2-methyl-5-ht has been researched along with bemesetron in 22 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (4.55) | 18.7374 |
1990's | 19 (86.36) | 18.2507 |
2000's | 2 (9.09) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Baker, R; Beer, M; Herbert, R; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, GI; Swain, CJ | 1 |
Baker, R; Beer, M; Kneen, C; Moseley, J; Saunders, J; Seward, EM; Stanton, J; Stevenson, G; Swain, CJ; Watling, K | 1 |
Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Cervo, L; Dalla Valle, F; Fracasso, C; Gemma, S; Goegan, M; Greco, G; Hamon, M; Mennini, T; Morelli, E; Nacci, V; Novellino, E | 1 |
Edamura, N; Kizawa, Y; Maruyama, C; Murakami, H; Sano, M; Yamazaki, A | 1 |
Hille, B; Mathie, A; Yang, J | 1 |
Feniuk, W; Saxena, PR; Tadipatri, S | 1 |
Hannon, S; Heal, DJ; Martin, KF; Phillips, I | 1 |
Higgins, GA; Jones, BJ; Oakley, NR; Tyers, MB | 1 |
Miller, AD; Nonaka, S | 1 |
Beani, L; Bianchi, C; Siniscalchi, A | 1 |
Giordano, J | 2 |
Anderson, EG; Glaum, SR; Proudfit, HK | 1 |
Anderson, EG; Todorovic, SM | 1 |
Dalton, DW; Feniuk, W; Humphrey, PP | 1 |
Buchheit, KH; Buhl, T | 1 |
Deschaux, P; Ferrière, F; Khan, NA; Meyniel, JP | 1 |
González, AA; Puig, MM | 1 |
Bodelsson, G; Bodelsson, M; Karlsson, C; Stjernquist, M | 1 |
Hu, GY; Yang, HH; Yuan, YM | 1 |
Goto, F; Ishizaki, K; Obata, H; Sasaki, M | 1 |
Ho, Y; Huang, KH; Lai, YC; Tsai, LH | 1 |
22 other study(ies) available for 2-methyl-5-ht and bemesetron
Article | Year |
---|---|
Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).
Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Oxazoles; Rats; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction | 1992 |
Novel 5-HT3 antagonists. Indole oxadiazoles.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Electrochemistry; Indicators and Reagents; Indoles; Magnetic Resonance Spectroscopy; Male; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tropisetron | 1991 |
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.
Topics: Animals; Anti-Anxiety Agents; Anti-Inflammatory Agents, Non-Steroidal; Blood-Brain Barrier; Brain; Guanidine; Guinea Pigs; Hybrid Cells; In Vitro Techniques; Ligands; Male; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship | 1999 |
Possible site of action of 2-methylserotonin in inducing relaxation of acetylcholine-induced contraction in the molluscan (Mytilus edulis) smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Cyclic AMP; Cyclic GMP; Cyproheptadine; Dose-Response Relationship, Drug; Indoles; Ketanserin; Mianserin; Muscle Relaxation; Muscle, Smooth; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
5-HT3 receptor channels in dissociated rat superior cervical ganglion neurons.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Ganglia, Sympathetic; Indoles; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1992 |
Rabbit isolated renal artery contractions by some tryptamine derivatives, including 2-methyl-5-HT, are mediated by a 5-HT1-like receptor.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; In Vitro Techniques; Indoles; Muscle Contraction; Muscle, Smooth, Vascular; Prostaglandin Endoperoxides, Synthetic; Rabbits; Receptors, Serotonin; Renal Artery; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes; Tropisetron; Vasoconstriction | 1992 |
Opposing roles for 5-HT1B and 5-HT3 receptors in the control of 5-HT release in rat hippocampus in vivo.
Topics: Animals; Dialysis; Dose-Response Relationship, Drug; Hippocampus; Indoles; Injections, Intraperitoneal; Male; Methiothepin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes | 1992 |
Evidence that the amygdala is involved in the disinhibitory effects of 5-HT3 receptor antagonists.
