5-carboxamidotryptamine and ketanserin

5-carboxamidotryptamine has been researched along with ketanserin in 66 studies

Research

Studies (66)

Timeframe	Studies, this research(%)	All Research%
pre-1990	9 (13.64)	18.7374
1990's	46 (69.70)	18.2507
2000's	10 (15.15)	29.6817
2010's	1 (1.52)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Newman-Tancredi, A; Strange, PG; Wootton, R	1
Amlaiky, N; Boschert, U; Hen, R; Maroteaux, L; Plassat, JL; Saudou, F	1
Glennon, RA	2
Buckingham, J; Glen, RC; Hill, AP; Hyde, RM; Martin, GR; Robertson, AD; Salmon, JA; Woollard, PM	1
Bull, D; den Daas, I; Foord, S; Goodson, S; Kilpatrick, G; Lee, M; Rees, S	1
Baez, M; Kursar, JD; Nelson, DL; Wainscott, DB	1
Adham, N; Bard, JA; Branchek, TA; Vaysse, P; Weinshank, RL; Zgombick, J	1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR	1
Amlaiky, N; Hen, R; Plassat, JL	1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB	1
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R	1
Chang, DJ; Eglen, RM; Jasper, JR; Kosaka, A; To, ZP	1
Brown, AM; Collin, LL; Ellis, CE; Forbes, IT; Gittins, SA; Gloger, I; Hagan, J; Middlemiss, DN; Riley, G; Thomas, DR	1
Bach, T; Krobert, KA; Kvingedal, AM; Levy, FO; Syversveen, T	1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D	1
Berardi, F; Colabufo, NA; Contino, M; Lacivita, E; Leopoldo, M; Perrone, R	1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R	1
Benhamú, B; Berkels, R; Lauterbach, T; López-Rodríguez, ML; Marco, I; Martín-Fontecha, M; Ramos, JA; Valhondo, M; Vázquez-Villa, H	1
Gürdal, H; Onaran, HO; Tulunay, FC	1
Dhasmana, KM; Saxena, PR; Tadipatri, S; Villalón, CM; Zhu, YN	1
Greene, RW; McCarley, RW; Stevens, DR	1
Feniuk, W; Saxena, PR; Tadipatri, S; van Heuven-Nolsen, D	1
Cohen, ML; Killam, AL	1
Gürdal, H; Tulunay, FC	1
Fone, KC; Marsden, CA; Robinson, AJ	1
Hoyer, D; Sahin-Erdemli, I; Schoeffter, P; Seiler, MP; Stoll, A	1
Sumner, MJ	1
Hedberg, PA; Rutlen, DL	1
Okamura, T; Toda, N	1
Coote, JH; Lewis, DI	1
Boeckxstaens, GE; Bogers, JJ; Herman, AG; Pelckmans, PA; Rampart, M; Van Maercke, YM; Verbeuren, TJ	1
Adler-Graschinsky, E; Butta, NV; Elgoyhen, AB	1
Connor, HE; Feniuk, W	1
Boeynaems, JM; Demolle, D; Van Coevorden, A	1
Hashiba, Y; Ishikawa, N; Satake, T; Sumita, T; Takagi, K	1
Lawang, A; Saxena, PR	1
Feniuk, W; Humphrey, PP; Perren, MJ; Watts, AD	1
Connor, HE; Feniuk, W; Humphrey, PP; Perren, MJ	1
Gilbert, MJ; Newberry, NR	1
Mizuno, R; Ohhashi, T	1
Miyamoto, A; Nishio, A; Sakota, T	1
Chiba, S; Vhora, S	1
Sillar, KT; Wedderburn, JF	1
Descombes, JJ; Devys, M; Laubie, M; Verbeuren, TJ	1
Coote, JH; Lewis, DI; Sermasi, E	1
Edvinsson, L; Jansen, I; Olesen, J	1
Arneklo-Nobin, B; Bodelsson, M; Törnebrandt, K	1
Horisaka, K; Kimura, I; Sugimoto, Y; Takeuchi, N; Watanabe, Y; Yamada, J	1
Bobirnac, I; Schoeffter, P	1
Crick, H; Manuel, NA; Wallis, DI	1
Frölich, D; Göthert, M; Likungu, J; Molderings, GJ	1
Böing, C; Bühlen, M; Fink, K; Göthert, M	1
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J	1
Pearce, WJ; Purdy, R; Teng, GQ; Williams, J; Zhang, L	1
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM	1
Terrón, JA	1
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D	1
George, SR; Lee, SP; O'Dowd, BF; Xie, Z	1
Bult, H; Geerts, IS; Herman, AG; Matthys, KE	1
Kinkead, R; Mitchell, GS	1
Akita, H; Inoue, N; Ishida, T; Kawashima, S; Miwa, Y; Sakoda, T; Shimokawa, Y; Shiomi, M; Ueyama, T; Yokoyama, M	1
Ge, L; Naylor, RJ; Tuladhar, BR	1
Jähnichen, S; Pertz, HH; Radtke, OA	1
Caparrotta, L; Froldi, G; Nicoletti, P; Ragazzi, E	1
Cao, YX; Edvinsson, L; He, LC; Luo, GG; Xu, CB	1

Reviews

2 review(s) available for 5-carboxamidotryptamine and ketanserin

Article	Year
Central serotonin receptors as targets for drug research. Journal of medicinal chemistry, 1987, Volume: 30, Issue:1 Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin	1987
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7). Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14 Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists	2003

Other Studies

64 other study(ies) available for 5-carboxamidotryptamine and ketanserin

Article	Year
High-level stable expression of recombinant 5-HT1A 5-hydroxytryptamine receptors in Chinese hamster ovary cells. The Biochemical journal, 1992, Aug-01, Volume: 285 ( Pt 3) Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Binding, Competitive; Blotting, Northern; Cattle; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Gene Expression; Guanosine Triphosphate; Hippocampus; Humans; Receptors, Serotonin; Recombinant Proteins; Tetrahydronaphthalenes; Transfection	1992
