2-hydroxysaclofen and gamma-aminobutyric acid

2-hydroxysaclofen has been researched along with gamma-aminobutyric acid in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.17)18.7374
1990's28 (60.87)18.2507
2000's12 (26.09)29.6817
2010's4 (8.70)24.3611
2020's1 (2.17)2.80

Authors

AuthorsStudies
Angst, C; Bettler, B; Bischoff, S; Bittiger, H; Flor, PJ; Froestl, W; Heid, J; Huggel, K; Kaupmann, K; McMaster, G; Mickel, SJ1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Chen, TF; Doyle, PT; Ferguson, DR1
Berthelot, P; Debaert, M; Flouquet, N; Kerr, DI; Ong, J; Vaccher, C1
Gilbert, CD; Hirsch, JA1
Asprodini, EK; Rainnie, DG; Shinnick-Gallagher, P1
Calandra, RS; Campos, MB; Ritta, MN1
Segal, M1
Kohlenbach, A; Schlicker, E1
Collingridge, GL; Davies, CH; Davies, SN1
Abbenante, J; Johnston, GA; Kerr, DI; Ong, J; Prager, RH1
Hirota, A; Kamino, K; Momose-Sato, Y; Sakai, T; Sato, K1
Ashe, JH; Metherate, R1
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ1
Piguet, P1
Finch, DM; Gigg, J; Tan, AM1
Ebner, FF; Friedberg, MH; Lee, SM1
Michelson, HB; Wong, RK1
Lacaille, JC; Vachon, P; Williams, S1
De Koning, HP; Jenks, BG; Roubos, EW1
Mayfield, RD; Zahniser, NR1
Morrisett, RA; Swartzwelder, HS1
Fischer, Y; Parnas, I1
Matsumoto, K; Nguyen, TT; Watanabe, H1
Katz, LC; Roerig, B1
Ballanyi, K; Brockhaus, J1
Bunnett, NW; Grady, EF; Marvizón, JC; Mayer, EA; Stefani, E1
Adanina, V; Batueva, I; Buchanan, JT; Reperant, J; Rio, JP; Sagatelyan, A; Suderevskaya, E; Tsvetkov, E; Vesselkin, N1
Fuchs, JL; Ilyinsky, OB; Schwark, HD; Tennison, CF1
Chen, CL; Chiu, TH; Yang, YR1
Stein, EA; Xi, ZX1
Fischer, Y; Parnas, I; Rashkovan, G; Ravin, R1
Duffy, P; Jackson, D; Kalivas, PW; Romanidies, A; Wyndham, L1
Cupello, A; Scarrone, S1
Akerman, S; Goadsby, PJ; Storer, RJ1
Abraini, JH; Balon, N; Kriem, B; Risso, JJ; Rostain, JC1
Martinez, V; Piqueras, L1
Beverly, JL; Doane, DF; Kotz, CM; Sweet, DC; Thorpe, AJ1
Bocian, R; Konopacki, J1
Gardner, EL; Li, X; Xi, ZX1
Gjoni, T; Urwyler, S1
Bonaventura, MM; Crivello, M; Cymeryng, C; Ferreira, ML; Libertun, C; Lux-Lantos, VA; Repetto, M1
Hanafusa, N; Kawasaki, H; Okamoto, K; Takatori, S1
Budefeld, T; Carbone, D; Eitel, C; Handa, RJ; Majdic, G; Nash, C; Searcy, BT; Staros, M; Stratton, MS; Tobet, SA1
Chang, S; Choi, KH; Gwak, YS; Jang, EY; Jin, W; Kim, HY; Kim, JH; Kim, MS; Koo, H; Lee, BH; Lee, JG; Lee, JY; Ryu, YH; Steffensen, SC; Yang, CH; Yoon, SS1
Cao, K; Liang, H; Luo, W; Tan, D; Tan, Y; Tian, N; Wang, X; Zhang, Q1

Other Studies

46 other study(ies) available for 2-hydroxysaclofen and gamma-aminobutyric acid

ArticleYear
Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors.
    Nature, 1997, Mar-20, Volume: 386, Issue:6622

    Topics: Adenylyl Cyclases; Affinity Labels; Amino Acid Sequence; Animals; Azides; Benzoates; Cell Line; Central Nervous System; Cloning, Molecular; COS Cells; DNA, Complementary; Escherichia coli; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Situ Hybridization; Ligands; Molecular Sequence Data; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Recombinant Proteins; RNA, Messenger; Sequence Alignment

1997
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Inhibitory role of gamma-amino-butyric acid in the rabbit urinary bladder.
    British journal of urology, 1992, Volume: 69, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Carbachol; Depression, Chemical; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Rabbits; Receptors, GABA-A; Urinary Bladder

