4-butyrolactone has been researched along with dihydroxyphenylalanine in 57 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 44 (77.19) | 18.7374 |
1990's | 10 (17.54) | 18.2507 |
2000's | 3 (5.26) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Roth, RH; Walters, JR | 1 |
Morgenroth, VH; Roth, RH; Walters, JR | 1 |
Persson, SA | 2 |
Nowycky, MC; Roth, RH | 1 |
Morgenroth, VH; Nowycky, MC; Roth, RH; Walters, JR | 1 |
Engel, J; Liljequist, S | 3 |
Biswas, B; Carlsson, A | 1 |
Kehr, W; Speckenbach, W; Zimmermann, R | 1 |
Demarest, KT; Moore, KE | 1 |
Carboni, E; Di Chiara, G; Tanda, G | 1 |
Waldmeier, PC | 1 |
De Vries, JB; Duran, R; Westerink, BH | 1 |
Ali, SF; Gough, BJ; Holson, RR; Newport, GD; Scalzo, FM | 1 |
Greiner, HE; Haase, AF; Seyfried, CA | 1 |
Pettibone, DJ; Pfleuger, AB; Totaro, JA | 1 |
Galloway, MP; Roth, RH; Wolf, ME | 2 |
Barton, AC; Demarest, KT; Moore, KE | 1 |
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Namba, Y | 1 |
Dijkstra, D; Horn, AS; Vermue, NA | 1 |
Bean, AJ; Bunney, BS; Nestler, EJ; Roth, RH; Shepard, PD | 1 |
Andersson, B; Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, AM; Sanchez, D; Svensson, K; Wikström, H | 1 |
Kaneno, S; Takahashi, R; Watanabe, A | 1 |
Gunnet, JW; Lindley, SE; Lookingland, KJ; Moore, KE | 1 |
Anderson, CM; Ely, TD; Kilts, CD; Nishita, JK | 1 |
Nakagawa, K; Sekihara, S; Somei, M; Watanabe, H; Yamada, F | 1 |
De Vries, JB; Dijkstra, D; Hazelhoff, B; Horn, AS; Mulder, TB | 1 |
Esposito, E; Samanin, R; Spampinato, U | 1 |
Howard, HR; Kelly, TR; Koe, BK; Sarges, R | 1 |
Tissari, AH | 1 |
Spaan, SJ; van Es, TP; Westerink, BH | 1 |
Demarest, KT; Lawson-Wendling, KL; Moore, KE | 1 |
Dijkstra, D; Horn, AS; Houwing, HA; Van Oene, JC | 1 |
Frau, MI; Gessa, GL; Meloni, M; Rossetti, ZL; Tissari, AH | 1 |
Andén, NE; Grabowska-Andén, M; Liljenberg, B | 1 |
Fadda, F; Gessa, GL; Marcou, M; Mosca, E; Rossetti, Z | 1 |
Feenstra, MG; Horn, AS; Westerink, BH; Wirix, E | 1 |
De Vries, JB; Dijkstra, D; Horn, AS; Renkema, RJ; Tepper, PG; Van Oene, JC | 1 |
Marek, KL; Roth, RH | 1 |
Bannon, MJ; Bunney, EB; Roth, RH; Skirboll, LR; Zigun, JR | 1 |
Bannon, MJ; Michaud, RL; Roth, RH | 1 |
Fernstrom, J; Sved, A | 1 |
Kummer, P; Stock, G | 1 |
Argiolas, A; Fadda, F; Gessa, GL; Marcou, M; Melis, MR; Porceddu, ML | 1 |
Hirose, T; Kikuchi, T; Miwa, T; Morita, S; Oshiro, Y; Tottori, K; Uwahodo, Y | 1 |
Akunne, HC; Cooke, LW; Davis, MD; DeMattos, SB; Georgic, LM; MacKenzie, RG; Rugsley, TA; Shih, YH; van Leeuwen, DH; Whetzel, SZ | 1 |
Baldessarini, RJ; Huston-Lyons, D; Marsh, ER | 1 |
Bartoszyk, GD; Seyfried, CA | 1 |
Bristow, LJ; Cook, GP; Gay, JC; Hutson, PH; Kulagowski, JJ; Landon, L; Murray, F; Saywell, KL; Young, L | 1 |
Kikuchi, T; Kurahashi, N; Nishi, T; Oshiro, Y; Sato, S; Tanaka, T; Tottori, K; Uwahodo, Y | 1 |
Carr, KD; Garcia-Espana, A; Goldstein, M; Haycock, JW; Lee, KY; Lew, JY; Meller, E | 1 |
Ahlenius, S; Ericson, E; Florvall, L; Hillegaart, V; Jiménez, P; Wijkström, A | 1 |
Bettler, B; Bräuner-Osborne, H; Cryan, JF; Froestl, W; Kaupmann, K; Klebs, K; Mombereau, C; Mosbacher, J; Sansig, G; Schmutz, M; van der Putten, H; Waldmeier, P; Wellendorph, P | 1 |
Bongiovanni, R; Jaskiw, GE; Newbould, E; Young, D | 1 |
3 review(s) available for 4-butyrolactone and dihydroxyphenylalanine
Article | Year |
---|---|