Mouse 5HT1B serotonin receptor: cloning, functional expression, and localization in motor control centers. Proceedings of the National Academy of Sciences of the United States of America, 1992, Apr-01, Volume: 89, Issue:7 Topics: 3T3 Cells; Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cerebellum; Corpus Striatum; Gene Expression; Genes; GTP-Binding Proteins; Mice; Molecular Sequence Data; Nucleic Acid Hybridization; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Purkinje Cells; Receptors, Serotonin; RNA, Messenger; Serotonin	1992
Computer-aided design and synthesis of 5-substituted tryptamines and their pharmacology at the 5-HT1D receptor: discovery of compounds with potential anti-migraine properties. Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18 Topics: Animals; Aorta; Computer-Aided Design; Drug Design; Haplorhini; In Vitro Techniques; Migraine Disorders; Models, Chemical; Rabbits; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Saphenous Vein; Serotonin Receptor Agonists; Structure-Activity Relationship; Tryptamines	1995
Cloning and characterisation of the human 5-HT5A serotonin receptor. FEBS letters, 1994, Dec-05, Volume: 355, Issue:3 Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Cloning, Molecular; Genome, Human; GTP-Binding Proteins; Humans; Mice; Molecular Sequence Data; Radioligand Assay; Receptors, Serotonin; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid; Serotonin; Tissue Distribution; Transfection	1994
Molecular cloning, functional expression, and mRNA tissue distribution of the human 5-hydroxytryptamine2B receptor. Molecular pharmacology, 1994, Volume: 46, Issue:2 Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; DNA, Complementary; Humans; Molecular Sequence Data; Open Reading Frames; Protein Conformation; Rats; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution	1994
Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase. The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31 Topics: Adenylyl Cyclases; Base Sequence; Cloning, Molecular; DNA Primers; Humans; Molecular Sequence Data; Receptors, Serotonin; Sequence Alignment; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction	1993
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype. The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24 Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection	1993
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase. Molecular pharmacology, 1993, Volume: 44, Issue:2 Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Cyclic AMP; DNA; Drosophila; Enzyme Activation; Humans; Intestinal Mucosa; Mice; Molecular Sequence Data; Myocardium; Receptors, Serotonin; Sequence Homology, Amino Acid; Serotonin Antagonists; Serotonin Receptor Agonists	1993
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor. Molecular pharmacology, 1993, Volume: 43, Issue:3 Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature	1993
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin Molecular pharmacology, 1996, Volume: 50, Issue:6 Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents	1996
Cloning, expression and pharmacology of a truncated splice variant of the human 5-HT7 receptor (h5-HT7b). British journal of pharmacology, 1997, Volume: 122, Issue:1 Topics: Alternative Splicing; Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; Cyclic AMP; DNA, Complementary; Humans; Molecular Sequence Data; Placenta; Radioligand Assay; Rats; Receptors, Serotonin; RNA, Messenger; Sequence Homology, Amino Acid; Sequence Homology, Nucleic Acid	1997
Functional characterisation of the human cloned 5-HT7 receptor (long form); antagonist profile of SB-258719. British journal of pharmacology, 1998, Volume: 124, Issue:6 Topics: Adenylyl Cyclases; Cell Line; Cloning, Molecular; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Piperidines; Protein Binding; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Sulfonamides	1998
The cloned human 5-HT7 receptor splice variants: a comparative characterization of their pharmacology, function and distribution. Naunyn-Schmiedeberg's archives of pharmacology, 2001, Volume: 363, Issue:6 Topics: Adenylyl Cyclases; Alternative Splicing; Binding, Competitive; Brain; Cell Line; Cloning, Organism; Genetic Variation; Humans; Radioligand Assay; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution	2001
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors. Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2 Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists	2004
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2. Journal of medicinal chemistry, 2007, Aug-23, Volume: 50, Issue:17 Topics: Amides; Animals; Cell Line; Guinea Pigs; Humans; Ileum; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship; Tetrahydronaphthalenes	2007
