5-fluorowillardiine has been researched along with alanine in 21 studies
Studies (5-fluorowillardiine) | Trials (5-fluorowillardiine) | Recent Studies (post-2010) (5-fluorowillardiine) | Studies (alanine) | Trials (alanine) | Recent Studies (post-2010) (alanine) |
---|---|---|---|---|---|
29 | 0 | 8 | 24,468 | 512 | 5,581 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 10 (47.62) | 18.2507 |
2000's | 7 (33.33) | 29.6817 |
2010's | 3 (14.29) | 24.3611 |
2020's | 1 (4.76) | 2.80 |
Authors | Studies |
---|---|
Cox, AJ; Lee, RK; Nitsch, RM; Wurtman, RJ | 1 |
Beaver, KM; Hawkins, LM; Jane, DE; Roberts, PJ; Sunter, DC; Taylor, PM | 1 |
Beart, PM; Cheung, NS; Larm, JA | 1 |
Dev, KK; Henley, JM; Roberts, PJ | 1 |
Butterworth, RF; Michalak, A | 1 |
Espitia, SA; Hawkinson, JE | 1 |
Henley, JM; Olivera, S; Rodriguez-Ithurralde, D | 3 |
Ashworth-Preece, MA; Chen, F; Jarrott, B; Lawrence, AJ | 1 |
Archibald, K; Henley, JM; Molnár, E | 1 |
Chen, F; Jarrott, B; Lawrence, AJ | 1 |
Arai, A; Kessler, M; Rogers, G | 1 |
Brotchie, JM; Crossman, AR; Silverdale, MA | 1 |
Hesp, BR; Kerr, DS; Mullaney, I; Wrightson, T | 1 |
Arai, AC; Kessler, M | 1 |
Arai, AC; Kessler, M; Montgomery, K; Suzuki, E | 1 |
Chebli, M; Eibl, C; Plested, A; Salazar, H | 1 |
Babaev, AA; Epifanova, EA; Tarabykin, VS; Turovskaya, MV; Turovsky, EA; Zinchenko, VP | 1 |
Konakov, MV; Levin, SG; Nenov, MN; Teplov, IY | 1 |
Berríos-Cartagena, N; De Cardona-Juliá, EA; Feliciano-Bonilla, MM; Ortiz, JG; Rivera-Delgado, I; Rubio-Dávila, MM | 1 |
21 other study(ies) available for 5-fluorowillardiine and alanine
Article | Year |
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Amyloid precursor protein processing is stimulated by metabotropic glutamate receptors.
Topics: Alanine; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Animals; Cell Line; Chelating Agents; Cycloleucine; Embryo, Mammalian; Fetus; Glioma; Glutamic Acid; Hippocampus; Humans; Indoles; Kidney; Kinetics; Maleimides; N-Methylaspartate; Neuroblastoma; Neurons; Neurotoxins; PC12 Cells; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Protein Kinase C; Protein Processing, Post-Translational; Pyrimidines; Quinacrine; Quisqualic Acid; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1995 |
Characterization of the pharmacology and regional distribution of (S)-[3H]-5-fluorowillardiine binding in rat brain.
Topics: Alanine; Animals; Autoradiography; Brain; Excitatory Amino Acid Agonists; In Vitro Techniques; Male; Pyrimidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Synaptic Membranes; Tissue Distribution | 1995 |
(S)-5-fluorowillardiine-mediated neurotoxicity in cultured murine cortical neurones occurs via AMPA and kainate receptors.
Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cells, Cultured; Excitatory Amino Acid Agonists; Mice; Neurons; Pyrimidines; Receptors, Kainic Acid | 1996 |
Characterisation of the interaction between guanyl nucleotides and AMPA receptors in rat brain.
Topics: Alanine; Animals; Autoradiography; Brain Chemistry; Excitatory Amino Acid Agonists; Female; Guanine Nucleotides; Guanosine Triphosphate; In Vitro Techniques; Membranes; Pyrimidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Thiocyanates | 1996 |
Selective loss of binding sites for the glutamate receptor ligands [3H]kainate and (S)-[3H]5-fluorowillardiine in the brains of rats with acute liver failure.
Topics: Alanine; Animals; Binding Sites; Brain; Cerebellum; Cerebral Cortex; Dizocilpine Maleate; Hepatic Encephalopathy; Hippocampus; Kainic Acid; Male; Pyrimidines; Rats; Rats, Sprague-Dawley | 1997 |
Effects of thiocyanate and AMPA receptor ligands on (S)-5-fluorowillardiine, (S)-AMPA and (R,S)-AMPA binding.
Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Binding, Competitive; Brain; Excitatory Amino Acid Agonists; In Vitro Techniques; Ligands; Male; Pyrimidines; Rats; Receptors, AMPA; Stereoisomerism; Thiocyanates | 1997 |
Acetylcholinesterase potentiates [3H]fluorowillardiine and [3H]AMPA binding to rat cortical membranes.
Topics: Acetylcholinesterase; Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Blotting, Western; Cerebral Cortex; Cholinesterase Inhibitors; Drug Synergism; Electrophoresis, Polyacrylamide Gel; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; In Vitro Techniques; Male; Pyrimidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA | 1999 |
Visualisation of AMPA binding sites in the brain stem of normotensive and hypertensive rats.
Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Binding Sites; Brain Stem; Denervation; Hypertension; Male; Neurons, Afferent; Nodose Ganglion; Pyrimidines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Reference Values; Solitary Nucleus; Tissue Distribution; Vagus Nerve | 1999 |
Differential changes in the subcellular distribution of alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate and N-methyl-D-aspartate receptors in neonate and adult rat cortex.
