5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole has been researched along with quipazine in 12 studies
Studies (5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole) | Trials (5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole) | Recent Studies (post-2010) (5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole) | Studies (quipazine) | Trials (quipazine) | Recent Studies (post-2010) (quipazine) |
---|---|---|---|---|---|
218 | 0 | 12 | 658 | 0 | 41 |
Protein | Taxonomy | 5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole (IC50) | quipazine (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 3E | Homo sapiens (human) | 0.0004 | |
5-hydroxytryptamine receptor 3B | Homo sapiens (human) | 0.0004 | |
5-hydroxytryptamine receptor 1A | Homo sapiens (human) | 1.4454 | |
5-hydroxytryptamine receptor 2C | Rattus norvegicus (Norway rat) | 0.47 | |
5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | 1.4 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 2.7 | |
5-hydroxytryptamine receptor 2C | Homo sapiens (human) | 0.0617 | |
5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | 3.7297 | |
5-hydroxytryptamine receptor 3A | Rattus norvegicus (Norway rat) | 0.0035 | |
5-hydroxytryptamine receptor 3A | Homo sapiens (human) | 0.0004 | |
5-hydroxytryptamine receptor 1D | Sus scrofa (pig) | 3.7153 | |
Adenylate cyclase type 5 | Rattus norvegicus (Norway rat) | 1.4454 | |
5-hydroxytryptamine receptor 3D | Homo sapiens (human) | 0.0004 | |
5-hydroxytryptamine receptor 2A | Bos taurus (cattle) | 3.4674 | |
5-hydroxytryptamine receptor 3C | Homo sapiens (human) | 0.0004 | |
5-hydroxytryptamine receptor 3B | Rattus norvegicus (Norway rat) | 0.0035 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (66.67) | 18.7374 |
1990's | 3 (25.00) | 18.2507 |
2000's | 1 (8.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Glennon, RA | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Eide, PK | 1 |
Hollingsworth, PJ; Smith, CB; Walker, EA; Woods, JH; Yamamoto, T | 1 |
Cooper, SJ; Neill, JC | 1 |
Amoroso, S; Annunziato, L; Basile, V; Canzoniero, L; Di Renzo, G; Fatatis, A; Taglialatela, M | 1 |
Fedele, E; Maura, G; Raiteri, M | 1 |
Goodwin, GM; Green, AR | 1 |
Middlemiss, DN | 1 |
Balestre, MN; Bockaert, J; Cory, RN; Guillon, G; Rouot, B; Sladeczek, F | 1 |
Boddeke, HW; Kalkman, HO; Timmermans, PB; Van Zwieten, PA | 1 |
1 review(s) available for 5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole and quipazine
Article | Year |
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Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
11 other study(ies) available for 5-methoxy 3-(1,2,3,6-tetrahydro-4-pyridinyl)1h indole and quipazine
Article | Year |
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Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Stimulation of 5-HT1 receptors in the spinal cord changes substance P-induced behaviour.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Analgesia; Animals; Indoles; Injections, Spinal; Male; Mice; Mice, Inbred Strains; Nerve Endings; Neurons; Pain; Piperazines; Quipazine; Receptors, Serotonin; Reference Values; Serotonin; Serotonin Antagonists; Spinal Cord; Stereotyped Behavior; Substance P | 1992 |
Discriminative-stimulus effects of quipazine and l-5-hydroxytryptophan in relation to serotonin binding sites in the pigeon.
Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Binding Sites; Binding, Competitive; Brain; Columbidae; Discrimination Learning; Dose-Response Relationship, Drug; Indoles; Ketanserin; Kinetics; Male; Pyrimidines; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Tritium | 1991 |
Selective reduction by serotonergic agents of hypertonic saline consumption in rats: evidence for possible 5-HT1C receptor mediation.
Topics: Animals; Dose-Response Relationship, Drug; Drinking Behavior; Fenfluramine; Fluoxetine; Hypertonic Solutions; Indoles; Male; Piperazines; Pyrazines; Quinoxalines; Quipazine; Rats; Receptors, Serotonin; Serotonin | 1989 |
Pharmacological characterization of serotonin receptors involved in the control of prolactin secretion.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Fenfluramine; Indoles; Male; Piperidines; Prolactin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes | 1989 |
Acetylcholine release from rat hippocampal slices is modulated by 5-hydroxytryptamine.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Electric Stimulation; Fenfluramine; Hippocampus; In Vitro Techniques; Indoles; Male; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes | 1989 |
A behavioural and biochemical study in mice and rats of putative selective agonists and antagonists for 5-HT1 and 5-HT2 receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Body Temperature; Brain Chemistry; Histamine H2 Antagonists; Hydroxyindoleacetic Acid; Indoles; Kinetics; Male; Methoxydimethyltryptamines; Mice; Mice, Inbred C57BL; Motor Activity; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Species Specificity; Tetrahydronaphthalenes | 1985 |
The putative 5-HT1 receptor agonist, RU 24969, inhibits the efflux of 5-hydroxytryptamine from rat frontal cortex slices by stimulation of the 5-HT autoreceptor.
Topics: Animals; Cerebral Cortex; Dioxanes; Idazoxan; In Vitro Techniques; Indoles; Male; Methiothepin; Potassium; Propranolol; Quipazine; Rats; Receptors, Serotonin; Serotonin | 1985 |
The 5-hydroxytryptamine (5-HT2) receptor stimulates inositol phosphate formation in intact and broken WRK1 cells: determination of occupancy-response relationships for 5-HT agonists.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bufotenin; Cell Line; Dibenzylchlorethamine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine Triphosphate; Indoles; Inositol Phosphates; Kinetics; Mammary Neoplasms, Experimental; Mathematics; N,N-Dimethyltryptamine; Piperazines; Quipazine; Rats; Receptors, Serotonin; Sugar Phosphates; Tetrahydronaphthalenes; Tryptamines | 1987 |
Calcium-dependency of the pressor responses to selective 5-hydroxytryptamine receptor agonists in pithed rats.
Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Calcium; Indoles; Methoxydimethyltryptamines; Piperazines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord; Yohimbine | 1983 |