Dopaminergic neurons - alteration in the sensitivity of tyrosine hydroxylase to inhibition by endovenous dopamine after cessation of impulse flow.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Haloperidol; Male; Neurons; Rats; Receptors, Adrenergic; Synapses; Synaptic Transmission; Tyrosine 3-Monooxygenase | 1976 |
The effect of chronic ethanol administration on central neurotransmitter mechanisms.
Topics: 4-Butyrolactone; Animals; Aromatic-L-Amino-Acid Decarboxylases; Behavior, Animal; Brain; Catecholamines; Dihydroxyphenylalanine; Dopamine; Ethanol; gamma-Aminobutyric Acid; Humans; Male; Mice; Neurons; Neurotransmitter Agents; Norepinephrine; Propranolol; Rats; Receptors, Cholinergic; Receptors, Dopamine; Substance Withdrawal Syndrome; Synaptic Transmission; Time Factors | 1979 |
Interaction of haloperidol and gamma-butyrolactone with (+)-amphetamine-induced changes in monoamine synthesis and metabolism in rat brain.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; Amphetamine; Animals; Biogenic Amines; Brain; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Drug Interactions; Furans; Haloperidol; Limbic System; Male; Rats; Tyramine | 1977 |
54 other study(ies) available for 4-butyrolactone and dihydroxyphenylalanine
Article | Year |
---|---|
Dopaminergic neurons--alteration in the kinetic properties of tyrosine hydroxylase after cessation of impulse flow.
Topics: 4-Butyrolactone; Animals; Apomorphine; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Egtazic Acid; Female; Kinetics; Male; Median Eminence; Neurons; Olfactory Bulb; Piperazines; Pterins; Rats; Receptors, Adrenergic; Substantia Nigra; Synapses; Synaptic Transmission; Tyrosine 3-Monooxygenase | 1976 |
The effect of LSD and 2-bromo LSD on the striatal DOPA accumulation after decarboxylase inhibition in rats.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Corpus Striatum; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Lysergic Acid Diethylamide; Male; Neural Pathways; Rats; Reserpine; Substantia Nigra; Time Factors | 1977 |
Nonstriatal dopaminergic neurons: role of presynaptic receptors in the modulation of transmitter synthesis.
Topics: 4-Butyrolactone; Animals; Apomorphine; Calcium; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Kinetics; Limbic System; Neurons; Rats; Receptors, Dopamine; Synapses; Tyrosine 3-Monooxygenase | 1977 |
gamma-Hydroxybutyrate: effects on nonstriatal dopaminergic neurons.
Topics: 4-Butyrolactone; Animals; Brain; Dihydroxyphenylalanine; Dopamine; Egtazic Acid; Hydroxybutyrates; Kinetics; Neurons; Picrotoxin; Rats; Tyrosine 3-Monooxygenase | 1977 |
On the mode of action of diazepam on brain catecholamine metabolism.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; Anesthesia; Animals; Brain; Catecholamines; Diazepam; Dihydroxyphenylalanine; Dopamine; gamma-Aminobutyric Acid; Male; Rats | 1978 |
Effect of morphine on the accumulation of DOPA after decarboxylase inhibition in the rat.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Dihydroxyphenylalanine; DNA; Haloperidol; Male; Morphine; Naloxone; Rats; Receptors, Drug; Reserpine; Time Factors | 1979 |
Attenuation of the gamma-butyrolactone-induced increase in DOPA accumulation by chronic ethanol administration.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Corpus Striatum; Dihydroxyphenylalanine; Ethanol; Furans; Limbic System; Male; Rats | 1979 |
Comparison of dopamine synthesis regulation in the terminals of nigrostriatal, mesolimbic, tuberoinfundibular and tuberohypophyseal neurons.
