2-methyl-5-ht and biguanides

2-methyl-5-ht has been researched along with biguanides in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19902 (10.53)18.7374
1990's12 (63.16)18.2507
2000's5 (26.32)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ashby, CR; Edwards, E; Wang, RY1
Boess, FG; Lummis, SC; Martin, IL; SepĂșlveda, MI1
Ashby, CR; Edwards, E; Minabe, Y; Wang, RY1
Miller, AD; Nonaka, S1
Lummis, SC; Martin, IL; SepĂșlveda, MI1
Ashby, CR; Edwards, E; Harkins, K; Wang, RY1
Black, CK; Schmidt, CJ1
Ireland, SJ; Tyers, MB1
Chiba, S; Fujiwara, T1
Gorzalka, BB; Tanco, SA; Watson, NV1
Blier, P; Bouchard, C1
Ashby, CR; Edwards, E; Hampton, E; Wang, RY; Zhang, J1
Kreikamp, AP; van Hooft, JA; Vijverberg, HP1
Lummis, SC; Niemeyer, MI1
Furuichi, K; Miyake, A; Mochizuki, S; Saito, M; Watanabe, T1
Akuzawa, S; Ito, H; Iwaoka, K; Kamato, T; Kiso, T; Miyata, K; Nagakura, Y; Naitoh, Y; Sakai, H; Suzuki, M; Yamaguchi, T; Yamano, M; Yuki, H1
Morales, M; Oz, M; Zhang, L1
Davies, PA; Hales, TG; Kirkness, EF; Safa, P; Stewart, A1
Fukushima, T; Hori, Y; Ohtsubo, T; Tsuda, M; Yanagawa, Y1

Other Studies

19 other study(ies) available for 2-methyl-5-ht and biguanides

ArticleYear
Biochemical characterization of phosphoinositide hydrolysis stimulated by 5-HT3 receptor agonists.
    Neuroreport, 1992, Volume: 3, Issue:12

    Topics: Animals; Arachidonate 5-Lipoxygenase; Arachidonic Acids; Biguanides; Hydrolysis; Hypoglycemic Agents; Male; Neuromuscular Depolarizing Agents; Neurons; Neurotransmitter Agents; Phosphatidylinositols; Prostaglandin-Endoperoxide Synthases; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists; Stimulation, Chemical

1992
5-HT3 receptors in NG108-15 neuroblastoma x glioma cells: effect of the novel agonist 1-(m-chlorophenyl)-biguanide.
    Neuropharmacology, 1992, Volume: 31, Issue:6

    Topics: Animals; Biguanides; Binding, Competitive; Evoked Potentials; Glioma; Hybrid Cells; Imidazoles; Indoles; Kinetics; Mice; Neuroblastoma; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1992
5-HT3-like receptors in the rat medial prefrontal cortex: an electrophysiological study.
    Brain research, 1991, Jun-07, Volume: 550, Issue:2

    Topics: Action Potentials; Animals; Benzamides; Biguanides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Evoked Potentials; Glutamates; Glutamic Acid; Hypoglycemic Agents; Magnesium Chloride; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1991
Mechanisms of vomiting induced by serotonin-3 receptor agonists in the cat: effect of vagotomy, splanchnicectomy or area postrema lesion.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Animals; Biguanides; Cats; Cerebral Ventricles; Female; Male; Serotonin; Serotonin Antagonists; Splanchnic Nerves; Tropanes; Vagotomy; Vomiting

1992
The agonist properties of m-chlorophenylbiguanide and 2-methyl-5-hydroxytryptamine on 5-HT3 receptors in N1E-115 neuroblastoma cells.
    British journal of pharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Biguanides; Membrane Potentials; Mice; Neuroblastoma; Neurons; Radioligand Assay; Receptors, Serotonin; Serotonin; Tumor Cells, Cultured

1991
Effect of 5-hydroxytryptamine3 receptor agonists on phosphoinositides hydrolysis in the rat fronto-cingulate and entorhinal cortices.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:3

    Topics: Animals; Biguanides; Brain; Hydrolysis; Hypoglycemic Agents; Male; Phosphatidylinositols; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1991
The putative 5-HT3 agonist phenylbiguanide induces carrier-mediated release of [3H]dopamine.
    European journal of pharmacology, 1989, Aug-22, Volume: 167, Issue:2

    Topics: Animals; Biguanides; Corpus Striatum; Dopamine; Drug Carriers; In Vitro Techniques; Rats; Serotonin

1989
Pharmacological characterization of 5-hydroxytryptamine-induced depolarization of the rat isolated vagus nerve.
    British journal of pharmacology, 1987, Volume: 90, Issue:1

    Topics: Animals; Biguanides; Cocaine; In Vitro Techniques; Male; Piperazines; Quipazine; Rats; Serotonin; Serotonin Antagonists; Vagus Nerve

1987
2-Methyl-5-HT-induced vasoconstrictions mediated via alpha 1-adrenoceptors in rabbit common carotid arteries.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Biguanides; Carotid Artery, Common; Guanethidine; Hypoglycemic Agents; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Rabbits; Receptors, Adrenergic, alpha-1; Serotonin; Vasoconstriction

