2-hydroxysaclofen and baclofen

2-hydroxysaclofen has been researched along with baclofen in 140 studies

Research

Studies (140)

TimeframeStudies, this research(%)All Research%
pre-19904 (2.86)18.7374
1990's93 (66.43)18.2507
2000's28 (20.00)29.6817
2010's13 (9.29)24.3611
2020's2 (1.43)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Chen, TF; Doyle, PT; Ferguson, DR1
Redman, SJ; Stuart, GJ1
Harrison, NL; Lambert, NA; Lovinger, DM1
Bernardini, MC; Blandizzi, C; Del Tacca, M; Martinotti, E; Natale, G1
Cao, Z; Clark, S; Hosford, DA; Huin, A; Lin, FH; Morrisett, RA; Wilson, WA1
Douglas, WW; Kongsamut, S; Shibuya, I2
Kunos, G; Varga, K1
Fromm, GH; Nakata, M; Sato, K1
Santiago, M; Westerink, BH1
Berthelot, P; Debaert, M; Flouquet, N; Kerr, DI; Ong, J; Vaccher, C1
Hahner, L; Harris, RA; McQuilkin, S1
Akema, T; Kimura, F1
Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Gilbert, CD; Hirsch, JA1
Lewis, DV; Mott, DD1
Asprodini, EK; Rainnie, DG; Shinnick-Gallagher, P1
Lewis, DV; Morrisett, RA; Mott, DD; Swartzwelder, HS; Wilson, WA1
Calandra, RS; Campos, MB; Ritta, MN1
Aran, S; Hammond, DL1
Florentino, A; Kunos, G; Varga, K1
Jensen, MS; Lambert, JD; Nathan, T1
Segal, M1
Kohlenbach, A; Schlicker, E1
Collingridge, GL; Davies, CH; Davies, SN1
al-Dahan, MI; Tehrani, MH; Thalmann, RH1
Harrison, NL; Kerr, DI; Lambert, NA; Lovinger, DM; Ong, J; Prager, R; Teyler, TJ1
Harrison, NL; Kerr, DI; Lambert, NA; Ong, J; Prager, RH; Teyler, TJ1
Abbenante, J; Johnston, GA; Kerr, DI; Ong, J; Prager, RH2
Beattie, DT; Curtis, DR; Gynther, BD; Kerr, DI; Prager, RH1
Herrero, JF1
Gustafsson, B; Karpefors, M; Wigström, H; Xiao, MY1
Ishibashi, Y; Nakagawa, Y; Tagashira, E; Yoshii, T1
Kodsi, MH; Swerdlow, NR1
Humeniuk, RE; Kerr, DI; Ong, J; White, JM1
Hirota, A; Kamino, K; Momose-Sato, Y; Sakai, T; Sato, K1
Anderson, DR; Martin, LP; Tepper, JM1
Ashe, JH; Metherate, R1
Caddick, SJ; Chad, JE; Stanford, IM1
Humeniuk, RE; Kerr, DI; Ong, J1
Goudreau, JL; Lookingland, KJ; Moore, KE; Wagner, EJ1
Slaughter, MM; Tian, N1
Piguet, P1
Finch, DM; Gigg, J; Tan, AM1
Ebner, FF; Friedberg, MH; Lee, SM1
Michelson, HB; Wong, RK1
Crunelli, V; Emri, Z; Juhász, G; Kékesi, KA; Salfay, O1
Bekenstein, JW; Lothman, EW1
Lacaille, JC; Vachon, P; Williams, S1
Lewis, DV; Mott, DD; Swartzwelder, HS; Wilson, WA; Xie, CW1
Jefferys, JG; Watts, AE; Whittington, MA1
Lacaille, JC; Samulack, DD1
Pitzer, MR; Stratford, TR; Wirtshafter, D1
Avanzino, GL; Blanchi, D; Cogo, CE; Ermirio, R; Ruggeri, P; Weaver, LC1
Anderson, JJ; Chase, TN; Engber, TM; Kuo, S1
Capek, R; Esplin, B1
De Koning, HP; Jenks, BG; Roubos, EW1
Gayet, J; Ginefri-Gayet, M1
Mayfield, RD; Zahniser, NR1
Bal, T; McCormick, DA; von Krosigk, M1
Higgins, MJ; Stone, TW1
Morrisett, RA; Swartzwelder, HS1
Fischer, Y; Parnas, I1
Doolette, DJ; Kerr, DI; Ong, J; Prager, RH; Schafer, K1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Komatsu, Y1
Snead, OC1
Crunelli, V; Dobolyi, A; Emri, Z; Juhász, G; Kékesi, KA; Nyitrai, G1
Ikeda, Y; Katsuki, H; Nishiyama, N; Saito, H1
Bowery, NG; Connelly, ST; daSilva, HM; Grobaski, KC; Ping, H; Shepard, PD1
Schulz, PE1
Matsumoto, K; Nguyen, TT; Watanabe, H1
Katz, LC; Roerig, B1
Batini, C; Vigot, R1
Chub, N; O'Donovan, MJ1
Izumi, F; Shibuya, I; Toyohira, Y; Ueda, Y; Ueno, S; Uezono, Y; Yamashita, H; Yanagihara, N1
Błaszczyk, M; Eckersdorf, B; Gołebiewski, H; Grabowski, R; Konopacki, J1
Funahashi, M; Stewart, M1
Ferreira, SA; Hileman, SM; Jackson, GL; Kuehl, DE1
Akihara, M; Izumi, F; Kaibara, M; Kawano, C; Shibuya, I; Taniyama, K; Toyohira, Y; Ueda, Y; Uezono, Y; Yamashita, H; Yanagihara, N1
Kremer, E; Lev-Tov, A1
Stein, EA; Xi, ZX2
Dun, NJ; Lin, HH1
Jefferys, JG; Traub, RD1
Choi, IG; Huh, SO; Ihn, BM; Jung, JS; Kim, YH; Song, DK; Suh, HW1
Ballanyi, K; Brockhaus, J1
Chitravanshi, VC; Sapru, HN1
Bunnett, NW; Grady, EF; Marvizón, JC; Mayer, EA; Stefani, E1
Kerr, DI; Ong, J; Parnas, I; Rashkovan, G1
Browning, DA; Ferreira, SA; Jackson, GL; Kuehl, DE; Scott, CJ1
Paladini, CA; Tepper, JM1
Adanina, V; Batueva, I; Buchanan, JT; Reperant, J; Rio, JP; Sagatelyan, A; Suderevskaya, E; Tsvetkov, E; Vesselkin, N1
Fuchs, JL; Ilyinsky, OB; Schwark, HD; Tennison, CF1
Obrietan, K; van den Pol, AN1
Chiang, CY; Hu, JW; Kwan, CL; Sessle, BJ1
Chen, CL; Chiu, TH; Yang, YR1
Bieger, D; Dong, H; Loomis, CW1
Coderre, E; Cui, LN; Renaud, LP1
Kolaj, M; Renaud, LP; Yang, CR1
Fischer, Y; Parnas, I; Rashkovan, G; Ravin, R1
Remmers, JE; Straus, C; Wilson, RJ1
Kulinskii, VI; Mikhel'son, GV1
Duffy, P; Jackson, D; Kalivas, PW; Romanidies, A; Wyndham, L1
Cupello, A; Scarrone, S1
Kudoh, M; Seki, K; Shibuki, K1
Akerman, S; Goadsby, PJ; Storer, RJ1
Guido, W; Lo, FS; Ziburkus, J1
Li, ZW; Wei, JB; Yang, Q1
Balerio, GN; Rubio, MC1
Abraini, JH; Balon, N; Kriem, B; Risso, JJ; Rostain, JC1
Lisman, JE; Otmakhova, NA1
Martinez, V; Piqueras, L1
Ikemoto, S1
Henderson, Z; Jones, GA1
Beverly, JL; Doane, DF; Kotz, CM; Sweet, DC; Thorpe, AJ1
Chang, FC; Chen, YC; Tsai, CH; Yi, PL1
Bocian, R; Konopacki, J1
Backes, EN; Hemby, SE1
Gardner, EL; Li, X; Xi, ZX1
Aono, Y; Cools, AR; Iwakami, T; Koshikawa, N; Mizoguchi, N; Oi, Y; Saigusa, T; Takada, K; Ueda, K1
Gjoni, T; Urwyler, S1
Cedillo, LN; Jiménez, JC; Millán-Mejía, P; Miranda, F; Sánchez-Castillo, H; Sandoval-Sánchez, A; Velázquez-Martínez, DN1
Bonaventura, MM; Crivello, M; Cymeryng, C; Ferreira, ML; Libertun, C; Lux-Lantos, VA; Repetto, M1
Balerio, GN; Varani, AP1
Hanafusa, N; Kawasaki, H; Okamoto, K; Takatori, S1
Bocian, R; Caban, B; Konopacki, J; Kowalczyk, T1
Callera, JC; De Oliveira, LB; Kimura, EH; Menani, JV1
Kazmierska, P; Konopacki, J1
Balerio, GN; Bettler, B; Pedrón, VT; Varani, AP1
Aso, E; Balerio, GN; Maldonado, R; Varani, AP1
Budefeld, T; Carbone, D; Eitel, C; Handa, RJ; Majdic, G; Nash, C; Searcy, BT; Staros, M; Stratton, MS; Tobet, SA1
Baker, DA; Blacktop, JM; Mantsch, JR; Mayer, M; Van Hoof, M; Vranjkovic, O1
Chang, S; Choi, KH; Gwak, YS; Jang, EY; Jin, W; Kim, HY; Kim, JH; Kim, MS; Koo, H; Lee, BH; Lee, JG; Lee, JY; Ryu, YH; Steffensen, SC; Yang, CH; Yoon, SS1
Aono, Y; Ishikawa, M; Kuboyama, N; Saigusa, T; Waddington, JL; Watanabe, Y1
Kovaleva, TE; Vedyasova, OA1
Cao, K; Liang, H; Luo, W; Tan, D; Tan, Y; Tian, N; Wang, X; Zhang, Q1
Bailey, BJ; Broxmeyer, HE; Cooper, SH; Cox, BJ; Elujoba-Bridenstine, A; Pajcini, KV; Pollok, KE; Sanchez, LM; Shao, L; Sims, EC; Sinn, AL; Tamplin, OJ; Zink, KE1

