Page last updated: 2024-08-16

5-methylurapidil and dihydropyridines

5-methylurapidil has been researched along with dihydropyridines in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19902 (15.38)18.7374
1990's10 (76.92)18.2507
2000's1 (7.69)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Insel, PA; Jackson, CA; Michel, MC1
Atkinson, B; Minneman, KP1
Han, CD; Minneman, KP1
Gross, G; Ravens, U; Wang, XL; Wettwer, E1
Boer, R; Glossman, H; Graziadei, I; Zernig, G1
Gross, G; Hanft, G; Mehdorn, HM1
Duan, D; Fermini, B; Nattel, S1
Esbenshade, TA; Hirasawa, A; Minneman, KP; Murphy, TJ; Tanaka, T; Tsujimoto, G; Yano, J1
Brodde, OE; Büscher, R; Michel, MC; Philipp, T1
Han, C; Xu, K; Zhang, Y1
Kocić, I; Korolkiewicz, KZ1
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM1
Gaivin, RJ; Gonzalez-Cabrera, P; Perez, DM; Ross, SA; Waugh, DJ; Yun, J; Zuscik, MJ1

Other Studies

13 other study(ies) available for 5-methylurapidil and dihydropyridines

ArticleYear
Expression of renal alpha 1-adrenergic receptor subtypes in established hypertension.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:6

    Topics: Animals; Dihydropyridines; Hypertension; In Vitro Techniques; Kidney; Kidney Medulla; Male; Membranes; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic, alpha

1992
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor-mediated second messenger responses in rat brain.
    Molecular pharmacology, 1991, Volume: 40, Issue:4

    Topics: Adrenergic alpha-Antagonists; Alkylation; Animals; Brain; Calcium Channel Blockers; Cells, Cultured; Cyclic AMP; Dihydropyridines; Dioxanes; Female; Inositol Phosphates; Male; Piperazines; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Second Messenger Systems; Tritium

1991
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor binding sites in rat tissues.
    Molecular pharmacology, 1991, Volume: 40, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dioxanes; Kinetics; Male; Membranes; Phentolamine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Time Factors

1991
Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect?
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dihydropyridines; Electrophysiology; Heart; Membrane Potentials; Myocardium; Phenylephrine; Piperazines; Propranolol; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical

1991
Stereoselective binding of niguldipine enantiomers to alpha 1A-adrenoceptors labeled with [3H]5-methyl-urapidil.
    European journal of pharmacology, 1989, Oct-17, Volume: 172, Issue:4-5

    Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; In Vitro Techniques; Male; Membranes; Piperazines; Potassium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Stereoisomerism

1989
Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue.
    European journal of pharmacology, 1989, Oct-10, Volume: 169, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Humans; In Vitro Techniques; Phenethylamines; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Tetralones

1989
Alpha-adrenergic control of volume-regulated Cl- currents in rabbit atrial myocytes. Characterization of a novel ionic regulatory mechanism.
    Circulation research, 1995, Volume: 77, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Atrial Function; Autonomic Nervous System; Calcium Channel Blockers; Chloride Channels; Dihydropyridines; Electrophysiology; Heart Atria; In Vitro Techniques; Ion Channels; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical

1995
Cloning of the human alpha 1d-adrenergic receptor and inducible expression of three human subtypes in SK-N-MC cells.
    Molecular pharmacology, 1995, Volume: 47, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Base Sequence; Cell Line; Cloning, Molecular; Dihydropyridines; DNA Primers; DNA, Complementary; Gene Expression; Humans; Isopropyl Thiogalactoside; Molecular Sequence Data; Phenethylamines; Piperazines; Polymerase Chain Reaction; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Restriction Mapping; Tetralones; Transfection

1995
Alpha 1A and alpha 1B-adrenoceptors enhance inositol phosphate generation in rat renal cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Dihydropyridines; Inositol Phosphates; Kidney Cortex; Kinetics; Male; Methoxamine; Norepinephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Substrate Specificity; Tritium

1993
Alterations of cardiac alpha 1-adrenoceptor subtypes in hypothyroid rats.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:7

    Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Dihydropyridines; Dioxanes; DNA Primers; Heart Atria; Hypothyroidism; Male; Myocardial Contraction; Norepinephrine; Phenethylamines; Piperazines; Polymerase Chain Reaction; Protein Binding; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; RNA, Messenger; Tetralones; Thiouracil

1997
Negative inotropic action of alpha-1a adrenoceptor blocking agents: role of adenosine and ATP-sensitive K+ channels.
    General pharmacology, 1998, Volume: 30, Issue:3

    Topics: Adenosine; Adrenergic alpha-Antagonists; Animals; Depression, Chemical; Dihydropyridines; Dioxanes; Female; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Piperazines; Potassium Channels; Receptors, Adrenergic, alpha-1

1998
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured

1999
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists.
    The Journal of biological chemistry, 2001, Jul-06, Volume: 276, Issue:27

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cell Membrane; Clonidine; Conserved Sequence; Cricetinae; Dihydropyridines; Dioxanes; Humans; Imidazoles; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Phenylalanine; Piperazines; Prazosin; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship

2001