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5-methylurapidil and 8-hydroxy-2-(di-n-propylamino)tetralin

5-methylurapidil has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Flores, CM; Hulihan-Giblin, BA; Kellar, KJ; Lumpkin, MD; Mulroney, SE1
Buisson-Defferier, S; Van den Buuse, M1
Kow, LM; Pfaff, DW; Tsai, YF; Wang, L1
Fischer, G; Grohs, JG; Huber, S; Raberger, G1
Bolaños, FJ; Gozlan, H; Hamon, M; Laporte, AM; Schechter, LE; Vergé, D1
Gross, G; Hanft, G; Schüttler, K; Xin, X1
Singer, EA; Valenta, B1
Beller, KD; Boer, R; Sanders, KH; Walter, B1
Buisson-Defferier, S; Hibert, M; van den Buuse, M1
Boeijinga, PH; Galvan, M; Leishman, DJ1
Dakshinamurti, K; Lal, KJ1

Other Studies

11 other study(ies) available for 5-methylurapidil and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
Stimulation of serotonin1A receptors increases release of prolactin in the rat.
    Neuropharmacology, 1992, Volume: 31, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Male; Metergoline; Methysergide; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Time Factors

1992
Cardiovascular effects of the 5-HT1A receptor ligand, MDL 73005EF, in conscious spontaneously hypertensive rats.
    European journal of pharmacology, 1992, Nov-17, Volume: 223, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Buspirone; Dioxins; Heart Rate; Hypertension; Male; Pindolol; Piperazines; Rats; Rats, Inbred SHR; Receptors, Serotonin; Serotonin Receptor Agonists; Spiro Compounds; Vasodilator Agents

1992
Electrophysiological analyses of serotonergic actions on neurons in hypothalamic ventromedial nucleus in vitro: receptor subtypes involved and implications for regulation of feeding and lordosis behaviors.
    The Chinese journal of physiology, 1992, Volume: 35, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Electrophysiology; Feeding Behavior; Female; In Vitro Techniques; Indoles; Neural Inhibition; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sexual Behavior, Animal; Tropisetron; Ventromedial Hypothalamic Nucleus

1992
Alpha 1-adrenoceptor blockade and/or 5-HT1A agonism during treadmill exercise in dogs.
    Journal of autonomic pharmacology, 1991, Volume: 11, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Heart Rate; Hemodynamics; Physical Exertion; Piperazines; Receptors, Serotonin; Sympathetic Nervous System; Tetrahydronaphthalenes; Vagus Nerve

1991
[3H]5-methyl-urapidil labels 5-HT1A receptors and alpha 1-adrenoceptors in the rat CNS. In vitro binding and autoradiographic studies.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding, Competitive; Brain; In Vitro Techniques; Kinetics; Male; Membranes; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1991
Urapidil analogues are potent ligands of the 5-HT1A receptor.
    Journal of cardiovascular pharmacology, 1990, Volume: 15 Suppl 7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Guanosine Triphosphate; In Vitro Techniques; Ligands; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1990
Hypotensive effects of 8-hydroxy-2-(di-n-propylamino)tetralin and 5-methylurapidil following stereotaxic microinjection into the ventral medulla of the rat.
    British journal of pharmacology, 1990, Volume: 99, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Blood Pressure; Dioxanes; Dopamine Antagonists; Heart Rate; Male; Medulla Oblongata; Microinjections; Naphthalenes; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Spiperone; Spiro Compounds; Stereotaxic Techniques; Tetrahydronaphthalenes

1990
Is blockade of alpha 1-adrenoceptors favourable in hypotension induced by stimulation of serotonin1A receptors in conscious dogs?
    Drugs, 1990, Volume: 40 Suppl 4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Heart Rate; Male; Piperazines; Prazosin; Rats; Receptors, Serotonin; Stimulation, Chemical; Swine; Tetrahydronaphthalenes

1990
Differential cardiovascular effects of 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT), flesinoxan, 5-methyl-urapidil and MDL 75,608A in conscious spontaneously hypertensive rats.
    Fundamental & clinical pharmacology, 1993, Volume: 7, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Dioxanes; Heart Rate; Hypertension; Injections, Intraventricular; Male; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Spiro Compounds

1993
Differential effects of centrally-active antihypertensives on 5-HT1A receptors in rat dorso-lateral septum, rat hippocampus and guinea-pig hippocampus.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Antihypertensive Agents; Electrophysiology; Guinea Pigs; Hippocampus; Male; Neurons; Piperazines; Prosencephalon; Pyramidal Cells; Rats; Receptors, Serotonin; Serotonin; Signal Transduction; Tetrodotoxin; Tryptamines

1994
Hypotensive action of 5-HT receptor agonists in the vitamin B6-deficient hypertensive rat.
    European journal of pharmacology, 1993, Apr-06, Volume: 234, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antihypertensive Agents; Blood Pressure; Cerebral Cortex; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Male; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Riboflavin Deficiency; Serotonin; Serotonin Receptor Agonists; Yohimbine

1993