Physical binding pocket induction for affinity prediction. Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19 Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A	2009
New serotonin 5-HT1A receptor agonists endowed with antinociceptive activity in vivo. Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20 Topics: Analgesics; Animals; Binding, Competitive; Cyclic AMP; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP2D6 Inhibitors; HeLa Cells; Heterocyclic Compounds, 2-Ring; Humans; Hydantoins; Kinetics; Ligands; Male; Mice; Models, Chemical; Molecular Structure; Pain; Pain Measurement; Piperazines; Pyridines; Radioligand Assay; Rats; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists	2013
Role of alpha-adrenoceptors in the effects of buspirone and 5-carboxamidotryptamine in rabbit isolated thoracic aorta. General pharmacology, 1992, Volume: 23, Issue:1 Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Cystamine; Dose-Response Relationship, Drug; Drug Interactions; Ketanserin; Methysergide; Phenylephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Serotonin; Serotonin; Vasoconstriction	1992
Role of 5-HT1-like receptors in the increase in intragastric pressure induced by 5-hydroxytryptamine in the rat. European journal of pharmacology, 1992, Mar-24, Volume: 213, Issue:2 Topics: Animals; Atropine; Catecholamines; Female; Indoles; Ketanserin; Male; Methiothepin; Methysergide; Pressure; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stomach; Tropisetron	1992
Serotonin1 and serotonin2 receptors hyperpolarize and depolarize separate populations of medial pontine reticular formation neurons in vitro. Neuroscience, 1992, Volume: 47, Issue:3 Topics: Animals; Brain Stem; Electrophysiology; Female; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Potentials; Neurons; Pons; Potassium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reticular Formation; Serotonin; Serotonin Antagonists; Tetrodotoxin	1992
Analysis of the 5-HT receptors mediating contractions in the rabbit isolated renal artery. British journal of pharmacology, 1991, Volume: 104, Issue:4 Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cocaine; In Vitro Techniques; Indoles; Ketanserin; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxidopamine; Phentolamine; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan; Sympathectomy; Tetrahydronaphthalenes; Tyramine; Vasoconstrictor Agents; Vasodilation	1991
Characterization of rat platelet serotonin receptors with tryptamine agonists and the antagonists: ketanserin and SCH 23390. Thrombosis research, 1991, Nov-01, Volume: 64, Issue:3 Topics: Animals; Benzazepines; Blood Platelets; Citrates; Citric Acid; Ketanserin; Male; Platelet Aggregation; Platelet Aggregation Inhibitors; Rats; Rats, Inbred WKY; Receptors, Serotonin; Serotonin	1991
Heterogeneous inhibitory effect of nitrendipine on 5-HT-responses in rabbit vascular tissues. General pharmacology, 1991, Volume: 22, Issue:6 Topics: Animals; Aorta, Thoracic; Carotid Arteries; In Vitro Techniques; Ketanserin; Kinetics; Muscle Contraction; Muscle, Smooth, Vascular; Nitrendipine; Phenoxybenzamine; Pulmonary Artery; Rabbits; Serotonin; Serotonin Antagonists	1991
Characterization of the 5-HT receptor subtypes involved in the motor behaviours produced by intrathecal administration of 5-HT agonists in rats. British journal of pharmacology, 1991, Volume: 103, Issue:2 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Clorgyline; Fluoxetine; Injections, Spinal; Ketanserin; Male; Motor Activity; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes	1991
5-HT1-like receptors mediate 5-hydroxytryptamine-induced contraction of guinea-pig isolated iliac artery. British journal of pharmacology, 1991, Volume: 102, Issue:2 Topics: Animals; Guinea Pigs; Iliac Artery; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Receptors, Serotonin; Serotonin; Sulfonamides; Sumatriptan; Tropisetron; Vasoconstriction	1991
Characterization of the 5-HT receptor mediating endothelium-dependent relaxation in porcine vena cava. British journal of pharmacology, 1991, Volume: 102, Issue:4 Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; alpha-Methyltyrosine; Animals; Animals, Newborn; Arginine; Endothelium, Vascular; Ketanserin; Methyltyrosines; Muscle Relaxation; Muscle, Smooth, Vascular; omega-N-Methylarginine; Prostaglandin Endoperoxides, Synthetic; Receptors, Serotonin; Serotonin; Swine; Venae Cavae	1991
Influence of serotonin on total intravascular capacity in the anaesthetized dog. Acta physiologica Scandinavica, 1990, Volume: 139, Issue:4 Topics: Animals; Blood Volume; Dogs; Heart; Hemodynamics; Ketanserin; Receptors, Serotonin; Serotonin; Veins	1990
