ; Greengrass, PM; Kenny, BA; Naylor, AM; Read, AM; Wyllie, MG | 1 |
Lepor, H; Shapiro, E; Tang, R | 1 |
Hatano, A; Koizumi, T; Komeyama, T; Takahashi, H; Takeda, M; Tamaki, M; Tsutsui, T | 1 |
Drescher, P; Knes, JM; Madsen, PO; Rauch, D | 1 |
Vargas, HM; Zhou, L | 1 |
Chess-Williams, R; Furukawa, K; Uchiyama, T | 1 |
Haynes, JM; Hill, SJ | 1 |
Forster, C | 1 |
Deng, XF; Varma, DR | 1 |
Ibarra, M; López-Guerrero, JJ; Terrón, JA; Villalobos-Molina, R | 1 |
Andersen, GO; Enger, M; Osnes, JB; Skomedal, T | 1 |
Hussain, MB; Marshall, I | 2 |
Daniel, EE; Gaspar, V; Kwan, CY; Low, AM; Lu-Chao, H | 1 |
Hasegawa, Y; Ono, H; Wada, T | 1 |
Avkiran, M; Yasutake, M; Yokoyama, H | 1 |
Li, W; Wang, XL; Zhang, Y | 1 |
Errasti, AE; Rothlin, RP; Sardi, SP; Torres, RM; Velo, MP | 1 |
Davies, MG; Hagen, PO; Huynh, TT | 1 |
Berkowitz, DE; Booth, JV; Cozart, KL; D'Amico, EB; El-Moalem, H; Funk, BL; Marucci, L; Page, SO; Richardson, CD; Rudner, XL; Schwinn, DA; Winters, B | 1 |
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM | 1 |
Saxena, PR; Valdivia, LF; Villalón, CM; Willems, EW | 1 |
De Vries, P; Heiligers, JP; Kapoor, K; Saxena, PR; Tom, B; Villalón, CM; Willems, EW | 1 |
Hillier, C; Jarajapu, YP; MacDonald, A | 1 |
Koike, K; Yamamoto, Y | 1 |
Dyer, DC; Ioudina, MV | 1 |
Arévalo-León, LE; Gallardo-Ortíz, IA; Urquiza-Marín, H; Villalobos-Molina, R | 1 |
Chalothorn, D; Gonzalez-Cabrera, PJ; McCune, DF; Perez, DM; Piascik, MT; Rorabaugh, BR; Ross, SA; Yun, J | 1 |
Abdullah, NA; Armenia, A; Helmi, A; Johns, EJ; Munavvar, AS | 1 |
Baber, SR; Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD | 1 |
Ding, X; McCune, DF; Murray, PA; Perez, DM; Sohn, JT | 1 |
Gao, Y; Huang, Z; Wu, LL; Yu, GY; Zhang, YY | 1 |
Cunha, FQ; de Andrade, CR; de Godoy, MA; de Oliveira, AM; de Souza, HP; Eberlin, MN; Fukada, SY; Haddad, R; Laurindo, FR; Olivon, VC | 1 |
Doze, VA; Hillman, KL; Porter, JE | 1 |
Abdullah, NA; Johns, EJ; Khan, AH; Sattar, MA | 1 |
Akinaga, J; Buratini, J; Castilho, A; Kamikihara, SY; Lima, V; Mueller, A; Nojimoto, FD; Pupo, AS | 1 |
Cheevers, CV; Donello, JE; Gil, DW | 1 |
Abdullah, NA; Johns, EJ; Khan, MA; Sattar, MA | 1 |
Asbun-Bojalil, J; Castillo-Henkel, C; Castillo-Hernández, MC; Cervantes-Cruz, J; Cruz-Domínguez, MP; Miliar-García, A; Montes-Cortés, DH; Reséndiz-Ramírez, AC; Villalobos-Molina, R | 1 |
Abdullah, NA; Armenia, A; Johns, EJ; Khan, MA; Sattar, MA | 1 |
Clair, DK; García-Cazarín, ML; Piascik, MT; Smith, JL | 1 |
Doze, VA; Hillman, KL; Lei, S; Porter, JE | 1 |
Abdullah, NA; Johns, EJ; Kazi, RN; Khan, AH; Munavvar, AS | 1 |
Chu, CC; Lin, MT; Shieh, JP; Wang, JJ | 1 |
Baker, AJ; Cowley, PM; Myagmar, BE; Simpson, PC; Singh, A; Swigart, PM; Thomas, RC | 1 |
Johns, EJ; Kazi, RN; Sattar, MA | 1 |
61 other study(ies) available for 5-methylurapidil and phenylephrine
Article | Year |
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Pharmacological pleiotropism of the human recombinant alpha1A-adrenoceptor: implications for alpha1-adrenoceptor classification.