Other Studies

140 other study(ies) available for 2-hydroxysaclofen and baclofen

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Inhibitory role of gamma-amino-butyric acid in the rabbit urinary bladder.
    British journal of urology, 1992, Volume: 69, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Carbachol; Depression, Chemical; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Muscimol; Muscle Contraction; Rabbits; Receptors, GABA-A; Urinary Bladder

1992
The role of GABAA and GABAB receptors in presynaptic inhibition of Ia EPSPs in cat spinal motoneurones.
    The Journal of physiology, 1992, Volume: 447

    Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; Membrane Potentials; Motor Neurons; Receptors, GABA-A; Receptors, Neurotransmitter; Spinal Cord

1992
The actions of 3-aminopropanephosphinic acid at GABAB receptors in rat hippocampus.
    European journal of pharmacology, 1992, Feb-18, Volume: 211, Issue:3

    Topics: Action Potentials; Aging; Animals; Baclofen; GABA Antagonists; Hippocampus; Membrane Potentials; Organophosphorus Compounds; Rats; Receptors, GABA-A; Synapses; Synaptic Transmission

1992
Peripheral 2-hydroxy-saclofen-sensitive GABA-B receptors mediate both vagal-dependent and vagal-independent acid secretory responses in rats.
    Journal of autonomic pharmacology, 1992, Volume: 12, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Electric Stimulation; Gastric Acid; Gastric Mucosa; Male; Perfusion; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vagotomy; Vagus Nerve

1992
The role of GABAB receptor activation in absence seizures of lethargic (lh/lh) mice.
    Science (New York, N.Y.), 1992, Jul-17, Volume: 257, Issue:5068

    Topics: Animals; Anticonvulsants; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; Electroencephalography; Electrophysiology; Epilepsy, Absence; Hippocampus; In Vitro Techniques; Mice; Mice, Inbred Strains; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate

1992
Effectiveness of GABAB antagonists in inhibiting baclofen-induced reductions in cytosolic free Ca concentration in isolated melanotrophs of rat.
    British journal of pharmacology, 1992, Volume: 105, Issue:4

    Topics: Animals; Baclofen; Calcium; Cytosol; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Organophosphorus Compounds; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains

1992
Inhibition of baroreflex bradycardia by ethanol involves both GABAA and GABAB receptors in the brainstem of the rat.
    European journal of pharmacology, 1992, Apr-22, Volume: 214, Issue:2-3

    Topics: 3-Mercaptopropionic Acid; Animals; Baclofen; Bradycardia; Brain Stem; Electric Stimulation; Ethanol; Male; Pressoreceptors; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reflex; Vagus Nerve

1992
The action of GABAB antagonists in the trigeminal nucleus of the rat.
    Neuropharmacology, 1992, Volume: 31, Issue:5

    Topics: Animals; Baclofen; GABA-A Receptor Antagonists; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Trigeminal Nuclei

1992
The role of GABA receptors in the control of nigrostriatal dopaminergic neurons: dual-probe microdialysis study in awake rats.
    European journal of pharmacology, 1992, Aug-25, Volume: 219, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Acrylates; Animals; Baclofen; Bicuculline; Corpus Striatum; Dendrites; Dopamine; Male; Muscimol; Neurons; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Substantia Nigra

1992
Differing actions of beta-(2-thienyl)-gamma-aminobutyric acid in central and peripheral preparations.
    European journal of pharmacology, 1992, Oct-06, Volume: 221, Issue:1

    Topics: Animals; Baclofen; Brain; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Receptors, GABA-A; Structure-Activity Relationship; Thiophenes

1992
Cerebellar GABAB receptors modulate function of GABAA receptors.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1991, Volume: 5, Issue:10

    Topics: Animals; Baclofen; Barium; Calcium; Cells, Cultured; Cerebellum; Cerebral Cortex; Chlorine; Dose-Response Relationship, Drug; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Mice; Mice, Inbred ICR; Muscimol; Pyrrolidinones; Receptors, GABA-A; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Type C Phospholipases

1991
2-Hydroxysaclofen, a potent GABAB receptor antagonist, stimulates luteinizing hormone secretion in female rats.
    Brain research, 1991, Apr-12, Volume: 546, Issue:1

    Topics: Animals; Baclofen; Estrogens; Female; GABA-A Receptor Antagonists; Injections, Intraventricular; Luteinizing Hormone; Ovariectomy; Rats; Rats, Inbred Strains; Stimulation, Chemical

1991
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle-relaxant effect induced by baclofen.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Analgesics; Animals; Baclofen; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Morphine; Muscle Relaxation; Muscles; Organophosphorus Compounds; Oxotremorine; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time

1991
Synaptic physiology of horizontal connections in the cat's visual cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Bicuculline; Cats; Electric Stimulation; Electrophysiology; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Lidocaine; Receptors, GABA-A; Synapses; Visual Cortex

1991
Facilitation of the induction of long-term potentiation by GABAB receptors.
    Science (New York, N.Y.), 1991, Jun-21, Volume: 252, Issue:5013

    Topics: 2-Amino-5-phosphonovalerate; Baclofen; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Learning; Membrane Potentials; Neural Inhibition; Neuronal Plasticity; Receptors, GABA-A

1991
Studies on pituitary melanotrophs reveal the novel GABAB antagonist CGP 35-348 to be the first such compound effective on endocrine cells.
    Proceedings. Biological sciences, 1991, Feb-22, Volume: 243, Issue:1307

    Topics: Animals; Baclofen; Bicuculline; Darkness; GABA Antagonists; GABA-A Receptor Antagonists; Kinetics; Male; Melanocyte-Stimulating Hormones; Methionine; Muscimol; Organophosphorus Compounds; Pituitary Gland; Rats; Rats, Inbred Strains; Xenopus laevis

