5-methylurapidil has been researched along with dexniguldipine in 14 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (14.29) | 18.7374 |
1990's | 11 (78.57) | 18.2507 |
2000's | 1 (7.14) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ballard, S; Blagg, J; Fox, D; Kenny, B | 1 |
Insel, PA; Jackson, CA; Michel, MC | 1 |
Atkinson, B; Minneman, KP | 1 |
Han, CD; Minneman, KP | 1 |
Gross, G; Ravens, U; Wang, XL; Wettwer, E | 1 |
Boer, R; Glossman, H; Graziadei, I; Zernig, G | 1 |
Gross, G; Hanft, G; Mehdorn, HM | 1 |
Duan, D; Fermini, B; Nattel, S | 1 |
Esbenshade, TA; Hirasawa, A; Minneman, KP; Murphy, TJ; Tanaka, T; Tsujimoto, G; Yano, J | 1 |
Brodde, OE; Büscher, R; Michel, MC; Philipp, T | 1 |
Han, C; Xu, K; Zhang, Y | 1 |
Kocić, I; Korolkiewicz, KZ | 1 |
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM | 1 |
Gaivin, RJ; Gonzalez-Cabrera, P; Perez, DM; Ross, SA; Waugh, DJ; Yun, J; Zuscik, MJ | 1 |
1 review(s) available for 5-methylurapidil and dexniguldipine
Article | Year |
---|---|
Pharmacological options in the treatment of benign prostatic hyperplasia.
Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Controlled Clinical Trials as Topic; Endothelins; Enzyme Inhibitors; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Structure-Activity Relationship | 1997 |
13 other study(ies) available for 5-methylurapidil and dexniguldipine
Article | Year |
---|---|
Expression of renal alpha 1-adrenergic receptor subtypes in established hypertension.
Topics: Animals; Dihydropyridines; Hypertension; In Vitro Techniques; Kidney; Kidney Medulla; Male; Membranes; Piperazines; Prazosin; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic, alpha | 1992 |
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor-mediated second messenger responses in rat brain.
Topics: Adrenergic alpha-Antagonists; Alkylation; Animals; Brain; Calcium Channel Blockers; Cells, Cultured; Cyclic AMP; Dihydropyridines; Dioxanes; Female; Inositol Phosphates; Male; Piperazines; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Second Messenger Systems; Tritium | 1991 |
Interaction of subtype-selective antagonists with alpha 1-adrenergic receptor binding sites in rat tissues.
Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dioxanes; Kinetics; Male; Membranes; Phentolamine; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Time Factors | 1991 |
Reduction of cardiac outward currents by alpha-1 adrenoceptor stimulation: a subtype-specific effect?
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dihydropyridines; Electrophysiology; Heart; Membrane Potentials; Myocardium; Phenylephrine; Piperazines; Propranolol; Rats; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1991 |
Stereoselective binding of niguldipine enantiomers to alpha 1A-adrenoceptors labeled with [3H]5-methyl-urapidil.
Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; In Vitro Techniques; Male; Membranes; Piperazines; Potassium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Stereoisomerism | 1989 |
Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue.
Topics: Adrenergic alpha-Antagonists; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Dihydropyridines; Humans; In Vitro Techniques; Phenethylamines; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Tetralones | 1989 |
Alpha-adrenergic control of volume-regulated Cl- currents in rabbit atrial myocytes. Characterization of a novel ionic regulatory mechanism.
Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Atrial Function; Autonomic Nervous System; Calcium Channel Blockers; Chloride Channels; Dihydropyridines; Electrophysiology; Heart Atria; In Vitro Techniques; Ion Channels; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Protein Kinase C; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical | 1995 |
Cloning of the human alpha 1d-adrenergic receptor and inducible expression of three human subtypes in SK-N-MC cells.
Topics: Adrenergic alpha-Antagonists; Animals; Base Sequence; Cell Line; Cloning, Molecular; Dihydropyridines; DNA Primers; DNA, Complementary; Gene Expression; Humans; Isopropyl Thiogalactoside; Molecular Sequence Data; Phenethylamines; Piperazines; Polymerase Chain Reaction; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Restriction Mapping; Tetralones; Transfection | 1995 |
Alpha 1A and alpha 1B-adrenoceptors enhance inositol phosphate generation in rat renal cortex.
Topics: Adrenergic alpha-Antagonists; Animals; Dihydropyridines; Inositol Phosphates; Kidney Cortex; Kinetics; Male; Methoxamine; Norepinephrine; Piperazines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Substrate Specificity; Tritium | 1993 |
Alterations of cardiac alpha 1-adrenoceptor subtypes in hypothyroid rats.
Topics: Adrenergic alpha-Antagonists; Animals; Atrial Function; Binding, Competitive; Dihydropyridines; Dioxanes; DNA Primers; Heart Atria; Hypothyroidism; Male; Myocardial Contraction; Norepinephrine; Phenethylamines; Piperazines; Polymerase Chain Reaction; Protein Binding; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; RNA, Messenger; Tetralones; Thiouracil | 1997 |
Negative inotropic action of alpha-1a adrenoceptor blocking agents: role of adenosine and ATP-sensitive K+ channels.
Topics: Adenosine; Adrenergic alpha-Antagonists; Animals; Depression, Chemical; Dihydropyridines; Dioxanes; Female; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Piperazines; Potassium Channels; Receptors, Adrenergic, alpha-1 | 1998 |
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured | 1999 |
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cell Membrane; Clonidine; Conserved Sequence; Cricetinae; Dihydropyridines; Dioxanes; Humans; Imidazoles; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Phenylalanine; Piperazines; Prazosin; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship | 2001 |