3,5-dihydroxyphenylglycine has been researched along with 6-methyl-2-(phenylethynyl)pyridine in 32 studies
Studies (3,5-dihydroxyphenylglycine) | Trials (3,5-dihydroxyphenylglycine) | Recent Studies (post-2010) (3,5-dihydroxyphenylglycine) | Studies (6-methyl-2-(phenylethynyl)pyridine) | Trials (6-methyl-2-(phenylethynyl)pyridine) | Recent Studies (post-2010) (6-methyl-2-(phenylethynyl)pyridine) |
---|---|---|---|---|---|
301 | 1 | 61 | 543 | 0 | 185 |
22 | 0 | 10 | 543 | 0 | 185 |
Protein | Taxonomy | 3,5-dihydroxyphenylglycine (IC50) | 6-methyl-2-(phenylethynyl)pyridine (IC50) |
---|---|---|---|
Luciferin 4-monooxygenase | Photinus pyralis (common eastern firefly) | 6.2333 | |
Metabotropic glutamate receptor 5 | Rattus norvegicus (Norway rat) | 0.0129 | |
Metabotropic glutamate receptor 5 | Homo sapiens (human) | 0.0199 | |
Amine oxidase [flavin-containing] A | Mus musculus (house mouse) | 8 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (3.13) | 18.2507 |
2000's | 20 (62.50) | 29.6817 |
2010's | 10 (31.25) | 24.3611 |
2020's | 1 (3.13) | 2.80 |
Authors | Studies |
---|---|
Chapman, AG; Meldrum, BS; Nanan, K; Williams, M | 1 |
Hermans, E; Maloteaux, JM; Najimi, M; Page, G; Peeters, M | 1 |
Ahmadi, H; Croucher, MJ; Harris, JR; Lawrence, V; Thomas, LS | 1 |
Conn, PJ; Mannaioni, G; Marino, MJ; Traynelis, SF; Valenti, O | 1 |
Chamberlain, M; Johnson, MP; Kelly, G | 1 |
Croucher, MJ; Gasparini, F; Jane, DE; Thomas, LS | 1 |
Bernardi, G; Bonsi, P; Calabresi, P; Centonze, D; Conquet, F; Gubellini, P; Picconi, B; Pisani, A | 1 |
Merlin, LR | 1 |
Anderson, J; Correa, L; Lorrain, DS; Varney, M | 1 |
Frondaroli, A; Grassi, S; Pettorossi, VE | 1 |
Conn, PJ; Mannaioni, G; Poisik, OV; Smith, Y; Traynelis, S | 1 |
Berrino, L; Bianchi, R; de Novellis, V; Maione, S; Marabese, I; Palazzo, E; Rodella, L; Rossi, F | 1 |
Hou, L; Klann, E | 1 |
Andree, TH; Gong, X; Liu, F; Marquis, K; Reinhart, P; Zhang, G | 1 |
Azzi, M; Kougioumoutzakis, A; Lacaille, JC; Morin, F; Topolnik, L | 1 |
Chen, Y; Conn, PJ; de Paulis, T; Goudet, C; Hemstapat, K; Nong, Y; Pin, JP | 1 |
Carroll, FI; Dewey, WL; Gabra, BH; Navarro, HA; Smith, FL | 1 |
Baker, S; Brioni, JD; Chang, R; EI-Kouhen, O; Gauvin, DM; Hernandez, G; Hollingsworth, PR; Honore, P; Lehto, SG; Moreland, RB; Stewart, AO; Zheng, G; Zhu, CZ | 1 |
Chongthammakun, S; Viwatpinyo, K | 1 |
Araque, A; Navarrete, M | 1 |
Kullmann, DM; Le Duigou, C | 1 |
Huang, JQ; Lou, YJ; Pan, X; Zhang, YY; Zhou, LM; Zhu, DY | 1 |
Dell'anno, MT; Fisone, G; Pallottino, S | 1 |
Boccella, S; De Chiaro, M; de Novellis, V; Gatta, L; Giordano, C; Guida, F; Luongo, L; Maione, S; Marabese, I; Palazzo, E; Rossi, F; Siniscalco, D; Vita, D | 1 |
Arreola, AC; Kimmey, BA; Pierce, RC; Schmidt, HD | 1 |
Hsu, KS; Huang, CC; Lee, CC; Liang, YC | 1 |
Chen, A; Hu, WW; Jiang, XL; Li, H; Potegal, M | 1 |
Seki, K; Yashiro, S | 1 |
Chen, SR; Pan, HL; Xie, JD | 1 |
Berardo, C; Cagna, M; Di Pasqua, LG; Ferrigno, A; Richelmi, P; Siciliano, V; Vairetti, M | 1 |
Costantino, G; Macchiarulo, A; Pellicciari, R | 1 |
Bräuner-Osborne, H; Egebjerg, J; Krogsgaard-Larsen, P; Madsen, U; Nielsen, EO | 1 |
1 review(s) available for 3,5-dihydroxyphenylglycine and 6-methyl-2-(phenylethynyl)pyridine
Article | Year |
---|---|
Ligands for glutamate receptors: design and therapeutic prospects.