1992
Differing actions of beta-(2-thienyl)-gamma-aminobutyric acid in central and peripheral preparations.
    European journal of pharmacology, 1992, Oct-06, Volume: 221, Issue:1

    Topics: Animals; Baclofen; Brain; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Receptors, GABA-A; Structure-Activity Relationship; Thiophenes

1992
Synaptic physiology of horizontal connections in the cat's visual cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrophysiology; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Lidocaine; Receptors, GABA-A; Synapses; Visual Cortex

1991
Inhibitory transmission in the basolateral amygdala.
    Journal of neurophysiology, 1991, Volume: 66, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neural Inhibition; Pentobarbital; Potassium; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1991
Coexistence of gamma-aminobutyric acid type A and type B receptors in testicular interstitial cells.
    Journal of neurochemistry, 1991, Volume: 56, Issue:4

    Topics: Ammonium Chloride; Animals; Baclofen; Binding Sites; Detergents; gamma-Aminobutyric Acid; Male; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Testosterone

1991
A subset of local interneurons generate slow inhibitory postsynaptic potentials in hippocampal neurons.
    Brain research, 1990, Mar-12, Volume: 511, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Animals; Baclofen; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Rats; Receptors, GABA-A

1990
GABAB receptor-mediated inhibition of the neurogenic vasopressor response in the pithed rat.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Decerebrate State; Electric Stimulation; gamma-Aminobutyric Acid; Male; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine; Tubocurarine; Vascular Resistance

1990
Paired-pulse depression of monosynaptic GABA-mediated inhibitory postsynaptic responses in rat hippocampus.
    The Journal of physiology, 1990, Volume: 424

    Topics: Action Potentials; Animals; Baclofen; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Picrotoxin; Rats; Synapses; Synaptic Transmission; Tetrodotoxin

1990
Antagonism at GABAB receptors by saclofen and related sulphonic analogues of baclofen and GABA.
    Neuroscience letters, 1989, Dec-15, Volume: 107, Issue:1-3

    Topics: Animals; Baclofen; Cerebral Cortex; Evoked Potentials; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Receptors, GABA-A

1989
A novel gamma-aminobutyric acid response in the embryonic brainstem as revealed by voltage-sensitive dye recording.
    Neuroscience letters, 1995, May-26, Volume: 191, Issue:3

    Topics: Animals; Baclofen; Brain Stem; Chick Embryo; Coloring Agents; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Picrotoxin

1995
Facilitation of an NMDA receptor-mediated EPSP by paired-pulse stimulation in rat neocortex via depression of GABAergic IPSPs.
    The Journal of physiology, 1994, Dec-01, Volume: 481 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Auditory Cortex; Baclofen; Cerebral Cortex; Cesium; Electric Stimulation; Electrophysiology; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Thalamus

1994
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
    Brain research, 1994, Oct-03, Volume: 659, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1994
GABAA- and GABAB-mediated inhibition in the rat dentate gyrus in vitro.
    Epilepsy research, 1993, Volume: 16, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Electric Stimulation; Epilepsy; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synapses

1993
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
    Hippocampus, 1994, Volume: 4, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus

1994
The role of GABA-mediated inhibition in the rat ventral posterior medial thalamus. II. Differential effects of GABAA and GABAB receptor antagonists on responses of VPM neurons.
    Journal of neurophysiology, 1994, Volume: 71, Issue:5

    Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Brain Mapping; Evoked Potentials, Somatosensory; Female; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neural Inhibition; Rats; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamic Nuclei; Vibrissae

1994
Synchronization of inhibitory neurones in the guinea-pig hippocampus in vitro.
    The Journal of physiology, 1994, May-15, Volume: 477, Issue:Pt 1

    Topics: 4-Aminopyridine; Animals; Baclofen; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Microelectrodes; Neurons; Picrotoxin; Pyramidal Cells; Synaptic Transmission

1994
Monosynaptic GABA-mediated inhibitory postsynaptic potentials in CA1 pyramidal cells of hyperexcitable hippocampal slices from kainic acid-treated rats.
    Neuroscience, 1993, Volume: 52, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

1993
Analysis of gamma-aminobutyric acidB receptor function in the in vitro and in vivo regulation of alpha-melanotropin-stimulating hormone secretion from melanotrope cells of Xenopus laevis.
    Endocrinology, 1993, Volume: 132, Issue:2

    Topics: alpha-MSH; Animals; Baclofen; Butylamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Homeostasis; In Vitro Techniques; Kinetics; Organophosphorus Compounds; Perfusion; Pituitary Gland, Posterior; Radioimmunoassay; Receptors, GABA-A; Xenopus laevis

1993
Endogenous GABA release from rat striatal slices: effects of the GABAB receptor antagonist 2-hydroxy-saclofen.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:1