Topics: Adrenergic Agents; Animals; CHO Cells; Cloning, Molecular; Cricetinae; Humans; Inositol Phosphates; Radioligand Assay; Receptors, Adrenergic, alpha-1; Recombinant Proteins | 1997 |
Role of alpha 1A adrenoceptor subtype in production of the positive inotropic effect mediated via myocardial alpha 1 adrenoceptors in the rabbit papillary muscle: influence of selective alpha 1A subtype antagonists WB 4101 and 5-methylurapidil.
Topics: Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1992 |
Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect?
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dihydropyridines; Electrophysiology; Heart; Membrane Potentials; Myocardium; Phenylephrine; Piperazines; Propranolol; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1991 |
Alpha 1A-adrenoceptors in rabbit bronchus.
Topics: Adrenergic alpha-Antagonists; Animals; Bronchi; Clonidine; Dioxanes; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Piperazines; Rabbits; Receptors, Adrenergic, alpha | 1991 |
Functional analyses of alpha 1-adrenoceptor subtypes in rat hypothalamic ventromedial nucleus neurons.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Female; Hypothalamus, Middle; In Vitro Techniques; Neurons; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 1995 |
Evidence for an alpha 1-adrenoceptor subtype mediating adrenergic vasoconstriction in Wistar normotensive and stroke-prone spontaneously hypertensive rat kidney.
Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Cerebrovascular Disorders; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Renal Circulation; Sympathetic Nervous System; Vasoconstriction | 1994 |
Alpha 1-adrenoceptor subtypes mediating adrenergic vasoconstriction in kidney, one-clip Goldblatt and deoxycorticosterone acetate-salt hypertensive rats.
Topics: Adrenergic alpha-Antagonists; Amlodipine; Animals; Clonidine; Desoxycorticosterone; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Hypertension, Renovascular; Kidney; Male; Methoxamine; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Vasoconstriction | 1994 |
Role of alpha 1A- and alpha 1B-adrenoceptors in phenylephrine-induced positive inotropic response in isolated rat left atrium.
Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart Atria; In Vitro Techniques; Inositol Phosphates; Male; Myocardial Contraction; Phenethylamines; Phenylephrine; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Tetralones | 1994 |
Alpha-adrenergic control of volume-regulated Cl- currents in rabbit atrial myocytes. Characterization of a novel ionic regulatory mechanism.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Atrial Function; Autonomic Nervous System; Calcium Channel Blockers; Chloride Channels; Dihydropyridines; Electrophysiology; Heart Atria; In Vitro Techniques; Ion Channels; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1995 |
Sustained negative inotropism mediated by alpha-adrenoceptors in adult mouse myocardia: developmental conversion from positive response in the neonate.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Animals, Newborn; Atropine; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Mice; Myocardial Contraction; Myocardium; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha; Yohimbine | 1995 |
Alpha 1A-adrenoceptor subtype mediates contraction of the rat urethra.
Topics: Aminoquinolines; Animals; Calcium; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Tetrahydroisoquinolines; Urethra | 1994 |
Functional identification of alpha 1-adrenoceptor subtypes in human prostate: comparison with those in rat vas deferens and spleen.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Animals; Clonidine; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens | 1994 |
Characterization of the alpha 1B-adrenergic receptors of chicken hepatocytes. Signal transduction and actions.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Chickens; Epinephrine; In Vitro Techniques; Liver; Membranes; Norepinephrine; Pertussis Toxin; Phenylephrine; Phosphatidylinositols; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Signal Transduction; Thermodynamics; Virulence Factors, Bordetella | 1993 |
Differential cardiovascular effects of 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT), flesinoxan, 5-methyl-urapidil and MDL 75,608A in conscious spontaneously hypertensive rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Dioxanes; Heart Rate; Hypertension; Injections, Intraventricular; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Spiro Compounds | 1993 |
Effect of alpha 1 adrenoceptor antagonists on prostatic pressure and blood pressure in the anesthetized dog.
