Compounds > 4-methylhistamine
Page last updated: 2024-08-23

4-methylhistamine and thioperamide

4-methylhistamine has been researched along with thioperamide in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (33.33)18.2507
2000's2 (22.22)29.6817
2010's4 (44.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Buschauer, A; Dove, S; Geyer, R; Igel, P; Seifert, R; Strasser, A1
Boonnak, R; de Esch, IJ; de Graaf, C; de Kloe, G; Istyastono, EP; Jongejan, A; Leurs, R; Lim, H; Nijmeijer, S; Smit, J; Smits, RA; Wijtmans, M; Zuiderveld, O1
Buschauer, A; Geyer, R; Nordemann, U; Strasser, A; Wittmann, HJ1
Ballabeni, V; Barocelli, E; Bordi, F; Caretta, A; Impicciatore, M; Morini, G; Silva, C1
KAMEI, CH1
Chlopicki, S; Grosicki, M; Kieć-Kononowicz, K; Wójcik, T1
Goto, A; Hida, H; Mouri, A; Nagai, T; Noda, Y; Ozaki, N; Tsubai, T; Ukigai, M; Yoshimi, A1

Reviews

1 review(s) available for 4-methylhistamine and thioperamide

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

8 other study(ies) available for 4-methylhistamine and thioperamide

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists.
    Journal of medicinal chemistry, 2009, Oct-22, Volume: 52, Issue:20

    Topics: Animals; Drug Discovery; Guanidine; Guanidines; Guanosine Triphosphate; Histamine Agonists; Humans; Hydrolysis; Isotope Labeling; Mice; Models, Molecular; Protein Conformation; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship; Substrate Specificity

2009
Triazole ligands reveal distinct molecular features that induce histamine H4 receptor affinity and subtly govern H4/H3 subtype selectivity.
    Journal of medicinal chemistry, 2011, Mar-24, Volume: 54, Issue:6

    Topics: Alkynes; Azides; Click Chemistry; HEK293 Cells; Humans; Imidazoles; Ligands; Models, Molecular; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Structure-Activity Relationship; Triazoles

2011
Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists.
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Animals; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); HEK293 Cells; Histamine Agonists; Humans; Imidazoles; Mice; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Protein Conformation; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Sf9 Cells; Spodoptera; Stereoisomerism; Structure-Activity Relationship

2016
Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2-, H3-receptors in guinea-pig.
    Agents and actions, 1993, Volume: 38, Issue:3-4

    Topics: Animals; Electric Stimulation; Female; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Ileum; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Piperidines; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3

1993
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:4

    Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P

1996
In vitro study of histamine and histamine receptor ligands influence on the adhesion of purified human eosinophils to endothelium.
    European journal of pharmacology, 2016, Apr-15, Volume: 777

    Topics: Cell Adhesion; Cell Communication; Cell Line; Cell Separation; Cell Survival; Drug Inverse Agonism; Endothelium; Eosinophils; Histamine; Histamine Agonists; Histamine H1 Antagonists; Humans; Indoles; Ligands; Methylhistamines; N-Formylmethionine Leucyl-Phenylalanine; Piperazines; Piperidines; Receptors, Histamine

2016
Involvement of the histamine H4 receptor in clozapine-induced hematopoietic toxicity: Vulnerability under granulocytic differentiation of HL-60 cells.
    Toxicology and applied pharmacology, 2016, 09-01, Volume: 306

    Topics: Antipsychotic Agents; Apoptosis; Cell Differentiation; Clozapine; Granulocytes; Histamine Antagonists; HL-60 Cells; Humans; Methylhistamines; Piperidines; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Tretinoin

2016