2-hydroxysaclofen has been researched along with gamma-aminobutyric acid in 46 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (2.17) | 18.7374 |
1990's | 28 (60.87) | 18.2507 |
2000's | 12 (26.09) | 29.6817 |
2010's | 4 (8.70) | 24.3611 |
2020's | 1 (2.17) | 2.80 |
Authors | Studies |
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Angst, C; Bettler, B; Bischoff, S; Bittiger, H; Flor, PJ; Froestl, W; Heid, J; Huggel, K; Kaupmann, K; McMaster, G; Mickel, SJ | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Chen, TF; Doyle, PT; Ferguson, DR | 1 |
Berthelot, P; Debaert, M; Flouquet, N; Kerr, DI; Ong, J; Vaccher, C | 1 |
Gilbert, CD; Hirsch, JA | 1 |
Asprodini, EK; Rainnie, DG; Shinnick-Gallagher, P | 1 |
Calandra, RS; Campos, MB; Ritta, MN | 1 |
Segal, M | 1 |
Kohlenbach, A; Schlicker, E | 1 |
Collingridge, GL; Davies, CH; Davies, SN | 1 |
Abbenante, J; Johnston, GA; Kerr, DI; Ong, J; Prager, RH | 1 |
Hirota, A; Kamino, K; Momose-Sato, Y; Sakai, T; Sato, K | 1 |
Ashe, JH; Metherate, R | 1 |
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ | 1 |
Piguet, P | 1 |
Finch, DM; Gigg, J; Tan, AM | 1 |
Ebner, FF; Friedberg, MH; Lee, SM | 1 |
Michelson, HB; Wong, RK | 1 |
Lacaille, JC; Vachon, P; Williams, S | 1 |
De Koning, HP; Jenks, BG; Roubos, EW | 1 |
Mayfield, RD; Zahniser, NR | 1 |
Morrisett, RA; Swartzwelder, HS | 1 |
Fischer, Y; Parnas, I | 1 |
Matsumoto, K; Nguyen, TT; Watanabe, H | 1 |
Katz, LC; Roerig, B | 1 |
Ballanyi, K; Brockhaus, J | 1 |
Bunnett, NW; Grady, EF; Marvizón, JC; Mayer, EA; Stefani, E | 1 |
Adanina, V; Batueva, I; Buchanan, JT; Reperant, J; Rio, JP; Sagatelyan, A; Suderevskaya, E; Tsvetkov, E; Vesselkin, N | 1 |
Fuchs, JL; Ilyinsky, OB; Schwark, HD; Tennison, CF | 1 |
Chen, CL; Chiu, TH; Yang, YR | 1 |
Stein, EA; Xi, ZX | 1 |
Fischer, Y; Parnas, I; Rashkovan, G; Ravin, R | 1 |
Duffy, P; Jackson, D; Kalivas, PW; Romanidies, A; Wyndham, L | 1 |
Cupello, A; Scarrone, S | 1 |
Akerman, S; Goadsby, PJ; Storer, RJ | 1 |
Abraini, JH; Balon, N; Kriem, B; Risso, JJ; Rostain, JC | 1 |
Martinez, V; Piqueras, L | 1 |
Beverly, JL; Doane, DF; Kotz, CM; Sweet, DC; Thorpe, AJ | 1 |
Bocian, R; Konopacki, J | 1 |
Gardner, EL; Li, X; Xi, ZX | 1 |
Gjoni, T; Urwyler, S | 1 |
Bonaventura, MM; Crivello, M; Cymeryng, C; Ferreira, ML; Libertun, C; Lux-Lantos, VA; Repetto, M | 1 |
Hanafusa, N; Kawasaki, H; Okamoto, K; Takatori, S | 1 |
Budefeld, T; Carbone, D; Eitel, C; Handa, RJ; Majdic, G; Nash, C; Searcy, BT; Staros, M; Stratton, MS; Tobet, SA | 1 |
Chang, S; Choi, KH; Gwak, YS; Jang, EY; Jin, W; Kim, HY; Kim, JH; Kim, MS; Koo, H; Lee, BH; Lee, JG; Lee, JY; Ryu, YH; Steffensen, SC; Yang, CH; Yoon, SS | 1 |
Cao, K; Liang, H; Luo, W; Tan, D; Tan, Y; Tian, N; Wang, X; Zhang, Q | 1 |
46 other study(ies) available for 2-hydroxysaclofen and gamma-aminobutyric acid
Article | Year |
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Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors.