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Benzyl Alcohols; Dihydroxyphenylalanine; Dopamine; Hydrazines; Hypothalamo-Hypophyseal System; Male; Median Eminence; Nialamide; Olfactory Bulb; Piribedil; Pituitary Gland, Posterior; Rats; Reserpine | 1979 |
Extracellular striatal concentrations of endogenous 3,4-dihydroxyphenylalanine in the absence of a decarboxylase inhibitor: a dynamic index of dopamine synthesis in vivo.
Topics: 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Carboxy-Lyases; Chromatography, High Pressure Liquid; Colorimetry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Extracellular Matrix; Haloperidol; Male; Methyltyrosines; Rats; Rats, Sprague-Dawley; Tetrodotoxin | 1992 |
The GABAB antagonist, CGP 35348, antagonizes the effects of baclofen, gamma-butyrolactone and HA 966 on rat striatal dopamine synthesis.
Topics: 4-Butyrolactone; Animals; Baclofen; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; GABA-A Receptor Antagonists; Haloperidol; Organophosphorus Compounds; Pyrrolidinones; Rats; Tetrabenazine | 1991 |
Use of microdialysis for monitoring tyrosine hydroxylase activity in the brain of conscious rats.
Topics: 1-Methyl-4-phenylpyridinium; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Apomorphine; Brain; Chromatography, High Pressure Liquid; Consciousness; Dialysis; Dihydroxyphenylalanine; Haloperidol; Male; Methyltyrosines; Monitoring, Physiologic; Rats; Rats, Inbred Strains; Tyrosine 3-Monooxygenase | 1990 |
Chronic prenatal haloperidol exposure: lack of effect on presynaptic dopamine autoreceptors.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain Chemistry; Caudate Nucleus; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Female; Haloperidol; Hydrazines; Nucleus Accumbens; Olfactory Bulb; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, Dopamine; Synapses | 1989 |
Biochemical and functional studies on EMD 49,980: a potent, selectively presynaptic D-2 dopamine agonist with actions on serotonin systems.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; Acetylcholine; Animals; Brain Chemistry; Dihydroxyphenylalanine; Dopamine Agents; Hippocampus; Hydroxydopamines; Indoles; Male; Oxidopamine; Oxindoles; p-Chloroamphetamine; Pyridines; Rats; Rats, Inbred Strains; Reserpine; Serotonin; Synaptosomes | 1989 |
Comparison of the effects of recently developed alpha 2-adrenergic antagonists with yohimbine and rauwolscine on monoamine synthesis in rat brain.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Biogenic Amines; Brain; Dihydroxyphenylalanine; Dioxanes; Idazoxan; Male; Mianserin; Norepinephrine; Quinolizines; Rats; Rats, Inbred Strains; Serotonin; Yohimbine | 1985 |
Regulation of dopamine synthesis in the medial prefrontal cortex: studies in brain slices.
Topics: 4-Butyrolactone; Animals; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Frontal Lobe; In Vitro Techniques; Indoles; Male; Models, Biological; Nomifensine; Potassium; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tyrosine 3-Monooxygenase | 1986 |
Differential action of bromocriptine on nigrostriatal versus mesolimbic dopaminergic neurons.
Topics: 4-Butyrolactone; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Ergolines; Limbic System; Male; Nucleus Accumbens; Olfactory Bulb; Prolactin; Rats; Time Factors | 1987 |
Relationship between receptor occupancy and response at striatal dopamine autoreceptors.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Homeostasis; Hydrazines; Levodopa; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
Pharmacological profile of a chromanamine analogue (DP-6OH-3CA) of the selective presynaptic dopamine agonist N,N-dipropyl-7-hydroxy-2-aminotetralin.
Topics: 4-Butyrolactone; Animals; Benzopyrans; Binding, Competitive; Cattle; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; In Vitro Techniques; Male; Mice; Motor Activity; Naphthalenes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Tetrahydronaphthalenes | 1988 |
The effects of pertussis toxin on autoreceptor-mediated inhibition of dopamine synthesis in the rat striatum.
