2-methyl-5-ht and granisetron

2-methyl-5-ht has been researched along with granisetron in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.88)18.7374
1990's13 (76.47)18.2507
2000's3 (17.65)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
King, GL1
Ashby, CR; Edwards, E; Harkins, K; Wang, RY1
Balestra, B; Candura, SM; Lucchelli, A; Messori, E; Rizzi, CA; Tonini, M1
Clark, R; Eglen, RM; Hegde, SS; Johnson, LG; Lee, CH; Smith, WL; Whiting, RL1
Brikas, P; Bueno, L; Fioramonti, J1
Batsche, K; Wang, RY; Zeise, ML1
Bley, KR; Eglen, RM; Wong, EH1
Brikas, P1
Blower, PR; Endo, T; Hamaue, N; Hirafuji, M; Minami, M; Ogawa, T; Tamakai, H; Yoshioka, M1
Hardcastle, J; Hardcastle, PT1
Akita, K; Blower, PR; Endo, T; Hamaue, N; Hirafuji, M; Minami, M; Ogawa, T1
Khan, NA; Poisson, JP1
Blower, PR; Endo, T; Hamaue, N; Hirafuji, M; Kitamura, N; Minami, M; Nemoto, M; Ogawa, T; Teramoto, Y; Yasuda, E1
Bertrand, PP; Bornstein, JC; Furness, JB; Kunze, WA1
Ge, L; Naylor, RJ; Tuladhar, BR1
Endo, T; Fukushi, E; Hamaue, N; Hirafuji, M; Kang, Y; Minami, M; Saito, M; Sato, H1

Other Studies

17 other study(ies) available for 2-methyl-5-ht and granisetron

ArticleYear
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
Emesis and defecations induced by the 5-hydroxytryptamine (5-HT3) receptor antagonist zacopride in the ferret.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Defecation; Dose-Response Relationship, Drug; Ferrets; Granisetron; Indazoles; Injections, Intravenous; Male; Metoclopramide; Pyrazoles; Serotonin; Serotonin Antagonists; Vagotomy; Vomiting

1990
Characterization of 5-hydroxytryptamine3 receptors in the medial prefrontal cortex: a microiontophoretic study.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: Animals; Cerebral Cortex; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Granisetron; Indazoles; Indoles; Iontophoresis; Magnesium Chloride; Male; Metergoline; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropisetron

1989
5-Hydroxytryptamine receptors that facilitate excitatory neuromuscular transmission in the guinea-pig isolated detrusor muscle.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Acetylcholine; Adenosine Triphosphate; Amphetamines; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Granisetron; Guinea Pigs; In Vitro Techniques; Indoles; Ketanserin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Urinary Bladder

1995
Pharmacological characterization of RS 25259-197, a novel and selective 5-HT3 receptor antagonist, in vivo.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Administration, Oral; Animals; Bradycardia; Dogs; Dose-Response Relationship, Drug; Duodenum; Female; Ferrets; Granisetron; Hemodynamics; Injections, Intravenous; Injections, Subcutaneous; Isoquinolines; Male; Ondansetron; Palonosetron; Quinuclidines; Random Allocation; Rats; Serotonin; Serotonin Antagonists; Stereoisomerism; Vomiting

1995
Types of serotonergic receptors involved in the control of reticulo-ruminal myoelectric activity in sheep.
    Journal of veterinary pharmacology and therapeutics, 1994, Volume: 17, Issue:5

    Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dioxanes; Dopamine Antagonists; Electromyography; Female; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Injections, Intraventricular; Microelectrodes; Receptors, Serotonin; Reticulum; Ritanserin; Rumen; Serotonin; Serotonin Receptor Agonists; Sheep; Spiro Compounds

1994
The 5-HT3 receptor agonist 2-methyl-5-HT reduces postsynaptic potentials in rat CA1 pyramidal neurons of the hippocampus in vitro.
    Brain research, 1994, Jul-18, Volume: 651, Issue:1-2

