5-bromowillardiine has been researched along with kainic acid in 4 studies
Studies (5-bromowillardiine) | Trials (5-bromowillardiine) | Recent Studies (post-2010) (5-bromowillardiine) | Studies (kainic acid) | Trials (kainic acid) | Recent Studies (post-2010) (kainic acid) |
---|---|---|---|---|---|
11 | 0 | 0 | 9,540 | 3 | 1,775 |
Protein | Taxonomy | 5-bromowillardiine (IC50) | kainic acid (IC50) |
---|---|---|---|
Glutamate receptor 1 | Rattus norvegicus (Norway rat) | 4.2857 | |
Glutamate receptor 2 | Rattus norvegicus (Norway rat) | 4.2857 | |
Glutamate receptor 3 | Rattus norvegicus (Norway rat) | 4.2857 | |
Glutamate receptor 4 | Rattus norvegicus (Norway rat) | 4.2857 | |
Glutamate receptor ionotropic, kainate 1 | Rattus norvegicus (Norway rat) | 0.0126 | |
Glutamate receptor ionotropic, kainate 1 | Homo sapiens (human) | 0.077 | |
Glutamate receptor ionotropic, kainate 2 | Rattus norvegicus (Norway rat) | 0.0126 | |
Glutamate receptor ionotropic, kainate 3 | Rattus norvegicus (Norway rat) | 0.0126 | |
Glutamate receptor ionotropic, kainate 4 | Rattus norvegicus (Norway rat) | 0.0126 | |
Glutamate receptor ionotropic, kainate 2 | Homo sapiens (human) | 0.077 | |
Glutamate receptor ionotropic, kainate 3 | Homo sapiens (human) | 0.077 | |
Glutamate receptor ionotropic, kainate 4 | Homo sapiens (human) | 0.077 | |
Glutamate receptor ionotropic, kainate 5 | Homo sapiens (human) | 0.077 | |
Glutamate receptor ionotropic, kainate 5 | Rattus norvegicus (Norway rat) | 0.0126 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (50.00) | 18.2507 |
2000's | 2 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bleakman, D; Deverill, M; Hoo, K; Jane, DE; Kamboj, R; Mandelzys, A | 1 |
Butini, S; Campiani, G; Christensen, JK; Coccone, SS; De Angelis, M; Fiorini, I; Gemma, S; Guarino, E; Morelli, E; Novellino, E; Pickering, DS; Schousboe, A; Trotta, F | 1 |
Bowie, D; Smart, TG | 1 |
Clippe, A; Gressens, P; Knoops, B; Plaisant, F; Vander Stricht, D | 1 |
4 other study(ies) available for 5-bromowillardiine and kainic acid
Article | Year |
---|---|
Synthesis of willardiine and 6-azawillardiine analogs: pharmacological characterization on cloned homomeric human AMPA and kainate receptor subtypes.
Topics: Alanine; Cell Line; Excitatory Amino Acid Agonists; Humans; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrimidinones; Radioligand Assay; Receptors, AMPA; Receptors, Kainic Acid; Recombinant Proteins; Triazines; Uracil | 1997 |
1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.
Topics: Animals; Cell Line; Electrophysiology; Excitatory Amino Acid Antagonists; Female; Humans; Ligands; Molecular Structure; Oocytes; Pyrimidinones; Rats; Receptors, Glutamate; Spodoptera; Structure-Activity Relationship; Thiophenes; Xenopus laevis | 2008 |
Interaction of 5-bromowillardiine with non-NMDA receptors expressed in Xenopus laevis oocytes injected with chick brain mRNA.
Topics: Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Brain; Chickens; Female; Ibotenic Acid; Injections; Kainic Acid; Membrane Potentials; Neuromuscular Depolarizing Agents; Oocytes; Quisqualic Acid; Receptors, Dopamine; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; RNA, Messenger; Xenopus laevis | 1991 |
Recombinant peroxiredoxin 5 protects against excitotoxic brain lesions in newborn mice.
Topics: Acetylcysteine; Alanine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Antioxidants; Brain; Catalase; Cell Death; Cells, Cultured; DNA, Complementary; Dose-Response Relationship, Drug; Electrons; Excitatory Amino Acid Agonists; Female; Humans; Kainic Acid; Male; Mice; Neurons; Peroxidases; Peroxiredoxins; Polyethylene Glycols; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Time Factors | 2003 |