1994
Effects of 5-HT3 agonists on reproductive behaviors in rats.
    Psychopharmacology, 1994, Volume: 115, Issue:1-2

    Topics: Animals; Biguanides; Ejaculation; Estradiol; Female; Hypoglycemic Agents; Injections, Intraventricular; Male; Ovariectomy; Posture; Progesterone; Rats; Serotonin; Serotonin Receptor Agonists; Sexual Behavior, Animal

1994
Functional characterization of a 5-HT3 receptor which modulates the release of 5-HT in the guinea-pig brain.
    British journal of pharmacology, 1993, Volume: 108, Issue:1

    Topics: Animals; Biguanides; Electric Stimulation; Frontal Lobe; Guinea Pigs; Hippocampus; Hypothalamus; In Vitro Techniques; Male; Paroxetine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1993
5-HT3-like receptors in the rat medial prefrontal cortex: further pharmacological characterization.
    Brain research, 1996, Sep-09, Volume: 733, Issue:1

    Topics: Animals; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Frontal Lobe; Glutamic Acid; Gyrus Cinguli; Hydrolysis; Indoles; Isomerism; Male; Neurons; Nicotinic Antagonists; Phosphatidylinositols; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tubocurarine

1996
Native serotonin 5-HT3 receptors expressed in Xenopus oocytes differ from homopentameric 5-HT3 receptors.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: Animals; Biguanides; Cell Differentiation; Dopamine; Female; Kinetics; Macromolecular Substances; Membrane Potentials; Mice; Neuroblastoma; Oocytes; Patch-Clamp Techniques; Plasmids; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; RNA, Messenger; Serotonin; Serotonin Receptor Agonists; Tumor Cells, Cultured; Xenopus

1997
Different efficacy of specific agonists at 5-HT3 receptor splice variants: the role of the extra six amino acid segment.
    British journal of pharmacology, 1998, Volume: 123, Issue:4

    Topics: Biguanides; Cell Line; Humans; Mutagenesis, Site-Directed; Radioligand Assay; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; RNA Splicing; Serotonin; Serotonin Receptor Agonists

1998
Cloning, expression, and characterization of ferret 5-HT(3) receptor subunit.
    European journal of pharmacology, 2000, Jul-07, Volume: 399, Issue:2-3

    Topics: Alternative Splicing; Amino Acid Sequence; Animals; Biguanides; Binding, Competitive; Cell Line; Cloning, Molecular; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Ferrets; Gene Expression; Humans; Imidazoles; Indoles; Kruppel-Like Factor 6; Kruppel-Like Transcription Factors; Membrane Potentials; Molecular Sequence Data; Ondansetron; Piperazines; Proto-Oncogene Proteins; Radioligand Assay; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; RNA, Messenger; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tissue Distribution; Trans-Activators; Tritium; Tubocurarine

2000
Pharmacological profile of YM-31636, a novel 5-HT3 receptor agonist, in vitro.
    European journal of pharmacology, 2000, Dec-08, Volume: 409, Issue:2

    Topics: Acetylcholine; Action Potentials; Animals; Anthraquinones; Atrial Function; Biguanides; Binding, Competitive; Colon; Dinoprostone; Dose-Response Relationship, Drug; Guinea Pigs; Heart Atria; Humans; In Vitro Techniques; Muscle Contraction; Myocardial Contraction; Pyrroles; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Receptor Agonists; Thiazoles

2000
Endogenous cannabinoid, anandamide, acts as a noncompetitive inhibitor on 5-HT3 receptor-mediated responses in Xenopus oocytes.
    Synapse (New York, N.Y.), 2002, Dec-01, Volume: 46, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Analysis of Variance; Animals; Arachidonic Acids; Biguanides; Cannabinoids; Chelating Agents; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Electrophysiology; Endocannabinoids; Enzyme Inhibitors; Female; Indazoles; Membrane Potentials; Oocytes; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Serotonin, 5-HT3; Rimonabant; RNA, Complementary; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin Receptor Agonists; Thionucleotides; Tropanes; Xenopus laevis

2002
Introduction of the 5-HT3B subunit alters the functional properties of 5-HT3 receptors native to neuroblastoma cells.
    Neuropharmacology, 2003, Volume: 44, Issue:2

    Topics: Animals; Biguanides; Calcium; Cell Differentiation; Cell Line; Dose-Response Relationship, Drug; Drug Interactions; Fluorescence; Gene Expression; Green Fluorescent Proteins; Luminescent Proteins; Mice; Molecular Sequence Data; Neuroblastoma; Ondansetron; Patch-Clamp Techniques; Protein Subunits; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

2003
Facilitatory actions of serotonin type 3 receptors on GABAergic inhibitory synaptic transmission in the spinal superficial dorsal horn.
    Journal of neurophysiology, 2009, Volume: 102, Issue:3

    Topics: Analysis of Variance; Animals; Biguanides; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Transgenic; Models, Biological; Neural Inhibition; Ondansetron; Patch-Clamp Techniques; Posterior Horn Cells; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

2009