Topics: Adenylyl Cyclases; Affinity Labels; Amino Acid Sequence; Animals; Azides; Benzoates; Cell Line; Central Nervous System; Cloning, Molecular; COS Cells; DNA, Complementary; Escherichia coli; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Situ Hybridization; Ligands; Molecular Sequence Data; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Recombinant Proteins; RNA, Messenger; Sequence Alignment | 1997 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Inhibitory role of gamma-amino-butyric acid in the rabbit urinary bladder.
Topics: Animals; Baclofen; Bicuculline; Carbachol; Depression, Chemical; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Rabbits; Receptors, GABA-A; Urinary Bladder | 1992 |
Differing actions of beta-(2-thienyl)-gamma-aminobutyric acid in central and peripheral preparations.
Topics: Animals; Baclofen; Brain; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Receptors, GABA-A; Structure-Activity Relationship; Thiophenes | 1992 |
Synaptic physiology of horizontal connections in the cat's visual cortex.
Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrophysiology; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Lidocaine; Receptors, GABA-A; Synapses; Visual Cortex | 1991 |
Inhibitory transmission in the basolateral amygdala.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neural Inhibition; Pentobarbital; Potassium; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission | 1991 |
Coexistence of gamma-aminobutyric acid type A and type B receptors in testicular interstitial cells.
Topics: Ammonium Chloride; Animals; Baclofen; Binding Sites; Detergents; gamma-Aminobutyric Acid; Male; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Testosterone | 1991 |
A subset of local interneurons generate slow inhibitory postsynaptic potentials in hippocampal neurons.
Topics: 4-Aminopyridine; Action Potentials; Animals; Baclofen; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Rats; Receptors, GABA-A | 1990 |
GABAB receptor-mediated inhibition of the neurogenic vasopressor response in the pithed rat.
Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Decerebrate State; Electric Stimulation; gamma-Aminobutyric Acid; Male; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine; Tubocurarine; Vascular Resistance | 1990 |
Paired-pulse depression of monosynaptic GABA-mediated inhibitory postsynaptic responses in rat hippocampus.
Topics: Action Potentials; Animals; Baclofen; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Picrotoxin; Rats; Synapses; Synaptic Transmission; Tetrodotoxin | 1990 |
Antagonism at GABAB receptors by saclofen and related sulphonic analogues of baclofen and GABA.
Topics: Animals; Baclofen; Cerebral Cortex; Evoked Potentials; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Receptors, GABA-A | 1989 |
A novel gamma-aminobutyric acid response in the embryonic brainstem as revealed by voltage-sensitive dye recording.
Topics: Animals; Baclofen; Brain Stem; Chick Embryo; Coloring Agents; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Picrotoxin | 1995 |
Facilitation of an NMDA receptor-mediated EPSP by paired-pulse stimulation in rat neocortex via depression of GABAergic IPSPs.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Auditory Cortex; Baclofen; Cerebral Cortex; Cesium; Electric Stimulation; Electrophysiology; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Thalamus | 1994 |
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures | 1994 |
GABAA- and GABAB-mediated inhibition in the rat dentate gyrus in vitro.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Electric Stimulation; Epilepsy; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synapses | 1993 |
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus | 1994 |
The role of GABA-mediated inhibition in the rat ventral posterior medial thalamus. II. Differential effects of GABAA and GABAB receptor antagonists on responses of VPM neurons.
Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Brain Mapping; Evoked Potentials, Somatosensory; Female; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neural Inhibition; Rats; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamic Nuclei; Vibrissae | 1994 |
Synchronization of inhibitory neurones in the guinea-pig hippocampus in vitro.
Topics: 4-Aminopyridine; Animals; Baclofen; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Microelectrodes; Neurons; Picrotoxin; Pyramidal Cells; Synaptic Transmission | 1994 |
Monosynaptic GABA-mediated inhibitory postsynaptic potentials in CA1 pyramidal cells of hyperexcitable hippocampal slices from kainic acid-treated rats.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses | 1993 |
Analysis of gamma-aminobutyric acidB receptor function in the in vitro and in vivo regulation of alpha-melanotropin-stimulating hormone secretion from melanotrope cells of Xenopus laevis.
