Page last updated: 2024-08-24

2-methoxyestradiol and 2-methoxyestradiol-3,17-o,o-bis(sulfamate)

2-methoxyestradiol has been researched along with 2-methoxyestradiol-3,17-o,o-bis(sulfamate) in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (44.44)29.6817
2010's3 (33.33)24.3611
2020's2 (22.22)2.80

Authors

AuthorsStudies
Bubert, C; Ferrandis, E; Ho, YT; Kasprzyk, PG; Leese, MP; Mahon, MF; Newman, SP; Potter, BV; Purohit, A; Reed, MJ; Regis-Lydi, S1
De Simone, G; Di Fiore, A; Ferrandis, E; Foster, PA; Gaukroger, K; Jourdan, FL; Leese, MP; Mahon, MF; Newman, SP; Potter, BV; Purohit, A; Reed, MJ; Regis-Lydi, S; Stengel, C; Supuran, CT1
Dohle, W; Ferrandis, E; Hamel, E; Jourdan, F; Leese, MP; Newman, SP; Potter, BV; Purohit, A; Reed, MJ1
Bai, R; Dohle, W; Ferrandis, E; Hamel, E; Jourdan, F; Kimberley, MR; Leese, MP; Potter, BV; Thomas, MP1
Potter, BV; Thomas, MP1
Day, JM; Foster, PA; Ho, YT; Judde, JG; Lassalle, M; Leese, MP; Newman, SP; Potter, BV; Prevost, G; Purohit, A; Reed, MJ; Stengel, C1
Chander, SK; Foster, PA; Jhalli, R; Leese, MP; Newman, SP; Parsons, MF; Potter, BV; Purohit, A; Reed, MJ1
Diercks, BP; Dohle, W; Flügel, A; Flügel, LT; Guse, AH; Hosang, L; Löhndorf, A; Marry, S; Müller-Kirschbaum, LC; Odoardi, F; Potter, BVL; Rosche, A1
Carvalho, LAC; da Silva, RO; de Moraes, MO; Dohle, W; Franco, YA; Lima, K; Machado-Neto, JA; Maria-Engler, SS; Noma, IHY; Potter, BVL1

Other Studies

9 other study(ies) available for 2-methoxyestradiol and 2-methoxyestradiol-3,17-o,o-bis(sulfamate)

ArticleYear
3,17-disubstituted 2-alkylestra-1,3,5(10)-trien-3-ol derivatives: synthesis, in vitro and in vivo anticancer activity.
    Journal of medicinal chemistry, 2007, Sep-06, Volume: 50, Issue:18

    Topics: Animals; Antineoplastic Agents; Carbamates; Cell Line, Tumor; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Estradiol; Female; Humans; Male; Mice; Mice, Nude; Models, Molecular; Molecular Structure; Neoplasm Transplantation; Structure-Activity Relationship; Sulfonic Acids

2007
Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Cell Line, Tumor; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Estradiol; Estrenes; Female; Humans; Mice; Mice, Nude; Models, Molecular; Molecular Conformation; Neoplasm Transplantation; Nitriles; Stereoisomerism; Steryl-Sulfatase; Structure-Activity Relationship; Transplantation, Heterologous; Tubulin Modulators

2008
Synthesis, antitubulin, and antiproliferative SAR of analogues of 2-methoxyestradiol-3,17-O,O-bis-sulfamate.
    Journal of medicinal chemistry, 2010, Apr-08, Volume: 53, Issue:7

    Topics: Animals; Antineoplastic Agents; Cattle; Cell Line, Tumor; Cell Proliferation; Colchicine; Estradiol; Humans; Inhibitory Concentration 50; Protein Multimerization; Protein Structure, Quaternary; Structure-Activity Relationship; Tubulin

2010
Steroidomimetic Tetrahydroisoquinolines for the Design of New Microtubule Disruptors.
    ACS medicinal chemistry letters, 2012, Jan-12, Volume: 3, Issue:1

    Topics:

2012
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators

2015
STX140 is efficacious in vitro and in vivo in taxane-resistant breast carcinoma cells.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2008, Jan-15, Volume: 14, Issue:2

    Topics: 2-Methoxyestradiol; Animals; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Drug Resistance, Neoplasm; Estradiol; Estrenes; Humans; Mice; Mice, Nude; Paclitaxel; Tubulin Modulators; Xenograft Model Antitumor Assays

2008
The in vivo properties of STX243: a potent angiogenesis inhibitor in breast cancer.
    British journal of cancer, 2008, Nov-04, Volume: 99, Issue:9

    Topics: 2-Methoxyestradiol; Angiogenesis Inhibitors; Animals; Breast Neoplasms; Cell Line, Tumor; Estradiol; Estrenes; Female; Humans; Mice; Mice, Inbred C57BL; Rats; Rats, Wistar; Sulfonic Acids

2008
2-Methoxyestradiol-3,17-O,O-bis-sulfamate inhibits store-operated Ca
    Biochimica et biophysica acta. Molecular cell research, 2023, Volume: 1870, Issue:6

    Topics: 2-Methoxyestradiol; Animals; Encephalomyelitis, Autoimmune, Experimental; Pharmaceutical Preparations; Rats; Rats, Inbred Lew; T-Lymphocytes

2023
2-Methoxyestradiol-3,17-
    International journal of molecular sciences, 2023, Jul-11, Volume: 24, Issue:14

    Topics: 2-Methoxyestradiol; Apoptosis; Cell Line, Tumor; Cell Proliferation; Estrenes; Humans; Melanoma

2023