Page last updated: 2024-08-26

2-methylhistamine and dimaprit

2-methylhistamine has been researched along with dimaprit in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19907 (43.75)18.7374
1990's7 (43.75)18.2507
2000's1 (6.25)29.6817
2010's1 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Buschauer, A; Dove, S; Igel, P1
Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Beaudoin, J; Beaulieu, L; Hébert, J; Jobin, M1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Jespersen, LT; Mikkelsen, E; Sakr, AM1
Davies, MG; Greaves, MW1
Baker, AP; Chakrin, LW; Holden, DA; Smith, WJ; Sung, CP1
Philippu, A; Wiedemann, K1
Nowak, JZ; Sek, B1
Braga, PC; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villani, P1
Fukuda, K; Matsumura, F; Tanaka, S1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Akaike, N; Ishibashi, H; Munakata, M; Sakata, T; Takeshita, Y; Watanabe, T1

Reviews

1 review(s) available for 2-methylhistamine and dimaprit

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Trials

1 trial(s) available for 2-methylhistamine and dimaprit

ArticleYear
Sensory responses of human skin to synthetic histamine analogues and histamine.
    British journal of clinical pharmacology, 1980, Volume: 9, Issue:5

    Topics: Adult; Chlorpheniramine; Dimaprit; Female; Histamine; Humans; Male; Methylhistamines; Pruritus; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea

1980

Other Studies

14 other study(ies) available for 2-methylhistamine and dimaprit

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Histamine H4 receptor agonists.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Animals; Benzimidazoles; Binding Sites; Clozapine; Guanidines; Humans; Ligands; Mice; Oximes; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2010
Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins

1992
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Effects of H1 and H2 receptor agonists on nonspecific proliferative response of human peripheral blood lymphocytes.
    International archives of allergy and applied immunology, 1986, Volume: 79, Issue:3

    Topics: Cimetidine; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Humans; Immunosuppressive Agents; Lymphocyte Activation; Methylhistamines; Phytohemagglutinins; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Studies on the effect of histamine in isolated human pulmonary arteries and veins.
    Acta pharmacologica et toxicologica, 1984, Volume: 54, Issue:2

    Topics: Aged; Dimaprit; Female; Histamine; Humans; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phentolamine; Potassium; Pulmonary Artery; Pulmonary Veins; Pyrilamine; Thiourea

1984
Effect of histamine agonists and antagonists on the production of murine reaginic antibodies.
    International journal of immunopharmacology, 1981, Volume: 3, Issue:4

    Topics: Animals; Antibody Formation; Dimaprit; Histamine; Histamine Antagonists; Immunoglobulin E; Male; Methylhistamines; Metiamide; Mice; Reagins; Receptors, Histamine; Thiourea

1981
Hypothalamic superfusion with histamine agonists and antagonists modifies the pressor response to hypothalamic stimulation.
    Journal of autonomic pharmacology, 1981, Volume: 1, Issue:2

    Topics: Animals; Blood Pressure; Cats; Dimaprit; Electric Stimulation; Female; Histamine; Histamine Antagonists; Hypothalamus; Male; Methylhistamines; Metiamide; Sympathomimetics; Thiourea; Time Factors

1981
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium

1994
Evidence for an inhibitory role of central histamine on carrageenin-induced hyperalgesia.
    Neuropharmacology, 1994, Volume: 33, Issue:2

    Topics: Animals; Carrageenan; Central Nervous System; Dimaprit; Histamine; Histamine Agonists; Hyperalgesia; Male; Methylhistamines; Rats; Rats, Sprague-Dawley

1994
Histamine H2 receptor mediates keratan sulfate secretion in rabbit chondrocytes: role of cAMP.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Animals; Bucladesine; Cartilage, Articular; Cells, Cultured; Cholera Toxin; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dinoprostone; Enzyme-Linked Immunosorbent Assay; Keratan Sulfate; Kinetics; Methylhistamines; Parathyroid Hormone; Proteoglycans; Rabbits; Receptors, Histamine H2; Sulfates; Sulfur Radioisotopes

1993
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus.
    Neuroscience, 1998, Volume: 87, Issue:4

    Topics: Animals; Calcium; Calcium Channels; Calcium Channels, N-Type; Depression, Chemical; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Ion Channel Gating; Mammillary Bodies; Methylhistamines; Nerve Tissue Proteins; Neurons; Nicardipine; omega-Agatoxin IVA; omega-Conotoxin GVIA; omega-Conotoxins; Patch-Clamp Techniques; Peptides; Pertussis Toxin; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3; Spider Venoms; Tuber Cinereum; Virulence Factors, Bordetella

1998