2-methyl-5-ht and bemesetron

2-methyl-5-ht has been researched along with bemesetron in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.55)18.7374
1990's19 (86.36)18.2507
2000's2 (9.09)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, R; Beer, M; Herbert, R; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, GI; Swain, CJ1
Baker, R; Beer, M; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, G; Swain, CJ; Watling, K1
Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Cervo, L; Dalla Valle, F; Fracasso, C; Gemma, S; Goegan, M; Greco, G; Hamon, M; Mennini, T; Morelli, E; Nacci, V; Novellino, E1
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A1
Hille, B; Mathie, A; Yang, J1
Feniuk, W; Saxena, PR; Tadipatri, S1
Hannon, S; Heal, DJ; Martin, KF; Phillips, I1
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB1
Miller, AD; Nonaka, S1
Beani, L; Bianchi, C; Siniscalchi, A1
Giordano, J2
Anderson, EG; Glaum, SR; Proudfit, HK1
Anderson, EG; Todorovic, SM1
Dalton, DW; Feniuk, W; Humphrey, PP1
Buchheit, KH; Buhl, T1
Deschaux, P; Ferrière, F; Khan, NA; Meyniel, JP1
González, AA; Puig, MM1
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M1
Hu, GY; Yang, HH; Yuan, YM1
Goto, F; Ishizaki, K; Obata, H; Sasaki, M1
Ho, Y; Huang, KH; Lai, YC; Tsai, LH1

Other Studies

22 other study(ies) available for 2-methyl-5-ht and bemesetron

ArticleYear
Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).
    Journal of medicinal chemistry, 1992, Mar-20, Volume: 35, Issue:6

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Oxazoles; Rats; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction

1992
Novel 5-HT3 antagonists. Indole oxadiazoles.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Electrochemistry; Indicators and Reagents; Indoles; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tropisetron

1991
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Blood-Brain Barrier; Brain; Guanidine; Guinea Pigs; Hybrid Cells; In Vitro Techniques; Ligands; Male; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

1999
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:2

    Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1992
5-HT3 receptor channels in dissociated rat superior cervical ganglion neurons.
    The Journal of physiology, 1992, Volume: 448

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Ganglia, Sympathetic; Indoles; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1992
Rabbit isolated renal artery contractions by some tryptamine derivatives, including 2-methyl-5-HT, are mediated by a 5-HT1-like receptor.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; In Vitro Techniques; Indoles; Muscle Contraction; Muscle, Smooth, Vascular; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron; Vasoconstriction

1992
Opposing roles for 5-HT1B and 5-HT3 receptors in the control of 5-HT release in rat hippocampus in vivo.
    British journal of pharmacology, 1992, Volume: 106, Issue:1

    Topics: Animals; Dialysis; Dose-Response Relationship, Drug; Hippocampus; Indoles; Injections, Intraperitoneal; Male; Methiothepin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes

1992
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron

1991
Mechanisms of vomiting induced by serotonin-3 receptor agonists in the cat: effect of vagotomy, splanchnicectomy or area postrema lesion.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Animals; Biguanides; Cats; Cerebral Ventricles; Female; Male; Serotonin; Serotonin Antagonists; Splanchnic Nerves; Tropanes; Vagotomy; Vomiting

1992
Influence of acute and chronic chlorimipramine treatment on the 5-HT receptor-mediated modulation of acetylcholine release from the cerebral cortex of freely moving guinea-pigs.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Cerebral Cortex; Clomipramine; Female; Guinea Pigs; Injections, Intraventricular; Male; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tropanes

1991
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
    European journal of pharmacology, 1991, Jun-25, Volume: 199, Issue:2

    Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes

1991
5-HT3 receptors modulate spinal nociceptive reflexes.
    Brain research, 1990, Feb-26, Volume: 510, Issue:1

    Topics: Animals; Indoles; Male; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Spinal Cord; Tropanes; Tropisetron

1990
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron

1990
An investigation into the mechanisms of the cardiovascular effects of 5-hydroxytryptamine in conscious normotensive and DOCA-salt hypertensive rats.
    Journal of autonomic pharmacology, 1986, Volume: 6, Issue:3

    Topics: Animals; Blood Pressure; Desoxycorticosterone; Heart Rate; Hemodynamics; Hypertension; Male; Rats; Serotonin; Serotonin Antagonists; Tropanes

1986
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron

1994
Antinociceptive effects of intrathecally administered 2-methylserotonin in developing rats.
    Brain research. Developmental brain research, 1997, Jan-02, Volume: 98, Issue:1

    Topics: Animals; Animals, Newborn; Dose-Response Relationship, Drug; Formaldehyde; Inflammation; Injections, Spinal; Male; Nociceptors; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes

1997
Identification of lymphocyte 5-HT3 receptor subtype and its implication in fish T-cell proliferation.
    Immunology letters, 1997, Volume: 55, Issue:3

    Topics: Animals; Cell Cycle; Indoles; Lymphocyte Activation; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Phytohemagglutinins; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Sodium; Time Factors; Tritium; Tropanes; Tropisetron

1997
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron

1997
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
    Gynecologic and obstetric investigation, 1999, Volume: 47, Issue:2

    Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries

1999
Tetraethylammonium and 4-aminopyridine enhancement of 5-HT3 receptor-mediated contraction of guinea pig ileum in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1998, Volume: 19, Issue:5

    Topics: 4-Aminopyridine; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Potassium Channels; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetraethylammonium; Tropanes

1998
Effects of 5-HT2 and 5-HT3 receptors on the modulation of nociceptive transmission in rat spinal cord according to the formalin test.
    European journal of pharmacology, 2001, Jul-13, Volume: 424, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dose-Response Relationship, Drug; Formaldehyde; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission; Tropanes

2001
Effects of serotonin on acid secretion in isolated rat stomach: the role of 5-HT3 receptors.
    The Chinese journal of physiology, 2009, Nov-30, Volume: 52, Issue:5 Suppl

    Topics: Animals; Enterochromaffin Cells; Gastric Acid; Histamine; In Vitro Techniques; Male; Oxotremorine; Pentagastrin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Stomach; Tropanes

2009