2-methyl-5-ht has been researched along with tropisetron in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (7.89) | 18.7374 |
1990's | 26 (68.42) | 18.2507 |
2000's | 8 (21.05) | 29.6817 |
2010's | 1 (2.63) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Baker, R; Beer, M; Herbert, R; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, GI; Swain, CJ | 1 |
Bryce, D; Chalabi, PM; Furman, J; Guarino, KJ; Ives, JL; McLean, S; Nagel, AA; Rosen, T; Roth, RW; Seeger, TF | 1 |
Daffeh, J; Guarino, K; Heym, J; McLean, S; Nagel, AA; Nowakowski, J; Rizzi, J; Rosen, T; Seeger, T; Vincent, LA | 1 |
Borrelli, G; Budriesi, R; Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Catalanotti, B; Chiarini, A; Coccone, SS; Colovic, M; Fattorusso, C; Fiorini, I; Fracasso, C; Gemma, S; Hamon, M; Ioan, P; Mennini, T; Morelli, E; Nacci, V; Novellino, E; Persico, M; Ros, S | 1 |
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A | 1 |
Cheshire, SH; Gilbert, MJ; Newberry, NR | 1 |
Hille, B; Mathie, A; Yang, J | 1 |
Feniuk, W; Saxena, PR; Tadipatri, S | 1 |
Dukat, M; Glennon, RA; Young, R | 1 |
Akaike, N; Furukawa, K; Kogure, K; Onodera, H | 1 |
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB | 1 |
Coffman, WJ; Cohen, ML; Wilson, H | 1 |
Bevan, S; Robertson, B | 1 |
Ishizawa, M | 2 |
Anderson, EG; Glaum, SR; Proudfit, HK | 1 |
Anderson, EG; Todorovic, SM | 1 |
Ashby, CR; Edwards, E; Harkins, K; Wang, RY | 1 |
Costall, B; Kelly, ME; Naylor, RJ; Tan, CC; Tattersall, FD | 1 |
Blandina, P; Goldfarb, J; Green, JP | 1 |
Buchheit, KH; Buhl, T | 1 |
Budhoo, MR; Kellum, JM; Siriwardena, AK; Smith, EP | 1 |
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J | 1 |
Deschaux, P; Ferrière, F; Khan, NA; Meyniel, JP | 1 |
Kandasamy, SB | 1 |
González, AA; Puig, MM | 1 |
Katz, LC; Roerig, B | 1 |
Bragadóttir, R; Jarkman, S; Kato, M | 1 |
Fu, LW; Longhurst, JC | 1 |
Alfaro, MJ; Goicoechea, C; Martín, MI; Ormazábal, MJ; Sánchez, E | 1 |
Arcuni, JC; Kellum, JM; Stoner, MC | 1 |
Bertrand, PP; Bornstein, JC; Furness, JB; Kunze, WA | 1 |
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V | 1 |
Bauzon, D; Bymaster, FP; Cohen, ML; DeLapp, NW; Falcone, JF; Kennedy, JS; Schenck, K | 1 |
Cairns, BE; Fujiwara, N; Hu, JW; Seo, K; Someya, G | 1 |
Gerstmann, H; Giordano, J | 1 |
Day, J; Haque, SM; Kellum, JM; King, B | 1 |
Alkam, T; Amos, B; Chebolu, S; Darmani, NA | 1 |
38 other study(ies) available for 2-methyl-5-ht and tropisetron
Article | Year |
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Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).
Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Oxazoles; Rats; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction | 1992 |
Synthesis, in vitro binding profile, and central nervous system penetrability of the highly potent 5-HT3 receptor antagonist [3H]-4-(2-methoxyphenyl)-2-[4(5)-methyl-5(4)-imidazolylmethyl]thiazole.
Topics: Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry; Glioma; Imidazoles; Mice; Molecular Structure; Neuroblastoma; Serotonin Antagonists; Thiazoles; Tumor Cells, Cultured | 1990 |
Aromatic thiazole derivatives: structurally novel and selective serotonin-3 receptor antagonists.
Topics: Animals; Binding, Competitive; Heart Rate; Molecular Structure; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured | 1990 |
Specific targeting of peripheral serotonin 5-HT(3) receptors. Synthesis, biological investigation, and structure-activity relationships.