Topics: Animals; Drug Design; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Humans; Ligands; N-Methylaspartate; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Synapses | 2000 |
31 other study(ies) available for 3,5-dihydroxyphenylglycine and 6-methyl-2-(phenylethynyl)pyridine
Article | Year |
---|---|
Anticonvulsant activity of two metabotropic glutamate group I antagonists selective for the mGlu5 receptor: 2-methyl-6-(phenylethynyl)-pyridine (MPEP), and (E)-6-methyl-2-styryl-pyridine (SIB 1893).
Topics: Animals; Anticonvulsants; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; Glycine; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred DBA; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Seizures; Sound; Time Factors | 2000 |
Modulation of the neuronal dopamine transporter activity by the metabotropic glutamate receptor mGluR5 in rat striatal synaptosomes through phosphorylation mediated processes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Carrier Proteins; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Indoles; Isoquinolines; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Phosphorylation; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Staurosporine; Sulfonamides; Synaptosomes; Tetradecanoylphorbol Acetate | 2001 |
Endogenous sulphur-containing amino acids: potent agonists at presynaptic metabotropic glutamate autoreceptors in the rat central nervous system.
Topics: Amino Acids, Sulfur; Animals; Aspartic Acid; Autoreceptors; Calcium; Central Nervous System; Cysteic Acid; Cysteine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glycine; Male; Neurotransmitter Agents; Presynaptic Terminals; Prosencephalon; Pyridines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Resorcinols; Tetrodotoxin; Tritium | 2001 |
Metabotropic glutamate receptors 1 and 5 differentially regulate CA1 pyramidal cell function.
Topics: Animals; Benzoates; Calcium; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Fluorescent Dyes; Glycine; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Patch-Clamp Techniques; Potassium Channels; Pyramidal Cells; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols; Synaptic Transmission | 2001 |
Changes in rat serum corticosterone after treatment with metabotropic glutamate receptor agonists or antagonists.
Topics: Adrenalectomy; Adrenocorticotropic Hormone; Amino Acids; Animals; Benzoates; Bridged Bicyclo Compounds; Corticosterone; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Male; Neuroprotective Agents; Paraventricular Hypothalamic Nucleus; Phenylacetates; Propionates; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Xanthenes | 2001 |
Glutamate release inhibiting properties of the novel mGlu(5) receptor antagonist 2-methyl-6-(phenylethynyl)-pyridine (MPEP): complementary in vitro and in vivo evidence.
Topics: Animals; Brain Chemistry; Electric Stimulation; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; In Vitro Techniques; Male; Microdialysis; Pyridines; Rats; Rats, Wistar; Receptors, Kainic Acid; Resorcinols | 2001 |
Metabotropic glutamate receptor 5 mediates the potentiation of N-methyl-D-aspartate responses in medium spiny striatal neurons.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Action Potentials; Animals; Anticonvulsants; Benzoates; Cyclopropanes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Mice; Mice, Knockout; Muscarine; Muscarinic Agonists; N-Methylaspartate; Neostriatum; Neurons; Phenylacetates; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols; Synaptic Transmission | 2001 |
Differential roles for mGluR1 and mGluR5 in the persistent prolongation of epileptiform bursts.
Topics: Animals; Benzoates; Convulsants; Dose-Response Relationship, Drug; Epilepsy; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Glycine; Guinea Pigs; Hippocampus; In Vitro Techniques; Membrane Potentials; Picrotoxin; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Time Factors | 2002 |
Activation of spinal group I metabotropic glutamate receptors in rats evokes local glutamate release and spontaneous nociceptive behaviors: effects of 2-methyl-6-(phenylethynyl)-pyridine pretreatment.
Topics: Animals; Behavior, Animal; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Extracellular Space; Glutamic Acid; Glycine; Male; Microdialysis; Pain; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Resorcinols; Spinal Cord; Time Factors | 2002 |
Different metabotropic glutamate receptors play opposite roles in synaptic plasticity of the rat medial vestibular nuclei.
Topics: Amino Acids; Animals; Chromones; Excitatory Amino Acid Antagonists; Glycine; Membrane Potentials; Neuronal Plasticity; Organ Culture Techniques; Phenylacetates; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Vestibular Nuclei; Xanthenes | 2002 |
Distinct functional roles of the metabotropic glutamate receptors 1 and 5 in the rat globus pallidus.
