4-aminopyridine and caffeine

4-aminopyridine has been researched along with caffeine in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-199016 (34.78)18.7374
1990's17 (36.96)18.2507
2000's8 (17.39)29.6817
2010's4 (8.70)24.3611
2020's1 (2.17)2.80

Authors

AuthorsStudies
Mirrlees, MS; Moulton, SJ; Murphy, CT; Taylor, PJ1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Sen, S; Sinha, N1
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN1
Gibbons, WR; Zygmunt, AC1
Deitmer, P; Lammel, E; Noack, T1
Antzelevitch, C; Di Diego, JM; Gintant, GA; Krishnan, SC; Litovsky, SH; Liu, DW; Lukas, A; Sicouri, S1
Barrett, EF; Morita, K1
Peracchia, C1
Hiraoka, M; Kawano, S2
Imaizumi, Y; Muraki, K; Watanabe, M1
Hoffman, BF; Tseng, GN1
Nishimura, M; Ohtani, H; Yagasaki, O1
Krnjevic, K; Leblond, J1
Savage, AO1
Rafuse, PE; Smith, PA; Zidichouski, JA1
Coraboeuf, E; Escande, D; Loisance, D; Planche, C1
Davis, JR; Gilmour, RF; Salata, JJ1
Delbono, O; Kotsias, BA1
Fujiwara, S; Kuriyama, H1
Anraku, M; Hashimura, S1
Carmeliet, E; Coraboeuf, E1
Herlofson, BB; Røed, A1
Feng, J; Fermini, B; Li, GR; Nattel, S; Wang, Z1
Cognard, C; Constantin, B; Raymond, G; Rivet-Bastide, M1
Chen, S; Inoue, R; Ito, Y1
Kokubun, S; Suda, N1
Gelband, CH; Hume, JR; Post, JM1
Zygmunt, AC1
Clausen, C; Goligorsky, MS; Gordienko, DV1
Harada, M; Konno, Y; Saito, K; Saito, S; Takagi, H; Yamamoto, M1
Akaike, N; Munakata, M; Uneyama, H1
Bonnet, P; Delpech, M; Vandier, C1
Garland, CJ; Mistry, DK1
Díaz, ME; Eisner, DA; Trafford, AW1
Chang, JP; Johnson, JD; Kwong, P; Wong, CJ; Yunker, WK1
Deitch, EA; Kim, SJ; Vatner, SF; Xu, DZ; Yatani, A1
Hong, Z; Kelly, RF; Lang, IM; Murar, J; Nelson, DP; Rezaie-Majd, S; Varghese, A; Weir, EK1
Hess, EJ; Raike, RS; Soria-Jasso, LE; Weisz, CJ1
Fujimoto, S; Kunimatsu, M; Mori, M; Tsushima, H1
Wang, SJ1
Boehm, S; Geier, P; Gupta, KD; Kubista, H; Lagler, M; Rubi, L; Schandl, U; Spies, D1
Pavón Arocas, O; Reichert, S; Rihel, J1
Aoki, Y; Ikeda, T; Ikeda-Murakami, K; Ishikawa, T; Tani, N1

Reviews

1 review(s) available for 4-aminopyridine and caffeine

ArticleYear
Heterogeneity within the ventricular wall. Electrophysiology and pharmacology of epicardial, endocardial, and M cells.
    Circulation research, 1991, Volume: 69, Issue:6

    Topics: 4-Aminopyridine; Action Potentials; Age Factors; Amiloride; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Coronary Disease; Dogs; Electric Conductivity; Endocardium; Flecainide; Heart Ventricles; Hot Temperature; Humans; In Vitro Techniques; Parasympathomimetics; Sodium Channels; Sympathomimetics; Ventricular Function

1991

Other Studies

45 other study(ies) available for 4-aminopyridine and caffeine

ArticleYear
Direct measurement of octanol-water partition coefficients by high-pressure liquid chromatography.
    Journal of medicinal chemistry, 1976, Volume: 19, Issue:5

    Topics: Chemistry, Physical; Chromatography, High Pressure Liquid; Kinetics; Octanols; Water

1976
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
    Chemical biology & drug design, 2016, Volume: 88, Issue:6

    Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain

2016
Properties of the calcium-activated chloride current in heart.
    The Journal of general physiology, 1992, Volume: 99, Issue:3

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Action Potentials; Animals; Cadmium; Caffeine; Calcium; Cell Membrane; Chlorides; Electric Conductivity; Heart; Ion Channels; Male; Nisoldipine; Rabbits; Ryanodine; Sodium