Topics: Animals; Baroreflex; Chemical Phenomena; Female; Guinea Pigs; Heart; Heart Atria; Male; Mice; Models, Molecular; Myocardium; Pyrroles; Quinoxalines; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin 5-HT3 Receptor Agonists; Structure-Activity Relationship | 2009 |
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Evidence that the 5-HT3 receptors of the rat, mouse and guinea-pig superior cervical ganglion may be different.
Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Ketanserin; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Superior Cervical Ganglion; Tropisetron; Tubocurarine | 1991 |
5-HT3 receptor channels in dissociated rat superior cervical ganglion neurons.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Ganglia, Sympathetic; Indoles; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Rabbit isolated renal artery contractions by some tryptamine derivatives, including 2-methyl-5-HT, are mediated by a 5-HT1-like receptor.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; In Vitro Techniques; Indoles; Muscle Contraction; Muscle, Smooth, Vascular; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron; Vasoconstriction | 1992 |
5-HT3 agonist 2-methylserotonin as a training drug in discrimination studies.
Topics: Animals; Discrimination, Psychological; Indoles; Male; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tropisetron | 1992 |
Expression of 5-HT3 receptors in PC12 cells treated with NGF and 8-Br-cAMP.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cations, Monovalent; Cell Membrane; Dose-Response Relationship, Drug; Indoles; Ketanserin; Kinetics; Membrane Potentials; Nerve Growth Factors; PC12 Cells; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Time Factors; Tropisetron | 1992 |
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron | 1991 |
5-Hydroxytryptamine3 receptors mediate tachycardia in conscious instrumented dogs.
Topics: Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Ergolines; Heart Rate; Hexamethonium; Hexamethonium Compounds; Imidazoles; Indoles; Male; Ondansetron; Receptors, Serotonin; Serotonin; Tropisetron | 1990 |
Properties of 5-hydroxytryptamine3 receptor-gated currents in adult rat dorsal root ganglion neurones.
Topics: Alkaloids; Animals; Calcium; Cations, Divalent; Choline; Culture Techniques; Ganglia, Spinal; Indoles; Ion Channel Gating; Membrane Potentials; Membranes; Neurons; Protein Kinase C; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Staurosporine; Tropisetron | 1991 |
Effect of 2-methyl-5-hydroxytryptamine on motility of the isolated guinea-pig colon.
Topics: Acetylcholine; Animals; Colon; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Indoles; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Receptors, Serotonin; Serotonin; Tropisetron | 1990 |
5-HT3 receptors modulate spinal nociceptive reflexes.
Topics: Animals; Indoles; Male; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Spinal Cord; Tropanes; Tropisetron | 1990 |
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron | 1990 |
Characterization of 5-hydroxytryptamine3 receptors in the medial prefrontal cortex: a microiontophoretic study.
Topics: Animals; Cerebral Cortex; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Granisetron; Indazoles; Indoles; Iontophoresis; Magnesium Chloride; Male; Metergoline; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron | 1989 |
5-Hydroxytryptamine M-receptor antagonism in the hypothalamus facilitates gastric emptying in the guinea-pig.
Topics: Animals; Gastric Emptying; Guinea Pigs; Hypothalamus; Indoles; Male; Methysergide; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Tropisetron | 1986 |
Activation of a 5-HT3 receptor releases dopamine from rat striatal slice.
Topics: Animals; Corpus Striatum; Dopamine; In Vitro Techniques; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropisetron | 1988 |
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron | 1994 |
A 5-HT3 receptor agonist induces neurally mediated chloride transport in rat distal colon.
Topics: Animals; Biological Transport; Chlorides; Colon; Electric Conductivity; Indoles; Intestinal Absorption; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium; Tetrodotoxin; Tropisetron | 1993 |
Inhibitory action of 5-hydroxytryptamine on propulsive activity of the guinea-pig isolated colon.
Topics: 5-Methoxytryptamine; Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Indomethacin; Ketanserin; Male; Muscle Contraction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron | 1996 |
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro?
Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron | 1996 |
Identification of lymphocyte 5-HT3 receptor subtype and its implication in fish T-cell proliferation.
Topics: Animals; Cell Cycle; Indoles; Lymphocyte Activation; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Phytohemagglutinins; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Sodium; Time Factors; Tritium; Tropanes; Tropisetron | 1997 |
Effect of ondansetron and ICS 205-930 on radiation-induced hypothermia in rats.