Topics: Animals; Cells, Cultured; Central Nervous System; Electric Conductivity; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Globus Pallidus; Glycine; Neurons; Parkinson Disease; Patch-Clamp Techniques; Phenotype; Protein Kinase C; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols | 2003 |
Group I metabotropic glutamate receptors modulate glutamate and gamma-aminobutyric acid release in the periaqueductal grey of rats.
Topics: Animals; Chromones; Dendrites; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Glutamates; Glycine; Male; Microdialysis; Microscopy, Electron; Periaqueductal Gray; Phenylacetates; Piperazines; Pyridines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Resorcinols; Tetrodotoxin | 2003 |
Activation of the phosphoinositide 3-kinase-Akt-mammalian target of rapamycin signaling pathway is required for metabotropic glutamate receptor-dependent long-term depression.
Topics: 3-Phosphoinositide-Dependent Protein Kinases; Androstadienes; Animals; Benzoates; Chromones; Dendrites; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Glycine; Hippocampus; Long-Term Synaptic Depression; Male; Mice; Mice, Inbred C57BL; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinases; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyramidal Cells; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Sirolimus; Synaptosomes; Tacrolimus; TOR Serine-Threonine Kinases; Wortmannin | 2004 |
The inhibition of glycogen synthase kinase 3beta by a metabotropic glutamate receptor 5 mediated pathway confers neuroprotection to Abeta peptides.
Topics: Amyloid beta-Peptides; Animals; Benzoates; Cells, Cultured; Chromones; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Hippocampus; In Vitro Techniques; Indoles; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Microtubule-Associated Proteins; Morpholines; Neurons; Oncogene Protein v-akt; Peptide Fragments; Phosphorylation; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Serine; Signal Transduction | 2005 |
mGluR1/5 subtype-specific calcium signalling and induction of long-term potentiation in rat hippocampal oriens/alveus interneurones.
Topics: Animals; Benzoates; Calcium; Calcium Signaling; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; In Vitro Techniques; Interneurons; Long-Term Potentiation; Membrane Potentials; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; src-Family Kinases; Synapses; Synaptic Transmission; TRPC Cation Channels | 2006 |
Interaction of novel positive allosteric modulators of metabotropic glutamate receptor 5 with the negative allosteric antagonist site is required for potentiation of receptor responses.
Topics: Allosteric Regulation; Allosteric Site; Animals; Benzamides; Binding, Competitive; Cell Line; Drug Synergism; Glycine; Humans; Male; Mutation; Neurons; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Substantia Nigra; Substrate Specificity; Subthalamic Nucleus | 2007 |
mGluR5 antagonists that block calcium mobilization in vitro also reverse (S)-3,5-DHPG-induced hyperalgesia and morphine antinociceptive tolerance in vivo.
Topics: Analgesics, Opioid; Animals; Calcium Signaling; Central Nervous System; Dose-Response Relationship, Drug; Drug Tolerance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Hyperalgesia; Male; Mice; Morphine; Nociceptors; Pain; Placebo Effect; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Synaptic Transmission | 2008 |
Analgesic activity of metabotropic glutamate receptor 1 antagonists on spontaneous post-operative pain in rats.
Topics: Analgesics, Non-Narcotic; Animals; Calcium; Cell Membrane; Cerebellum; Dimethylamines; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Exploratory Behavior; Fluorometry; Glycine; Heterocyclic Compounds, 3-Ring; Hindlimb; Male; Molecular Structure; Morphine; Pain, Postoperative; Pyridines; Pyrimidinones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Resorcinols; Rotarod Performance Test; Thiophenes; Tritium | 2008 |
Activation of group I metabotropic glutamate receptors leads to brain-derived neurotrophic factor expression in rat C6 cells.
Topics: Animals; Brain-Derived Neurotrophic Factor; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cell Line, Tumor; Chromones; Glycine; Protein Kinase C; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; RNA, Messenger; Signal Transduction | 2009 |
Endocannabinoids potentiate synaptic transmission through stimulation of astrocytes.
Topics: Animals; Animals, Newborn; Astrocytes; Benzoates; Biophysics; Calcium; Cannabinoid Receptor Modulators; Chelating Agents; Drug Interactions; Egtazic Acid; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; In Vitro Techniques; Mice; Mice, Inbred C57BL; Mice, Knockout; Patch-Clamp Techniques; Photolysis; Piperidines; Pyramidal Cells; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Resorcinols; Synaptic Transmission; Thapsigargin | 2010 |
Group I mGluR agonist-evoked long-term potentiation in hippocampal oriens interneurons.
