5-carboxamidotryptamine and pindolol

5-carboxamidotryptamine has been researched along with pindolol in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19902 (14.29)18.7374
1990's10 (71.43)18.2507
2000's2 (14.29)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Glennon, RA1
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B1
Chaput, C; Millan, MJ; Newman-Tancredi, A; Verrièle, L1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Miller, KJ; Teitler, M1
Connor, HE; Higgins, GA1
Borton, M; Docherty, JR1
Feuerstein, TJ; Hertting, G; Lupp, A1
Grisel, DA; Iben, LG; Parker, EM; Shapiro, RA1
Crick, H; Manuel, NA; Wallis, DI1
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM1
Barnes, NM; Stowe, RL1
Arnold, PB; Cardenas, CG; Cardenas, LM; Mar, LP; Scroggs, RS; Surmeier, DJ; Vysokanov, AV1

Reviews

1 review(s) available for 5-carboxamidotryptamine and pindolol

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987

Other Studies

13 other study(ies) available for 5-carboxamidotryptamine and pindolol

ArticleYear
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Affinity Labels; Animals; Binding, Competitive; CHO Cells; Cricetinae; Guanine Nucleotides; Hippocampus; Humans; Male; Membranes; Piperazines; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1998
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Quantitative autoradiography of 5-CT-sensitive (5-HT1D) and 5-CT-insensitive (5-HT1E) serotonin receptors in human brain.
    Neuroscience letters, 1992, Mar-02, Volume: 136, Issue:2

    Topics: Antiparkinson Agents; Autoradiography; Brain Chemistry; Ergolines; Humans; In Vitro Techniques; Pindolol; Receptors, Serotonin; Serotonin

1992
Cardiovascular effects of 5-HT1A receptor agonists injected into the dorsal raphe nucleus of conscious rats.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antihypertensive Agents; Atropine Derivatives; Behavior, Animal; Catheterization; Hemodynamics; Injections; Injections, Intravenous; Male; Pindolol; Piperazines; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1990
The effects of ageing on prejunctional 5-hydroxytryptamine receptors in the rat vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:2

    Topics: Aging; Animals; Electric Stimulation; In Vitro Techniques; Male; Muscle, Smooth; Myocardial Contraction; Pertussis Toxin; Pindolol; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vas Deferens; Virulence Factors, Bordetella; Yohimbine

1990
The serotonin (5-HT) autoreceptor in the hippocampus of the rabbit: role of 5-HT biophase concentration.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Mathematics; Metergoline; Methiothepin; Methoxydimethyltryptamines; Methysergide; Phentolamine; Pindolol; Quipazine; Rabbits; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1987
A single amino acid difference accounts for the pharmacological distinctions between the rat and human 5-hydroxytryptamine1B receptors.
    Journal of neurochemistry, 1993, Volume: 60, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Humans; Iodocyanopindolol; Mutagenesis, Insertional; Pindolol; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1993
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan

1995
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro.
    American journal of respiratory and critical care medicine, 1998, Volume: 158, Issue:5 Pt 1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron

1998
Selective labelling of 5-HT7 receptor recognition sites in rat brain using [3H]5-carboxamidotryptamine.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Brain; Clozapine; Indoles; Kinetics; Male; Pindolol; Piperazines; Pyridines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Recombinant Proteins; Serotonin; Sulfonamides; Tritium

1998
Serotonergic modulation of hyperpolarization-activated current in acutely isolated rat dorsal root ganglion neurons.
    The Journal of physiology, 1999, Jul-15, Volume: 518 ( Pt 2)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Cell Size; Cyclic Nucleotide-Gated Cation Channels; Dopamine Antagonists; Ganglia, Spinal; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Pindolol; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999