4-methylhistamine has been researched along with dimaprit in 29 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 20 (68.97) | 18.7374 |
1990's | 5 (17.24) | 18.2507 |
2000's | 2 (6.90) | 29.6817 |
2010's | 2 (6.90) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Timmerman, H | 1 |
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Buschauer, A; Dove, S; Igel, P | 1 |
Nowak, JZ; Sek, B | 2 |
Amerini, S; Cerbai, E; Mugelli, A | 1 |
Bugajski, J; Gadek-Michalska, A | 1 |
Cortijo, J; Esplugues, J; Morcillo, EJ; Orón, JD; Ortiz, JL; Perpiñá, M; Sanz, C | 1 |
Rising, TJ; Steward, A | 1 |
Knigge, U; Matzen, S; Warberg, J | 1 |
Cazzamalli, E; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I | 1 |
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I | 1 |
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K | 1 |
Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M | 1 |
Kim, LE; Oudart, N; Sercombe, R; Teste, JF | 1 |
Tomioka, K; Yamada, T | 1 |
Bielkiewicz, B; Cook, D | 1 |
Donoso, AO; Zárate, MB | 1 |
Bielkiewicz, B; Kordecka, A; Lebrecht, U; Maslinski, C; Nowak, JZ | 1 |
Bugajski, J; Gadek, A | 2 |
Barker, LA; Hough, LB | 1 |
Nishibori, M | 1 |
Davies, MG; Greaves, MW | 1 |
Baker, AP; Chakrin, LW; Holden, DA; Smith, WJ; Sung, CP | 1 |
Brink, C; Douglas, JS; Duncan, PG | 1 |
Fukuda, K; Matsumura, F; Tanaka, S | 1 |
Akagi, T; Iwagaki, H; Kubo, S; Mori, S; Morichika, T; Nishibori, M; Takahashi, HK; Tamura, R; Tanaka, N; Yoshino, T | 1 |
Ciz, M; Jancinova, V; Lojek, A; Nosal, R; Vasicek, O | 1 |
1 review(s) available for 4-methylhistamine and dimaprit
Article | Year |
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Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
1 trial(s) available for 4-methylhistamine and dimaprit
Article | Year |
---|---|
Sensory responses of human skin to synthetic histamine analogues and histamine.
Topics: Adult; Chlorpheniramine; Dimaprit; Female; Histamine; Humans; Male; Methylhistamines; Pruritus; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea | 1980 |
27 other study(ies) available for 4-methylhistamine and dimaprit
Article | Year |
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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Histamine H4 receptor agonists.
Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship | 2010 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
Histamine and abnormal automaticity in barium- and strophanthidin-treated sheep Purkinje fibers.
Topics: Animals; Barium; Dimaprit; Electrophysiology; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Membrane Potentials; Methylhistamines; Purkinje Fibers; Sheep; Strophanthidin; Thiourea | 1990 |
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea | 1989 |
Responses to histamine and selective H2-receptor agonists in lung parenchymal strips from normal and sensitized guinea-pigs.
Topics: Animals; Benzimidazoles; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; Isoproterenol; Lung; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine H2; Thiourea | 1989 |
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
Central effects of histamine H2-receptor agonists and antagonists on nociception in the rat.
Topics: Animals; Dimaprit; Histamine H2 Antagonists; Male; Methylhistamines; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiourea | 1988 |
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea | 1988 |
The effects of histamine and some related compounds on conditioned avoidance response in rats.
Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea | 1985 |
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Effects of histamine H2-receptor agonists and antagonists on isolated guinea-pig airway muscles.
Topics: Airway Resistance; Animals; Cimetidine; Dimaprit; Drug Interactions; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea | 1982 |
Are there excitatory H2 receptors in guinea-pig ileum?
Topics: Animals; Dimaprit; Guinea Pigs; Histamine H2 Antagonists; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Muscle, Smooth; Pyrimidinones; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1983 |
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea | 1983 |
Effects of the histamine H2-receptor agonists dimaprit and 4-methylhistamine on the central noradrenaline and serotonin system.
Topics: Animals; Behavior, Animal; Brain; Dimaprit; Female; Histamine; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Methylhistamines; Norepinephrine; Rats; Receptors, Histamine; Receptors, Histamine H2; Serotonin; Thiourea; Tranylcypromine | 1980 |
Central H1- and H2-histaminergic stimulation of pituitary-adrenocortical response under stress in rats.
Topics: Animals; Corticosterone; Dimaprit; Histamine; Histamine Antagonists; Male; Methylhistamines; Pituitary-Adrenal System; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stress, Physiological; Thiourea | 1983 |
Selectivity of 4-methylhistamine at H1- and H2-receptors in the guinea-pig isolated ileum.
Topics: Animals; Dibenzylchlorethamine; Dimaprit; Drug Interactions; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Effect of intracerebroventricular impromidine on pituitary-adrenocortical response to stress in rats.
Topics: Adrenal Cortex; Animals; Atropine; Cimetidine; Corticosterone; Dimaprit; Imidazoles; Impromidine; Injections, Intraventricular; Male; Methylhistamines; Pituitary Gland; Propranolol; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Sympatholytics; Thiourea | 1984 |
Cyclic AMP increase in canine parotid gland mediated by histamine H2-receptors.
Topics: Animals; Cyclic AMP; Dimaprit; Dogs; Female; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Parotid Gland; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1981 |
Effect of histamine agonists and antagonists on the production of murine reaginic antibodies.
Topics: Animals; Antibody Formation; Dimaprit; Histamine; Histamine Antagonists; Immunoglobulin E; Male; Methylhistamines; Metiamide; Mice; Reagins; Receptors, Histamine; Thiourea | 1981 |
Changes in the response of guinea-pig airways in vivo and in vitro to cimetidine and propranolol during development.
Topics: Aging; Airway Resistance; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Propranolol; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea | 1982 |
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium | 1994 |
Histamine H2 receptor mediates keratan sulfate secretion in rabbit chondrocytes: role of cAMP.
Topics: Animals; Bucladesine; Cartilage, Articular; Cells, Cultured; Cholera Toxin; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dinoprostone; Enzyme-Linked Immunosorbent Assay; Keratan Sulfate; Kinetics; Methylhistamines; Parathyroid Hormone; Proteoglycans; Rabbits; Receptors, Histamine H2; Sulfates; Sulfur Radioisotopes | 1993 |
Histamine downregulates CD14 expression via H2 receptors on human monocytes.
Topics: Cells, Cultured; Dimaprit; Down-Regulation; Histamine; Histamine Agonists; Histamine H2 Antagonists; Humans; Leukocytes, Mononuclear; Lipopolysaccharide Receptors; Lipopolysaccharides; Methylhistamines; Monocytes; Receptors, Histamine H2; Time Factors; Tumor Necrosis Factor-alpha | 2003 |
Role of histamine receptors in the effects of histamine on the production of reactive oxygen species by whole blood phagocytes.
Topics: Benzimidazoles; Dimaprit; Guanidines; Histamine; Histamine Agonists; Humans; Male; Methylhistamines; Phagocytes; Reactive Oxygen Species; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4; Thiourea | 2014 |