Topics: Adrenergic alpha-Antagonists; Affinity Labels; Anesthesia, Endotracheal; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Doxazosin; Male; Models, Biological; Phenylephrine; Piperazines; Prazosin; Pressure; Prostate; Quinazolines; Sulfonamides; Tamsulosin | 1994 |
The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Binding, Competitive; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylephrine; Piperazines; Prostate; Receptors, Adrenergic, alpha | 1993 |
Alpha 1-adrenoceptors in the human prostatic urethra are different from those of the human peripheral arteries.
Topics: Arteries; Atropine; Clonidine; Dioxanes; Humans; Iliac Artery; Isometric Contraction; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Propranolol; Receptors, Adrenergic, alpha-1; Urethra; Yohimbine | 1993 |
Contrast medium induced renal vasoconstriction, role of alpha receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Contrast Media; Dose-Response Relationship, Drug; Drug Interactions; Phenylephrine; Piperazines; Prazosin; Rabbits; Radiography; Receptors, Adrenergic, alpha-1; Renal Artery; Sulfonamides; Tamsulosin; Vasoconstriction; Vasoconstrictor Agents | 1995 |
alpha1-Adrenoceptor subtypes mediating antinatriuresis in Wistar and stroke-prone spontaneously hypertensive rats.
Topics: Animals; Clonidine; Diuresis; Hypertension; Male; Natriuresis; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1995 |
Vascular alpha 1D-adrenoceptors have a role in the pressor response to phenylephrine in the pithed rat.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Imidazoles; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes | 1996 |
Alpha 1B-adrenoceptor subtype mediating the phenylephrine-induced contractile response in rabbit corpus cavernosum penis.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Male; Penile Erection; Penis; Phenylephrine; Piperazines; Rabbits | 1996 |
Alpha-adrenoceptor mediated responses of the cauda epididymis of the guinea-pig.
Topics: Animals; Calcium; Cyclic AMP; Epididymis; Guinea Pigs; In Vitro Techniques; Inositol Phosphates; Male; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha; Xylazine | 1996 |
Interaction of 5-methyl-urapidil with alpha 1-adrenoceptors in canine blood vessels: impact of pacing-induced heart failure.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Cardiac Pacing, Artificial; Dogs; Heart Failure; Hindlimb; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Piperazines; Saphenous Vein; Vasoconstrictor Agents | 1996 |
Alpha 1D-adrenoceptors do not contribute to inotropic responses of neonatal rat myocardium.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Aorta; Cell Membrane; Cerebral Cortex; Heart Ventricles; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Phenylephrine; Piperazines; Prazosin; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstrictor Agents; Ventricular Function | 1997 |
Evidence for an age-dependent functional expression of alpha 1D-adrenoceptors in the rat vasculature.
Topics: Adrenergic alpha-Antagonists; Aging; Animals; Blood Pressure; Blood Vessels; Clonidine; Male; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 1997 |
Alpha 1-adrenoceptor mediated activation of Na/K/2Cl cotransport and K+ channels in the rat heart involves different receptor subtypes.
Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Bumetanide; Carrier Proteins; Chlorides; Clonidine; Heart; In Vitro Techniques; Male; Myocardium; Phenylephrine; Piperazines; Potassium; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sodium; Sodium-Potassium-Chloride Symporters | 1997 |
Characterization of alpha1-adrenoceptor subtypes mediating contractions to phenylephrine in rat thoracic aorta, mesenteric artery and pulmonary artery.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dioxanes; Dioxins; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Indoramin; Isometric Contraction; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Oxathiins; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spiro Compounds; Vasoconstrictor Agents | 1997 |
Characterization of alpha-adrenoceptors in canine mesenteric vein.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dogs; Female; Male; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Yohimbine | 1997 |
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord | 1997 |
Alpha1-adrenergic stimulation of sarcolemmal Na+-H+ exchanger activity in rat ventricular myocytes: evidence for selective mediation by the alpha1A-adrenoceptor subtype.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cattle; Clonidine; Dioxanes; Heart Ventricles; Humans; Imidazoles; Kinetics; Myocardium; Phenylephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Sarcolemma; Sodium-Hydrogen Exchangers; Tetrahydronaphthalenes | 1998 |
Altered alpha 1-adrenoceptor subtypes mediated cardiac function after treatment of propranolol to rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Clonidine; Heart Rate; Male; Myocardial Contraction; Phenylephrine; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Stimulation, Chemical | 1997 |
Characterization of alpha1-adrenoceptor subtypes mediating vasoconstriction in human umbilical vein.
