Compounds > 4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide
Page last updated: 2024-09-03

4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide and bisindolylmaleimide i

4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide has been researched along with bisindolylmaleimide i in 3 studies

Compound Research Comparison

Studies
(4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide)		Trials
(4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide)		Recent Studies (post-2010)
(4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide)		Studies
(bisindolylmaleimide i)		Trials
(bisindolylmaleimide i)		Recent Studies (post-2010) (bisindolylmaleimide i)
620141,1981174

Protein Interaction Comparison

ProteinTaxonomy4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide (IC50)bisindolylmaleimide i (IC50)
Chain A, Protein kinase C, iotaHomo sapiens (human)5.8
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)9
G2/mitotic-specific cyclin-B2Homo sapiens (human)2.3
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.5
Protein kinase C gamma typeHomo sapiens (human)0.03
Protein kinase C beta typeHomo sapiens (human)0.0054
Cyclin-dependent kinase 1Homo sapiens (human)2.3
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.068
Cyclin-dependent kinase 4Homo sapiens (human)0.99
G2/mitotic-specific cyclin-B1Homo sapiens (human)2.3
Lethal factorBacillus anthracis1.5
Protein kinase C alpha typeHomo sapiens (human)0.0055
Glycogen synthase kinase-3 betaRattus norvegicus (Norway rat)0.36
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoformOryctolagus cuniculus (rabbit)0.7
G1/S-specific cyclin-D1Homo sapiens (human)0.99
Protein kinase C eta typeHomo sapiens (human)0.0066
G1/S-specific cyclin-E1Homo sapiens (human)0.99
Cyclin-dependent kinase 2Homo sapiens (human)0.99
cAMP-dependent protein kinase catalytic subunit alpha Rattus norvegicus (Norway rat)2
Protein kinase C iota typeHomo sapiens (human)3.463
Glycogen synthase kinase-3 betaHomo sapiens (human)0.19
Protein kinase C epsilon typeHomo sapiens (human)0.0067
Protein kinase C theta typeHomo sapiens (human)0.0061
Protein kinase C zeta typeHomo sapiens (human)5.8
Protein kinase C delta typeHomo sapiens (human)0.0096
Peroxisome proliferator-activated receptor alphaHomo sapiens (human)0.006
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)7.3
G2/mitotic-specific cyclin-B3Homo sapiens (human)2.3
Serine/threonine-protein kinase LMTK3Homo sapiens (human)0.0001

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Jadhav, A; Kerns, E; Nguyen, K; Shah, P; Sun, H; Xu, X; Yan, Z; Yu, KR1
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR1
Kabir, M; Kerns, E; Neyra, J; Nguyen, K; Nguyễn, ÐT; Shah, P; Siramshetty, VB; Southall, N; Williams, J; Xu, X; Yu, KR1

Other Studies

3 other study(ies) available for 4-diethoxyphosphorylmethyl-n-(4-bromo-2-cyanophenyl)benzamide and bisindolylmaleimide i

ArticleYear
Highly predictive and interpretable models for PAMPA permeability.
    Bioorganic & medicinal chemistry, 2017, 02-01, Volume: 25, Issue:3

    Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Humans; Models, Biological; Organic Chemicals; Regression Analysis; Support Vector Machine

2017
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility

2019
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models.
    Scientific reports, 2020, 11-26, Volume: 10, Issue:1

    Topics: Animals; Computer Simulation; Databases, Factual; Drug Discovery; High-Throughput Screening Assays; Liver; Machine Learning; Male; Microsomes, Liver; National Center for Advancing Translational Sciences (U.S.); Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Retrospective Studies; United States

2020