1991
Inhibitory transmission in the basolateral amygdala.
    Journal of neurophysiology, 1991, Volume: 66, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Evoked Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Potentials; Neural Inhibition; Pentobarbital; Potassium; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1991
GABAB-receptor-mediated inhibition of the N-methyl-D-aspartate component of synaptic transmission in the rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1991, Volume: 11, Issue:1

    Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1991
Coexistence of gamma-aminobutyric acid type A and type B receptors in testicular interstitial cells.
    Journal of neurochemistry, 1991, Volume: 56, Issue:4

    Topics: Ammonium Chloride; Animals; Baclofen; Binding Sites; Detergents; gamma-Aminobutyric Acid; Male; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Testosterone

1991
Antagonism of baclofen-induced antinociception by intrathecal administration of phaclofen or 2-hydroxy-saclofen, but not delta-aminovaleric acid in the rat.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Amino Acids; Amino Acids, Neutral; Analgesia; Animals; Baclofen; Injections, Spinal; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Mechanism of the cardiovascular effects of GABAB receptor activation in the nucleus tractus solitarii of the rat.
    Brain research, 1990, Dec-10, Volume: 535, Issue:2

    Topics: Anesthesia; Animals; Baclofen; Blood Pressure; Dizocilpine Maleate; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Male; Medulla Oblongata; Microinjections; Pertussis Toxin; Pressoreceptors; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Urethane; Virulence Factors, Bordetella

1990
GABAB receptors play a major role in paired-pulse facilitation in area CA1 of the rat hippocampus.
    Brain research, 1990, Oct-29, Volume: 531, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Electric Stimulation; Evoked Potentials; Female; Hippocampus; In Vitro Techniques; Male; Pyramidal Tracts; Quinoxalines; Rats; Receptors, GABA-A

1990
A subset of local interneurons generate slow inhibitory postsynaptic potentials in hippocampal neurons.
    Brain research, 1990, Mar-12, Volume: 511, Issue:1

    Topics: 4-Aminopyridine; Action Potentials; Animals; Baclofen; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Rats; Receptors, GABA-A

1990
GABAB receptor-mediated inhibition of the neurogenic vasopressor response in the pithed rat.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Blood Pressure; Decerebrate State; Electric Stimulation; gamma-Aminobutyric Acid; Male; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine; Tubocurarine; Vascular Resistance

1990
Paired-pulse depression of monosynaptic GABA-mediated inhibitory postsynaptic responses in rat hippocampus.
    The Journal of physiology, 1990, Volume: 424

    Topics: Action Potentials; Animals; Baclofen; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Picrotoxin; Rats; Synapses; Synaptic Transmission; Tetrodotoxin

1990
Effect of 2-hydroxy-saclofen, an antagonist of GABAB action, upon the binding of baclofen and other receptor ligands in rat cerebrum.
    Brain research, 1990, Sep-03, Volume: 526, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Baclofen; Brain; GABA Antagonists; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1990
The actions of 2-hydroxy-saclofen at presynaptic GABAB receptors in the rat hippocampus.
    Neuroscience letters, 1990, Nov-13, Volume: 119, Issue:2

    Topics: Animals; Baclofen; Electrophysiology; Hippocampus; In Vitro Techniques; Neurons; Rats; Receptors, GABA-A; Synapses

1990
Blockade of the late IPSP in rat CA1 hippocampal neurons by 2-hydroxy-saclofen.
    Neuroscience letters, 1989, Dec-15, Volume: 107, Issue:1-3

    Topics: Action Potentials; Animals; Baclofen; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Neural Inhibition; Rats; Receptors, GABA-A

1989
Antagonism at GABAB receptors by saclofen and related sulphonic analogues of baclofen and GABA.
    Neuroscience letters, 1989, Dec-15, Volume: 107, Issue:1-3

    Topics: Animals; Baclofen; Cerebral Cortex; Evoked Potentials; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Receptors, GABA-A

1989
2-Hydroxy-saclofen: an improved antagonist at central and peripheral GABAB receptors.
    Neuroscience letters, 1988, Sep-23, Volume: 92, Issue:1

    Topics: Action Potentials; Animals; Baclofen; Cerebral Cortex; Ileum; In Vitro Techniques; Male; Motor Neurons; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vas Deferens

1988
Baclofen antagonism by 2-hydroxy-saclofen in the cat spinal cord.
    Neuroscience letters, 1988, Sep-23, Volume: 92, Issue:1

    Topics: Action Potentials; Animals; Baclofen; Cats; Electric Stimulation; Interneurons; Receptors, GABA-A; Spinal Cord

1988
GABAergic activity of quisqualamine and homoquisqualamine in hemisected spinal cord in vitro preparation.
    Revista espanola de fisiologia, 1994, Volume: 50, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Bicuculline; Decarboxylation; Evoked Potentials; GABA Agonists; Magnesium; Muscimol; Picrotoxin; Quisqualic Acid; Rats; Rats, Wistar; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Tetrodotoxin

1994
On the linkage between AMPA and NMDA receptor-mediated EPSPs in homosynaptic long-term depression in the hippocampal CA1 region of young rats.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Long-Term Potentiation; N-Methylaspartate; Neuronal Plasticity; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission; Time Factors

1995
Involvement of cholinergic systems in the deficit of place learning in Morris water maze task induced by baclofen in rats.
    Brain research, 1995, Jun-19, Volume: 683, Issue:2

    Topics: Animals; Baclofen; Cholinergic Fibers; GABA Agonists; GABA-B Receptor Agonists; Male; Maze Learning; Memory; Muscarinic Agonists; Oxotremorine; Rats; Rats, Wistar; Scopolamine

1995
Ventral pallidal GABA-A receptors regulate prepulse inhibition of acoustic startle.
    Brain research, 1995, Jun-26, Volume: 684, Issue:1

    Topics: Acoustic Stimulation; Animals; Baclofen; Corpus Striatum; Globus Pallidus; Injections; Male; Neural Inhibition; Picrotoxin; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Reflex, Startle

1995
Characterization of GABAB ligands in vivo.
    General pharmacology, 1995, Volume: 26, Issue:2

    Topics: Animals; Baclofen; beta-Alanine; Drug Interactions; Female; GABA Antagonists; GABA-B Receptor Antagonists; Ligands; Mice; Mice, Inbred BALB C; Muscle Relaxation; Organophosphorus Compounds

1995
A novel gamma-aminobutyric acid response in the embryonic brainstem as revealed by voltage-sensitive dye recording.
    Neuroscience letters, 1995, May-26, Volume: 191, Issue:3

    Topics: Animals; Baclofen; Brain Stem; Chick Embryo; Coloring Agents; Electrophysiology; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Picrotoxin

1995
GABAA receptor-mediated inhibition of rat substantia nigra dopaminergic neurons by pars reticulata projection neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Dopamine; Electric Stimulation; Evoked Potentials; Globus Pallidus; Kainic Acid; Kinetics; Male; Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substantia Nigra; Superior Colliculi; Thalamus; Time Factors

1995
Facilitation of an NMDA receptor-mediated EPSP by paired-pulse stimulation in rat neocortex via depression of GABAergic IPSPs.
    The Journal of physiology, 1994, Dec-01, Volume: 481 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Auditory Cortex; Baclofen; Cerebral Cortex; Cesium; Electric Stimulation; Electrophysiology; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Thalamus

1994
2-Hydroxy-saclofen causes a phaclofen-reversible reduction in population spike amplitude in the rat hippocampal slice.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Antagonists; Hippocampus; Male; Microelectrodes; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B; Synaptic Transmission

1995
Gamma-guanidinobaclofen is a peripheral GABAB receptor agonist.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: Animals; Baclofen; Cerebral Cortex; Corpus Callosum; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Sprague-Dawley

1994
GABAergic regulation of tuberoinfundibular dopaminergic neurons in the male rat.
    Brain research, 1994, Oct-03, Volume: 659, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isonicotinic Acids; Male; Neurons; Osmolar Concentration; Prolactin; Pyridazines; Rats; Rats, Inbred Strains; Seizures