1992
Characterization of membrane currents in single smooth muscle cells from the guinea-pig gastric antrum.
    The Journal of physiology, 1992, Volume: 451

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Caffeine; Calcium; Guinea Pigs; In Vitro Techniques; Kinetics; Membrane Potentials; Muscle, Smooth; Nifedipine; Potassium; Pyloric Antrum; Tetraethylammonium; Tetraethylammonium Compounds

1992
Evidence for two calcium-dependent potassium conductances in lizard motor nerve terminals.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1990, Volume: 10, Issue:8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Action Potentials; Animals; Apamin; Caffeine; Calcium; Charybdotoxin; Egtazic Acid; Electric Conductivity; Lizards; Motor Neurons; Muscle Contraction; Nerve Endings; Potassium; Procaine; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds

1990
Effects of the anesthetics heptanol, halothane and isoflurane on gap junction conductance in crayfish septate axons: a calcium- and hydrogen-independent phenomenon potentiated by caffeine and theophylline, and inhibited by 4-aminopyridine.
    The Journal of membrane biology, 1991, Volume: 121, Issue:1

    Topics: 4-Aminopyridine; Alcohols; Anesthetics; Animals; Astacoidea; Axons; Caffeine; Calcium; Electric Conductivity; Halothane; Heptanol; Hydrogen-Ion Concentration; Intercellular Junctions; Isoflurane; Kinetics; Membrane Potentials; Theophylline

1991
Mechanism of increased amplitude and duration of the plateau with sudden shortening of diastolic intervals in rabbit ventricular cells.
    Circulation research, 1987, Volume: 60, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Aminopyridines; Animals; Caffeine; Electric Conductivity; Guinea Pigs; Heart Rate; Heart Ventricles; In Vitro Techniques; Ion Channels; Membrane Potentials; Myocardial Contraction; Rabbits; Time Factors; Ventricular Function

1987
Ionic currents in single smooth muscle cells from the ureter of the guinea-pig.
    The Journal of physiology, 1989, Volume: 411

    Topics: 4-Aminopyridine; Action Potentials; Animals; Cadmium; Caffeine; Calcium Channel Blockers; Egtazic Acid; Guinea Pigs; In Vitro Techniques; Ion Channels; Lithium; Muscle, Smooth; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Ureter

1989
Two components of transient outward current in canine ventricular myocytes.
    Circulation research, 1989, Volume: 64, Issue:4

    Topics: 4-Aminopyridine; Action Potentials; Aminopyridines; Animals; Caffeine; Calcium; Cells, Cultured; Dogs; Electrophysiology; Heart Conduction System; Heart Ventricles; Kinetics; Manganese; Myocardium; Ryanodine; Sarcoplasmic Reticulum; Ventricular Function

1989
The influence of ouabain on twitch contractions in the presence of veratridine.
    General pharmacology, 1989, Volume: 20, Issue:1

    Topics: 4-Aminopyridine; Aconitine; Aminopyridines; Animals; Caffeine; Electric Stimulation; Male; Mice; Mice, Inbred Strains; Monensin; Muscle Contraction; Ouabain; Potassium Chloride; Respiratory Muscles; Tetraethylammonium Compounds; Tubocurarine; Veratridine; Veratrine

1989
Hypoxic changes in hippocampal neurons.
    Journal of neurophysiology, 1989, Volume: 62, Issue:1

    Topics: 4-Aminopyridine; Adenosine Triphosphate; Aminopyridines; Animals; Apamin; Caffeine; Calcium; Egtazic Acid; Electric Stimulation; Hippocampus; Hypoxia; Membrane Potentials; Neuroglia; Neuromuscular Depolarizing Agents; Neurons; Nitrogen; Quinine; Rats; Rats, Inbred Strains; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Tolbutamide

1989
Calcium-sensitive and insensitive transient outward current in rabbit ventricular myocytes.
    The Journal of physiology, 1989, Volume: 410

    Topics: 4-Aminopyridine; Action Potentials; Animals; Caffeine; Calcium; Egtazic Acid; Heart; In Vitro Techniques; Membrane Potentials; Potassium; Rabbits; Ryanodine; Tetrodotoxin

1989
A comparison of the actions of 4-aminopyridine, caffeine and quinine on the toad isolated rectus abdominis muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1989, Volume: 92, Issue:1

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Bufonidae; Caffeine; Egtazic Acid; In Vitro Techniques; Manganese; Muscle Contraction; Muscle, Smooth; Neuromuscular Depolarizing Agents; Potassium; Procaine; Quinine; Verapamil

1989
Examination of the role of calcium in the adrenaline-induced hyperpolarization of bullfrog sympathetic neurons.
    Neuroscience, 1988, Volume: 25, Issue:2

