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2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one and 2,5-dihydro-2-(4-methoxyphenyl)-3h-pyrazolo(4,3-c)quinolin-3-one

2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one has been researched along with 2,5-dihydro-2-(4-methoxyphenyl)-3h-pyrazolo(4,3-c)quinolin-3-one in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19906 (85.71)18.7374
1990's1 (14.29)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Braunwalder, A; Loo, P; Wood, PL1
Bennett, DA1
Shannon, HE; Thompson, WA1
Brown, C; Jones, B; Martin, I; Oakley, N1
Brown, CL; Martin, IL1
Herling, S; Shannon, HE1
Loew, GH; Maguire, PA; Perez, JJ; Schove, LT1

Reviews

1 review(s) available for 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one and 2,5-dihydro-2-(4-methoxyphenyl)-3h-pyrazolo(4,3-c)quinolin-3-one

ArticleYear
Pharmacology of the pyrazolo-type compounds: agonist, antagonist and inverse agonist actions.
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Hypnotics and Sedatives; Muscle Relaxants, Central; Pyrazoles; Rats; Receptors, GABA-A

1987

Other Studies

6 other study(ies) available for 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one and 2,5-dihydro-2-(4-methoxyphenyl)-3h-pyrazolo(4,3-c)quinolin-3-one

ArticleYear
Benzodiazepine receptor modulation of [35S]TBPS binding to the chloride channel. Noncompetitive inhibition of classical benzodiazepines and competitive inhibition of the partial agonist, CGS 9895, by CGS 8216.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Ion Channels; Pyrazoles; Rats; Receptors, GABA-A; Sulfur Radioisotopes

1987
Pyrazoloquinoline benzodiazepine receptor ligands: effects on schedule-controlled behavior in dogs.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:2

    Topics: Animals; Conditioning, Operant; Convulsants; Diazepam; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Female; Ligands; Male; Pyrazoles; Receptors, GABA-A; Reinforcement Schedule

1985
In vivo determination of efficacy of pyrazoloquinolinones at the benzodiazepine receptor.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain; Convulsants; Diazepam; Flunitrazepam; Male; Mice; Pentylenetetrazole; Pyrazoles; Receptors, GABA-A

1984
Modification of pyrazoloquinolinone affinity by GABA predicts efficacy at the benzodiazepine receptor.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: Animals; Diazepam; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kinetics; Male; Membranes; Mice; Mice, Inbred Strains; Pentylenetetrazole; Pyrazoles; Radioligand Assay; Receptors, GABA-A; Seizures

1984
Antagonism of the discriminative effects of diazepam by pyrazoloquinolines in rats.
    European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2

    Topics: Animals; Diazepam; Discrimination Learning; Male; Pyrazoles; Rats; Rats, Inbred F344; Receptors, Cell Surface; Receptors, GABA-A

1983
Comparison of a new class of pyrrole containing benzodiazepine ligands to the pyrazoloquinolinones CGS 9896, 9895, and 8216.
    Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents, 1994, Volume: 4, Issue:5

    Topics: Animals; Cerebellum; Chemistry, Pharmaceutical; Drug Design; GABA Agonists; GABA-A Receptor Agonists; Ligands; Models, Chemical; Pyrazoles; Rats; Spinal Cord; Structure-Activity Relationship

1994