Topics: Adrenergic Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Humans; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Umbilical Veins; Vasoconstriction; Vasoconstrictor Agents | 1999 |
Functional characterization of alpha1-adrenergic receptors in experimental vein grafts.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Carotid Artery, Common; Dioxanes; GTP-Binding Proteins; Jugular Veins; Male; Osmolar Concentration; Pertussis Toxin; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Virulence Factors, Bordetella | 1999 |
Subtype specific regulation of human vascular alpha(1)-adrenergic receptors by vessel bed and age.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Aging; Aorta; Arteries; Celiac Artery; Dopamine Antagonists; Female; Femoral Artery; Gene Expression; Hepatic Artery; Humans; Iliac Artery; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; Phenylephrine; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Renal Artery; RNA, Messenger; Saphenous Vein; Spiperone; Splenic Artery; Vasoconstriction | 1999 |
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured | 1999 |
Alpha(1)-adrenoceptor subtypes mediating contractions of the rat mesenteric artery.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Indoles; Indoramin; Male; Mesenteric Arteries; Methoxamine; Oxathiins; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents | 2000 |
The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Carotid Artery, External; Dogs; Female; Imidazoles; Indoles; Isoindoles; Male; Phenylephrine; Piperazines; Prazosin; Quinolizines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Regional Blood Flow; Vasoconstriction | 2001 |
Alpha1-adrenoceptor subtypes mediating vasoconstriction in the carotid circulation of anaesthetized pigs: possible avenues for antimigraine drug development.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dose-Response Relationship, Drug; Female; Hemodynamics; Infusions, Intra-Arterial; Migraine Disorders; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Swine; Vasoconstriction | 2001 |
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction | 2001 |
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction | 2001 |
Pharmacological characterization of alpha1-adrenoceptor subtypes in the bovine tail artery.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tail; Tetrahydronaphthalenes; Vasoconstriction | 2002 |
Evidence for the role of alpha1D- and alpha1A-adrenoceptors in contraction of the rat mesenteric artery.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxymetazoline; Phenylephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1 | 2003 |
The alpha(1B)-adrenergic receptor decreases the inotropic response in the mouse Langendorff heart model.
Topics: Adrenergic alpha-Antagonists; Animals; Female; Gene Expression; Heart; Male; Mice; Mice, Transgenic; Myocardial Contraction; Myocytes, Cardiac; Perfusion; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha-1; Stimulation, Chemical | 2003 |
The contribution of adrenoceptor subtype(s) in the renal vasculature of diabetic spontaneously hypertensive rats.
Topics: Animals; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Electric Stimulation; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intravenous; Kidney; Kidney Cortex; Malaysia; Male; Methoxamine; Muscle, Smooth, Vascular; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-1; Streptozocin; Time Factors; Vasoconstriction | 2004 |
Effects of norepinephrine on alpha-subtype receptors in the feline pulmonary vascular bed.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Angiotensin II; Animals; Cats; Clonidine; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation, Preclinical; Ephedrine; Female; Injections, Intra-Arterial; Injections, Intravenous; Male; Norepinephrine; Phenylephrine; Piperazines; Pulmonary Artery; Pulmonary Circulation; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstrictor Agents | 2004 |
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction.
Topics: Anesthetics, Intravenous; Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Fentanyl; Hydrogen-Ion Concentration; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Receptors, Adrenergic, alpha-1; Vasoconstriction | 2005 |
Functional alpha(1)-adrenoceptor subtypes in human submandibular glands.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aged; Blotting, Western; Calcium; Cells, Cultured; Female; Humans; Immunohistochemistry; In Situ Hybridization; Male; Middle Aged; Phenylephrine; Piperazines; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Submandibular Gland; Tissue Distribution | 2006 |
Alpha1D-adrenoceptor-induced relaxation on rat carotid artery is impaired during the endothelial dysfunction evoked in the early stages of hyperhomocysteinemia.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Hyperhomocysteinemia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Superoxides; Vasoconstriction; Vasodilation | 2006 |
Alpha1A-adrenergic receptors are functionally expressed by a subpopulation of cornu ammonis 1 interneurons in rat hippocampus.