    Topics: Animals; Baclofen; Calcium; Chromatography, High Pressure Liquid; Corpus Striatum; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nipecotic Acids; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Tiagabine

1993
Attenuation of hippocampal long-term potentiation by ethanol: a patch-clamp analysis of glutamatergic and GABAergic mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:5

    Topics: Animals; Baclofen; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Glutamine; Granulocytes; Hippocampus; Male; Midazolam; Neuronal Plasticity; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses

1993
Activation of GABAB receptors at individual release boutons of the crayfish opener neuromuscular junction produces presynaptic inhibition.
    Journal of neurophysiology, 1996, Volume: 75, Issue:4

    Topics: Animals; Astacoidea; Baclofen; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neural Conduction; Neural Inhibition; Neuromuscular Junction; Picrotoxin; Presynaptic Terminals

1996
Involvement of supraspinal GABA-ergic systems in clonidine-induced antinociception in the tail-pinch test in mice.
    Life sciences, 1997, Volume: 61, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Analgesics; Animals; Baclofen; Bicuculline; Clonidine; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Pain; Picrotoxin; Receptors, GABA; Tail

1997
Modulation of intrinsic circuits by serotonin 5-HT3 receptors in developing ferret visual cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Ferrets; gamma-Aminobutyric Acid; Indoles; Ligands; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Pyridinium Compounds; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Tropisetron; Virulence Factors, Bordetella; Visual Cortex

1997
Synaptic inhibition in the isolated respiratory network of neonatal rats.
    The European journal of neuroscience, 1998, Volume: 10, Issue:12

    Topics: Action Potentials; Animals; Animals, Newborn; Anti-Bacterial Agents; Baclofen; Bicarbonates; Bicuculline; Carbon Dioxide; Chloride Channel Agonists; Chloride Channels; Chlorides; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine Agents; Gramicidin; Medulla Oblongata; Microdialysis; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Receptors, GABA-B; Respiration; Strychnine; Synapses; Tetrodotoxin

1998
Substance P release in the dorsal horn assessed by receptor internalization: NMDA receptors counteract a tonic inhibition by GABA(B) receptors.
    The European journal of neuroscience, 1999, Volume: 11, Issue:2

    Topics: Animals; Baclofen; Dizocilpine Maleate; Down-Regulation; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Muscimol; Neural Inhibition; Organ Culture Techniques; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Substance P

1999
Physiological and morphological correlates of presynaptic inhibition in primary afferents of the lamprey spinal cord.
    Neuroscience, 1999, Volume: 88, Issue:3

    Topics: Afferent Pathways; Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Barium; Cadmium; Calcium Channels; Cell Membrane; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Lampreys; Membrane Potentials; Motor Neurons; Nerve Fibers; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Presynaptic Terminals; Species Specificity; Spinal Cord; Synapses

1999
Inhibitory influences on receptive field size in the dorsal column nuclei.
    Experimental brain research, 1999, Volume: 126, Issue:3

    Topics: Animals; Baclofen; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Male; Neural Inhibition; Neurons; Rats; Rats, Sprague-Dawley; Spinal Cord

1999
Activation of rat locus coeruleus neuron GABA(A) receptors by propofol and its potentiation by pentobarbital or alphaxalone.
    European journal of pharmacology, 1999, Dec-15, Volume: 386, Issue:2-3

    Topics: Anesthetics; Anesthetics, Intravenous; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazepam; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ionophores; Locus Coeruleus; Male; Neurons; Pentobarbital; Picrotoxin; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc Compounds

1999
Increased mesolimbic GABA concentration blocks heroin self-administration in the rat.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Animals; Baclofen; Behavior, Animal; Bicuculline; Enzyme Inhibitors; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Heroin; Injections, Intraventricular; Lateral Ventricles; Male; Microinjections; Narcotics; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Opioid-Related Disorders; Rats; Rats, Sprague-Dawley; Self Administration; Telencephalon; Ventral Tegmental Area; Vigabatrin

2000
Novel mechanism for presynaptic inhibition: GABA(A) receptors affect the release machinery.
    Journal of neurophysiology, 2000, Volume: 84, Issue:3

    Topics: Action Potentials; Animals; Astacoidea; Baclofen; Calcium; Dose-Response Relationship, Drug; Electric Stimulation; Fura-2; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Intracellular Fluid; Magnesium; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Picrotoxin; Presynaptic Terminals; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Temperature

2000
Involvement of pallidothalamic circuitry in working memory.
    Neuroscience, 2001, Volume: 104, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics, Opioid; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Maze Learning; Mediodorsal Thalamic Nucleus; Memory, Short-Term; Motor Activity; Neural Inhibition; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-B; Receptors, Opioid, mu

