2-methyl-5-ht and ondansetron

2-methyl-5-ht has been researched along with ondansetron in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-19902 (5.71)18.7374
1990's26 (74.29)18.2507
2000's7 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, R; Beer, M; Herbert, R; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, GI; Swain, CJ1
Baker, R; Beer, M; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, G; Swain, CJ; Watling, K1
Bryce, D; Chalabi, PM; Furman, J; Guarino, KJ; Ives, JL; McLean, S; Nagel, AA; Rosen, T; Roth, RW; Seeger, TF1
Daffeh, J; Guarino, K; Heym, J; McLean, S; Nagel, AA; Nowakowski, J; Rizzi, J; Rosen, T; Seeger, T; Vincent, LA1
Calderó, JM; del Río, J; García, E; Lasheras, B; Monge, A; Palop, JA; Peña, MC; Roca, J; Romero, G1
Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Cervo, L; Dalla Valle, F; Fracasso, C; Gemma, S; Goegan, M; Greco, G; Hamon, M; Mennini, T; Morelli, E; Nacci, V; Novellino, E1
Alton, EW; Geddes, DM; Graham, A1
Coleman, J; Lattimer, N; Rhodes, KF1
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
Abe, M; Ikeda, T; Saito, H; Togashi, H; Yoshioka, M1
Coffman, WJ; Cohen, ML; Wilson, H1
Fox, A; Morton, IK1
Barnes, JM; Barnes, NM; Costall, B; Naylor, RJ; Tyers, MB1
Butler, A; Hill, JM; Ireland, SJ; Jordan, CC; Tyers, MB1
Blier, P; Bouchard, C; Monroe, PJ; Smith, DJ; Smith, DL1
Clark, R; Eglen, RM; Hegde, SS; Johnson, LG; Lee, CH; Smith, WL; Whiting, RL1
Fone, KC; Scott, MA1
Desai, KM; Vane, JR; Warner, TD1
Blier, P; De Montigny, C; Mongeau, R1
Levy, AD; Li, Q; Rittenhouse, PA; Van de Kar, LD1
Gillies, DM; Jackson, DM; Mylecharane, EJ1
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J1
Bourin, M; Redrobe, JP1
Kandasamy, SB1
Alcalde, AI; Rodríguez-Yoldi, MC; Rodríguez-Yoldi, MJ; Salvador, MT1
González, AA; Puig, MM1
Bagdy, E; Harsing, LG; Solyom, S1
Blower, PR; Endo, T; Hamaue, N; Hirafuji, M; Kitamura, N; Minami, M; Nemoto, M; Ogawa, T; Teramoto, Y; Yasuda, E1
Furuichi, K; Miyake, A; Mochizuki, S; Saito, M; Watanabe, T1
Chen, X; Martin, SM; Pittman, QJ; Poulin, P; Takahashi, Y; Wilson, BC1
Bauzon, D; Bymaster, FP; Cohen, ML; DeLapp, NW; Falcone, JF; Kennedy, JS; Schenck, K1
Davies, PA; Hales, TG; Kirkness, EF; Safa, P; Stewart, A1
Chuaychoo, B; Kollarik, M; Lee, MG; Undem, BJ1
Day, J; Haque, SM; Kellum, JM; King, B1
Fukushima, T; Hori, Y; Ohtsubo, T; Tsuda, M; Yanagawa, Y1

Other Studies

35 other study(ies) available for 2-methyl-5-ht and ondansetron

ArticleYear
Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).
    Journal of medicinal chemistry, 1992, Mar-20, Volume: 35, Issue:6

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Oxazoles; Rats; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction

1992
Novel 5-HT3 antagonists. Indole oxadiazoles.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Electrochemistry; Indicators and Reagents; Indoles; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tropisetron

1991
Synthesis, in vitro binding profile, and central nervous system penetrability of the highly potent 5-HT3 receptor antagonist [3H]-4-(2-methoxyphenyl)-2-[4(5)-methyl-5(4)-imidazolylmethyl]thiazole.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:11