Topics: Animals; Body Temperature; Dose-Response Relationship, Drug; Indoles; Male; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Tropisetron | 1997 |
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron | 1997 |
Modulation of intrinsic circuits by serotonin 5-HT3 receptors in developing ferret visual cortex.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Ferrets; gamma-Aminobutyric Acid; Indoles; Ligands; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Pyridinium Compounds; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Tropisetron; Virulence Factors, Bordetella; Visual Cortex | 1997 |
Serotonin elevates the c-wave of the electroretinogram of the rabbit eye by increasing the transepithelial potential.
Topics: 5-Methoxytryptamine; Animals; Dose-Response Relationship, Drug; Electroretinography; Ergolines; Indoles; Membrane Potentials; Pigment Epithelium of Eye; Rabbits; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1997 |
Role of 5-HT3 receptors in activation of abdominal sympathetic C fibre afferents during ischaemia in cats.
Topics: Adrenergic Fibers; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cats; Electrophysiology; Female; Ganglia, Sympathetic; Indoles; Indomethacin; Ischemia; Male; Neurons, Afferent; Pain; Prostaglandins; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Splanchnic Circulation; Tropisetron; Viscera | 1998 |
Study of mechanisms of calcitonin analgesia in mice. Involvement of 5-HT3 receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Brain Chemistry; Calcitonin; Dose-Response Relationship, Drug; Indoles; Indophenol; Ketanserin; Male; Mice; Mice, Inbred Strains; Nociceptors; Pain; Pain Measurement; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1999 |
Vasoactive intestinal peptide is a neuropeptide mediator of the secretory response to serotonin in rat.
Topics: Animals; Chlorides; Drug Combinations; Indoles; Male; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Vasoactive Intestinal Peptide | 2000 |
The terminals of myenteric intrinsic primary afferent neurons of the guinea-pig ileum are excited by 5-hydroxytryptamine acting at 5-hydroxytryptamine-3 receptors.
Topics: 5-Methoxytryptamine; Action Potentials; Animals; Dioxanes; Granisetron; Guinea Pigs; Ileum; Indoles; Myenteric Plexus; Neurons, Afferent; Piperidines; Presynaptic Terminals; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Signal Transduction; Tropisetron | 2000 |
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron | 2001 |
Potent antagonism of 5-HT(3) and 5-HT(6) receptors by olanzapine.
Topics: Animals; Benzodiazepines; Binding, Competitive; Clozapine; Dibenzothiazepines; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Haloperidol; HeLa Cells; Humans; Ileum; In Vitro Techniques; Indoles; Lysergic Acid; Muscle Contraction; Olanzapine; Ondansetron; Pirenzepine; Quetiapine Fumarate; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Risperidone; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfur Radioisotopes; Tritium; Tropisetron | 2001 |
Intrathecal administration of 5-HT(3) receptor agonist modulates jaw muscle activity evoked by injection of mustard oil into the temporomandibular joint in the rat.
Topics: Afferent Pathways; Animals; Dose-Response Relationship, Drug; Drug Interactions; Efferent Pathways; Electromyography; Indoles; Male; Masticatory Muscles; Muscle Contraction; Mustard Plant; Neurons, Afferent; Nociceptors; Plant Extracts; Plant Oils; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Temporomandibular Joint; Trigeminal Caudal Nucleus; Tropisetron | 2002 |
Patterns of serotonin- and 2-methylserotonin-induced pain may reflect 5-HT3 receptor sensitization.
Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Indoles; Male; Mice; Pain; Pain Measurement; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Tropisetron | 2004 |
A nonneuronal 5-hydroxytryptamine receptor 3 induces chloride secretion in the rat distal colonic mucosa.
Topics: Analysis of Variance; Animals; Chlorides; Colon; In Vitro Techniques; Indoles; Intestinal Mucosa; Ion Transport; Male; Membrane Potentials; Ondansetron; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Tetrodotoxin; Tropisetron | 2005 |
Synergistic antiemetic interactions between serotonergic 5-HT3 and tachykininergic NK1-receptor antagonists in the least shrew (Cryptotis parva).
Topics: Analysis of Variance; Animals; Antiemetics; Dose-Response Relationship, Drug; Drug Synergism; Female; Indoles; Male; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Shrews; Substance P; Tropisetron; Vomiting | 2011 |