1994
Pharmacology of the GABAB receptor in amphibian retina.
    Brain research, 1994, Oct-17, Volume: 660, Issue:2

    Topics: Ambystoma; Animals; Baclofen; Butylamines; Evoked Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Necturus; Organophosphorus Compounds; Propylamines; Receptors, GABA-B; Retina; Retinal Ganglion Cells; Stereoisomerism; Structure-Activity Relationship

1994
GABAA- and GABAB-mediated inhibition in the rat dentate gyrus in vitro.
    Epilepsy research, 1993, Volume: 16, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Electric Stimulation; Epilepsy; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synapses

1993
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
    Hippocampus, 1994, Volume: 4, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus

1994
The role of GABA-mediated inhibition in the rat ventral posterior medial thalamus. II. Differential effects of GABAA and GABAB receptor antagonists on responses of VPM neurons.
    Journal of neurophysiology, 1994, Volume: 71, Issue:5

    Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Brain Mapping; Evoked Potentials, Somatosensory; Female; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Neural Inhibition; Rats; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Thalamic Nuclei; Vibrissae

1994
Synchronization of inhibitory neurones in the guinea-pig hippocampus in vitro.
    The Journal of physiology, 1994, May-15, Volume: 477, Issue:Pt 1

    Topics: 4-Aminopyridine; Animals; Baclofen; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Interneurons; Membrane Potentials; Microelectrodes; Neurons; Picrotoxin; Pyramidal Cells; Synaptic Transmission

1994
Blockade of thalamic GABAB receptors decreases EEG synchronization.
    Neuroscience letters, 1994, May-19, Volume: 172, Issue:1-2

    Topics: Animals; Baclofen; Cats; Cortical Synchronization; Electroencephalography; Electromyography; Electrooculography; GABA-B Receptor Antagonists; Microdialysis; Organophosphorus Compounds; Sleep; Thalamus; Wakefulness

1994
Dormancy of inhibitory interneurons in a model of temporal lobe epilepsy.
    Science (New York, N.Y.), 1993, Jan-01, Volume: 259, Issue:5091

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Electric Stimulation; Epilepsy, Temporal Lobe; Evoked Potentials; Hippocampus; In Vitro Techniques; Interneurons; Male; Membrane Potentials; Picrotoxin; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Status Epilepticus

1993
Monosynaptic GABA-mediated inhibitory postsynaptic potentials in CA1 pyramidal cells of hyperexcitable hippocampal slices from kainic acid-treated rats.
    Neuroscience, 1993, Volume: 52, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Evoked Potentials; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Neurons; Pyramidal Tracts; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

1993
GABAB autoreceptors mediate activity-dependent disinhibition and enhance signal transmission in the dentate gyrus.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Culture Techniques; GABA-A Receptor Antagonists; Hippocampus; Male; Membrane Potentials; Nerve Fibers; Neural Inhibition; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Theta Rhythm

1993
Epileptic focus induced in rat by intrahippocampal cholera toxin: neuronal properties in vitro.
    Neuroscience, 1993, Volume: 55, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Cholera Toxin; Chronic Disease; Epilepsy; Hippocampus; Injections; Male; Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission

1993
Hyperpolarizing synaptic potentials evoked in CA1 pyramidal cells by glutamate stimulation of interneurons from the oriens/alveus border of rat hippocampal slices. II. Sensitivity to GABA antagonists.
    Hippocampus, 1993, Volume: 3, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Electrophysiology; Evoked Potentials; GABA Antagonists; Glutamates; Glutamic Acid; Hippocampus; In Vitro Techniques; Interneurons; Neural Inhibition; Neurons; Rats; Synapses

1993
Studies on the behavioral activation produced by stimulation of GABAB receptors in the median raphe nucleus.
    Behavioural brain research, 1993, Dec-31, Volume: 59, Issue:1-2

    Topics: Animals; Baclofen; Behavior, Animal; Brain Mapping; Dopamine; Drinking; Eating; Fenclonine; Injections; Male; Motor Activity; Prosencephalon; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Serotonin; Stereoisomerism

1993
GABAB receptor-mediated mechanisms in the RVLM studied by microinjections of two GABAB receptor antagonists.
    The American journal of physiology, 1994, Volume: 266, Issue:5 Pt 2

    Topics: Animals; Baclofen; Blood Pressure; Electrocardiography; Functional Laterality; GABA-B Receptor Antagonists; Heart Rate; Homeostasis; Male; Medulla Oblongata; Microinjections; Muscimol; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B

1994
GABAA and GABAB receptors differentially regulate striatal acetylcholine release in vivo.
    Neuroscience letters, 1993, Oct-01, Volume: 160, Issue:2

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Corpus Striatum; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Kinetics; Male; Microdialysis; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Stereotaxic Techniques; Time Factors

1993
Frequency-dependent enhancement of hippocampal inhibition by GABA uptake blockers.
    Epilepsy research, 1993, Volume: 16, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Nicotinic Acids; Nipecotic Acids; Pyramidal Tracts; Rats; Rats, Sprague-Dawley; Time Factors

1993
Analysis of gamma-aminobutyric acidB receptor function in the in vitro and in vivo regulation of alpha-melanotropin-stimulating hormone secretion from melanotrope cells of Xenopus laevis.
    Endocrinology, 1993, Volume: 132, Issue:2

    Topics: alpha-MSH; Animals; Baclofen; Butylamines; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Homeostasis; In Vitro Techniques; Kinetics; Organophosphorus Compounds; Perfusion; Pituitary Gland, Posterior; Radioimmunoassay; Receptors, GABA-A; Xenopus laevis

1993
Hypothermia induced by infusion of methionine sulfoximine into the dorsal raphe nucleus of the rat: involvement of 5-HT1A and GABAB receptors.
    European journal of pharmacology, 1993, Apr-28, Volume: 235, Issue:2-3

    Topics: 4-Aminobutyrate Transaminase; Aminocaproates; Animals; Baclofen; Bicuculline; Body Temperature Regulation; Hypothermia; Infusions, Parenteral; Ketanserin; Male; Methionine Sulfoximine; Nipecotic Acids; Pindolol; Proline; Raphe Nuclei; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Vigabatrin

1993
Endogenous GABA release from rat striatal slices: effects of the GABAB receptor antagonist 2-hydroxy-saclofen.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:1

    Topics: Animals; Baclofen; Calcium; Chromatography, High Pressure Liquid; Corpus Striatum; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nipecotic Acids; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Tiagabine

1993
Cellular mechanisms of a synchronized oscillation in the thalamus.
    Science (New York, N.Y.), 1993, Jul-16, Volume: 261, Issue:5119

    Topics: Animals; Baclofen; Bicuculline; Calcium; Epilepsy, Absence; Ferrets; Geniculate Bodies; In Vitro Techniques; Membrane Potentials; Neurons; Potassium; Receptors, Amino Acid; Receptors, GABA-A; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate

1993
Bicuculline-resistant paired-pulse inhibition in the rat hippocampal slice.
    British journal of pharmacology, 1993, Volume: 109, Issue:4

    Topics: Adenosine; Animals; Baclofen; Bicuculline; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, GABA

1993
Attenuation of hippocampal long-term potentiation by ethanol: a patch-clamp analysis of glutamatergic and GABAergic mechanisms.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:5

    Topics: Animals; Baclofen; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Glutamine; Granulocytes; Hippocampus; Male; Midazolam; Neuronal Plasticity; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses

1993
Activation of GABAB receptors at individual release boutons of the crayfish opener neuromuscular junction produces presynaptic inhibition.
    Journal of neurophysiology, 1996, Volume: 75, Issue:4

    Topics: Animals; Astacoidea; Baclofen; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neural Conduction; Neural Inhibition; Neuromuscular Junction; Picrotoxin; Presynaptic Terminals

