Page last updated: 2024-09-05

4-methoxyphenylboronic acid and benzeneboronic acid

4-methoxyphenylboronic acid has been researched along with benzeneboronic acid in 6 studies

Compound Research Comparison

Studies
(4-methoxyphenylboronic acid)
Trials
(4-methoxyphenylboronic acid)
Recent Studies (post-2010)
(4-methoxyphenylboronic acid)
Studies
(benzeneboronic acid)
Trials
(benzeneboronic acid)
Recent Studies (post-2010) (benzeneboronic acid)
10066880485

Protein Interaction Comparison

ProteinTaxonomy4-methoxyphenylboronic acid (IC50)benzeneboronic acid (IC50)
Fatty-acid amide hydrolase 1Rattus norvegicus (Norway rat)2.6
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2Homo sapiens (human)10

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (16.67)18.2507
2000's2 (33.33)29.6817
2010's3 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baquero, F; Blázquez, J; Shoichet, BK; Weston, GS1
Käsnänen, H; Leppänen, J; Minkkilä, A; Nevalainen, T; Poso, A; Saario, SM1
Hall, RA; Innocenti, A; Mühlschlegel, FA; Scozzafava, A; Supuran, CT; Winum, JY1
Belitsky, JM1
Bouillon, A; Cresteil, T; Fontaine, F; Hequet, A; Jolivalt, C; Lesnard, A; Rault, S; Voisin-Chiret, AS1
Cole, DC; Hixon, MS; Istratiy, Y; Jennings, A; Klein, MG; Lanier, M; Schwartz, PA; Tjhen, R1

Other Studies

6 other study(ies) available for 4-methoxyphenylboronic acid and benzeneboronic acid

ArticleYear
Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase.
    Journal of medicinal chemistry, 1998, Nov-05, Volume: 41, Issue:23

    Topics: Anti-Bacterial Agents; Bacterial Proteins; beta-Lactam Resistance; beta-Lactamase Inhibitors; beta-Lactamases; Binding Sites; Boronic Acids; Crystallography, X-Ray; Drug Synergism; Enterobacter cloacae; Enzyme Inhibitors; Escherichia coli; Microbial Sensitivity Tests; Models, Molecular; Structure-Activity Relationship; Thiophenes

1998
Discovery of boronic acids as novel and potent inhibitors of fatty acid amide hydrolase.
    Journal of medicinal chemistry, 2008, Nov-27, Volume: 51, Issue:22

    Topics: Amidohydrolases; Boronic Acids; Dose-Response Relationship, Drug; Drug Discovery; Enzyme Inhibitors; Molecular Structure; Stereoisomerism; Structure-Activity Relationship

2008
Carbonic anhydrase inhibitors. Inhibition of the fungal beta-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids.
    Bioorganic & medicinal chemistry letters, 2009, May-15, Volume: 19, Issue:10

    Topics: Boronic Acids; Candida albicans; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Cryptococcus neoformans; Humans; Structure-Activity Relationship

2009
Aryl boronic acid inhibition of synthetic melanin polymerization.
    Bioorganic & medicinal chemistry letters, 2010, Aug-01, Volume: 20, Issue:15

    Topics: Boronic Acids; Catechols; Levodopa; Melanins; Structure-Activity Relationship

2010
First identification of boronic species as novel potential inhibitors of the Staphylococcus aureus NorA efflux pump.
    Journal of medicinal chemistry, 2014, Mar-27, Volume: 57, Issue:6

    Topics: Anti-Bacterial Agents; Antineoplastic Agents; Bacterial Proteins; Boronic Acids; Cell Survival; Ciprofloxacin; Culture Media; Drug Resistance, Bacterial; Drug Screening Assays, Antitumor; Humans; Indicators and Reagents; KB Cells; Microbial Sensitivity Tests; Multidrug Resistance-Associated Proteins; Staphylococcus aureus; Structure-Activity Relationship

2014
Repurposing Suzuki Coupling Reagents as a Directed Fragment Library Targeting Serine Hydrolases and Related Enzymes.
    Journal of medicinal chemistry, 2017, 06-22, Volume: 60, Issue:12

    Topics: Boronic Acids; Crystallography, X-Ray; Drug Evaluation, Preclinical; Humans; Nitriles; Phosphoric Diester Hydrolases; Serine Endopeptidases; Serine Proteinase Inhibitors; Small Molecule Libraries; Structure-Activity Relationship; Surface Plasmon Resonance

2017