Topics: Amygdala; Animals; Anxiety; Conflict, Psychological; Granisetron; Imidazoles; Indazoles; Indoles; Lighting; Male; Ondansetron; Raphe Nuclei; Rats; Serotonin; Serotonin Antagonists; Social Behavior; Tropanes; Tropisetron | 1991 |
Mechanisms of vomiting induced by serotonin-3 receptor agonists in the cat: effect of vagotomy, splanchnicectomy or area postrema lesion.
Topics: Animals; Biguanides; Cats; Cerebral Ventricles; Female; Male; Serotonin; Serotonin Antagonists; Splanchnic Nerves; Tropanes; Vagotomy; Vomiting | 1992 |
Influence of acute and chronic chlorimipramine treatment on the 5-HT receptor-mediated modulation of acetylcholine release from the cerebral cortex of freely moving guinea-pigs.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Cerebral Cortex; Clomipramine; Female; Guinea Pigs; Injections, Intraventricular; Male; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tropanes | 1991 |
Analgesic profile of centrally administered 2-methylserotonin against acute pain in rats.
Topics: Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Injections, Intraventricular; Injections, Spinal; Ketanserin; Male; Mianserin; Motor Activity; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Serotonin; Respiration; Serotonin; Serotonin Antagonists; Tropanes | 1991 |
5-HT3 receptors modulate spinal nociceptive reflexes.
Topics: Animals; Indoles; Male; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Serotonin; Spinal Cord; Tropanes; Tropisetron | 1990 |
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron | 1990 |
An investigation into the mechanisms of the cardiovascular effects of 5-hydroxytryptamine in conscious normotensive and DOCA-salt hypertensive rats.
Topics: Animals; Blood Pressure; Desoxycorticosterone; Heart Rate; Hemodynamics; Hypertension; Male; Rats; Serotonin; Serotonin Antagonists; Tropanes | 1986 |
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron | 1994 |
Antinociceptive effects of intrathecally administered 2-methylserotonin in developing rats.
Topics: Animals; Animals, Newborn; Dose-Response Relationship, Drug; Formaldehyde; Inflammation; Injections, Spinal; Male; Nociceptors; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Tropanes | 1997 |
Identification of lymphocyte 5-HT3 receptor subtype and its implication in fish T-cell proliferation.
Topics: Animals; Cell Cycle; Indoles; Lymphocyte Activation; Lymphocytes; Metoclopramide; Oncorhynchus mykiss; Phytohemagglutinins; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Sodium; Time Factors; Tritium; Tropanes; Tropisetron | 1997 |
Ondansetron facilitates neuromuscular transmission in the guinea-pig ileum.
Topics: 5-Methoxytryptamine; Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Ondansetron; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tropanes; Tropisetron | 1997 |
Characterization of 5-hydroxytryptamine receptors mediating circular smooth muscle contraction in the human umbilical artery.
Topics: Adolescent; Adult; Female; Humans; Ketanserin; Methiothepin; Muscle Contraction; Muscle, Smooth; Pregnancy; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tropanes; Umbilical Arteries | 1999 |
Tetraethylammonium and 4-aminopyridine enhancement of 5-HT3 receptor-mediated contraction of guinea pig ileum in vitro.
Topics: 4-Aminopyridine; Animals; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Potassium Channels; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetraethylammonium; Tropanes | 1998 |
Effects of 5-HT2 and 5-HT3 receptors on the modulation of nociceptive transmission in rat spinal cord according to the formalin test.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dose-Response Relationship, Drug; Formaldehyde; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission; Tropanes | 2001 |
Effects of serotonin on acid secretion in isolated rat stomach: the role of 5-HT3 receptors.
Topics: Animals; Enterochromaffin Cells; Gastric Acid; Histamine; In Vitro Techniques; Male; Oxotremorine; Pentagastrin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Stomach; Tropanes | 2009 |