Topics: alpha-MSH; Animals; Baclofen; Butylamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Homeostasis; In Vitro Techniques; Kinetics; Organophosphorus Compounds; Perfusion; Pituitary Gland, Posterior; Radioimmunoassay; Receptors, GABA-A; Xenopus laevis | 1993 |
Endogenous GABA release from rat striatal slices: effects of the GABAB receptor antagonist 2-hydroxy-saclofen.
Topics: Animals; Baclofen; Calcium; Chromatography, High Pressure Liquid; Corpus Striatum; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nipecotic Acids; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Tiagabine | 1993 |
Attenuation of hippocampal long-term potentiation by ethanol: a patch-clamp analysis of glutamatergic and GABAergic mechanisms.
Topics: Animals; Baclofen; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Glutamine; Granulocytes; Hippocampus; Male; Midazolam; Neuronal Plasticity; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses | 1993 |
Activation of GABAB receptors at individual release boutons of the crayfish opener neuromuscular junction produces presynaptic inhibition.
Topics: Animals; Astacoidea; Baclofen; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neural Conduction; Neural Inhibition; Neuromuscular Junction; Picrotoxin; Presynaptic Terminals | 1996 |
Involvement of supraspinal GABA-ergic systems in clonidine-induced antinociception in the tail-pinch test in mice.
Topics: Adrenergic alpha-2 Receptor Agonists; Analgesics; Animals; Baclofen; Bicuculline; Clonidine; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Pain; Picrotoxin; Receptors, GABA; Tail | 1997 |
Modulation of intrinsic circuits by serotonin 5-HT3 receptors in developing ferret visual cortex.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Ferrets; gamma-Aminobutyric Acid; Indoles; Ligands; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Pyridinium Compounds; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Tropisetron; Virulence Factors, Bordetella; Visual Cortex | 1997 |
Synaptic inhibition in the isolated respiratory network of neonatal rats.
Topics: Action Potentials; Animals; Animals, Newborn; Anti-Bacterial Agents; Baclofen; Bicarbonates; Bicuculline; Carbon Dioxide; Chloride Channel Agonists; Chloride Channels; Chlorides; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine Agents; Gramicidin; Medulla Oblongata; Microdialysis; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Receptors, GABA-B; Respiration; Strychnine; Synapses; Tetrodotoxin | 1998 |
Substance P release in the dorsal horn assessed by receptor internalization: NMDA receptors counteract a tonic inhibition by GABA(B) receptors.
Topics: Animals; Baclofen; Dizocilpine Maleate; Down-Regulation; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Muscimol; Neural Inhibition; Organ Culture Techniques; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Substance P | 1999 |
Physiological and morphological correlates of presynaptic inhibition in primary afferents of the lamprey spinal cord.
Topics: Afferent Pathways; Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Barium; Cadmium; Calcium Channels; Cell Membrane; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Lampreys; Membrane Potentials; Motor Neurons; Nerve Fibers; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Presynaptic Terminals; Species Specificity; Spinal Cord; Synapses | 1999 |
Inhibitory influences on receptive field size in the dorsal column nuclei.
Topics: Animals; Baclofen; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Male; Neural Inhibition; Neurons; Rats; Rats, Sprague-Dawley; Spinal Cord | 1999 |
Activation of rat locus coeruleus neuron GABA(A) receptors by propofol and its potentiation by pentobarbital or alphaxalone.
Topics: Anesthetics; Anesthetics, Intravenous; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazepam; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ionophores; Locus Coeruleus; Male; Neurons; Pentobarbital; Picrotoxin; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc Compounds | 1999 |
Increased mesolimbic GABA concentration blocks heroin self-administration in the rat.
Topics: 4-Aminobutyrate Transaminase; Animals; Baclofen; Behavior, Animal; Bicuculline; Enzyme Inhibitors; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Heroin; Injections, Intraventricular; Lateral Ventricles; Male; Microinjections; Narcotics; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Opioid-Related Disorders; Rats; Rats, Sprague-Dawley; Self Administration; Telencephalon; Ventral Tegmental Area; Vigabatrin | 2000 |
Novel mechanism for presynaptic inhibition: GABA(A) receptors affect the release machinery.