Comparison of the response to 5-carboxamidotryptamine and serotonin in isolated human, monkey and dog coronary arteries. The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2 Topics: Animals; Coronary Vessels; Dogs; Drug Interactions; Female; Humans; Ketanserin; Macaca; Male; Methysergide; Muscle, Smooth, Vascular; Serotonin; Serotonin Antagonists; Species Specificity; Vasoconstriction	1990
The influence of 5-hydroxytryptamine agonists and antagonists on identified sympathetic preganglionic neurones in the rat, in vivo. British journal of pharmacology, 1990, Volume: 99, Issue:4 Topics: Anesthesia; Animals; Electric Stimulation; Ergolines; Ganglia, Sympathetic; Homocysteine; Indoles; Iontophoresis; Ketanserin; Male; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron	1990
Pharmacological characterization of 5-hydroxytryptamine receptors in the canine terminal ileum and ileocolonic junction. The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2 Topics: Animals; Colon; Culture Techniques; Dogs; Female; Ileum; Indoles; Intestinal Mucosa; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron	1990
Different receptor subtypes mediate the dual presynaptic effects of 5-hydroxytryptamine on peripheral sympathetic neurones. Journal of autonomic pharmacology, 1989, Volume: 9, Issue:1 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cats; Cyproheptadine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Ketanserin; Male; Membranes; Metoclopramide; Neurons; Norepinephrine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes; Tropanes	1989
Influence of the endothelium on contractile effects of 5-hydroxytryptamine and selective 5-HT agonists in canine basilar artery. British journal of pharmacology, 1989, Volume: 96, Issue:1 Topics: Animals; Basilar Artery; Detergents; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Microscopy, Electron, Scanning; Octoxynol; Polyethylene Glycols; Potassium Chloride; Serotonin; Serotonin Antagonists; Sulfonamides; Sumatriptan	1989
Stimulation of aortic smooth muscle prostacyclin by serotonin: role of distinct receptors in contractile and synthetic states. Circulation research, 1989, Volume: 64, Issue:4 Topics: Animals; Aorta, Thoracic; Cattle; Cells, Cultured; Epoprostenol; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Serotonin; Stimulation, Chemical	1989
5-Hydroxytryptamine receptor subtypes participating in pulmonary edema in dogs. European journal of pharmacology, 1989, May-02, Volume: 164, Issue:1 Topics: Animals; Capillary Permeability; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Methysergide; Perfusion; Pulmonary Circulation; Pulmonary Edema; Receptors, Serotonin; Serotonin; Vascular Resistance	1989
A comparison of cardiovascular and smooth muscle effects of 5-hydroxytryptamine and 5-carboxamidotryptamine, a selective agonist of 5-HT1 receptors. Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 277, Issue:2 Topics: Airway Resistance; Animals; Cyproheptadine; Guinea Pigs; Heart Rate; Hemodynamics; Ileum; In Vitro Techniques; Ketanserin; Male; Mecamylamine; Methysergide; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Urinary Bladder	1985
A comparison of 5-hydroxytryptamine receptors mediating contraction in rabbit aorta and dog saphenous vein: evidence for different receptor types obtained by use of selective agonists and antagonists. British journal of pharmacology, 1985, Volume: 86, Issue:3 Topics: Animals; Aorta; Dogs; In Vitro Techniques; Ketanserin; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Piperidines; Rabbits; Receptors, Serotonin; Saphenous Vein; Serotonin; Serotonin Antagonists; Spiperone	1985
5-Carboxamidotryptamine is a selective agonist at 5-hydroxytryptamine receptors mediating vasodilatation and tachycardia in anaesthetized cats. British journal of pharmacology, 1986, Volume: 87, Issue:2 Topics: Animals; Blood Pressure; Cats; Female; Heart Rate; Ketanserin; Male; Methiothepin; Methysergide; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasodilation	1986
A 5-HT1-like receptor mediates a sympathetic ganglionic hyperpolarization. European journal of pharmacology, 1987, Dec-15, Volume: 144, Issue:3 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ganglia, Sympathetic; In Vitro Techniques; Ketanserin; Membrane Potentials; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tropanes	1987