2001
Pretreatment of rat brain synaptosomes with GABA increases subsequent GABA uptake via GABA(B) receptor activation.
    Neurochemical research, 2001, Volume: 26, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Baclofen; Brain; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synaptosomes; Up-Regulation

2001
GABA receptors modulate trigeminovascular nociceptive neurotransmission in the trigeminocervical complex.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Muscimol; Neurons; Nociceptors; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors; Trigeminal Nuclei

2001
Gamma-aminobutyric acid neuropharmacological investigations on narcosis produced by nitrogen, argon, or nitrous oxide.
    Anesthesia and analgesia, 2003, Volume: 96, Issue:3

    Topics: Anesthesia, Inhalation; Animals; Argon; Baclofen; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Motor Activity; Nitrogen; Nitrous Oxide; Pyridazines; Rats; Rats, Sprague-Dawley

2003
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy

2004
Orexin A in the rostrolateral hypothalamic area induces feeding by modulating GABAergic transmission.
    Brain research, 2006, Dec-13, Volume: 1125, Issue:1

    Topics: Analysis of Variance; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; Eating; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Microdialysis; Muscimol; Neuropeptides; Orexins; Rats; Rats, Sprague-Dawley; Time Factors

2006
Posterior hypothalamic GABAergic mediation of hippocampal theta in the cat.
    Brain research bulletin, 2007, Jul-12, Volume: 73, Issue:4-6

    Topics: Animals; Baclofen; Bicuculline; Cats; Electroencephalography; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus, Posterior; Muscimol; Rats; Theta Rhythm

2007
The metabotropic glutamate receptor 7 (mGluR7) allosteric agonist AMN082 modulates nucleus accumbens GABA and glutamate, but not dopamine, in rats.
    Neuropharmacology, 2008, Volume: 54, Issue:3

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Baclofen; Benzhydryl Compounds; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Nucleus Accumbens; Phosphoserine; Rats; Rats, Long-Evans; Tetrodotoxin

2008
Changes in the properties of allosteric and orthosteric GABAB receptor ligands after a continuous, desensitizing agonist pretreatment.
    European journal of pharmacology, 2009, Jan-28, Volume: 603, Issue:1-3

    Topics: Allosteric Regulation; Animals; Baclofen; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclopentanes; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Ligands; Pyrimidines; Rats; Receptors, GABA-B

2009
Effects of GABAB receptor agonists and antagonists on glycemia regulation in mice.
    European journal of pharmacology, 2012, Feb-29, Volume: 677, Issue:1-3

    Topics: Animals; Baclofen; Basal Metabolism; Blood Glucose; Body Weight; Eating; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Glucose Tolerance Test; Homeostasis; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred BALB C; Protein Subunits; Receptors, GABA-B; RNA, Messenger; Time Factors

2012
Involvement of hypothalamic periventricular GABAergic nerves in the central pressor response to clonidine in freely-moving conscious rats.
    Journal of pharmacological sciences, 2012, Volume: 118, Issue:3

    Topics: Animals; Antihypertensive Agents; Baclofen; Bicuculline; Blood Pressure; Clonidine; Excitatory Amino Acid Antagonists; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Heart Rate; Hypothalamus; Kynurenic Acid; Male; Muscimol; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Receptors, Glutamate

2012
Embryonic GABA(B) receptor blockade alters cell migration, adult hypothalamic structure, and anxiety- and depression-like behaviors sex specifically in mice.
    PloS one, 2014, Volume: 9, Issue:8

    Topics: Animals; Anxiety; Baclofen; Cell Movement; Depression; Embryo, Mammalian; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Hypothalamo-Hypophyseal System; Immobilization; Male; Maze Learning; Mice; Mice, Transgenic; Paraventricular Hypothalamic Nucleus; Phosphinic Acids; Pituitary-Adrenal System; Pregnancy; Propanolamines; Protein Subunits; Psychomotor Agitation; Receptors, GABA-B; Sex Factors; Stress, Psychological; Tissue Culture Techniques

2014
Acupuncture reduces relapse to cocaine-seeking behavior via activation of GABA neurons in the ventral tegmental area.
    Addiction biology, 2018, Volume: 23, Issue:1

    Topics: Acupuncture; Animals; Baclofen; Behavior, Animal; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Electrophysiological Phenomena; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Locomotion; Microdialysis; Nucleus Accumbens; Rats; Ventral Tegmental Area

2018
GABA consumption during early pregnancy impairs endometrial receptivity and embryo development in mice.
    Journal of biochemical and molecular toxicology, 2020, Volume: 34, Issue:5

    Topics: Administration, Oral; Animals; Baclofen; Cadherins; Dose-Response Relationship, Drug; Embryo Implantation; Embryonic Development; Endometrium; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Homeobox A10 Proteins; Leukemia Inhibitory Factor; Mice; Pregnancy; Signal Transduction

2020