Page last updated: 2024-09-05

4-aminospiroperidol and domperidone

4-aminospiroperidol has been researched along with domperidone in 1 studies

*Domperidone: A specific blocker of dopamine receptors. It speeds gastrointestinal peristalsis, causes prolactin release, and is used as antiemetic and tool in the study of dopaminergic mechanisms. [MeSH]

*Domperidone: A specific blocker of dopamine receptors. It speeds gastrointestinal peristalsis, causes prolactin release, and is used as antiemetic and tool in the study of dopaminergic mechanisms. [MeSH]

Compound Research Comparison

Studies
(4-aminospiroperidol)
Trials
(4-aminospiroperidol)
Recent Studies (post-2010)
(4-aminospiroperidol)
Studies
(domperidone)
Trials
(domperidone)
Recent Studies (post-2010) (domperidone)
191181,977275468

Protein Interaction Comparison

ProteinTaxonomy4-aminospiroperidol (IC50)domperidone (IC50)
Solute carrier family 22 member 2Homo sapiens (human)7.9
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.332
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)2.614
Alpha-2A adrenergic receptorHomo sapiens (human)2.74
D(2) dopamine receptorHomo sapiens (human)0.0026
Alpha-2B adrenergic receptorHomo sapiens (human)2.125
Alpha-2C adrenergic receptorHomo sapiens (human)1.011
Sodium-dependent noradrenaline transporter Homo sapiens (human)2.614
Alpha-1D adrenergic receptorHomo sapiens (human)1.065
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.037
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.332
Sodium-dependent serotonin transporterHomo sapiens (human)3.055
Histamine H1 receptorHomo sapiens (human)1.344
Mu-type opioid receptorHomo sapiens (human)4.218
D(3) dopamine receptorHomo sapiens (human)0.018
Kappa-type opioid receptorHomo sapiens (human)6.994
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.6
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0052
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.1447
Multidrug and toxin extrusion protein 1Homo sapiens (human)2.3

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19901 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Korner, M; Luedtke, RR; Molinoff, PB; Neve, KA1

Other Studies

1 other study(ies) available for 4-aminospiroperidol and domperidone

ArticleYear
Monoclonal antibodies with high affinity for spiroperidol.
    Journal of neurochemistry, 1988, Volume: 50, Issue:4

    Topics: Animals; Antibodies, Monoclonal; Antibody Specificity; Antigens; Binding Sites, Antibody; Domperidone; Female; Haptens; Hemocyanins; Hybridomas; Immune Sera; Immunization; Mice; Mice, Inbred BALB C; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1988