Topics: Aging; Alanine; Animals; Animals, Newborn; Cerebral Cortex; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Female; Microsomes; Pyrimidines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synaptosomes | 1999 |
Up-regulation of cortical AMPA receptor binding in the fawn-hooded rat following ethanol withdrawal.
Topics: Alanine; Alcohol Drinking; Animals; Autoradiography; Behavior, Animal; Binding, Competitive; Brain; Central Nervous System Depressants; Cerebral Cortex; Drinking Behavior; Ethanol; Female; Male; Pyrimidines; Rats; Rats, Inbred WKY; Receptors, AMPA; Species Specificity; Substance Withdrawal Syndrome; Tritium; Up-Regulation; Water | 1999 |
The norbornenyl moiety of cyclothiazide determines the preference for flip-flop variants of AMPA receptor subunits.
Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Alternative Splicing; Animals; Antihypertensive Agents; Benzothiadiazines; Binding Sites; Binding, Competitive; Cells, Cultured; Excitatory Amino Acid Agonists; Humans; Kidney; Pyrimidines; Rats; Receptors, AMPA; Tritium | 2000 |
Regional localization and developmental profile of acetylcholinesterase-evoked increases in [(3)H]-5-fluororwillardiine binding to AMPA receptors in rat brain.
Topics: Acetylcholinesterase; Aging; Alanine; Animals; Autoradiography; Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide; Binding, Competitive; Brain; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Hippocampus; Kainic Acid; Pyrimidines; Rats; Rats, Wistar; Receptors, AMPA; Solubility; Tritium | 2001 |
Striatal AMPA receptor binding is unaltered in the MPTP-lesioned macaque model of Parkinson's disease and dyskinesia.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Alanine; Animals; Apomorphine; Autoradiography; Binding, Competitive; Corpus Striatum; Disease Models, Animal; Dyskinesia, Drug-Induced; Excitatory Amino Acid Agonists; Female; Ligands; Macaca mulatta; Male; Organ Specificity; Parkinson Disease, Secondary; Pyrimidines; Radioligand Assay; Receptors, AMPA | 2002 |
AMPA receptor potentiation by acetylcholinesterase is age-dependently upregulated at synaptogenesis sites of the rat brain.
Topics: Acetylcholinesterase; Aging; Alanine; Animals; Animals, Newborn; Binding Sites; Brain; Drug Synergism; Male; Neuronal Plasticity; Pyrimidines; Rats; Rats, Wistar; Receptors, AMPA; Reproducibility of Results; Sensitivity and Specificity; Synapses; Synaptic Membranes; Up-Regulation | 2003 |
Kainate receptor agonists and antagonists mediate tolerance to kainic acid and reduce high-affinity GTPase activity in young, but not aged, rat hippocampus.
Topics: Action Potentials; Age Factors; Alanine; Animals; Dose-Response Relationship, Drug; Drug Tolerance; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; GTP Phosphohydrolases; Hippocampus; In Vitro Techniques; Kainic Acid; Male; Pyrimidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Kainic Acid | 2004 |
Use of [3H]fluorowillardiine to study properties of AMPA receptor allosteric modulators.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Alanine; Allosteric Site; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Membranes; Peptides, Cyclic; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tritium | 2006 |
Factors affecting guanine nucleotide binding to rat AMPA receptors.
Topics: Alanine; Amino Acid Substitution; Animals; Cell Line; DNA, Complementary; Guanine Nucleotides; Guanosine Diphosphate; Humans; Lysine; Mutagenesis; Plasmids; Purinergic Antagonists; Pyrimidines; Rats; Receptors, AMPA; Receptors, Purinergic; Transfection | 2007 |
Mechanism of partial agonism in AMPA-type glutamate receptors.
Topics: Alanine; Animals; Cross-Linking Reagents; Crystallography, X-Ray; Excitatory Amino Acid Agonists; HEK293 Cells; Humans; Kainic Acid; Models, Molecular; Protein Conformation; Protein Domains; Protein Multimerization; Pyrimidines; Rats; Receptors, AMPA; Receptors, Glutamate | 2017 |
Mutation in the Sip1 transcription factor leads to a disturbance of the preconditioning of AMPA receptors by episodes of hypoxia in neurons of the cerebral cortex due to changes in their activity and subunit composition. The protective effects of interleu
Topics: Alanine; Animals; Calcium; Calcium Signaling; Cerebral Cortex; Enzyme Activation; Excitatory Amino Acid Agonists; Hypoxia; Interleukin-10; Mice; Microscopy, Fluorescence; Mutation; Nerve Tissue Proteins; Neurons; Phosphatidylinositol 3-Kinases; Pyrimidines; Receptors, AMPA | 2018 |
Interleukin-10 Facilitates Glutamatergic Synaptic Transmission and Homeostatic Plasticity in Cultured Hippocampal Neurons.
Topics: Alanine; Animals; Cells, Cultured; Hippocampus; Interleukin-10; Microscopy, Fluorescence; Neuronal Plasticity; Neurons; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Tetrodotoxin | 2019 |
Effects of Zinc, Mercury, or Lead on [
Topics: Alanine; Animals; Dizocilpine Maleate; Lead; Mercury; Neuroprotective Agents; Pyrimidines; Rats; Synaptic Membranes; Zinc | 2021 |