1996
The (S)-enantiomer of 2-hydroxysaclofen is the active GABAB receptor antagonist in central and peripheral preparations.
    European journal of pharmacology, 1995, Dec-12, Volume: 287, Issue:2

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Guinea Pigs; Hippocampus; Ileum; Male; Membrane Potentials; Muscle Contraction; Rats; Rats, Sprague-Dawley; Receptors, GABA-B

1995
Role of peripheral GABAB receptors in the regulation of pepsinogen secretion in anaesthetized rats.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Anesthesia; Animals; Baclofen; Capsaicin; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gastric Mucosa; Male; Organophosphorus Compounds; p-Methoxy-N-methylphenethylamine; Pepsinogens; Perfusion; Rats; Rats, Wistar; Receptors, GABA-B; Vagotomy

1995
GABAB receptors, monoamine receptors, and postsynaptic inositol trisphosphate-induced Ca2+ release are involved in the induction of long-term potentiation at visual cortical inhibitory synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Oct-15, Volume: 16, Issue:20

    Topics: Animals; Baclofen; Calcium; Dose-Response Relationship, Drug; GABA Antagonists; Inositol 1,4,5-Trisphosphate; Long-Term Potentiation; Rats; Rats, Sprague-Dawley; Receptors, Amino Acid; Receptors, GABA-B; Synapses; Time Factors; Visual Cortex

1996
Antiabsence seizure activity of specific GABAB and gamma-Hydroxybutyric acid receptor antagonists.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:1

    Topics: Animals; Anticonvulsants; Baclofen; Benzocycloheptenes; Electroencephalography; Epilepsy, Absence; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Injections, Intraventricular; Isomerism; Male; Pentylenetetrazole; Rats; Rats, Sprague-Dawley

1996
In vivo blockade of thalamic GABA(B) receptors increases excitatory amino-acid levels.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: Animals; Aspartic Acid; Baclofen; GABA-B Receptor Antagonists; Glutamic Acid; Male; Microdialysis; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Taurine; Thalamus

1996
GABAA receptor stimulation promotes survival of embryonic rat striatal neurons in culture.
    Brain research. Developmental brain research, 1997, Feb-20, Volume: 98, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Calcium Channel Blockers; Cell Survival; Cells, Cultured; Corpus Striatum; Embryo, Mammalian; GABA Antagonists; Neurons; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Stimulation, Chemical

1997
Responses of rat substantia nigra dopamine-containing neurones to (-)-HA-966 in vitro.
    British journal of pharmacology, 1997, Volume: 120, Issue:4

    Topics: Animals; Baclofen; Dopamine; Electrophysiology; Excitatory Amino Acid Agonists; GABA Agonists; Male; Neurons; Organophosphorus Compounds; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Substantia Nigra

1997
Long-term potentiation involves increases in the probability of neurotransmitter release.
    Proceedings of the National Academy of Sciences of the United States of America, 1997, May-27, Volume: 94, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Cadmium Chloride; Calcium Channel Blockers; Evoked Potentials; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Neurotransmitter Agents; omega-Conotoxin GVIA; Peptides; Probability; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission; Time Factors

1997
Involvement of supraspinal GABA-ergic systems in clonidine-induced antinociception in the tail-pinch test in mice.
    Life sciences, 1997, Volume: 61, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Analgesics; Animals; Baclofen; Bicuculline; Clonidine; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Pain; Picrotoxin; Receptors, GABA; Tail

1997
Modulation of intrinsic circuits by serotonin 5-HT3 receptors in developing ferret visual cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Ferrets; gamma-Aminobutyric Acid; Indoles; Ligands; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Pyridinium Compounds; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Tropisetron; Virulence Factors, Bordetella; Visual Cortex

1997
GABA(B) receptor activation of Purkinje cells in cerebellar slices.
    Neuroscience research, 1997, Volume: 29, Issue:2

    Topics: Animals; Baclofen; Cerebellum; Dose-Response Relationship, Drug; Electric Conductivity; Female; GABA Agonists; GABA Antagonists; In Vitro Techniques; Male; Neural Inhibition; Phosphinic Acids; Potassium; Propanolamines; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synapses

1997
Blockade and recovery of spontaneous rhythmic activity after application of neurotransmitter antagonists to spinal networks of the chick embryo.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jan-01, Volume: 18, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Chick Embryo; Cholinergic Antagonists; Dihydro-beta-Erythroidine; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glycine; Glycine Agents; Mecamylamine; Motor Neurons; Neuronal Plasticity; Neurotransmitter Agents; Nicotinic Antagonists; Periodicity; Spinal Cord; Strychnine

1998
Enhancement by baclofen of the Gs-coupled receptor-mediated cAMP production in Xenopus oocytes expressing rat brain cortex poly (A)+ RNA: a role of G-protein beta gamma subunits.
    Biochemical and biophysical research communications, 1997, Dec-18, Volume: 241, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Baclofen; Cerebral Cortex; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; GABA Agonists; GABA Antagonists; Genes, Reporter; GTP-Binding Protein alpha Subunits, Gs; Isoproterenol; Oocytes; Rats; Receptors, GABA-B; RNA, Messenger; Vasoactive Intestinal Peptide; Xenopus

1997
Theta-like activity in hippocampal formation slices: the effect of strong disinhibition of GABAA and GABAB receptors.
    Brain research, 1997, Nov-14, Volume: 775, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Carbachol; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Muscarinic Agonists; Neurons; Rats; Rats, Wistar; Receptors, Muscarinic; Theta Rhythm

1997
GABA receptor-mediated post-synaptic potentials in the retrohippocampal cortices: regional, laminar and cellular comparisons.
    Brain research, 1998, Mar-16, Volume: 787, Issue:1

    Topics: Animals; Baclofen; Electric Stimulation; Entorhinal Cortex; Evoked Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Neural Inhibition; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA

1998
Effects of dialyzing gamma-aminobutyric acid receptor antagonists into the medial preoptic and arcuate ventromedial region on luteinizing hormone release in male sheep.
    Biology of reproduction, 1998, Volume: 58, Issue:4

    Topics: Animals; Arcuate Nucleus of Hypothalamus; Baclofen; Bicuculline; GABA Antagonists; Luteinizing Hormone; Male; Microdialysis; Orchiectomy; Phosphinic Acids; Preoptic Area; Propanolamines; Receptors, GABA; Sheep; Testosterone

1998
Activation of inwardly rectifying K+ channels by GABA-B receptors expressed in Xenopus oocytes.
    Neuroreport, 1998, Mar-09, Volume: 9, Issue:4

    Topics: Animals; Baclofen; Cerebellum; Female; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Antagonists; GTP-Binding Proteins; Membrane Potentials; Muscimol; Oocytes; Organophosphorus Compounds; Patch-Clamp Techniques; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Receptors, GABA-B; Recombinant Proteins; Xenopus laevis

1998
GABA-receptor-independent dorsal root afferents depolarization in the neonatal rat spinal cord.
    Journal of neurophysiology, 1998, Volume: 79, Issue:5

    Topics: Action Potentials; Afferent Pathways; Amino Acids, Dicarboxylic; Aminobutyrates; Animals; Animals, Newborn; Baclofen; Bicuculline; Excitatory Amino Acid Antagonists; GABA Agonists; Ganglia, Spinal; Glycine Agents; Ion Transport; Isethionic Acid; Methysergide; N-Methylaspartate; Neurons, Afferent; Potassium; Rats; Receptors, GABA; Receptors, Glutamate; Serotonin; Serotonin Antagonists; Spinal Cord; Strychnine; Synaptic Transmission

1998
Nucleus accumbens dopamine release modulation by mesolimbic GABAA receptors-an in vivo electrochemical study.
    Brain research, 1998, Jul-06, Volume: 798, Issue:1-2

    Topics: Animals; Baclofen; Dopamine; Electrochemistry; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; Limbic System; Male; Muscimol; Nucleus Accumbens; Rats; Rats, Inbred Strains; Receptors, GABA-A; Self Administration

1998
Post- and presynaptic GABA(B) receptor activation in neonatal rat rostral ventrolateral medulla neurons in vitro.
    Neuroscience, 1998, Volume: 86, Issue:1

