Page last updated: 2024-09-03

5-fluorowillardiine and gyki 53655

5-fluorowillardiine has been researched along with gyki 53655 in 2 studies

Compound Research Comparison

Studies
(5-fluorowillardiine)
Trials
(5-fluorowillardiine)
Recent Studies (post-2010)
(5-fluorowillardiine)
Studies
(gyki 53655)
Trials
(gyki 53655)
Recent Studies (post-2010) (gyki 53655)
2908111022

Protein Interaction Comparison

ProteinTaxonomy5-fluorowillardiine (IC50)gyki 53655 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)1
Glutamate receptor 2Rattus norvegicus (Norway rat)1
Glutamate receptor 3Rattus norvegicus (Norway rat)1
Glutamate receptor 4Rattus norvegicus (Norway rat)1

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
England, PM; Fleming, JJ1
Arai, AC; Kessler, M1

Other Studies

2 other study(ies) available for 5-fluorowillardiine and gyki 53655

ArticleYear
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
    Bioorganic & medicinal chemistry, 2010, Feb-15, Volume: 18, Issue:4

    Topics: Allosteric Regulation; Animals; Binding Sites; Ligands; Receptors, AMPA

2010
Use of [3H]fluorowillardiine to study properties of AMPA receptor allosteric modulators.
    Brain research, 2006, Mar-03, Volume: 1076, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Membranes; Peptides, Cyclic; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tritium

2006