2-methyl-5-ht has been researched along with ketanserin in 27 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (3.70) | 18.7374 |
1990's | 23 (85.19) | 18.2507 |
2000's | 3 (11.11) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Calderó, JM; del Río, J; García, E; Lasheras, B; Monge, A; Palop, JA; Peña, MC; Roca, J; Romero, G | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Gommeren, W; Haegeman, G; Heylen, L; Lesage, AS; Leysen, JE; Luyten, WH; Schotte, A; Van de Weyer, I; Van Gompel, P; Vanhoenacker, P; Wouters, R | 1 |
Glennon, RA | 1 |
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A | 1 |
Cheshire, SH; Gilbert, MJ; Newberry, NR | 1 |
Kagami, Y; Shigenobu, S; Watanabe, S | 1 |
Akaike, N; Furukawa, K; Kogure, K; Onodera, H | 1 |
Giordano, J | 1 |
Bunce, KT; Burridge, J; Butler, A; Elswood, CJ; Ireland, SJ; Kilpatrick, GJ; Tyers, MB | 1 |
Salonen, RO; Webber, SE; Widdicombe, JG | 1 |
Anderson, EG; Todorovic, SM | 1 |
Bunce, KT; Higgins, GA; Jones, BJ; Kilpatrick, GJ; Tyers, MB | 1 |
Balestra, B; Candura, SM; Lucchelli, A; Messori, E; Rizzi, CA; Tonini, M | 1 |
Davis, EA; Haynes, JM; Hodgson, WC; James, GM | 1 |
Ishizawa, M | 1 |
Masek, K; Ruzicka, V; Sevcík, J; Slánsky, J | 1 |
Horisaka, K; Sugimoto, Y; Yamada, J; Yoshikawa, T | 1 |
Horisaka, K; Noma, T; Sugimoto, Y; Yamada, J; Yoshikawa, T | 1 |
Bourin, M; Redrobe, JP | 1 |
Deschaux, P; Ferriere, F; Khan, NA; Meyniel, JP | 1 |
Briejer, MR; Mathis, C; Schuurkes, JA | 1 |
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M | 1 |
Bard, JA; Branchek, T; Edvinsson, L; Longmore, J; Nilsson, T; Pantev, E; Shaw, D | 1 |
Alfaro, MJ; Goicoechea, C; Martín, MI; Ormazábal, MJ; Sánchez, E | 1 |
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V | 1 |
Ge, L; Naylor, RJ; Tuladhar, BR | 1 |
1 review(s) available for 2-methyl-5-ht and ketanserin
Article | Year |
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Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists | 2003 |
26 other study(ies) available for 2-methyl-5-ht and ketanserin
Article | Year |
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Synthesis of 2-piperazinylbenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT3 antagonist and 5-HT4 agonist properties.
Topics: Animals; Benzothiazoles; Binding, Competitive; Cerebral Cortex; Female; Gastric Emptying; Granisetron; Guinea Pigs; Ileum; Male; Molecular Structure; Mucous Membrane; Ondansetron; Piperazines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles | 1994 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Alniditan, a new 5-hydroxytryptamine1D agonist and migraine-abortive agent: ligand-binding properties of human 5-hydroxytryptamine1D alpha, human 5-hydroxytryptamine1D beta, and calf 5-hydroxytryptamine1D receptors investigated with [3H]5-hydroxytryptamin
Topics: Animals; Benzopyrans; Cattle; Cloning, Molecular; Glioma; HeLa Cells; Humans; Mice; Migraine Disorders; Propylamines; Protein Binding; Pyrimidines; Radioligand Assay; Receptors, Serotonin; Serotonin Receptor Agonists; Signal Transduction; Tritium; Tumor Cells, Cultured; Vasoconstrictor Agents | 1996 |
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Evidence that the 5-HT3 receptors of the rat, mouse and guinea-pig superior cervical ganglion may be different.
Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Ketanserin; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Superior Cervical Ganglion; Tropisetron; Tubocurarine | 1991 |
Neuroprotective effect of 5-HT3 receptor antagonist on ischemia-induced decrease in CA1 field potential in rat hippocampal slices.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain Ischemia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Hippocampus; Hypoglycemia; Hypoxia; In Vitro Techniques; Ketanserin; Membrane Potentials; Oxazines; Rats; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1992 |
Expression of 5-HT3 receptors in PC12 cells treated with NGF and 8-Br-cAMP.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cations, Monovalent; Cell Membrane; Dose-Response Relationship, Drug; Indoles; Ketanserin; Kinetics; Membrane Potentials; Nerve Growth Factors; PC12 Cells; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spiperone; Time Factors; Tropisetron | 1992 |
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes | 1991 |
The pharmacological characterization of 5-HT3 receptors in three isolated preparations derived from guinea-pig tissues.