    Topics: Animals; Animals, Newborn; Baclofen; Calcium; Chelating Agents; Egtazic Acid; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; Guanosine Diphosphate; In Vitro Techniques; Medulla Oblongata; Neurons; Organophosphorus Compounds; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Tetraethylammonium; Tetrodotoxin; Thionucleotides

1998
'Dormant' inhibitory neurons: do they exist and what is their functional impact?
    Epilepsy research, 1998, Volume: 32, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Computer Simulation; Epilepsy; GABA Antagonists; Hippocampus; In Vitro Techniques; Interneurons; Male; Models, Neurological; Neurons; Pyramidal Cells; Rats; Tetanus Toxin

1998
Central GABAA and GABAB receptor modulation of basal and stress-induced plasma interleukin-6 levels in mice.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:1

    Topics: Animals; Baclofen; Brain; Dizocilpine Maleate; GABA Modulators; Injections, Intraventricular; Interleukin-6; Male; Mice; Mice, Inbred ICR; Muscimol; Oxidopamine; Pyridazines; Receptors, GABA-A; Receptors, GABA-B; Stress, Physiological

1998
Synaptic inhibition in the isolated respiratory network of neonatal rats.
    The European journal of neuroscience, 1998, Volume: 10, Issue:12

    Topics: Action Potentials; Animals; Animals, Newborn; Anti-Bacterial Agents; Baclofen; Bicarbonates; Bicuculline; Carbon Dioxide; Chloride Channel Agonists; Chloride Channels; Chlorides; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine Agents; Gramicidin; Medulla Oblongata; Microdialysis; Muscimol; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Receptors, GABA-B; Respiration; Strychnine; Synapses; Tetrodotoxin

1998
GABA receptors in the phrenic nucleus of the rat.
    The American journal of physiology, 1999, Volume: 276, Issue:2

    Topics: Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; Male; Microinjections; Muscimol; Neurons; Phrenic Nerve; Rats; Rats, Wistar; Receptors, GABA; Spinal Cord

1999
Substance P release in the dorsal horn assessed by receptor internalization: NMDA receptors counteract a tonic inhibition by GABA(B) receptors.
    The European journal of neuroscience, 1999, Volume: 11, Issue:2

    Topics: Animals; Baclofen; Dizocilpine Maleate; Down-Regulation; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Muscimol; Neural Inhibition; Organ Culture Techniques; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Substance P

1999
Tonic activation of presynaptic GABAB receptors in the opener neuromuscular junction of crayfish.
    Journal of neurophysiology, 1999, Volume: 81, Issue:3

    Topics: Animals; Astacoidea; Axons; Baclofen; GABA Agonists; GABA Antagonists; Logistic Models; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Pronase; Quantum Theory; Receptors, GABA-B; Receptors, Presynaptic

1999
Effect of infusing gamma-aminobutyric acid receptor agonists and antagonists into the medial preoptic area and ventromedial hypothalamus on prolactin secretion in male sheep.
    Endocrine, 1998, Volume: 9, Issue:3

    Topics: Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; Male; Muscimol; Phosphinic Acids; Preoptic Area; Prolactin; Propanolamines; Sheep; Ventromedial Hypothalamic Nucleus

1998
GABA(A) and GABA(B) antagonists differentially affect the firing pattern of substantia nigra dopaminergic neurons in vivo.
    Synapse (New York, N.Y.), 1999, Jun-01, Volume: 32, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Bicuculline; Dopamine; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Kinetics; Male; Neurons; Phosphinic Acids; Picrotoxin; Propanolamines; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Substantia Nigra

1999
Physiological and morphological correlates of presynaptic inhibition in primary afferents of the lamprey spinal cord.
    Neuroscience, 1999, Volume: 88, Issue:3

    Topics: Afferent Pathways; Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Barium; Cadmium; Calcium Channels; Cell Membrane; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Lampreys; Membrane Potentials; Motor Neurons; Nerve Fibers; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Presynaptic Terminals; Species Specificity; Spinal Cord; Synapses

1999
Inhibitory influences on receptive field size in the dorsal column nuclei.
    Experimental brain research, 1999, Volume: 126, Issue:3

    Topics: Animals; Baclofen; Bicuculline; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Male; Neural Inhibition; Neurons; Rats; Rats, Sprague-Dawley; Spinal Cord

1999
GABAB receptor-mediated regulation of glutamate-activated calcium transients in hypothalamic and cortical neuron development.
    Journal of neurophysiology, 1999, Volume: 82, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Baclofen; Bicuculline; Calcium; Cells, Cultured; Cerebral Cortex; Cytarabine; Drug Synergism; Embryo, Mammalian; Excitatory Amino Acid Antagonists; GABA Antagonists; Glutamic Acid; Hypothalamus, Middle; Membrane Potentials; Neurons; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Tetrodotoxin; Virulence Factors, Bordetella

1999
Effects of GABA receptor antagonist on trigeminal caudalis nociceptive neurons in normal and neonatally capsaicin-treated rats.
    Journal of neurophysiology, 1999, Volume: 82, Issue:5

    Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Brain Mapping; Capsaicin; Functional Laterality; GABA Antagonists; GABA-A Receptor Antagonists; Male; Medulla Oblongata; Microinjections; Neuronal Plasticity; Neurons; Nociceptors; Pain; Physical Stimulation; Rats; Rats, Sprague-Dawley; Touch; Trigeminal Nerve

1999
Activation of rat locus coeruleus neuron GABA(A) receptors by propofol and its potentiation by pentobarbital or alphaxalone.
    European journal of pharmacology, 1999, Dec-15, Volume: 386, Issue:2-3

    Topics: Anesthetics; Anesthetics, Intravenous; Animals; Baclofen; Barium Compounds; Bicuculline; Chlorides; Diazepam; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Ionophores; Locus Coeruleus; Male; Neurons; Pentobarbital; Picrotoxin; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zinc Compounds

1999
Distal and deglutitive inhibition in the rat esophagus: role of inhibitory neurotransmission in the nucleus tractus solitarii.
    Gastroenterology, 2000, Volume: 118, Issue:2

    Topics: Animals; Baclofen; Bicuculline; Deglutition; Esophagus; GABA-A Receptor Antagonists; Male; Models, Biological; Muscle, Smooth; Propylamines; Rats; Rats, Sprague-Dawley; Solitary Nucleus; Strychnine; Synaptic Transmission

2000
GABA(B) presynaptically modulates suprachiasmatic input to hypothalamic paraventricular magnocellular neurons.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2000, Volume: 278, Issue:5

    Topics: Animals; Baclofen; Electric Conductivity; Electric Stimulation; Ethylmaleimide; GABA Agonists; GABA Antagonists; In Vitro Techniques; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Pertussis Toxin; Rats; Rats, Long-Evans; Receptors, GABA-A; Receptors, GABA-B; Suprachiasmatic Nucleus; Synapses; Virulence Factors, Bordetella

2000
Presynaptic GABA(B) receptors modulate organum vasculosum lamina terminalis-evoked postsynaptic currents in rat hypothalamic supraoptic neurons.
    Neuroscience, 2000, Volume: 98, Issue:1

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; In Vitro Techniques; Male; Patch-Clamp Techniques; Presynaptic Terminals; Rats; Rats, Long-Evans; Receptors, GABA-B; Supraoptic Nucleus; Water-Electrolyte Balance

2000
Increased mesolimbic GABA concentration blocks heroin self-administration in the rat.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Animals; Baclofen; Behavior, Animal; Bicuculline; Enzyme Inhibitors; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Heroin; Injections, Intraventricular; Lateral Ventricles; Male; Microinjections; Narcotics; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Opioid-Related Disorders; Rats; Rats, Sprague-Dawley; Self Administration; Telencephalon; Ventral Tegmental Area; Vigabatrin

2000
Novel mechanism for presynaptic inhibition: GABA(A) receptors affect the release machinery.
    Journal of neurophysiology, 2000, Volume: 84, Issue:3

