2-methyl-5-ht and ketanserin

2-methyl-5-ht has been researched along with ketanserin in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.70)18.7374
1990's23 (85.19)18.2507
2000's3 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Calderó, JM; del Río, J; García, E; Lasheras, B; Monge, A; Palop, JA; Peña, MC; Roca, J; Romero, G1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R1
Glennon, RA1
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A1
Cheshire, SH; Gilbert, MJ; Newberry, NR1
Kagami, Y; Shigenobu, S; Watanabe, S1
Akaike, N; Furukawa, K; Kogure, K; Onodera, H1
Giordano, J1
Bunce, KT; Burridge, J; Butler, A; Elswood, CJ; Ireland, SJ; Kilpatrick, GJ; Tyers, MB1
Salonen, RO; Webber, SE; Widdicombe, JG1
Anderson, EG; Todorovic, SM1
Bunce, KT; Higgins, GA; Jones, BJ; Kilpatrick, GJ; Tyers, MB1
Balestra, B; Candura, SM; Lucchelli, A; Messori, E; Rizzi, CA; Tonini, M1
Davis, EA; Haynes, JM; Hodgson, WC; James, GM1
Ishizawa, M1
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J1
Horisaka, K; Sugimoto, Y; Yamada, J; Yoshikawa, T1
Horisaka, K; Noma, T; Sugimoto, Y; Yamada, J; Yoshikawa, T1
Bourin, M; Redrobe, JP1
Deschaux, P; Ferriere, F; Khan, NA; Meyniel, JP1
Briejer, MR; Mathis, C; Schuurkes, JA1
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M1
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D1
Alfaro, MJ; Goicoechea, C; Martín, MI; Ormazábal, MJ; Sánchez, E1
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V1
Ge, L; Naylor, RJ; Tuladhar, BR1

Reviews

1 review(s) available for 2-methyl-5-ht and ketanserin

ArticleYear
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

26 other study(ies) available for 2-methyl-5-ht and ketanserin

ArticleYear
Synthesis of 2-piperazinylbenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT3 antagonist and 5-HT4 agonist properties.
    Journal of medicinal chemistry, 1994, Apr-29, Volume: 37, Issue:9

    Topics: Animals; Benzothiazoles; Binding, Competitive; Cerebral Cortex; Female; Gastric Emptying; Granisetron; Guinea Pigs; Ileum; Male; Molecular Structure; Mucous Membrane; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

1994
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
    Molecular pharmacology, 1996, Volume: 50, Issue:6

    Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents

1996
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:2

    Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1992
Evidence that the 5-HT3 receptors of the rat, mouse and guinea-pig superior cervical ganglion may be different.
    British journal of pharmacology, 1991, Volume: 102, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Ketanserin; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Superior Cervical Ganglion; Tropisetron; Tubocurarine

1991
Neuroprotective effect of 5-HT3 receptor antagonist on ischemia-induced decrease in CA1 field potential in rat hippocampal slices.
    European journal of pharmacology, 1992, Nov-24, Volume: 224, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Animals; Brain Ischemia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Hippocampus; Hypoglycemia; Hypoxia; In Vitro Techniques; Ketanserin; Membrane Potentials; Oxazines; Rats; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1992
Expression of 5-HT3 receptors in PC12 cells treated with NGF and 8-Br-cAMP.
    Journal of neurophysiology, 1992, Volume: 67, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cations, Monovalent; Cell Membrane; Dose-Response Relationship, Drug; Indoles; Ketanserin; Kinetics; Membrane Potentials; Nerve Growth Factors; PC12 Cells; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Time Factors; Tropisetron

1992
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes

1991
The pharmacological characterization of 5-HT3 receptors in three isolated preparations derived from guinea-pig tissues.
    British journal of pharmacology, 1990, Volume: 101, Issue:3

    Topics: Animals; Colon; Female; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Receptors, Serotonin; Serotonin; Vagus Nerve

1990
Receptors mediating the effects of 5-hydroxytryptamine on the tracheal vasculature and smooth muscle of sheep.
    British journal of pharmacology, 1990, Volume: 99, Issue:1

    Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle Tonus; Muscle, Smooth; Perfusion; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep; Trachea

1990
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron

1990
5-HT3 receptor antagonists injected into the area postrema inhibit cisplatin-induced emesis in the ferret.
    British journal of pharmacology, 1989, Volume: 97, Issue:1

    Topics: Animals; Apomorphine; Autoradiography; Brain Chemistry; Carnivora; Cisplatin; Female; Ferrets; Injections, Intraventricular; Ketanserin; Male; Methiothepin; Serotonin; Serotonin Antagonists; Vomiting

1989
5-Hydroxytryptamine receptors that facilitate excitatory neuromuscular transmission in the guinea-pig isolated detrusor muscle.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Acetylcholine; Adenosine Triphosphate; Amphetamines; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Urinary Bladder

1995
Attenuated 5-hydroxytryptamine receptor-mediated responses in aortae from streptozotocin-induced diabetic rats.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Animals; Aorta; Arginine; Blood Glucose; Diabetes Mellitus, Experimental; Endothelium, Vascular; Insulin; Ketanserin; Male; Nitroarginine; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Vasoconstriction

1994
Inhibitory action of 5-hydroxytryptamine on propulsive activity of the guinea-pig isolated colon.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1996, Volume: 114, Issue:1

    Topics: 5-Methoxytryptamine; Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Indomethacin; Ketanserin; Male; Muscle Contraction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron

1996
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro?
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:7

    Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron

1996
The effects of peripheral serotonin2 (5-HT2) and serotonin3 (5-HT3) receptor agonists on blood glucose levels in rats.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:10

    Topics: Animals; Blood Glucose; Glucagon; Insulin; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists

1996
Effects of peripheral 5-HT2 and 5-HT3 receptor agonists on food intake in food-deprived and 2-deoxy-D-glucose-treated rats.
    European journal of pharmacology, 1996, Nov-28, Volume: 316, Issue:1

    Topics: Adrenal Medulla; Adrenalectomy; Animals; Deoxyglucose; Eating; Epinephrine; Food Deprivation; Hyperphagia; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Partial role of 5-HT2 and 5-HT3 receptors in the activity of antidepressants in the mouse forced swimming test.
    European journal of pharmacology, 1997, May-01, Volume: 325, Issue:2-3

    Topics: Amphetamines; Animals; Antidepressive Agents; Behavior, Animal; Citalopram; Desipramine; Drug Interactions; Fluoxetine; Fluvoxamine; Imipramine; Ketanserin; Male; Maprotiline; Mice; Ondansetron; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

1997
5-Hydroxytryptamine-induced calcium-channel gating in rainbow trout (Oncorhynchus mykiss) peripheral blood lymphocytes.
    The Biochemical journal, 1997, Apr-01, Volume: 323 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium Channels; Dopamine Antagonists; Ion Channel Gating; Ionomycin; Ionophores; Ketanserin; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulpiride

1997
5-HT receptor types in the rat ileum longitudinal muscle: focus on 5-HT2 receptors mediating contraction.
    Neurogastroenterology and motility, 1997, Volume: 9, Issue:4

    Topics: 5-Methoxytryptamine; Animals; Female; Gastrointestinal Motility; Ileum; In Vitro Techniques; Ketanserin; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1997
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
    Gynecologic and obstetric investigation, 1999, Volume: 47, Issue:2

    Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries

1999
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction

1999
Study of mechanisms of calcitonin analgesia in mice. Involvement of 5-HT3 receptors.
    Brain research, 1999, Oct-23, Volume: 845, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Brain Chemistry; Calcitonin; Dose-Response Relationship, Drug; Indoles; Indophenol; Ketanserin; Male; Mice; Mice, Inbred Strains; Nociceptors; Pain; Pain Measurement; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1999
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
    American journal of physiology. Lung cellular and molecular physiology, 2001, Volume: 281, Issue:4

    Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron

2001
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003