    Topics: Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry; Glioma; Imidazoles; Mice; Molecular Structure; Neuroblastoma; Serotonin Antagonists; Thiazoles; Tumor Cells, Cultured

1990
Aromatic thiazole derivatives: structurally novel and selective serotonin-3 receptor antagonists.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Binding, Competitive; Heart Rate; Molecular Structure; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured

1990
Synthesis of 2-piperazinylbenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT3 antagonist and 5-HT4 agonist properties.
    Journal of medicinal chemistry, 1994, Apr-29, Volume: 37, Issue:9

    Topics: Animals; Benzothiazoles; Binding, Competitive; Cerebral Cortex; Female; Gastric Emptying; Granisetron; Guinea Pigs; Ileum; Male; Molecular Structure; Mucous Membrane; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

1994
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Blood-Brain Barrier; Brain; Guanidine; Guinea Pigs; Hybrid Cells; In Vitro Techniques; Ligands; Male; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

1999
Effects of 5-hydroxytryptamine and 5-hydroxytryptamine receptor agonists on ion transport across mammalian airway epithelia.
    Clinical science (London, England : 1979), 1992, Volume: 83, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amiloride; Animals; Bronchi; Buspirone; Dose-Response Relationship, Drug; Epithelium; Humans; In Vitro Techniques; Ondansetron; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Sheep; Sodium Channels; Trachea

1992
A component of 5-HT-evoked depolarization of the rat isolated vagus nerve is mediated by a putative 5-HT4 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:5

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Male; Neuromuscular Depolarizing Agents; Ondansetron; Potentiometry; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vagus Nerve

1992
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
Effect of 5-hydroxytryptamine on external carotid nerve activity and its blockade by GR38032F in anesthetized rats.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 74, Issue:1

    Topics: Analysis of Variance; Animals; Dose-Response Relationship, Drug; Imidazoles; Male; Ondansetron; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Sympathetic Nervous System

1991
5-Hydroxytryptamine3 receptors mediate tachycardia in conscious instrumented dogs.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:2

    Topics: Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Ergolines; Heart Rate; Hexamethonium; Hexamethonium Compounds; Imidazoles; Indoles; Male; Ondansetron; Receptors, Serotonin; Serotonin; Tropisetron

1990
An examination of the 5-HT3 receptor mediating contraction and evoked [3H]-acetylcholine release in the guinea-pig ileum.
    British journal of pharmacology, 1990, Volume: 101, Issue:3

    Topics: Acetylcholine; Animals; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Ondansetron; Receptors, Serotonin; Serotonin

1990
5-HT3 receptors mediate inhibition of acetylcholine release in cortical tissue.
    Nature, 1989, Apr-27, Volume: 338, Issue:6218

    Topics: Acetylcholine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Female; Imidazoles; Metoclopramide; Ondansetron; Potassium; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1989
Pharmacological properties of GR38032F, a novel antagonist at 5-HT3 receptors.
    British journal of pharmacology, 1988, Volume: 94, Issue:2

    Topics: Animals; Ganglia, Spinal; Guinea Pigs; Heart; Heart Rate; Imidazoles; In Vitro Techniques; Male; Muscle, Smooth; Ondansetron; Rabbits; Rats; Receptors, Serotonin; Serotonin; Vagus Nerve

1988
5-HT3 receptors which modulate [3H]5-HT release in the guinea pig hypothalamus are not autoreceptors.
    Synapse (New York, N.Y.), 1993, Volume: 15, Issue:2

    Topics: Animals; Autoreceptors; Guinea Pigs; Hydroxyindoleacetic Acid; Hypothalamus; In Vitro Techniques; Male; Ondansetron; Potassium; Presynaptic Terminals; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptosomes; Tetrodotoxin