    Topics: Action Potentials; Animals; Astacoidea; Baclofen; Calcium; Dose-Response Relationship, Drug; Electric Stimulation; Fura-2; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Intracellular Fluid; Magnesium; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; Picrotoxin; Presynaptic Terminals; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Temperature

2000
Developmental disinhibition: turning off inhibition turns on breathing in vertebrates.
    Journal of neurobiology, 2000, Nov-05, Volume: 45, Issue:2

    Topics: Action Potentials; Aging; Animals; Baclofen; Brain Stem; Efferent Pathways; GABA Antagonists; Metamorphosis, Biological; Nerve Net; Neural Inhibition; Neurons; Rana catesbeiana; Receptors, GABA-B; Respiration; Respiratory Physiological Phenomena; Respiratory System

2000
Additivity and independence of neuroprotective effects of GABAA and GABAB receptor agonists in complete global cerebral ischemia.
    Bulletin of experimental biology and medicine, 2000, Volume: 130, Issue:8

    Topics: Animals; Baclofen; Bicuculline; Brain Ischemia; Drug Interactions; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoxazoles; Male; Mice; Mice, Inbred CBA; Muscimol; Neuroprotective Agents; Picrotoxin

2000
Involvement of pallidothalamic circuitry in working memory.
    Neuroscience, 2001, Volume: 104, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analgesics, Opioid; Animals; Baclofen; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Agonists; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Maze Learning; Mediodorsal Thalamic Nucleus; Memory, Short-Term; Motor Activity; Neural Inhibition; Neural Pathways; Neurons; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, GABA-B; Receptors, Opioid, mu

2001
Pretreatment of rat brain synaptosomes with GABA increases subsequent GABA uptake via GABA(B) receptor activation.
    Neurochemical research, 2001, Volume: 26, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Baclofen; Brain; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Synaptosomes; Up-Regulation

2001
Sequence dependence of post-tetanic potentiation after sequential heterosynaptic stimulation in the rat auditory cortex.
    The Journal of physiology, 2001, Jun-01, Volume: 533, Issue:Pt 2

    Topics: Animals; Auditory Cortex; Baclofen; Bicuculline; Calcium; Electric Stimulation; Excitatory Postsynaptic Potentials; Female; Fluorescent Dyes; GABA Antagonists; Heterocyclic Compounds, 3-Ring; Long-Term Potentiation; Male; Organ Culture Techniques; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Wistar; Synapses

2001
GABA receptors modulate trigeminovascular nociceptive neurotransmission in the trigeminocervical complex.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Muscimol; Neurons; Nociceptors; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors; Trigeminal Nuclei

2001
Synaptic mechanisms regulating the activation of a Ca(2+)-mediated plateau potential in developing relay cells of the LGN.
    Journal of neurophysiology, 2002, Volume: 87, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Baclofen; Bicuculline; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Geniculate Bodies; Neurons; Nitrendipine; Rats; Rats, Sprague-Dawley; Receptors, GABA; Synapses

2002
[Current responses mediated by endogenous GABA(B) and GABA(C) receptors in Xenopus oocytes].
    Sheng li xue bao : [Acta physiologica Sinica], 2001, Volume: 53, Issue:4

    Topics: Animals; Baclofen; Female; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Receptors, GABA; Receptors, GABA-B; Xenopus

2001
Baclofen analgesia: involvement of the GABAergic system.
    Pharmacological research, 2002, Volume: 46, Issue:3

    Topics: Analgesics; Animals; Baclofen; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; Injections, Intraperitoneal; Male; Mice; Muscle Relaxation; Receptors, GABA

2002
Gamma-aminobutyric acid neuropharmacological investigations on narcosis produced by nitrogen, argon, or nitrous oxide.
    Anesthesia and analgesia, 2003, Volume: 96, Issue:3

    Topics: Anesthesia, Inhalation; Animals; Argon; Baclofen; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Motor Activity; Nitrogen; Nitrous Oxide; Pyridazines; Rats; Rats, Sprague-Dawley

2003
Contribution of Ih and GABAB to synaptically induced afterhyperpolarizations in CA1: a brake on the NMDA response.
    Journal of neurophysiology, 2004, Volume: 92, Issue:4

    Topics: Animals; Baclofen; Calcium; Electrophysiology; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Ion Channels; Patch-Clamp Techniques; Perforant Pathway; Picrotoxin; Potassium Channel Blockers; Potassium Channels; Pyrimidines; Rats; Rats, Long-Evans; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Synapses

2004
Peripheral GABAB agonists stimulate gastric acid secretion in mice.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Animals; Antibodies, Monoclonal; Atropine; Baclofen; Deoxyglucose; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Gastric Acid; Gastrins; Imidazoles; Injections, Intravenous; Male; Mice; Mice, Knockout; Muscimol; Organophosphorus Compounds; Pentagastrin; Peptides, Cyclic; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Somatostatin; Somatostatin; Time Factors; Vagotomy

2004
The supramammillary nucleus mediates primary reinforcement via GABA(A) receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:6

    Topics: Animals; Baclofen; Benzazepines; Bicuculline; Discrimination, Psychological; Dopamine Antagonists; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; Male; Mammillary Bodies; Microinjections; Muscimol; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Reinforcement, Psychology; Reward; Self Administration

2005
GABAB receptors in the medial septum/diagonal band slice from 16-25 day rat.
    Neuroscience, 2005, Volume: 132, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Baclofen; Bicuculline; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; In Vitro Techniques; Kainic Acid; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-A; Septum Pellucidum; Sodium Channel Blockers; Tetrodotoxin; Time Factors; Valine

2005
Orexin A in the rostrolateral hypothalamic area induces feeding by modulating GABAergic transmission.
    Brain research, 2006, Dec-13, Volume: 1125, Issue:1

    Topics: Analysis of Variance; Animals; Baclofen; Behavior, Animal; Bicuculline; Dose-Response Relationship, Drug; Drug Interactions; Eating; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamic Area, Lateral; Intracellular Signaling Peptides and Proteins; Male; Microdialysis; Muscimol; Neuropeptides; Orexins; Rats; Rats, Sprague-Dawley; Time Factors

2006
Gamma-aminobutyric acid (GABA) receptor mediates suanzaorentang, a traditional Chinese herb remedy, -induced sleep alteration.
    Journal of biomedical science, 2007, Volume: 14, Issue:2

    Topics: Administration, Oral; Animals; Baclofen; Bicuculline; Drugs, Chinese Herbal; GABA Antagonists; Male; Plant Extracts; Rats; Rats, Sprague-Dawley; Receptors, GABA; Sleep Stages; Starch

2007
Posterior hypothalamic GABAergic mediation of hippocampal theta in the cat.
    Brain research bulletin, 2007, Jul-12, Volume: 73, Issue:4-6

    Topics: Animals; Baclofen; Bicuculline; Cats; Electroencephalography; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus, Posterior; Muscimol; Rats; Theta Rhythm

2007
Contribution of ventral tegmental GABA receptors to cocaine self-administration in rats.
    Neurochemical research, 2008, Volume: 33, Issue:3

    Topics: Animals; Baclofen; Cocaine-Related Disorders; Conditioning, Operant; Dose-Response Relationship, Drug; Food; GABA Agonists; GABA Antagonists; Immunohistochemistry; Male; Muscimol; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Reinforcement, Psychology; Self Administration; Ventral Tegmental Area

2008
The metabotropic glutamate receptor 7 (mGluR7) allosteric agonist AMN082 modulates nucleus accumbens GABA and glutamate, but not dopamine, in rats.
    Neuropharmacology, 2008, Volume: 54, Issue:3

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Baclofen; Benzhydryl Compounds; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Microdialysis; Nucleus Accumbens; Phosphoserine; Rats; Rats, Long-Evans; Tetrodotoxin

2008
Role of GABA B receptors in the endomorphin-1-, but not endomorphin-2-, induced dopamine efflux in the nucleus accumbens of freely moving rats.
    European journal of pharmacology, 2008, Mar-10, Volume: 581, Issue:3

