2-hydroxysaclofen has been researched along with cgp 35348 in 17 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 17 (100.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Angst, C; Bettler, B; Bischoff, S; Bittiger, H; Flor, PJ; Froestl, W; Heid, J; Huggel, K; Kaupmann, K; McMaster, G; Mickel, SJ | 1 |
| Cao, Z; Clark, S; Hosford, DA; Huin, A; Lin, FH; Morrisett, RA; Wilson, WA | 1 |
| Douglas, WW; Kongsamut, S; Shibuya, I | 2 |
| Fromm, GH; Nakata, M; Sato, K | 1 |
| Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P | 1 |
| Humeniuk, RE; Kerr, DI; Ong, J; White, JM | 1 |
| Slaughter, MM; Tian, N | 1 |
| Finch, DM; Gigg, J; Tan, AM | 1 |
| Crunelli, V; Emri, Z; Juhász, G; Kékesi, KA; Salfay, O | 1 |
| Lewis, DV; Mott, DD; Swartzwelder, HS; Wilson, WA; Xie, CW | 1 |
| Avanzino, GL; Blanchi, D; Cogo, CE; Ermirio, R; Ruggeri, P; Weaver, LC | 1 |
| Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G | 1 |
| Crunelli, V; Dobolyi, A; Emri, Z; Juhász, G; Kékesi, KA; Nyitrai, G | 1 |
| Bowery, NG; Connelly, ST; daSilva, HM; Grobaski, KC; Ping, H; Shepard, PD | 1 |
| Akihara, M; Izumi, F; Kaibara, M; Kawano, C; Shibuya, I; Taniyama, K; Toyohira, Y; Ueda, Y; Uezono, Y; Yamashita, H; Yanagihara, N | 1 |
| Dun, NJ; Lin, HH | 1 |
17 other study(ies) available for 2-hydroxysaclofen and cgp 35348
| Article | Year |
|---|---|
Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors.
Topics: Adenylyl Cyclases; Affinity Labels; Amino Acid Sequence; Animals; Azides; Benzoates; Cell Line; Central Nervous System; Cloning, Molecular; COS Cells; DNA, Complementary; Escherichia coli; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Situ Hybridization; Ligands; Molecular Sequence Data; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Recombinant Proteins; RNA, Messenger; Sequence Alignment | 1997 |
The role of GABAB receptor activation in absence seizures of lethargic (lh/lh) mice.
Topics: Animals; Anticonvulsants; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; Electroencephalography; Electrophysiology; Epilepsy, Absence; Hippocampus; In Vitro Techniques; Mice; Mice, Inbred Strains; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate | 1992 |
Effectiveness of GABAB antagonists in inhibiting baclofen-induced reductions in cytosolic free Ca concentration in isolated melanotrophs of rat.
Topics: Animals; Baclofen; Calcium; Cytosol; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Organophosphorus Compounds; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains | 1992 |
The action of GABAB antagonists in the trigeminal nucleus of the rat.
Topics: Animals; Baclofen; GABA-A Receptor Antagonists; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Trigeminal Nuclei | 1992 |
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle-relaxant effect induced by baclofen.
Topics: Analgesics; Animals; Baclofen; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Morphine; Muscle Relaxation; Muscles; Organophosphorus Compounds; Oxotremorine; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time | 1991 |
Studies on pituitary melanotrophs reveal the novel GABAB antagonist CGP 35-348 to be the first such compound effective on endocrine cells.
Topics: Animals; Baclofen; Bicuculline; Darkness; GABA Antagonists; GABA-A Receptor Antagonists; Kinetics; Male; Melanocyte-Stimulating Hormones; Methionine; Muscimol; Organophosphorus Compounds; Pituitary Gland; Rats; Rats, Inbred Strains; Xenopus laevis | 1991 |
Characterization of GABAB ligands in vivo.
Topics: Animals; Baclofen; beta-Alanine; Drug Interactions; Female; GABA Antagonists; GABA-B Receptor Antagonists; Ligands; Mice; Mice, Inbred BALB C; Muscle Relaxation; Organophosphorus Compounds | 1995 |
Pharmacology of the GABAB receptor in amphibian retina.
Topics: Ambystoma; Animals; Baclofen; Butylamines; Evoked Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Necturus; Organophosphorus Compounds; Propylamines; Receptors, GABA-B; Retina; Retinal Ganglion Cells; Stereoisomerism; Structure-Activity Relationship | 1994 |
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus | 1994 |
Blockade of thalamic GABAB receptors decreases EEG synchronization.
Topics: Animals; Baclofen; Cats; Cortical Synchronization; Electroencephalography; Electromyography; Electrooculography; GABA-B Receptor Antagonists; Microdialysis; Organophosphorus Compounds; Sleep; Thalamus; Wakefulness | 1994 |
GABAB autoreceptors mediate activity-dependent disinhibition and enhance signal transmission in the dentate gyrus.
Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Culture Techniques; GABA-A Receptor Antagonists; Hippocampus; Male; Membrane Potentials; Nerve Fibers; Neural Inhibition; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Theta Rhythm | 1993 |
GABAB receptor-mediated mechanisms in the RVLM studied by microinjections of two GABAB receptor antagonists.
Topics: Animals; Baclofen; Blood Pressure; Electrocardiography; Functional Laterality; GABA-B Receptor Antagonists; Heart Rate; Homeostasis; Male; Medulla Oblongata; Microinjections; Muscimol; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B | 1994 |
Role of peripheral GABAB receptors in the regulation of pepsinogen secretion in anaesthetized rats.
Topics: Anesthesia; Animals; Baclofen; Capsaicin; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gastric Mucosa; Male; Organophosphorus Compounds; p-Methoxy-N-methylphenethylamine; Pepsinogens; Perfusion; Rats; Rats, Wistar; Receptors, GABA-B; Vagotomy | 1995 |
In vivo blockade of thalamic GABA(B) receptors increases excitatory amino-acid levels.
Topics: Animals; Aspartic Acid; Baclofen; GABA-B Receptor Antagonists; Glutamic Acid; Male; Microdialysis; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Taurine; Thalamus | 1996 |
Responses of rat substantia nigra dopamine-containing neurones to (-)-HA-966 in vitro.
Topics: Animals; Baclofen; Dopamine; Electrophysiology; Excitatory Amino Acid Agonists; GABA Agonists; Male; Neurons; Organophosphorus Compounds; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Substantia Nigra | 1997 |
Activation of inwardly rectifying K+ channels by GABA-B receptors expressed in Xenopus oocytes.
Topics: Animals; Baclofen; Cerebellum; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Antagonists; GTP-Binding Proteins; Membrane Potentials; Muscimol; Oocytes; Organophosphorus Compounds; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, GABA-B; Recombinant Proteins; Xenopus laevis | 1998 |
Post- and presynaptic GABA(B) receptor activation in neonatal rat rostral ventrolateral medulla neurons in vitro.
Topics: Animals; Animals, Newborn; Baclofen; Calcium; Chelating Agents; Egtazic Acid; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Guanosine Diphosphate; In Vitro Techniques; Medulla Oblongata; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Tetraethylammonium; Tetrodotoxin; Thionucleotides | 1998 |