Page last updated: 2024-08-24

2-fluoroestradiol and 4-fluoroestradiol

2-fluoroestradiol has been researched along with 4-fluoroestradiol in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19904 (44.44)18.7374
1990's3 (33.33)18.2507
2000's0 (0.00)29.6817
2010's1 (11.11)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Heiman, DF; Katzenellenbogen, JA; Neeley, RJ; Senderoff, SG1
Cortés-Benítez, F; Dutour, R; Poirier, D; Roy, J1
Bulman-Page, PC; Hussain, F; Maggs, JL; Morgan, P; Park, BK1
Dey, SK; Johnson, DC; Liehr, JG; Pakrasi, PL1
Barnea, E; Krey, LC; Loriaux, DL; MacLusky, NJ; Merriam, GR; Naftolin, F; Pfeiffer, DG1
Krey, LC; Loriaux, DL; MacLusky, NJ; Merriam, GR; Naftolin, F; Parsons, B; Pfeiffer, DG1
Gilchrist, TL; Maggs, JL; Park, BK; Stalford, AC1
Ashburn, SP; Han, X; Liehr, JG1
Itoh, S; Jinno, H; Okamoto, Y; Shibutani, S1

Other Studies

9 other study(ies) available for 2-fluoroestradiol and 4-fluoroestradiol

ArticleYear
Estrogen receptor based imaging agents. 1. Synthesis and receptor binding affinity of some aromatic and D-ring halogenated estrogens.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:9

    Topics: Animals; Breast Neoplasms; Estradiol Congeners; Estrogens, Non-Steroidal; Female; In Vitro Techniques; Radionuclide Imaging; Receptors, Estrogen; Sheep; Structure-Activity Relationship; Uterus

1980
Targeting cytochrome P450 (CYP) 1B1 with steroid derivatives.
    Bioorganic & medicinal chemistry letters, 2016, 11-01, Volume: 26, Issue:21

    Topics: Cytochrome P-450 CYP1B1; Cytochrome P-450 Enzyme Inhibitors; Estrogens; Humans; Inhibitory Concentration 50; Molecular Docking Simulation; Structure-Activity Relationship

2016
The metabolism of 2- and 4-fluoro-17 beta-oestradiol in the rat and its implications for oestrogen carcinogenesis.
    Biochemical pharmacology, 1992, Mar-03, Volume: 43, Issue:5

    Topics: Animals; Bile; Biotransformation; Chromatography, High Pressure Liquid; Estradiol; Female; Glucuronates; Inactivation, Metabolic; Male; Mass Spectrometry; Rats; Rats, Inbred Strains

1992
Estrogens with reduced catechol-forming capacity fail to induce implantation in the rat.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1986, Volume: 181, Issue:2

    Topics: Animals; Embryo Implantation; Embryo Implantation, Delayed; Estradiol; Estrogens, Catechol; Female; Organ Size; Pregnancy; Rats; Uterus

1986
Are catechol oestrogens obligatory mediators of oestrogen action in the central nervous system? I. Characterization of pharmacological probes with different receptor binding affinities and catechol oestrogen formation rates.
    The Journal of endocrinology, 1986, Volume: 110, Issue:3

    Topics: Animals; Central Nervous System; Chromatography, High Pressure Liquid; Cytosol; Estradiol; Estrogens, Catechol; Ethinyl Estradiol; Female; Hydroxylation; Ovariectomy; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Estrogen

1986
Are catechol oestrogens obligatory mediators of oestrogen action in the central nervous system? II. Potencies of natural and synthetic oestrogens for induction of gonadotrophin release and female sexual behaviour in the rat.
    The Journal of endocrinology, 1986, Volume: 110, Issue:3

    Topics: Animals; Central Nervous System; Estradiol; Estrogens; Estrogens, Catechol; Ethinyl Estradiol; Female; Luteinizing Hormone; Ovariectomy; Progesterone; Rats; Rats, Inbred Strains; Sexual Behavior, Animal

1986
Catecholestrogens as mediators of carcinogenesis: correlation of aromatic hydroxylation of estradiol and its fluorinated analogs with tumor induction in Syrian hamsters.
    Molecular pharmacology, 1994, Volume: 45, Issue:6

    Topics: Animals; Bile; Carcinogens; Cricetinae; Estradiol; Estrogens, Catechol; Hydroxylation; Kidney Neoplasms; Male; Mesocricetus; Tritium

1994
Microsomal hydroxylation of 2- and 4-fluoroestradiol to catechol metabolites and their conversion to methyl ethers: catechol estrogens as possible mediators of hormonal carcinogenesis.
    Molecular pharmacology, 1993, Volume: 43, Issue:4

    Topics: Animals; Carcinogens; Catechol O-Methyltransferase; Cricetinae; DNA; Estradiol; Estrogens, Catechol; Hydroxylation; In Vitro Techniques; Kidney; Male; Mesocricetus; Methylation; Microsomes; Microsomes, Liver

1993
Carcinogenic potential of fluorinated estrogens in mammary tumorigenesis.
    Toxicology letters, 2020, Volume: 318

    Topics: Animals; Breast Neoplasms; Cell Transformation, Neoplastic; Estradiol; Female; Organ Size; Rats, Inbred ACI; Risk Assessment; Uterus

2020