    Topics: Analgesics, Opioid; Animals; Baclofen; Dopamine; GABA Agonists; GABA Antagonists; Male; Microdialysis; Nucleus Accumbens; Oligopeptides; Rats; Rats, Sprague-Dawley; Receptors, GABA-B

2008
Changes in the properties of allosteric and orthosteric GABAB receptor ligands after a continuous, desensitizing agonist pretreatment.
    European journal of pharmacology, 2009, Jan-28, Volume: 603, Issue:1-3

    Topics: Allosteric Regulation; Animals; Baclofen; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Cyclopentanes; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Ligands; Pyrimidines; Rats; Receptors, GABA-B

2009
The GABA-B antagonist 2-hydroxysaclofen reverses the effects of baclofen on the discriminative stimulus effects of D-amphetamine in the conditioned taste aversion procedure.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 93, Issue:1

    Topics: Animals; Baclofen; Central Nervous System Stimulants; Conditioning, Psychological; Dextroamphetamine; Discrimination, Psychological; Disease Models, Animal; GABA Antagonists; GABA-B Receptor Antagonists; Male; Rats; Rats, Wistar; Receptors, GABA-B; Substance-Related Disorders; Synaptic Transmission; Taste Perception

2009
Effects of GABAB receptor agonists and antagonists on glycemia regulation in mice.
    European journal of pharmacology, 2012, Feb-29, Volume: 677, Issue:1-3

    Topics: Animals; Baclofen; Basal Metabolism; Blood Glucose; Body Weight; Eating; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Glucose Tolerance Test; Homeostasis; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred BALB C; Protein Subunits; Receptors, GABA-B; RNA, Messenger; Time Factors

2012
GABA(B) receptors involvement in the effects induced by nicotine on anxiety-related behaviour in mice.
    Pharmacological research, 2012, Volume: 65, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Baclofen; Behavior, Animal; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Maze Learning; Mice; Motor Activity; Nicotine; Receptors, GABA-B; Tobacco Use Disorder

2012
Involvement of hypothalamic periventricular GABAergic nerves in the central pressor response to clonidine in freely-moving conscious rats.
    Journal of pharmacological sciences, 2012, Volume: 118, Issue:3

    Topics: Animals; Antihypertensive Agents; Baclofen; Bicuculline; Blood Pressure; Clonidine; Excitatory Amino Acid Antagonists; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Heart Rate; Hypothalamus; Kynurenic Acid; Male; Muscimol; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Receptors, Glutamate

2012
Theta-related gating cells in hippocampal formation: in vivo and in vitro study.
    Hippocampus, 2013, Volume: 23, Issue:1

    Topics: Anesthesia; Animals; Baclofen; Bicuculline; CA1 Region, Hippocampal; CA3 Region, Hippocampal; Carbachol; Cholinergic Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Male; Neurons; Organ Culture Techniques; Rats; Rats, Wistar; Theta Rhythm

2013
Baclofen into the lateral parabrachial nucleus induces hypertonic sodium chloride intake during cell dehydration.
    Behavioral and brain functions : BBF, 2013, May-03, Volume: 9

    Topics: Animals; Arterial Pressure; Baclofen; Dehydration; Drinking; Functional Laterality; GABA Agonists; GABA Antagonists; Heart Rate; Male; Osmolar Concentration; Pons; Rats; Rats, Wistar; Saline Solution, Hypertonic

2013
Development of NMDA-induced theta rhythm in hippocampal formation slices.
    Brain research bulletin, 2013, Volume: 98

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Bicuculline; Carbachol; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agents; Hippocampus; In Vitro Techniques; Male; Muscimol; N-Methylaspartate; Rats; Theta Rhythm; Time Factors

2013
Involvement of GABAB receptors in biochemical alterations induced by anxiety-related responses to nicotine in mice: genetic and pharmacological approaches.
    Neuropharmacology, 2014, Volume: 81

    Topics: Analysis of Variance; Animals; Anxiety; Baclofen; Disease Models, Animal; Dorsal Raphe Nucleus; Dose-Response Relationship, Drug; GABA-B Receptor Antagonists; Gene Expression Regulation; Male; Mice; Mice, Knockout; Neurotransmitter Agents; Nicotine; Nicotinic Agonists; Proto-Oncogene Proteins c-fos; Receptors, GABA-B; Septal Nuclei

2014
Baclofen and 2-hydroxysaclofen modify acute hypolocomotive and antinociceptive effects of nicotine.
    European journal of pharmacology, 2014, Sep-05, Volume: 738

    Topics: Analgesics; Animals; Baclofen; Drug Interactions; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Mice; Motor Activity; Nicotine

2014
Embryonic GABA(B) receptor blockade alters cell migration, adult hypothalamic structure, and anxiety- and depression-like behaviors sex specifically in mice.
    PloS one, 2014, Volume: 9, Issue:8

    Topics: Animals; Anxiety; Baclofen; Cell Movement; Depression; Embryo, Mammalian; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Hypothalamo-Hypophyseal System; Immobilization; Male; Maze Learning; Mice; Mice, Transgenic; Paraventricular Hypothalamic Nucleus; Phosphinic Acids; Pituitary-Adrenal System; Pregnancy; Propanolamines; Protein Subunits; Psychomotor Agitation; Receptors, GABA-B; Sex Factors; Stress, Psychological; Tissue Culture Techniques

2014
Antagonism of GABA-B but not GABA-A receptors in the VTA prevents stress- and intra-VTA CRF-induced reinstatement of extinguished cocaine seeking in rats.
    Neuropharmacology, 2016, Volume: 102

    Topics: Animals; Baclofen; Bicuculline; Cocaine; Corticotropin-Releasing Hormone; Drug-Seeking Behavior; Extinction, Psychological; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Male; Rats; Rats, Sprague-Dawley; Self Administration; Ventral Tegmental Area

2016
Acupuncture reduces relapse to cocaine-seeking behavior via activation of GABA neurons in the ventral tegmental area.
    Addiction biology, 2018, Volume: 23, Issue:1

    Topics: Acupuncture; Animals; Baclofen; Behavior, Animal; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Electrophysiological Phenomena; GABA-B Receptor Antagonists; GABAergic Neurons; gamma-Aminobutyric Acid; Locomotion; Microdialysis; Nucleus Accumbens; Rats; Ventral Tegmental Area

2018
In vivo neurochemical evidence that stimulation of accumbal GABA
    Synapse (New York, N.Y.), 2019, Volume: 73, Issue:4

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Dopamine; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Movement; Muscimol; Nucleus Accumbens; Rats; Rats, Sprague-Dawley

2019
Participation of GABA
    Bulletin of experimental biology and medicine, 2019, Volume: 168, Issue:1

    Topics: Animals; Baclofen; Electroencephalography; GABA-B Receptor Agonists; Pulmonary Ventilation; Rats; Receptors, GABA-B; Respiration; Tidal Volume

2019
GABA consumption during early pregnancy impairs endometrial receptivity and embryo development in mice.
    Journal of biochemical and molecular toxicology, 2020, Volume: 34, Issue:5

    Topics: Administration, Oral; Animals; Baclofen; Cadherins; Dose-Response Relationship, Drug; Embryo Implantation; Embryonic Development; Endometrium; Female; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Homeobox A10 Proteins; Leukemia Inhibitory Factor; Mice; Pregnancy; Signal Transduction

2020
The neurotransmitter receptor Gabbr1 regulates proliferation and function of hematopoietic stem and progenitor cells.
    Blood, 2021, 02-11, Volume: 137, Issue:6

    Topics: Animals; B-Lymphocytes; Baclofen; Bone Marrow; Bone Marrow Transplantation; Cell Division; Cell Lineage; Female; Gene Expression Regulation; Hematopoietic Stem Cells; Human Umbilical Vein Endothelial Cells; Humans; Lymphopenia; Male; Mice; Mice, Inbred C57BL; Mice, Inbred NOD; Mice, Knockout; Mice, SCID; Radiation Chimera; Receptors, GABA-B; Stem Cell Niche

2021