Topics: Action Potentials; Animals; Astacoidea; Baclofen; Calcium; Dose-Response Relationship, Drug; Electric Stimulation; Fura-2; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Intracellular Fluid; Magnesium; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Picrotoxin; Presynaptic Terminals; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Temperature | 2000 |
Involvement of pallidothalamic circuitry in working memory.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics, Opioid; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Maze Learning; Mediodorsal Thalamic Nucleus; Memory, Short-Term; Motor Activity; Neural Inhibition; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-B; Receptors, Opioid, mu | 2001 |
Pretreatment of rat brain synaptosomes with GABA increases subsequent GABA uptake via GABA(B) receptor activation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Baclofen; Brain; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synaptosomes; Up-Regulation | 2001 |
GABA receptors modulate trigeminovascular nociceptive neurotransmission in the trigeminocervical complex.
Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Muscimol; Neurons; Nociceptors; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors; Trigeminal Nuclei | 2001 |
Gamma-aminobutyric acid neuropharmacological investigations on narcosis produced by nitrogen, argon, or nitrous oxide.
Topics: Anesthesia, Inhalation; Animals; Argon; Baclofen; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Motor Activity; Nitrogen; Nitrous Oxide; Pyridazines; Rats; Rats, Sprague-Dawley | 2003 |
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy | 2004 |
Orexin A in the rostrolateral hypothalamic area induces feeding by modulating GABAergic transmission.
Topics: Analysis of Variance; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; Eating; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Microdialysis; Muscimol; Neuropeptides; Orexins; Rats; Rats, Sprague-Dawley; Time Factors | 2006 |
Posterior hypothalamic GABAergic mediation of hippocampal theta in the cat.
Topics: Animals; Baclofen; Bicuculline; Cats; Electroencephalography; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus, Posterior; Muscimol; Rats; Theta Rhythm | 2007 |
The metabotropic glutamate receptor 7 (mGluR7) allosteric agonist AMN082 modulates nucleus accumbens GABA and glutamate, but not dopamine, in rats.
Topics: Analysis of Variance; Anesthetics, Local; Animals; Baclofen; Benzhydryl Compounds; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Nucleus Accumbens; Phosphoserine; Rats; Rats, Long-Evans; Tetrodotoxin | 2008 |
Changes in the properties of allosteric and orthosteric GABAB receptor ligands after a continuous, desensitizing agonist pretreatment.
Topics: Allosteric Regulation; Animals; Baclofen; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclopentanes; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Ligands; Pyrimidines; Rats; Receptors, GABA-B | 2009 |
Effects of GABAB receptor agonists and antagonists on glycemia regulation in mice.
Topics: Animals; Baclofen; Basal Metabolism; Blood Glucose; Body Weight; Eating; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Glucose Tolerance Test; Homeostasis; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred BALB C; Protein Subunits; Receptors, GABA-B; RNA, Messenger; Time Factors | 2012 |
Involvement of hypothalamic periventricular GABAergic nerves in the central pressor response to clonidine in freely-moving conscious rats.
Topics: Animals; Antihypertensive Agents; Baclofen; Bicuculline; Blood Pressure; Clonidine; Excitatory Amino Acid Antagonists; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Heart Rate; Hypothalamus; Kynurenic Acid; Male; Muscimol; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Receptors, Glutamate | 2012 |
Embryonic GABA(B) receptor blockade alters cell migration, adult hypothalamic structure, and anxiety- and depression-like behaviors sex specifically in mice.
Topics: Animals; Anxiety; Baclofen; Cell Movement; Depression; Embryo, Mammalian; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Hypothalamo-Hypophyseal System; Immobilization; Male; Maze Learning; Mice; Mice, Transgenic; Paraventricular Hypothalamic Nucleus; Phosphinic Acids; Pituitary-Adrenal System; Pregnancy; Propanolamines; Protein Subunits; Psychomotor Agitation; Receptors, GABA-B; Sex Factors; Stress, Psychological; Tissue Culture Techniques | 2014 |
Acupuncture reduces relapse to cocaine-seeking behavior via activation of GABA neurons in the ventral tegmental area.
Topics: Acupuncture; Animals; Baclofen; Behavior, Animal; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Electrophysiological Phenomena; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Locomotion; Microdialysis; Nucleus Accumbens; Rats; Ventral Tegmental Area | 2018 |
GABA consumption during early pregnancy impairs endometrial receptivity and embryo development in mice.
Topics: Administration, Oral; Animals; Baclofen; Cadherins; Dose-Response Relationship, Drug; Embryo Implantation; Embryonic Development; Endometrium; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Homeobox A10 Proteins; Leukemia Inhibitory Factor; Mice; Pregnancy; Signal Transduction | 2020 |