Page last updated: 2024-08-23

4-methylhistamine and dimaprit

4-methylhistamine has been researched along with dimaprit in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199020 (68.97)18.7374
1990's5 (17.24)18.2507
2000's2 (6.90)29.6817
2010's2 (6.90)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Buschauer, A; Dove, S; Igel, P1
Nowak, JZ; Sek, B2
Amerini, S; Cerbai, E; Mugelli, A1
Bugajski, J; Gadek-Michalska, A1
Cortijo, J; Esplugues, J; Morcillo, EJ; Orón, JD; Ortiz, JL; Perpiñá, M; Sanz, C1
Rising, TJ; Steward, A1
Knigge, U; Matzen, S; Warberg, J1
Cazzamalli, E; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I1
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Tomioka, K; Yamada, T1
Bielkiewicz, B; Cook, D1
Donoso, AO; Zárate, MB1
Bielkiewicz, B; Kordecka, A; Lebrecht, U; Maslinski, C; Nowak, JZ1
Bugajski, J; Gadek, A2
Barker, LA; Hough, LB1
Nishibori, M1
Davies, MG; Greaves, MW1
Baker, AP; Chakrin, LW; Holden, DA; Smith, WJ; Sung, CP1
Brink, C; Douglas, JS; Duncan, PG1
Fukuda, K; Matsumura, F; Tanaka, S1
Akagi, T; Iwagaki, H; Kubo, S; Mori, S; Morichika, T; Nishibori, M; Takahashi, HK; Tamura, R; Tanaka, N; Yoshino, T1
Ciz, M; Jancinova, V; Lojek, A; Nosal, R; Vasicek, O1

Reviews

1 review(s) available for 4-methylhistamine and dimaprit

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Trials

1 trial(s) available for 4-methylhistamine and dimaprit

ArticleYear
Sensory responses of human skin to synthetic histamine analogues and histamine.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:5

    Topics: Adult; Chlorpheniramine; Dimaprit; Female; Histamine; Humans; Male; Methylhistamines; Pruritus; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea

1980

Other Studies

27 other study(ies) available for 4-methylhistamine and dimaprit

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Histamine H4 receptor agonists.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2010
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Histamine and abnormal automaticity in barium- and strophanthidin-treated sheep Purkinje fibers.
    Agents and actions, 1990, Volume: 31, Issue:1-2

    Topics: Animals; Barium; Dimaprit; Electrophysiology; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Membrane Potentials; Methylhistamines; Purkinje Fibers; Sheep; Strophanthidin; Thiourea

1990
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Responses to histamine and selective H2-receptor agonists in lung parenchymal strips from normal and sensitized guinea-pigs.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Animals; Benzimidazoles; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; Histamine; Imidazoles; Impromidine; Isoproterenol; Lung; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine H2; Thiourea

1989
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1986
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
Central effects of histamine H2-receptor agonists and antagonists on nociception in the rat.
    Agents and actions, 1988, Volume: 23, Issue:3-4

    Topics: Animals; Dimaprit; Histamine H2 Antagonists; Male; Methylhistamines; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiourea

1988
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
    Acta endocrinologica, 1988, Volume: 119, Issue:4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea

1988
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
    International archives of allergy and applied immunology, 1986, Volume: 79, Issue:3

    Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Effects of histamine H2-receptor agonists and antagonists on isolated guinea-pig airway muscles.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 255, Issue:1

    Topics: Airway Resistance; Animals; Cimetidine; Dimaprit; Drug Interactions; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1982
Are there excitatory H2 receptors in guinea-pig ileum?
    Proceedings of the Western Pharmacology Society, 1983, Volume: 26

    Topics: Animals; Dimaprit; Guinea Pigs; Histamine H2 Antagonists; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Muscle, Smooth; Pyrimidinones; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1983
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
    Experimental brain research, 1983, Volume: 52, Issue:2

    Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea

1983
Effects of the histamine H2-receptor agonists dimaprit and 4-methylhistamine on the central noradrenaline and serotonin system.
    Agents and actions, 1980, Volume: 10, Issue:1 Pt 2