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Apamin; Bufonidae; Caffeine; Calcium; Dantrolene; Electrophysiology; Epinephrine; Gallic Acid; Neurons; Potassium; Quinidine; Sympathetic Nervous System; Tetraethylammonium Compounds; Tubocurarine

1988
Age-related changes of action potential plateau shape in isolated human atrial fibers.
    The American journal of physiology, 1985, Volume: 249, Issue:4 Pt 2

    Topics: 4-Aminopyridine; Action Potentials; Adult; Aged; Aging; Aminopyridines; Atrial Function; Caffeine; Heart Atria; Humans; Infant; Middle Aged

1985
Effects of 4-aminopyridine on rate-related depression of cardiac action potentials.
    The American journal of physiology, 1986, Volume: 251, Issue:2 Pt 2

    Topics: 4-Aminopyridine; Action Potentials; Aminopyridines; Animals; Caffeine; Cats; Cesium; Chlorides; Dogs; Female; Heart; Heart Atria; Isoproterenol; Male; Papillary Muscles; Purkinje Fibers; Rats; Rats, Inbred Strains

1986
Relation between action potential duration and mechanical activity on rat diaphragm fibers. Effects of 3,4-diaminopyridine and tetraethylammonium.
    Pflugers Archiv : European journal of physiology, 1987, Volume: 410, Issue:4-5

    Topics: 4-Aminopyridine; Action Potentials; Amifampridine; Aminopyridines; Animals; Caffeine; In Vitro Techniques; Muscle Contraction; Potassium; Rats; Rats, Inbred Strains; Respiratory Muscles; Tetraethylammonium Compounds

1987
Effects of agents that modulate potassium permeability on smooth muscle cells of the guinea-pig basilar artery.
    British journal of pharmacology, 1983, Volume: 79, Issue:1

    Topics: 4-Aminopyridine; Acetylcholine; Aminopyridines; Animals; Basilar Artery; Caffeine; Diltiazem; Female; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth, Vascular; Permeability; Potassium; Procaine; Tetraethylammonium; Tetraethylammonium Compounds

1983
Contraction of the frog muscle in 4-aminopyridine by rapid cooling.
    The Japanese journal of physiology, 1981, Volume: 31, Issue:3

    Topics: 4-Aminopyridine; Acetylcholine; Aminopyridines; Animals; Caffeine; Cold Temperature; Dose-Response Relationship, Drug; In Vitro Techniques; Manganese; Membrane Potentials; Muscle Contraction; Neuromuscular Depolarizing Agents; Rana catesbeiana; Tetrodotoxin; Tubocurarine

1981
Existence of two transient outward currents in sheep cardiac Purkinje fibers.
    Pflugers Archiv : European journal of physiology, 1982, Volume: 392, Issue:4

    Topics: 4-Aminopyridine; Action Potentials; Aminopyridines; Animals; Caffeine; Cardiovascular Agents; Electrophysiology; Heart; Heart Conduction System; Purkinje Fibers; Sheep

1982
Inhibitory effects of HgCl2 on excitation-secretion coupling at the motor nerve terminal and excitation-contraction coupling in the muscle cell.
    Cellular and molecular neurobiology, 1994, Volume: 14, Issue:6

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Caffeine; Calcium; Dantrolene; Diaphragm; Electric Stimulation; In Vitro Techniques; Lidocaine; Magnesium; Mercuric Chloride; Methylmercury Compounds; Motor Neurons; Muscle Contraction; Muscle, Skeletal; Nerve Endings; Phrenic Nerve; Potassium Chloride; Rats; Rats, Wistar; Ruthenium Red; Tetraethylammonium; Tetraethylammonium Compounds

1994
Comparative mechanisms of 4-aminopyridine-resistant Ito in human and rabbit atrial myocytes.
    The American journal of physiology, 1995, Volume: 269, Issue:2 Pt 2

    Topics: 4-Aminopyridine; Animals; Atrial Function; Caffeine; Calcium; Chlorides; Drug Resistance; Electrophysiology; Humans; Myocardium; Patch-Clamp Techniques; Potassium Channels; Rabbits

1995
Activation of a slow outward current by the calcium released during contraction of cultured rat skeletal muscle cells.
    Pflugers Archiv : European journal of physiology, 1993, Volume: 423, Issue:3-4

    Topics: 4-Aminopyridine; Animals; Apamin; Caffeine; Calcium; Cells, Cultured; Cesium; Charybdotoxin; Egtazic Acid; Electric Conductivity; Electric Stimulation; Membrane Potentials; Muscle Contraction; Muscles; Nifedipine; Potassium; Rats; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds

1993
Pharmacological characterization of muscarinic receptor-activated cation channels in guinea-pig ileum.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Caffeine; Calcium Channels; Diphenylamine; Egtazic Acid; Electrophysiology; Female; Flufenamic Acid; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Ileum; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Muscle, Smooth; Nystatin; Procaine; Quinine; Receptors, Muscarinic; Tetraethylammonium Compounds

1993
The effect of extracellular Ca2+ concentration on the negative staircase of Ca2+ transient in field-stimulated rat ventricular cells.
    Pflugers Archiv : European journal of physiology, 1994, Volume: 429, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Animals; Caffeine; Calcium; Electric Stimulation; Extracellular Space; Fura-2; Heart Ventricles; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Rats; Sarcolemma; Sarcoplasmic Reticulum; Ventricular Function

1994
[Ca2+]i inhibition of K+ channels in canine pulmonary artery. Novel mechanism for hypoxia-induced membrane depolarization.
    Circulation research, 1995, Volume: 77, Issue:1

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Calcium Channels; Cell Hypoxia; Dogs; Electrophysiology; In Vitro Techniques; Membrane Potentials; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Potassium Channels; Pulmonary Artery

1995
Intracellular calcium activates a chloride current in canine ventricular myocytes.
    The American journal of physiology, 1994, Volume: 267, Issue:5 Pt 2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; Animals; Caffeine; Calcimycin; Calcium; Calcium Channels; Calcium Chloride; Cells, Cultured; Diacetyl; Dogs; Egtazic Acid; Electrophysiology; Female; Heart; Heart Ventricles; Isoproterenol; Kinetics; Male; Meglumine; Membrane Potentials; Time Factors

1994
Ionic currents and endothelin signaling in smooth muscle cells from rat renal resistance arteries.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: 4-Aminopyridine; Animals; Arterioles; Caffeine; Calcium; Cell Membrane; Cobalt; Egtazic Acid; Electric Conductivity; Endothelins; Fluorescent Dyes; Fura-2; In Vitro Techniques; Kidney; Male; Membrane Potentials; Muscle, Smooth, Vascular; Nifedipine; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Renal Circulation; Signal Transduction; Spectrometry, Fluorescence; Tetraethylammonium; Tetraethylammonium Compounds; Vascular Resistance

1994
Muscle relaxant action of dantrolene sodium in rats.
    Research communications in chemical pathology and pharmacology, 1993, Volume: 81, Issue:3

    Topics: 4-Aminopyridine; Animals; Caffeine; Dantrolene; Drug Interactions; Electric Stimulation; Injections, Intravenous; Male; Muscle Relaxation; Neuromuscular Junction; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Synaptic Transmission

1993
Caffeine response in pyramidal neurons freshly dissociated from rat hippocampus.
    Brain research, 1993, Feb-26, Volume: 604, Issue:1-2

    Topics: 4-Aminopyridine; Animals; Apamin; Barium; Caffeine; Calcimycin; Calcium; Electrophysiology; Hippocampus; In Vitro Techniques; Kinetics; Neurons; Nystatin; Potassium Channels; Procaine; Pyramidal Tracts; Rats; Rats, Wistar; Ryanodine; Tetraethylammonium; Tetraethylammonium Compounds

1993
Spontaneous transient outward currents and delayed rectifier K+ current: effects of hypoxia.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Cell Hypoxia; Cells, Cultured; Delayed Rectifier Potassium Channels; Female; Male; Membrane Potentials; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Pulmonary Artery; Rabbits; Ryanodine; Tetraethylammonium; Thapsigargin; Time Factors

1998
The influence of phenylephrine outward potassium currents in single smooth muscle cells from the rabbit mesenteric artery.
    General pharmacology, 1999, Volume: 33, Issue:5

    Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Amifampridine; Animals; Caffeine; Calcium; Chelating Agents; Drug Interactions; Egtazic Acid; Female; In Vitro Techniques; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Potassium; Potassium Channels; Prazosin; Rabbits; Tetraethylammonium; Vasoconstrictor Agents

1999
Coordinated control of cell Ca(2+) loading and triggered release from the sarcoplasmic reticulum underlies the rapid inotropic response to increased L-type Ca(2+) current.
    Circulation research, 2001, Feb-02, Volume: 88, Issue:2