Topics: 4-Butyrolactone; Adenosine Diphosphate Ribose; Animals; Apomorphine; Chromatography, High Pressure Liquid; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; GTP-Binding Proteins; Hydrazines; Male; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Virulence Factors, Bordetella | 1988 |
Regulation of dopamine synthesis in the medial prefrontal cortex is mediated by release modulating autoreceptors: studies in vivo.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Feedback; Frontal Lobe; Hydrazines; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
(+)-UH 232 and (+)-UH 242: novel stereoselective dopamine receptor antagonists with preferential action on autoreceptors.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Male; Motor Activity; Naphthalenes; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Serotonin; Stereoisomerism; Tetrahydronaphthalenes | 1986 |
Alteration of striatal dopaminergic functions implicated in methamphetamine-induced reverse tolerance in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Behavior, Animal; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Drug Tolerance; Homovanillic Acid; Male; Methamphetamine; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
Effect of electrical stimulation of the arcuate nucleus on neurochemical estimates of tuberoinfundibular and tuberohypophysial dopaminergic neuronal activities.
Topics: 4-Butyrolactone; 5-Hydroxytryptophan; Animals; Arcuate Nucleus of Hypothalamus; Dihydroxyphenylalanine; Dopamine; Electric Stimulation; Male; Median Eminence; Neurons; Osmolar Concentration; Pituitary Gland, Posterior; Prolactin; Rats; Rats, Inbred Strains | 1987 |
Absence of synthesis-modulating nerve terminal autoreceptors on mesoamygdaloid and other mesolimbic dopamine neuronal populations.
Topics: 4-Butyrolactone; Amygdala; Animals; Apomorphine; Dihydroxyphenylalanine; Dopamine; Hydrazines; Limbic System; Male; Medial Forebrain Bundle; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
Dopamine receptor stimulating effects of chanoclavine analogues, tricyclic ergot alkaloids, in the brain.
Topics: 4-Butyrolactone; Animals; Binding, Competitive; Brain; Catechols; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Ergot Alkaloids; In Vitro Techniques; Male; Mice; Rats; Rats, Inbred Strains; Receptors, Dopamine; Rotation; Spiperone; Stereotyped Behavior; Time Factors | 1987 |
N-methyl,N-propargyl-2-aminotetralins:novel dopamine agonists with monoamine oxidase inhibiting properties.
Topics: 4-Butyrolactone; Alkynes; Animals; Apomorphine; Brain; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Female; Humans; In Vitro Techniques; Mice; Monoamine Oxidase Inhibitors; Motor Activity; Naphthalenes; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Tetrahydronaphthalenes | 1985 |
Serotonin agonists reduce dopamine synthesis in the striatum only when the impulse flow of nigro-striatal neurons is intact.
Topics: 4-Butyrolactone; Animals; Benserazide; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Male; Methoxydimethyltryptamines; Neurons; Piperazines; Rats; Serotonin Antagonists; Substantia Nigra | 1985 |
Synthesis and dopamine autoreceptor activity of a 5-(methylmercapto)methyl-substituted derivative of (+/-)-3-PPP (3-(3-hydroxyphenyl)-1-n-propylpiperidine).
Topics: 4-Butyrolactone; Animals; Chemical Phenomena; Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Mice; Piperidines; Rats; Receptors, Dopamine; Structure-Activity Relationship | 1985 |
Increase of dopamine synthesis in synaptosomes from rats treated with neuroleptics or reserpine.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Haloperidol; Kinetics; Male; Rats; Rats, Inbred Strains; Reserpine; Sulpiride; Synaptosomes; Temperature; Tyrosine 3-Monooxygenase | 1982 |
Effects of drugs interfering with dopamine and noradrenaline biosynthesis on the endogenous 3,4-dihydroxyphenylalanine levels in rat brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Apomorphine; Brain; Chlorpromazine; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dopamine; Female; Homovanillic Acid; Norepinephrine; Rats; Rats, Inbred Strains; Tissue Distribution; Tyrosine 3-Monooxygenase | 1982 |
d-Amphetamine and gamma-butyrolactone alteration of dopamine synthesis in the terminals of nigrostriatal and mesolimbic neurons. Possible role of various autoreceptor sensitivities.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain Chemistry; Corpus Striatum; Dextroamphetamine; Dihydroxyphenylalanine; Dopamine; Furans; Haloperidol; Limbic System; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra | 1983 |
trans-N-n-Propyl-7-hydroxy-octahydrobenzo(f)quinoline, a rigid 3-PPP analogue with greater potency but lack of selectivity for dopamine autoreceptors.