Topics: Action Potentials; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electrophysiology; Hippocampus; In Vitro Techniques; Interneurons; Isoproterenol; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 2007 |
Influence of cisplatin-induced renal failure on the alpha(1)-adrenoceptor subtype causing vasoconstriction in the kidney of the rat.
Topics: Amlodipine; Animals; Cisplatin; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Injections, Intraperitoneal; Kidney; Male; Methoxamine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Renal Insufficiency; Vasoconstriction; Vasodilator Agents | 2007 |
alpha1-Adrenoceptors in proximal segments of tail arteries from control and reserpinised rats.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Buspirone; Gene Expression; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Oxymetazoline; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reserpine; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sympathectomy; Tail; Tetrahydronaphthalenes | 2007 |
Transient allodynia pain models in mice for early assessment of analgesic activity.
Topics: Adrenergic alpha-Antagonists; Amines; Amitriptyline; Analgesics; Animals; Clonidine; Cyclohexanecarboxylic Acids; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Excitatory Amino Acid Antagonists; Gabapentin; gamma-Aminobutyric Acid; Hyperalgesia; Injections, Intraperitoneal; Injections, Spinal; Male; Memantine; Mice; Mice, Inbred C57BL; Morphine; N-Methylaspartate; Pain; Peripheral Nervous System; Phenylephrine; Piperazines; Prostaglandin Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, N-Methyl-D-Aspartate; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Reproducibility of Results; Spinal Cord; Spinal Nerves; Time Factors | 2008 |
Alpha1A- and alpha1D-adrenoceptors are the major functional subtypes of renal alpha1-adrenoceptors in streptozotocin-induced diabetic and normal Sprague-Dawley rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Kidney; Male; Methoxamine; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Renal Artery; Renal Circulation; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents | 2008 |
Evidence of alpha1-adrenoceptor functional changes in omental arteries of patients with end-stage renal disease.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Arteries; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Female; Humans; Imines; Kidney Failure, Chronic; Male; Middle Aged; Omentum; Phenylephrine; Piperazines; Piperidines; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Vasoconstriction; Vasoconstrictor Agents | 2008 |
Functional subtypes of renal alpha1-adrenoceptor in diabetic and non-diabetic 2K1C Goldblatt renovascular hypertension.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Clonidine; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension, Renovascular; Kidney; Male; Methoxamine; Nitrendipine; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Sprague-Dawley; Vasoconstriction | 2008 |
The alpha1D-adrenergic receptor induces vascular smooth muscle apoptosis via a p53-dependent mechanism.
Topics: Acetophenones; Adrenergic alpha-1 Receptor Antagonists; Anthracenes; Aorta; Apoptosis; Benzothiazoles; Cells, Cultured; Culture Media, Serum-Free; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitochondria; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Pyridines; Reactive Oxygen Species; Receptors, Adrenergic, alpha-1; Time Factors; Toluene; Tumor Suppressor Protein p53 | 2008 |
Alpha-1A adrenergic receptor activation increases inhibitory tone in CA1 hippocampus.
Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Dose-Response Relationship, Drug; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Phenylephrine; Picrotoxin; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sodium Channel Blockers; Somatostatin; Tetrodotoxin; Time Factors | 2009 |
Influence of high dietary sodium intake on the functional subtypes of alpha-adrenoceptors in the renal cortical vasculature of Wistar-Kyoto rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Body Weight; Clonidine; Drinking; Hydroxylamines; Kidney Cortex; Male; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Sodium; Sodium, Dietary; Urine; Vasoconstriction; Vasoconstrictor Agents | 2009 |
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Anesthesia, Local; Anesthetics, Local; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Methoxamine; Nifedipine; Nitroglycerin; Pain Measurement; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1 | 2009 |
The Alpha-1A Adrenergic Receptor in the Rabbit Heart.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Blood Pressure; Brain; Heart Ventricles; Isoproterenol; Liver; Male; Myocardium; Phenylephrine; Piperazines; Protein Binding; Rabbits; Receptors, Adrenergic, alpha-1 | 2016 |
Antidiuretic and antinatriuretic response to high salt load in normotensive Wistar-Kyoto rats: Role of alpha-1A-adrenoreceptors.
Topics: Animals; Antidiuretic Agents; Arterial Pressure; Insulin; Male; Natriuretic Agents; Phenylephrine; Piperazines; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Renal Circulation; Sodium Chloride, Dietary | 2017 |