Topics: Animals; Colon; Female; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Kinetics; Male; Methysergide; Receptors, Serotonin; Serotonin; Vagus Nerve | 1990 |
Receptors mediating the effects of 5-hydroxytryptamine on the tracheal vasculature and smooth muscle of sheep.
Topics: Animals; Female; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscle Tonus; Muscle, Smooth; Perfusion; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep; Trachea | 1990 |
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron | 1990 |
5-HT3 receptor antagonists injected into the area postrema inhibit cisplatin-induced emesis in the ferret.
Topics: Animals; Apomorphine; Autoradiography; Brain Chemistry; Carnivora; Cisplatin; Female; Ferrets; Injections, Intraventricular; Ketanserin; Male; Methiothepin; Serotonin; Serotonin Antagonists; Vomiting | 1989 |
5-Hydroxytryptamine receptors that facilitate excitatory neuromuscular transmission in the guinea-pig isolated detrusor muscle.
Topics: Acetylcholine; Adenosine Triphosphate; Amphetamines; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Urinary Bladder | 1995 |
Attenuated 5-hydroxytryptamine receptor-mediated responses in aortae from streptozotocin-induced diabetic rats.
Topics: Animals; Aorta; Arginine; Blood Glucose; Diabetes Mellitus, Experimental; Endothelium, Vascular; Insulin; Ketanserin; Male; Nitroarginine; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Vasoconstriction | 1994 |
Inhibitory action of 5-hydroxytryptamine on propulsive activity of the guinea-pig isolated colon.
Topics: 5-Methoxytryptamine; Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Indomethacin; Ketanserin; Male; Muscle Contraction; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron | 1996 |
Which type of 5-hydroxytryptamine receptor mediates relaxation of the longitudinal muscle of guinea pig proximal colon in vitro?
Topics: Animals; Colon; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Metergoline; Methiothepin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropisetron | 1996 |
The effects of peripheral serotonin2 (5-HT2) and serotonin3 (5-HT3) receptor agonists on blood glucose levels in rats.
Topics: Animals; Blood Glucose; Glucagon; Insulin; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists | 1996 |
Effects of peripheral 5-HT2 and 5-HT3 receptor agonists on food intake in food-deprived and 2-deoxy-D-glucose-treated rats.
Topics: Adrenal Medulla; Adrenalectomy; Animals; Deoxyglucose; Eating; Epinephrine; Food Deprivation; Hyperphagia; Ketanserin; Male; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1996 |
Partial role of 5-HT2 and 5-HT3 receptors in the activity of antidepressants in the mouse forced swimming test.
Topics: Amphetamines; Animals; Antidepressive Agents; Behavior, Animal; Citalopram; Desipramine; Drug Interactions; Fluoxetine; Fluvoxamine; Imipramine; Ketanserin; Male; Maprotiline; Mice; Ondansetron; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming | 1997 |
5-Hydroxytryptamine-induced calcium-channel gating in rainbow trout (Oncorhynchus mykiss) peripheral blood lymphocytes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Calcium Channels; Dopamine Antagonists; Ion Channel Gating; Ionomycin; Ionophores; Ketanserin; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulpiride | 1997 |
5-HT receptor types in the rat ileum longitudinal muscle: focus on 5-HT2 receptors mediating contraction.
Topics: 5-Methoxytryptamine; Animals; Female; Gastrointestinal Motility; Ileum; In Vitro Techniques; Ketanserin; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1997 |
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries | 1999 |
Characterisation of 5-HT receptors in human coronary arteries by molecular and pharmacological techniques.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Cardiovascular System; Coronary Vessels; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Vitro Techniques; Ketanserin; Methiothepin; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tissue Distribution; Tryptamines; Vasoconstriction | 1999 |
Study of mechanisms of calcitonin analgesia in mice. Involvement of 5-HT3 receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesics; Animals; Brain Chemistry; Calcitonin; Dose-Response Relationship, Drug; Indoles; Indophenol; Ketanserin; Male; Mice; Mice, Inbred Strains; Nociceptors; Pain; Pain Measurement; Piperazines; Pyridines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1999 |
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron | 2001 |
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides | 2003 |