Topics: 4-Butyrolactone; Animals; Corpus Striatum; Dihydroxyphenylalanine; Female; Hydroxyquinolines; Male; Mice; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine | 1983 |
Autoreceptors mediate the inhibition of dopamine synthesis by bromocriptine and lisuride in rats.
Topics: 4-Butyrolactone; Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Brain Chemistry; Bromocriptine; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Ergolines; Lisuride; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Time Factors | 1983 |
Demonstration of autoreceptors on dopamine neurons in different brain regions of rats treated with gammabutyrolactone.
Topics: 3,4-Dihydroxyphenylacetic Acid; 4-Butyrolactone; Animals; Azepines; Brain; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Furans; Haloperidol; Limbic System; Male; Norepinephrine; Nucleus Accumbens; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1983 |
Evidence for dopamine autoreceptors in mesocortical dopamine neurons.
Topics: 4-Butyrolactone; Adrenergic Fibers; Animals; Apomorphine; Caudate Nucleus; Dihydroxyphenylalanine; Frontal Lobe; Haloperidol; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1984 |
Certain dopamine agonists increase dopamine synthesis in the striatum of rat brain.
Topics: 4-Butyrolactone; Animals; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Female; Haloperidol; Kinetics; Olfactory Bulb; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes | 1984 |
In vivo dopamine autoreceptor selectivity appears to be critically dependent upon the aromatic hydroxyl position in a series of N,N-disubstituted 2-aminotetralins.
Topics: 4-Butyrolactone; Animals; Apomorphine; Aromatic Amino Acid Decarboxylase Inhibitors; Dihydroxyphenylalanine; Female; Male; Mice; Motor Activity; Naphthalenes; Piribedil; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Structure-Activity Relationship; Tetrahydronaphthalenes | 1984 |
Ergot alkaloids: interaction with presynaptic dopamine receptors in the neostriatum and olfactory tubercles.
Topics: 4-Butyrolactone; Animals; Caudate Nucleus; Dihydroxyphenylalanine; Ergot Alkaloids; Haloperidol; Male; Neurons; Olfactory Bulb; Putamen; Rats; Receptors, Dopamine | 1980 |
Presynaptic dopamine receptors: insensitivity to kainic acid and the development of supersensitivity following chronic haloperidol.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Haloperidol; Kainic Acid; Male; Pyrrolidines; Rats; Receptors, Dopamine | 1980 |
Altered response to cessation of nerve impulse flow in dopamine neurons after chronic ethanol administration.
Topics: 4-Butyrolactone; Animals; Brain; Dihydroxyphenylalanine; Dopamine; Ethanol; Neurons; Rats; Receptors, Dopamine | 1980 |
Mesocortical dopamine neurons. Lack of autoreceptors modulating dopamine synthesis.
Topics: 4-Butyrolactone; Animals; Cerebral Cortex; Dihydroxyphenylalanine; Dopamine; In Vitro Techniques; Male; Methyltyrosines; Monoamine Oxidase Inhibitors; Neurons; Rats; Receptors, Dopamine | 1981 |
Tyrosine availability and dopamine synthesis in the striatum: studies with gamma-butyrolactone.
Topics: 4-Butyrolactone; Animals; Benzyl Alcohols; Carboxy-Lyases; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Furans; Hydrazines; Hydroxylation; Male; Rats; Rats, Inbred Strains; Tyrosine | 1981 |
Long-term application of haloperidol: effects on dopamine and acetylcholine receptors.
Topics: 4-Butyrolactone; Animals; Benztropine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Drug Interactions; Haloperidol; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Dopamine; Time Factors | 1981 |
Delayed inhibition of dopamine synthesis by gamma-butyrolactone and baclofen: dopamine autoreceptor supersensitivity?