1993
Pharmacological characterization of RS 25259-197, a novel and selective 5-HT3 receptor antagonist, in vivo.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Oral; Animals; Bradycardia; Dogs; Dose-Response Relationship, Drug; Duodenum; Female; Ferrets; Granisetron; Hemodynamics; Injections, Intravenous; Injections, Subcutaneous; Isoquinolines; Male; Ondansetron; Palonosetron; Quinuclidines; Random Allocation; Rats; Serotonin; Serotonin Antagonists; Stereoisomerism; Vomiting

1995
Modulation of calcitonin gene-related peptide release from dorsal thoraco-lumbar spinal cord slices by 5-HT3 receptors.
    Neuroscience letters, 1994, Jul-04, Volume: 175, Issue:1-2

    Topics: Calcitonin Gene-Related Peptide; Calcium; Capsaicin; In Vitro Techniques; Ondansetron; Potassium; Radioimmunoassay; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord

1994
5-HT3 receptors do not mediate vagally-induced relaxation or contraction of the isolated stomach of the guinea-pig.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Animals; Dimethylphenylpiperazinium Iodide; Electric Stimulation; In Vitro Techniques; Male; Metoclopramide; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitroglycerin; Ondansetron; Receptors, Serotonin; Serotonin; Stomach; Vagus Nerve

1994
Activation of 5-HT3 receptors enhances the electrically evoked release of [3H]noradrenaline in rat brain limbic structures.
    European journal of pharmacology, 1994, May-02, Volume: 256, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Animals; Drug Interactions; Evoked Potentials; Limbic System; Male; Norepinephrine; Ondansetron; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1994
Investigation of the role of 5-HT3 receptors in the secretion of prolactin, ACTH and renin.
    Neuroendocrinology, 1993, Volume: 58, Issue:1

    Topics: Adrenocorticotropic Hormone; Animals; Cerebral Ventricles; Infusions, Parenteral; Male; Ondansetron; p-Chloroamphetamine; Prolactin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Renin; Serotonin

1993
Effects of 5-HT3 receptor-selective agents on locomotor activity in rats following injection into the nucleus accumbens and the ventral tegmental area.
    European journal of pharmacology, 1996, May-06, Volume: 303, Issue:1-2

    Topics: Animals; Central Nervous System Stimulants; Dextroamphetamine; Dose-Response Relationship, Drug; Injections, Intraventricular; Male; Motor Activity; Nucleus Accumbens; Ondansetron; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Agents; Ventral Tegmental Area

1996
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro?
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:7

    Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron

1996
Partial role of 5-HT2 and 5-HT3 receptors in the activity of antidepressants in the mouse forced swimming test.
    European journal of pharmacology, 1997, May-01, Volume: 325, Issue:2-3

    Topics: Amphetamines; Animals; Antidepressive Agents; Behavior, Animal; Citalopram; Desipramine; Drug Interactions; Fluoxetine; Fluvoxamine; Imipramine; Ketanserin; Male; Maprotiline; Mice; Ondansetron; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

1997
Effect of ondansetron and ICS 205-930 on radiation-induced hypothermia in rats.
    Radiation research, 1997, Volume: 147, Issue:6

    Topics: Animals; Body Temperature; Dose-Response Relationship, Drug; Indoles; Male; Ondansetron; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Tropisetron

1997
5-HT receptor subtypes involved in the serotonin-induced inhibition of L-leucine absorption in rabbit jejunum.
    Life sciences, 1997, Volume: 61, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Indoles; Intestinal Absorption; Jejunum; Leucine; Male; Ondansetron; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

1997
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron

1997
Feedback stimulation of somatodendritic serotonin release: a 5-HT3 receptor-mediated effect in the raphe nuclei of the rat.
    Brain research bulletin, 1998, Volume: 45, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Animals; Bridged Bicyclo Compounds, Heterocyclic; Dendrites; Electric Stimulation; Feedback; Fluoxetine; In Vitro Techniques; Male; Neural Pathways; Ondansetron; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reserpine; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

