Page last updated: 2024-09-03

4-bromo-a-23187 and thapsigargin

4-bromo-a-23187 has been researched along with thapsigargin in 6 studies

Compound Research Comparison

Studies
(4-bromo-a-23187)
Trials
(4-bromo-a-23187)
Recent Studies (post-2010)
(4-bromo-a-23187)
Studies
(thapsigargin)
Trials
(thapsigargin)
Recent Studies (post-2010) (thapsigargin)
63055,2343918

Protein Interaction Comparison

ProteinTaxonomy4-bromo-a-23187 (IC50)thapsigargin (IC50)
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1Oryctolagus cuniculus (rabbit)0.002

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's3 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Loh, TT; Zhu, WH1
Gillies, RJ; Gomez, A; Hendrix, MJ; Martinez, GM; Martínez-Zaguilán, R1
Chapman, SW; Cleary, JD; Kramer, RE; Rogers, PD1
Gylfe, E; Hellman, B; Tengholm, A1
Ali, Z; Kargacin, GJ; Kargacin, ME; Pollock, NS; Ward, CA1
Kiemer, AK; Vollmar, AM1

Other Studies

6 other study(ies) available for 4-bromo-a-23187 and thapsigargin

ArticleYear
Differential effects of phorbol ester on apoptosis in HL-60 promyelocytic leukemia cells.
    Biochemical pharmacology, 1996, May-03, Volume: 51, Issue:9

    Topics: Apoptosis; Calcimycin; Calcium; Down-Regulation; Enzyme Inhibitors; HL-60 Cells; Homeostasis; Humans; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1996
Distinct regulation of pHin and [Ca2+]in in human melanoma cells with different metastatic potential.
    Journal of cellular physiology, 1998, Volume: 176, Issue:1

    Topics: Ammonium Chloride; Anti-Bacterial Agents; Benzopyrans; Calcimycin; Calcium; Calcium-Transporting ATPases; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Homeostasis; Humans; Hydrogen-Ion Concentration; Indoles; Ionophores; Macrolides; Melanoma; Naphthols; Neoplasm Metastasis; Proton-Translocating ATPases; Rhodamines; Thapsigargin; Tumor Cells, Cultured

1998
Amphotericin B-induced interleukin-1beta expression in human monocytic cells is calcium and calmodulin dependent.
    The Journal of infectious diseases, 1999, Volume: 180, Issue:4

    Topics: Amphotericin B; Calcimycin; Calcium; Calmodulin; Cell Line; Enzyme Inhibitors; Gene Expression Regulation; Humans; Imidazoles; Interleukin-1; Kinetics; Monocytes; Thapsigargin

1999
Mobilization of Ca2+ stores in individual pancreatic beta-cells permeabilized or not with digitonin or alpha-toxin.
    Cell calcium, 2000, Volume: 27, Issue:1

    Topics: Adenosine Diphosphate Ribose; Adenosine Triphosphate; Animals; Bacterial Toxins; Caffeine; Calcimycin; Calcium; Calcium-Transporting ATPases; Cell Compartmentation; Cell Membrane Permeability; Cyclic ADP-Ribose; Cytoplasm; Digitonin; Enzyme Inhibitors; Hemolysin Proteins; Inositol 1,4,5-Trisphosphate; Ionophores; Islets of Langerhans; Mice; Mice, Obese; NADP; Organelles; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin

2000
Tamoxifen inhibits Ca2+ uptake by the cardiac sarcoplasmic reticulum.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 440, Issue:4

    Topics: Animals; Caffeine; Calcimycin; Calcium; Calcium Channels; Calcium-Transporting ATPases; Estrogen Antagonists; Ionophores; Male; Myocardium; Potassium Channels; Rats; Rats, Sprague-Dawley; Sarcoplasmic Reticulum; Tamoxifen; Thapsigargin

2000
Elevation of intracellular calcium levels contributes to the inhibition of nitric oxide production by atrial natriuretic peptide.
    Immunology and cell biology, 2001, Volume: 79, Issue:1

    Topics: Aniline Compounds; Animals; Atrial Natriuretic Factor; Calcimycin; Calcium; Cells, Cultured; Dibutyryl Cyclic GMP; Fluorescent Dyes; Guanylate Cyclase; Lipopolysaccharides; Macrophages; Mice; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Polysaccharides; Receptors, Atrial Natriuretic Factor; Thapsigargin; Xanthenes

2001