2-chloroadenosine has been researched along with cv 1808 in 13 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (30.77) | 18.7374 |
1990's | 5 (38.46) | 18.2507 |
2000's | 3 (23.08) | 29.6817 |
2010's | 1 (7.69) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Jacobson, KA; van Galen, PJ; Williams, M | 1 |
Contardo, N; deJesus, R; Dotson, R; Francis, JE; Ghai, GR; Hutchison, AJ; Moskal, MA; Rovinski, SL; Webb, RL; Yokoyama, R | 1 |
Arroyo, LH; Olsson, RA; Thompson, RD; Ueeda, M | 1 |
Bruns, RF; Trivedi, BK | 1 |
Bristol, JA; Bruns, RF; Haleen, SJ; Steffen, RP; Trivedi, BK | 1 |
Arslan, G; Fredholm, BB; Kull, B; Lorenzen, A; Nilsson, C; Owman, C; Schwabe, U | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
de Lera Ruiz, M; Lim, YH; Zheng, J | 1 |
Barclay, BW; McNeal, RB; Webb, RL; Yasay, GD | 1 |
Franklin, PH; Murray, TF; Tripp, ED; Zhang, G | 1 |
Taylor, DA; Williams, M | 1 |
Carneiro, FS; Giachini, FR; Inscho, EW; Leite, R; Tostes, RC; Webb, RC | 1 |
2 review(s) available for 2-chloroadenosine and cv 1808
Article | Year |
---|---|
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship | 1992 |
Adenosine A2A receptor as a drug discovery target.
Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Crystallography, X-Ray; Drug Discovery; Humans; Ligands; Protein Conformation; Receptor, Adenosine A2A; Signal Transduction | 2014 |
11 other study(ies) available for 2-chloroadenosine and cv 1808
Article | Year |
---|---|
Highly selective adenosine A2 receptor agonists in a series of N-alkylated 2-aminoadenosines.
Topics: Adenosine; Alkylation; Animals; Antihypertensive Agents; Blood Pressure; Chemical Phenomena; Chemistry; Cyclohexanes; Heart Rate; Hypertension; Male; Molecular Structure; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Purinergic | 1991 |
2-Alkoxyadenosines: potent and selective agonists at the coronary artery A2 adenosine receptor.
Topics: Adenosine; Animals; Atrioventricular Node; Coronary Vessels; Guinea Pigs; Heart; In Vitro Techniques; Models, Molecular; Molecular Conformation; Molecular Structure; Muscle, Smooth, Vascular; Rats; Receptors, Purinergic; Structure-Activity Relationship | 1991 |
C2,N6-disubstituted adenosines: synthesis and structure-activity relationships.
Topics: Adenosine; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Rats; Receptors, Purinergic; Structure-Activity Relationship | 1989 |
N6-(arylalkyl)adenosines. Identification of N6-(9-fluorenylmethyl)adenosine as a highly potent agonist for the adenosine A2 receptor.
Topics: Adenosine; Animals; Brain; Cell Membrane; Coronary Circulation; Fluorenes; Heart Rate; In Vitro Techniques; Indicators and Reagents; Kinetics; Rats; Receptors, Purinergic; Structure-Activity Relationship | 1988 |
Differences in the order of potency for agonists but not antagonists at human and rat adenosine A2A receptors.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Humans; Kinetics; PC12 Cells; Phenethylamines; Polymerase Chain Reaction; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Recombinant Proteins; RNA, Messenger; Transcription, Genetic; Transfection; Triazoles; Tritium | 1999 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Hemodynamic effects of adenosine agonists in the conscious spontaneously hypertensive rat.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Heart Rate; Hydralazine; Injections, Intravenous; Male; Rats; Rats, Inbred SHR; Receptors, Purinergic; Renin; Vascular Resistance; Vasodilator Agents | 1990 |
Adenosine A1 receptor activation mediates suppression of (-) bicuculline methiodide-induced seizures in rat prepiriform cortex.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Autoradiography; Bicuculline; Cerebral Cortex; Dose-Response Relationship, Drug; Male; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Seizures | 1989 |
Interaction of 2-phenylaminoadenosine (CV 1808) with adenosine systems in rat tissues.
Topics: 2-Chloroadenosine; Adenosine; Animals; Dipyridamole; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Vas Deferens; Vasodilator Agents | 1982 |
Determination of adenosine effects and adenosine receptors in murine corpus cavernosum.
Topics: 2-Chloroadenosine; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Atropine; Bretylium Tosylate; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Penile Erection; Phenylephrine; Prazosin; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Pyrimidines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Triazoles | 2007 |