1998
Effects of various 5-HT3 receptor antagonists, granisetron, ondansetron, ramosetron and azasetron on serotonin (5-HT) release from the ferret isolated ileum.
    Research communications in molecular pathology and pharmacology, 1999, Volume: 104, Issue:2

    Topics: Animals; Benzimidazoles; Dose-Response Relationship, Drug; Drug Interactions; Ferrets; Granisetron; Ileum; Male; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1999
Cloning, expression, and characterization of ferret 5-HT(3) receptor subunit.
    European journal of pharmacology, 2000, Jul-07, Volume: 399, Issue:2-3

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Biguanides; Binding, Competitive; Cell Line; Cloning, Molecular; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Ferrets; Gene Expression; Humans; Imidazoles; Indoles; Kruppel-Like Factor 6; Kruppel-Like Transcription Factors; Membrane Potentials; Molecular Sequence Data; Ondansetron; Piperazines; Proto-Oncogene Proteins; Radioligand Assay; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution; Trans-Activators; Tritium; Tubocurarine

2000
Vagal CCK and 5-HT(3) receptors are unlikely to mediate LPS or IL-1beta-induced fever.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 279, Issue:3

    Topics: Animals; Body Temperature; Devazepide; Fever; Hormone Antagonists; Interleukin-1; Lipopolysaccharides; Male; Ondansetron; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sincalide; Vagus Nerve

2000
Potent antagonism of 5-HT(3) and 5-HT(6) receptors by olanzapine.
    European journal of pharmacology, 2001, Nov-02, Volume: 430, Issue:2-3

    Topics: Animals; Benzodiazepines; Binding, Competitive; Clozapine; Dibenzothiazepines; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Haloperidol; HeLa Cells; Humans; Ileum; In Vitro Techniques; Indoles; Lysergic Acid; Muscle Contraction; Olanzapine; Ondansetron; Pirenzepine; Quetiapine Fumarate; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Risperidone; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfur Radioisotopes; Tritium; Tropisetron

2001
Introduction of the 5-HT3B subunit alters the functional properties of 5-HT3 receptors native to neuroblastoma cells.
    Neuropharmacology, 2003, Volume: 44, Issue:2

    Topics: Animals; Biguanides; Calcium; Cell Differentiation; Cell Line; Dose-Response Relationship, Drug; Drug Interactions; Fluorescence; Gene Expression; Green Fluorescent Proteins; Luminescent Proteins; Mice; Molecular Sequence Data; Neuroblastoma; Ondansetron; Patch-Clamp Techniques; Protein Subunits; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

2003
Effect of 5-hydroxytryptamine on vagal C-fiber subtypes in guinea pig lungs.
    Pulmonary pharmacology & therapeutics, 2005, Volume: 18, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Lung; Male; Membrane Potentials; Nerve Fibers, Unmyelinated; Nodose Ganglion; Ondansetron; Patch-Clamp Techniques; Serotonin; Serotonin Agents; Serotonin Antagonists; Vagus Nerve

2005
A nonneuronal 5-hydroxytryptamine receptor 3 induces chloride secretion in the rat distal colonic mucosa.
    American journal of surgery, 2005, Volume: 190, Issue:5

    Topics: Analysis of Variance; Animals; Chlorides; Colon; In Vitro Techniques; Indoles; Intestinal Mucosa; Ion Transport; Male; Membrane Potentials; Ondansetron; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Tetrodotoxin; Tropisetron

2005
Facilitatory actions of serotonin type 3 receptors on GABAergic inhibitory synaptic transmission in the spinal superficial dorsal horn.
    Journal of neurophysiology, 2009, Volume: 102, Issue:3

    Topics: Analysis of Variance; Animals; Biguanides; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Transgenic; Models, Biological; Neural Inhibition; Ondansetron; Patch-Clamp Techniques; Posterior Horn Cells; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

2009