    Topics: Animals; Granisetron; Hippocampus; Rats; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission

1994
Characterization of 5-hydroxytryptamine-induced depolarizations in rat isolated vagus nerve.
    European journal of pharmacology, 1994, Aug-01, Volume: 260, Issue:2-3

    Topics: 5-Methoxytryptamine; 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Electrophysiology; Granisetron; In Vitro Techniques; Indoles; Male; Methiothepin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Regression Analysis; Serotonin; Serotonin Antagonists; Sulfonamides; Temperature; Vagus Nerve

1994
Motor-modifying properties of 5-HT3 and 5-HT4 receptor agonists on ovine abomasum.
    Zentralblatt fur Veterinarmedizin. Reihe A, 1994, Volume: 41, Issue:2

    Topics: 5-Methoxytryptamine; Abomasum; Animals; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electromyography; Female; Granisetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sheep

1994
Chemical modulation of 5-HT3 and 5-HT4 receptors affects the release of 5-hydroxytryptamine from the ferret and rat intestine.
    Research communications in molecular pathology and pharmacology, 1995, Volume: 89, Issue:2

    Topics: 5-Methoxytryptamine; Animals; Ferrets; Granisetron; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Evidence that the secretory response of rat intestine to 5-hydroxytryptamine in-vivo involves more than one 5-hydroxytryptamine-receptor subtype.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:9

    Topics: 5-Methoxytryptamine; Action Potentials; Animals; Blood Pressure; Chlorides; Colon; Electrodes; Granisetron; Intestine, Small; Male; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists

1995
Granisetron, a 5-HT3 receptor antagonist, inhibited cisplatin-induced 5-hydroxytryptamine release in the isolated ileum of ferrets.
    Research communications in molecular pathology and pharmacology, 1998, Volume: 100, Issue:3

    Topics: Animals; Cisplatin; Ferrets; Granisetron; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Tetrodotoxin

1998
5-HT3 receptor-channels coupled with Na+ influx in human T cells: role in T cell activation.
    Journal of neuroimmunology, 1999, Sep-01, Volume: 99, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium Signaling; Cell Cycle; Enzyme Activation; Granisetron; Humans; Ion Channel Gating; Ion Transport; Jurkat Cells; Lymphocyte Activation; Metoclopramide; Neoplasm Proteins; Phytohemagglutinins; Piperazines; Protein Kinase C; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Ryanodine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sodium Channels; T-Lymphocytes; Thapsigargin

1999
Effects of various 5-HT3 receptor antagonists, granisetron, ondansetron, ramosetron and azasetron on serotonin (5-HT) release from the ferret isolated ileum.
    Research communications in molecular pathology and pharmacology, 1999, Volume: 104, Issue:2

    Topics: Animals; Benzimidazoles; Dose-Response Relationship, Drug; Drug Interactions; Ferrets; Granisetron; Ileum; Male; Ondansetron; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1999
The terminals of myenteric intrinsic primary afferent neurons of the guinea-pig ileum are excited by 5-hydroxytryptamine acting at 5-hydroxytryptamine-3 receptors.
    Neuroscience, 2000, Volume: 101, Issue:2

    Topics: 5-Methoxytryptamine; Action Potentials; Animals; Dioxanes; Granisetron; Guinea Pigs; Ileum; Indoles; Myenteric Plexus; Neurons, Afferent; Piperidines; Presynaptic Terminals; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Signal Transduction; Tropisetron

2000
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003
Functional roles of 5-hydroxytryptamine 3/4 receptors in neurons of rat dorsal motor nucleus of the vagus.
    Neuroscience, 2006, Aug-25, Volume: 141, Issue:2

    Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Animals, Newborn; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Granisetron; In Vitro Techniques; Medulla Oblongata; Membrane Potentials; Neurons; para-Aminobenzoates; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vagus Nerve

2006