Topics: 4-Butyrolactone; Animals; Apomorphine; Baclofen; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Furans; Haloperidol; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors | 1982 |
7-(4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butyloxy)-3,4-dihydro-2(1H)-quinolinone (OPC-14597), a new putative antipsychotic drug with both presynaptic dopamine autoreceptor agonistic activity and postsynaptic D2 receptor antagonistic activity.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Aripiprazole; Catalepsy; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxidopamine; Piperazines; Presynaptic Terminals; Quinolones; Radioligand Assay; Rats; Reserpine; Spiperone; Stereotyped Behavior; Synapses; Tritium | 1995 |
CI-1007, a dopamine partial agonist and potential antipsychotic agent. I. Neurochemical effects.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 4-Butyrolactone; Acetylcholine; Adenylyl Cyclases; Animals; Antipsychotic Agents; Autoreceptors; CHO Cells; Cricetinae; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Guinea Pigs; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Serotonin | 1995 |
Effects of dopamine partial-agonist aminoergolines on dopamine metabolism in limbic and extrapyramidal regions of rat brain.
Topics: 4-Butyrolactone; Animals; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Extrapyramidal Tracts; Hydrazines; Limbic System; Male; Rats; Rats, Sprague-Dawley | 1994 |
Sensitivity of dopamine D2 receptors following long-term treatment with roxindole.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agents; Down-Regulation; Drug Interactions; Haloperidol; Indoles; Injections, Intraperitoneal; Male; Oxindoles; Pyridines; Rats; Rats, Wistar; Receptors, Dopamine D2; Stereotyped Behavior | 1994 |
The behavioural and neurochemical profile of the putative dopamine D3 receptor agonist, (+)-PD 128907, in the rat.
Topics: 4-Butyrolactone; Animals; Apomorphine; Behavior, Animal; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Male; Nucleus Accumbens; Oxazines; Rats; Rats, Sprague-Dawley | 1996 |
Novel antipsychotic agents with dopamine autoreceptor agonist properties: synthesis and pharmacology of 7-[4-(4-phenyl-1-piperazinyl)butoxy]-3,4-dihydro-2(1H)-quinolinone derivatives.
Topics: 4-Butyrolactone; Animals; Antipsychotic Agents; Apomorphine; Aripiprazole; Brain; Catalepsy; Dihydroxyphenylalanine; Dopamine Agonists; Dopamine Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; Molecular Structure; Piperazines; Quinolones; Rats; Stereotyped Behavior; Structure-Activity Relationship | 1998 |
Increased site-specific phosphorylation of tyrosine hydroxylase accompanies stimulation of enzymatic activity induced by cessation of dopamine neuronal activity.
Topics: 4-Butyrolactone; Animals; Apomorphine; Binding Sites; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Enzyme Activation; GABA Modulators; Hydroxylation; In Vitro Techniques; Male; Neurons; Phosphorylation; Rats; Rats, Sprague-Dawley; Tyrosine; Tyrosine 3-Monooxygenase | 1999 |
In vivo characterization of novel full and partial 2-(4-aminophenyl)-N,N-dipropylethylamine dopamine D(2) receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 4-Butyrolactone; alpha-Methyltyrosine; Animals; Brain Chemistry; Catecholamines; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Ethylamines; Fluorobenzenes; GABA Modulators; Male; Monoamine Oxidase Inhibitors; Motor Activity; Pargyline; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine; Sympatholytics | 2000 |
Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA(B)(1)-deficient mice.
Topics: 4-Butyrolactone; Adjuvants, Anesthesia; Animals; Anticonvulsants; Autoradiography; Baclofen; Behavior, Animal; Benzocycloheptenes; Binding, Competitive; Body Weight; Brain; Cell Membrane; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; Electroencephalography; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Guanosine 5'-O-(3-Thiotriphosphate); Mice; Mice, Inbred BALB C; Mice, Knockout; Motor Activity; Organophosphorus Compounds; Phenols; Radioligand Assay; Receptors, GABA-B; Sodium Oxybate; Time Factors | 2003 |
Increased striatal dopamine synthesis is associated with decreased tissue levels of tyrosine.
Topics: 4-Butyrolactone; Amino Acids; Animals; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Antagonists; Down-Regulation; Extracellular Fluid; Haloperidol; Hydroxylation; Male; Microdialysis; Neurons; Prefrontal Cortex; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Solvents; Tyrosine; Tyrosine 3-Monooxygenase; Up-Regulation | 2006 |