3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan and enkephalin, leucine-2-alanine

3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan has been researched along with enkephalin, leucine-2-alanine in 1 studies

Compound Research Comparison

Studies (3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan)	Trials (3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan)	Recent Studies (post-2010) (3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan)	Studies (enkephalin, leucine-2-alanine)	Trials (enkephalin, leucine-2-alanine)	Recent Studies (post-2010) (enkephalin, leucine-2-alanine)
75	0	24	1,581	23	74

Protein Interaction Comparison

Protein	Taxonomy	enkephalin, leucine-2-alanine (IC50)
Delta-type opioid receptor	Mus musculus (house mouse)	0.0915
Delta-type opioid receptor	Rattus norvegicus (Norway rat)	0.0017
Kappa-type opioid receptor	Mus musculus (house mouse)	0.009
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	0.0419
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	1.4691
Mu-type opioid receptor	Mus musculus (house mouse)	0.009

Research

Studies (1)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	1 (100.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Davis, P; Hruby, VJ; Lai, J; Ma, SW; Moye, S; Nair, P; Navratilova, E; Porreca, F; Tumati, S; Vanderah, TW; Yamamoto, T; Yamamura, HI	1

Other Studies

1 other study(ies) available for 3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan and enkephalin, leucine-2-alanine

Article	Year
Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists. Journal of medicinal chemistry, 2007, Jun-14, Volume: 50, Issue:12 Topics: Analgesics; Animals; Cell Line; Drug Design; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Vas Deferens	2007

Article

Year

Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists.

Journal of medicinal chemistry, 2007, Jun-14, Volume: 50, Issue:12

Topics: Analgesics; Animals; Cell Line; Drug Design; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship; Vas Deferens

2007