5-Hydroxytryptamine-induced NO-dependent relaxation in isolated strips of monkey popliteal lymph nodes. The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 2 Topics: Animals; Arginine; Aspirin; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Lymph Nodes; Macaca; Male; Methiothepin; Methylene Blue; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; omega-N-Methylarginine; Serotonin; Serotonin Receptor Agonists	1995
Characterization of 5-hydroxytryptamine receptors on the isolated pig basilar artery by functional and radioligand binding studies. Japanese journal of pharmacology, 1994, Volume: 65, Issue:3 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Basilar Artery; Binding, Competitive; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Radioligand Assay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Swine	1994
Functional 5-HT receptor subtypes in the isolated canine common carotid artery. Heart and vessels, 1994, Volume: 9, Issue:5 Topics: Adrenergic alpha-Antagonists; Animals; Carotid Artery, Common; Diltiazem; Dogs; Female; Ketanserin; Male; Methysergide; Norepinephrine; Potassium Chloride; Quinazolines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spiperone; Vasoconstriction	1994
Modulation of rhythmic swimming activity in post-embryonic Xenopus laevis tadpoles by 5-hydroxytryptamine acting at 5HT1a receptors. Proceedings. Biological sciences, 1994, Jul-22, Volume: 257, Issue:1348 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Cyproheptadine; Ergolines; Ketanserin; Metamorphosis, Biological; Methysergide; Motor Activity; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming; Xenopus laevis	1994
Endothelial thromboxane production plays a role in the contraction caused by 5-hydroxytryptamine in rat basilar arteries. European journal of pharmacology, 1993, Oct-19, Volume: 243, Issue:2 Topics: Animals; Basilar Artery; Dioxanes; Endothelium, Vascular; In Vitro Techniques; Isometric Contraction; Ketanserin; Male; Metergoline; Muscle, Smooth, Vascular; Pentanoic Acids; Pyridines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thromboxane-A Synthase; Thromboxanes	1993
Excitatory and indirect inhibitory actions of 5-hydroxytryptamine on sympathetic preganglionic neurones in the neonate rat spinal cord in vitro. Brain research, 1993, May-07, Volume: 610, Issue:2 Topics: Action Potentials; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Female; Fluoxetine; Glycine; In Vitro Techniques; Interneurons; Ketanserin; Male; Membrane Potentials; Neurons; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists; Spinal Cord; Strychnine; Sympathetic Nervous System	1993
5-Hydroxytryptamine receptor characterization of human cerebral, middle meningeal and temporal arteries: regional differences. Acta physiologica Scandinavica, 1993, Volume: 147, Issue:2 Topics: 5-Methoxytryptamine; Cerebral Arteries; Humans; Indoles; Ketanserin; Meningeal Arteries; Methiothepin; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Temporal Arteries; Vasoconstriction; Vasoconstrictor Agents	1993
Endothelial relaxing 5-hydroxytryptamine receptors in the rat jugular vein: similarity with the 5-hydroxytryptamine1C receptor. The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Endothelium, Vascular; Female; In Vitro Techniques; Jugular Veins; Ketanserin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Vasodilation	1993
Peripherally administered serotonin induces hyperglucagonemia in mice. Life sciences, 1993, Volume: 52, Issue:23 Topics: Animals; Glucagon; Indoles; Injections, Intraperitoneal; Ketanserin; Male; Methysergide; Mice; Mice, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron	1993
5-Hydroxytryptamine 5-HT1D receptors mediating inhibition of cyclic AMP accumulation in Madin-Darby canine kidney (MDCK) cells. Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprostadil; Animals; Cells, Cultured; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Epithelium; Ketanserin; Kidney Cortex; Methiothepin; Oxadiazoles; Pertussis Toxin; Piperazines; Propranolol; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Virulence Factors, Bordetella; Yohimbine	1995
Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord. British journal of pharmacology, 1995, Volume: 116, Issue:6 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Depression, Chemical; Dioxanes; Dopamine Antagonists; Drug Interactions; Female; Ketanserin; Male; Motor Neurons; Oxadiazoles; Pindolol; Piperazines; Propranolol; Rats; Rats, Wistar; Receptors, Serotonin; Reflex, Monosynaptic; Serotonin; Serotonin Antagonists; Spinal Cord; Spiro Compounds; Sumatriptan	1995
Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium. Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3 Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cisapride; Corticosterone; Desipramine; Heart Atria; Humans; Indoles; Ketanserin; Male; Middle Aged; Norepinephrine; Oxadiazoles; Piperidines; Receptors, Presynaptic; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tritium; Tryptamines	1996
Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in the guinea-pig brain cortex. Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3 Topics: Animals; Autoreceptors; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Ketanserin; Male; Methiothepin; Oxadiazoles; Oxymetazoline; Potassium; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Synaptosomes; Tritium; Tryptamines	1996
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro? Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:7 Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron	1996
Effects of maturation, artery size, and chronic hypoxia on 5-HT receptor type in ovine cranial arteries. The American journal of physiology, 1998, Volume: 275, Issue:3 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aging; Animals; Carotid Artery, Common; Cerebral Arteries; Female; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth, Vascular; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sheep	1998
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro. American journal of respiratory and critical care medicine, 1998, Volume: 158, Issue:5 Pt 1 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron	1998
Antagonism of the relaxant 5-HT receptor in the dog basilar artery by the high-affinity 5-HT7 receptor ligand, LY215840. Proceedings of the Western Pharmacology Society, 1998, Volume: 41 Topics: Animals; Basilar Artery; Dinoprost; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Ketanserin; Lysergic Acid; Muscle Relaxation; Muscle, Smooth, Vascular; Oxadiazoles; Piperazines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists	1998
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques. European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction	1999
Serotonin 5-HT1B and 5-HT1D receptors form homodimers when expressed alone and heterodimers when co-expressed. FEBS letters, 1999, Jul-30, Volume: 456, Issue:1 Topics: Animals; Benzamides; Binding, Competitive; Cell Membrane; Cells, Cultured; Dimerization; Gene Expression; Immunoblotting; Ketanserin; Molecular Weight; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists	1999
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery. British journal of pharmacology, 1999, Volume: 127, Issue:6 Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction	1999
Time-dependent hypoxic ventilatory responses in rats: effects of ketanserin and 5-carboxamidotryptamine. The American journal of physiology, 1999, Volume: 277, Issue:3 Topics: Animals; Hypoxia; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Respiratory Mechanics; Serotonin; Serotonin Receptor Agonists; Time Factors	1999
Serotonin-induced hypercontraction through 5-hydroxytryptamine 1B receptors in atherosclerotic rabbit coronary arteries. Circulation, 2001, Mar-06, Volume: 103, Issue:9 Topics: Animals; Arteriosclerosis; Calcium; Coronary Vessels; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Ketanserin; Male; Oxadiazoles; Phenylephrine; Piperazines; Rabbits; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Vasoconstriction	2001
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum. British journal of pharmacology, 2003, Volume: 138, Issue:7 Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides	2003
Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery. Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:1 Topics: Animals; Benzamides; Brain; Carbazoles; Dinoprost; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Endothelium, Vascular; Female; Forecasting; Guinea Pigs; Iliac Artery; Indoles; Ketanserin; Male; Muscle Contraction; Muscle, Smooth; Oxadiazoles; Oxazolidinones; Piperazines; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sumatriptan; Triazoles; Tryptamines	2004
5-HT receptors mediating contraction in the rat-tail artery. Advances in experimental medicine and biology, 2003, Volume: 527 Topics: Animals; Arteries; Ketanserin; Male; Piperidones; Prazosin; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Vasoconstriction	2003
Enhanced transcription of contractile 5-hydroxytryptamine 2A receptors via extracellular signal-regulated kinase 1/2 after organ culture of rat mesenteric artery. Basic & clinical pharmacology & toxicology, 2005, Volume: 96, Issue:4 Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Ketanserin; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; RNA, Messenger; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Time Factors; Transcription, Genetic; Up-Regulation; Vasoconstriction	2005