    Topics: Animals; Behavior, Animal; Brain; Dimaprit; Female; Histamine; Hydroxyindoleacetic Acid; Methoxyhydroxyphenylglycol; Methylhistamines; Norepinephrine; Rats; Receptors, Histamine; Receptors, Histamine H2; Serotonin; Thiourea; Tranylcypromine

1980
Central H1- and H2-histaminergic stimulation of pituitary-adrenocortical response under stress in rats.
    Neuroendocrinology, 1983, Volume: 36, Issue:6

    Topics: Animals; Corticosterone; Dimaprit; Histamine; Histamine Antagonists; Male; Methylhistamines; Pituitary-Adrenal System; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stress, Physiological; Thiourea

1983
Selectivity of 4-methylhistamine at H1- and H2-receptors in the guinea-pig isolated ileum.
    British journal of pharmacology, 1983, Volume: 80, Issue:1

    Topics: Animals; Dibenzylchlorethamine; Dimaprit; Drug Interactions; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Effect of intracerebroventricular impromidine on pituitary-adrenocortical response to stress in rats.
    Agents and actions, 1984, Volume: 14, Issue:5-6

    Topics: Adrenal Cortex; Animals; Atropine; Cimetidine; Corticosterone; Dimaprit; Imidazoles; Impromidine; Injections, Intraventricular; Male; Methylhistamines; Pituitary Gland; Propranolol; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Sympatholytics; Thiourea

1984
Cyclic AMP increase in canine parotid gland mediated by histamine H2-receptors.
    European journal of pharmacology, 1981, Dec-17, Volume: 76, Issue:4

    Topics: Animals; Cyclic AMP; Dimaprit; Dogs; Female; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Parotid Gland; Pyridines; Receptors, Histamine; Receptors, Histamine H2; Thiourea

1981
Effect of histamine agonists and antagonists on the production of murine reaginic antibodies.
    International journal of immunopharmacology, 1981, Volume: 3, Issue:4

    Topics: Animals; Antibody Formation; Dimaprit; Histamine; Histamine Antagonists; Immunoglobulin E; Male; Methylhistamines; Metiamide; Mice; Reagins; Receptors, Histamine; Thiourea

1981
Changes in the response of guinea-pig airways in vivo and in vitro to cimetidine and propranolol during development.
    British journal of pharmacology, 1982, Volume: 75, Issue:3

    Topics: Aging; Airway Resistance; Animals; Bronchi; Cimetidine; Dimaprit; Female; Guanidines; Guinea Pigs; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Propranolol; Receptors, Histamine; Receptors, Histamine H2; Thiourea; Trachea

1982
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium

1994
Histamine H2 receptor mediates keratan sulfate secretion in rabbit chondrocytes: role of cAMP.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Animals; Bucladesine; Cartilage, Articular; Cells, Cultured; Cholera Toxin; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dinoprostone; Enzyme-Linked Immunosorbent Assay; Keratan Sulfate; Kinetics; Methylhistamines; Parathyroid Hormone; Proteoglycans; Rabbits; Receptors, Histamine H2; Sulfates; Sulfur Radioisotopes

1993
Histamine downregulates CD14 expression via H2 receptors on human monocytes.
    Clinical immunology (Orlando, Fla.), 2003, Volume: 108, Issue:3

    Topics: Cells, Cultured; Dimaprit; Down-Regulation; Histamine; Histamine Agonists; Histamine H2 Antagonists; Humans; Leukocytes, Mononuclear; Lipopolysaccharide Receptors; Lipopolysaccharides; Methylhistamines; Monocytes; Receptors, Histamine H2; Time Factors; Tumor Necrosis Factor-alpha

2003
Role of histamine receptors in the effects of histamine on the production of reactive oxygen species by whole blood phagocytes.
    Life sciences, 2014, Mar-28, Volume: 100, Issue:1

    Topics: Benzimidazoles; Dimaprit; Guanidines; Histamine; Histamine Agonists; Humans; Male; Methylhistamines; Phagocytes; Reactive Oxygen Species; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4; Thiourea

2014