    Topics: 4-Aminopyridine; Action Potentials; Aniline Compounds; Animals; Barium; Caffeine; Calcium; Calcium Channels, L-Type; Cells, Cultured; Electric Stimulation; Ferrets; Fluorescent Dyes; Intracellular Fluid; Myocardial Contraction; Patch-Clamp Techniques; Potassium Channel Blockers; Rats; Sarcoplasmic Reticulum; Sodium-Calcium Exchanger; Systole; Xanthenes

2001
Modulation of gonadotropin II release by K+ channel blockers in goldfish gonadotropes: a novel stimulatory action of 4-aminopyridine.
    Journal of neuroendocrinology, 2001, Volume: 13, Issue:11

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Fluorescent Dyes; Fura-2; Goldfish; Gonadotropins, Pituitary; Phosphodiesterase Inhibitors; Pituitary Gland; Potassium Channel Blockers; Tetraethylammonium; Verapamil

2001
Mesenteric lymph from rats with thermal injury prolongs the action potential and increases Ca2+ transient in rat ventricular myocytes.
    Shock (Augusta, Ga.), 2003, Volume: 20, Issue:5

    Topics: 4-Aminopyridine; Action Potentials; Animals; Burns; Caffeine; Calcium; Calcium Channels, T-Type; Egtazic Acid; Electrophysiology; Lithium; Lymph; Male; Mesentery; Myocytes, Cardiac; Patch-Clamp Techniques; Potassium; Potassium Channels; Rats; Rats, Sprague-Dawley; Sarcoplasmic Reticulum; Sodium-Calcium Exchanger

2003
Increased release of serotonin from rat ileum due to dexfenfluramine.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2004, Volume: 287, Issue:5

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Chromatography, High Pressure Liquid; Cytosol; Dexfenfluramine; Fluoxetine; Hypertension, Pulmonary; Ileum; Male; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

2004
Potassium channel blockers inhibit the triggers of attacks in the calcium channel mouse mutant tottering.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-20, Volume: 25, Issue:16

    Topics: 4-Aminopyridine; Analysis of Variance; Animals; Behavior, Animal; Caffeine; Calcium Channels, N-Type; Calcium Channels, P-Type; Calcium Channels, Q-Type; Cerebellum; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesias; Mice; Mice, Inbred C57BL; Mice, Neurologic Mutants; Microinjections; Mutation; Potassium Channel Blockers

2005
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Apamin; Barium; Benzopyrans; Caffeine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Charybdotoxin; Diclofenac; Dimethyl Sulfoxide; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanethidine; Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nitroarginine; Papaverine; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Protein Serine-Threonine Kinases; Pyrazoles; Receptor, Cannabinoid, CB1; rho-Associated Kinases; Tetraethylammonium; Vasodilator Agents

2006
Caffeine facilitation of glutamate release from rat cerebral cortex nerve terminals (synaptosomes) through activation protein kinase C pathway: an interaction with presynaptic adenosine A1 receptors.
    Synapse (New York, N.Y.), 2007, Volume: 61, Issue:6

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Calcium Signaling; Cerebral Cortex; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Presynaptic Terminals; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Synaptic Membranes; Synaptic Transmission; Synaptosomes

2007
Raised activity of L-type calcium channels renders neurons prone to form paroxysmal depolarization shifts.
    Neuromolecular medicine, 2013, Volume: 15, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Anthracenes; Caffeine; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Dimethyl Sulfoxide; Epilepsy; Excitatory Postsynaptic Potentials; Hippocampus; Hydrogen Peroxide; Isradipine; Magnesium; Neurons; Oxidative Stress; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley

2013
The Neuropeptide Galanin Is Required for Homeostatic Rebound Sleep following Increased Neuronal Activity.
    Neuron, 2019, 10-23, Volume: 104, Issue:2

    Topics: 4-Aminopyridine; Aconitine; Animals; Caffeine; Extracellular Signal-Regulated MAP Kinases; GABA Antagonists; Galanin; Homeostasis; Mutation; Neurons; Pentylenetetrazole; Phosphorylation; Potassium Channel Blockers; Preoptic Area; Purinergic P1 Receptor Antagonists; Sleep; Sleep Deprivation; Voltage-Gated Sodium Channel Agonists; Wakefulness; Zebrafish

2019
Central Nervous System Stimulants Limit Caffeine Transport at the Blood-Cerebrospinal Fluid Barrier.
    International journal of molecular sciences, 2022, Feb-07, Volume: 23, Issue:3

    Topics: 4-Aminopyridine; Autopsy; Biological Transport; Blood-Brain Barrier; Caffeine; Case-Control Studies; Cells, Cultured; Central Nervous System Stimulants; Cerebrospinal Fluid; Choroid Plexus; Endothelial Cells; Endothelium, Vascular; Humans; Models, Biological

2022