Topics: Animals; Benzoates; Electric Stimulation; Electrodes, Implanted; Electrophysiological Phenomena; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Interneurons; Long-Term Potentiation; Male; Phenylacetates; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Metabotropic Glutamate; Resorcinols | 2011 |
Involvement of metabotropic glutamate receptor 5 in cardiomyocyte differentiation from mouse embryonic stem cells.
Topics: Animals; Calcium Channels, L-Type; Calcium Channels, T-Type; Calcium Signaling; Carrier Proteins; Cell Differentiation; Cell Line; Cell Survival; Coculture Techniques; Embryoid Bodies; Female; Gene Expression; Gene Knockdown Techniques; Glycine; GTP Phosphohydrolases; Homer Scaffolding Proteins; Male; Mice; Mice, Inbred ICR; Myocytes, Cardiac; Nerve Tissue Proteins; Phosphatidylinositol 3-Kinases; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; RNA Interference | 2012 |
mGlu5R promotes glutamate AMPA receptor phosphorylation via activation of PKA/DARPP-32 signaling in striatopallidal medium spiny neurons.
Topics: Animals; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Dopamine and cAMP-Regulated Phosphoprotein 32; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Phosphorylation; Purinergic P1 Receptor Antagonists; Pyridines; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Triazines; Triazoles | 2013 |
Role of metabotropic glutamate receptor 1 in the basolateral amygdala-driven prefrontal cortical deactivation in inflammatory pain in the rat.
Topics: Action Potentials; Amygdala; Animals; Bicuculline; Carrageenan; Chromones; Disease Models, Animal; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Formaldehyde; GABA Antagonists; Gene Expression; Glycine; Male; Neural Inhibition; Neural Pathways; Neuronal Plasticity; Pain; Physical Stimulation; Prefrontal Cortex; Pyramidal Cells; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols | 2013 |
Group I metabotropic glutamate receptor-mediated activation of PKC gamma in the nucleus accumbens core promotes the reinstatement of cocaine seeking.
Topics: Animals; Benzimidazoles; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Nucleus Accumbens; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles | 2015 |
Cocaine Withdrawal Impairs mGluR5-Dependent Long-Term Depression in Nucleus Accumbens Shell Neurons of Both Direct and Indirect Pathways.
Topics: Animals; Benzamides; Chromones; Cocaine; Cocaine-Related Disorders; Dopaminergic Neurons; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Genes, Reporter; Glycine; Imidazoles; Long-Term Synaptic Depression; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Tissue Proteins; Nucleus Accumbens; Pyrazoles; Pyridazines; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Dopamine D1; Receptors, Dopamine D2; Resorcinols; Substance Withdrawal Syndrome | 2015 |
Molecular mechanisms of group I metabotropic glutamate receptor mediated LTP and LTD in basolateral amygdala in vitro.
Topics: Animals; Basolateral Nuclear Complex; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Long-Term Potentiation; Long-Term Synaptic Depression; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols | 2017 |
Association of social defeat stress-induced anhedonia-like symptoms with mGluR1-dependent decrease in membrane-bound AMPA-GluR1 in the mouse ventral midbrain.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Anhedonia; Animals; Glycine; Male; Mesencephalon; Methoxyhydroxyphenylglycol; Mice; Prefrontal Cortex; Pyridines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Resorcinols; Social Dominance; Stress, Psychological | 2017 |
Presynaptic mGluR5 receptor controls glutamatergic input through protein kinase C-NMDA receptors in paclitaxel-induced neuropathic pain.
Topics: Animals; Antineoplastic Agents, Phytogenic; Behavior, Animal; Cells, Cultured; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Injections, Spinal; Male; Nerve Tissue Proteins; Neuralgia; Neurons, Afferent; Paclitaxel; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, N-Methyl-D-Aspartate; Resorcinols; Spinal Cord Dorsal Horn; Synaptosomes | 2017 |
The selective blockade of metabotropic glutamate receptor-5 attenuates fat accumulation in an in vitro model of benign steatosis.
Topics: Fatty Liver; Glycine; Hep G2 Cells; Humans; PPAR alpha; Pyridines; Receptor, Metabotropic Glutamate 5; Resorcinols; Sterol Regulatory Element Binding Protein 1; Triglycerides | 2020 |
Modeling of amino-terminal domains of group I metabotropic glutamate receptors: structural motifs affecting ligand selectivity.
Topics: Amino Acid Sequence; Binding Sites; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Ligands; Models, Molecular; Molecular Sequence Data; Protein Conformation; Receptors, Metabotropic Glutamate; Sequence Homology, Amino Acid | 1999 |