Page last updated: 2024-08-26

5-iodotubercidin and epz004777

5-iodotubercidin has been researched along with epz004777 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Al-Awar, R; Arrowsmith, CH; Bolshan, Y; Brown, PJ; Fedorov, O; Knapp, S; Li, F; Nguyen, KT; Schapira, M; Smil, D; Tempel, W; Vedadi, M; Yu, W1
Anglin, JL; Song, Y1
Bayle, ED; Fish, PV; Li, F; Schapira, M; Spurr, SS; Tempel, W; Vedadi, M; Yu, W1

Reviews

1 review(s) available for 5-iodotubercidin and epz004777

ArticleYear
A medicinal chemistry perspective for targeting histone H3 lysine-79 methyltransferase DOT1L.
    Journal of medicinal chemistry, 2013, Nov-27, Volume: 56, Issue:22

    Topics: Animals; Chemistry, Pharmaceutical; Disease; Enzyme Inhibitors; Histones; Humans; Lysine; Methyltransferases

2013

Other Studies

2 other study(ies) available for 5-iodotubercidin and epz004777

ArticleYear
Bromo-deaza-SAH: a potent and selective DOT1L inhibitor.
    Bioorganic & medicinal chemistry, 2013, Apr-01, Volume: 21, Issue:7

    Topics: Crystallography, X-Ray; Halogenation; Histone-Lysine N-Methyltransferase; Humans; Leukemia; Methyltransferases; Models, Molecular; S-Adenosylhomocysteine

2013
New small molecule inhibitors of histone methyl transferase DOT1L with a nitrile as a non-traditional replacement for heavy halogen atoms.
    Bioorganic & medicinal chemistry letters, 2016, 09-15, Volume: 26, Issue:18

    Topics: Crystallography; Enzyme Inhibitors; Halogens; Histone-Lysine N-Methyltransferase; Methyltransferases; Nitriles; Small Molecule Libraries; Structure-Activity Relationship

2016